| DB01229 | Paclitaxel | approved, vet_approved | yes | inhibitor | Details |
| DB01248 | Docetaxel | approved, investigational | unknown | | Details |
| DB01367 | Rasagiline | approved | yes | activator | Details |
| DB05297 | Paclitaxel docosahexaenoic acid | investigational | unknown | | Details |
| DB08871 | Eribulin | approved, investigational | unknown | | Details |
| DB12340 | Navitoclax | investigational | yes | inhibitor | Details |
| DB06307 | Apoptone | investigational | unknown | | Details |
| DB12191 | Obatoclax | investigational | unknown | | Details |
| DB01050 | Ibuprofen | approved | unknown | modulator | Details |
| DB11581 | Venetoclax | approved, investigational | yes | antagonistinhibitor | Details |
| DB09213 | Dexibuprofen | approved, investigational | unknown | negative modulator | Details |
| DB12816 | Terpinen-4-ol | investigational | unknown | regulator | Details |
| DB05103 | AN-9 | investigational | yes | downregulator | Details |
| DB12843 | Oleandrin | experimental, investigational | unknown | downregulator | Details |