| DB00648 | Mitotane | approved | yes | inducer | Details |
| DB05667 | Levoketoconazole | approved, investigational | yes | inhibitor | Details |
| DB01011 | Metyrapone | approved, investigational | yes | inhibitor | Details |
| DB04630 | Aldosterone | experimental, investigational | unknown | substrate | Details |
| DB00501 | Cimetidine | approved, investigational | unknown | inhibitor | Details |
| DB00292 | Etomidate | approved | unknown | inhibitor | Details |
| DB00741 | Hydrocortisone | approved, vet_approved | unknown | substrate | Details |
| DB01026 | Ketoconazole | approved, investigational | unknown | inhibitor | Details |
| DB01011 | Metyrapone | approved, investigational | unknown | inhibitor | Details |
| DB01388 | Mibefradil | investigational, withdrawn | unknown | inhibitor | Details |
| DB01110 | Miconazole | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB00252 | Phenytoin | approved, vet_approved | no | inhibitor | Details |
| DB00421 | Spironolactone | approved | unknown | inducer | Details |
| DB14539 | Hydrocortisone acetate | approved, vet_approved | unknown | substrate | Details |
| DB14540 | Hydrocortisone butyrate | approved, vet_approved | unknown | substrate | Details |
| DB14543 | Hydrocortisone probutate | approved, vet_approved | unknown | substrate | Details |
| DB14544 | Hydrocortisone valerate | approved, vet_approved | unknown | substrate | Details |
| DB14545 | Hydrocortisone succinate | approved | no | substrate | Details |
| DB01234 | Dexamethasone | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB11837 | Osilodrostat | approved, investigational | yes | inhibitor | Details |
| DB14649 | Dexamethasone acetate | approved, investigational, vet_approved | unknown | inhibitor | Details |