Pharmaceutical Preparations

Name
Pharmaceutical Preparations
Accession Number
DBCAT000896
Description

Drugs intended for human or veterinary use, presented in their finished dosage form. Included here are materials used in the preparation and/or formulation of the finished dosage form.

Drugs
DrugDrug Description
Sodium tetradecyl sulfateAn anionic surfactant used to treat varicose veins of the lower extremities.
DimenhydrinateA medication used to prevent and treat nausea, vomiting, vertigo, and motion sickness.
TrimetrexateA folate antagonist used for the treatment of moderate-to-severe Pneumocystis carinii pneumonia (PCP) in immunocompromised patients as an alternative therapy in combination with leucovorin.
TetryzolineAn alpha-adrenergic agonist used in the temporary symptomatic relief of discomfort and redness of the eyes due to minor irritations, as well as alleviate nasal congestion.
Iron sucroseAn compound used as a source of iron in patients with iron deficiency anemia associated with chronic kidney disease (CKD).
Omega-3-acid ethyl estersA mixture of fatty acids used as an adjunct to diet to reduce triglyceride (TG) levels in adult patients with severe hypertriglyceridemia.
PetrolatumFor use as an over the counter skin protectant [FDA Label]. Commonly used to treat diaper rash and chapped lips [FDA Label] .
SennosidesA laxative used to treat constipation.
Ferrous sulfate anhydrousAn iron supplement used to prevent or treat iron deficiency anemia.
Ginkgo bilobaA herbal supplement found in over-the-counter or unapproved homeopathic products for various health conditions, such as cognitive, neurodegenerative, cardiovascular, and reproductive health disorders.
D-glucoseA most commonly occurring isomer of glucose used as a carbohydrate supplementation in case of nutrient deprivation and metabolic disorders, such as hypoglycemia.
FructoseNot Available
Polyethylene glycolA laxative used to treat constipation and used for bowel preparation before colonoscopies and other procedures.
LactitolAn orally administered osmotic laxative used to treat chronic idiopathic constipation.
Maritime pine extractA plant extract in nutritional supplements for healthy hair, skin, and nails.
Medical CannabisThe use of the plant species Cannabis sativa and Cannabis indica, popularly known as marijuana, has gained popularity in recent years for the management of a wide variety of medical...
Carboprost tromethamineA prostaglandin used to treat postpartum uterine hemorrhage due to atony when other methods of management have not been effective.
IrinotecanAn antineoplastic enzyme inhibitor used to treat metastatic carcinoma of the colon or rectum.
QuinidineA medication used to restore normal sinus rhythm, treat atrial fibrillation and flutter, and treat ventricular arrhythmias.
IbuprofenAn NSAID and non-selective COX inhibitor used to treat mild-moderate pain, fever, and inflammation.
AminophyllineA bronchodilator consisting of theophylline that is used for the treatment of bronchospasm due to asthma, emphysema and chronic bronchitis.
AlmitrineFor the treatment of chronic obstructive pulmonary disease.
EmbutramideNot Available
LiotrixMay be used to treat primary, secondary or tertiary hypothyroidism. May also be used to suppress thyroid stimulating hormone (TSH) secretion in patients with simple (nontoxic) goiter, subacute or chronic...
LucinactantIntended for the prevention of respiratory distress syndrome (RDS) in premature infants at high risk for RDS.
OMS-103HPInvestigated for use/treatment in inflammatory disorders (unspecified), knee replacement, orthopedic surgery, and pain (acute or chronic).
NOV-002Investigated for use/treatment in breast cancer, lung cancer, and ovarian cancer.
AviptadilNot Annotated
NorelgestrominA progestin used for the prevention of pregnancy in women who elect to use a transdermal patch as a method of contraception.
SpinosadA pediculicide used topically to treat head lice.
TAS-102TAS-102 (Taiho Pharma USA, Inc.) is an anti-cancer drug under development and in stage 3 clinical trials for the treatment of colorectal cancer. It is composed of the thymidine phosphorylase...
SacubitrilA neprilysin inhibitor used in combination with valsartan as an adjunct to reduce the risk of cardiovascular death and hospitalization for heart failure in patients with chronic heart failure (NYHA Class II-IV) and reduced ejection fraction.
FerumoxsilNot Annotated
GleptoferronColloid solution of ferric hydroxide, dextran & glucoheptonic acid.
BrexanoloneBrexanolone is a synthetic neuroactive steroid gamma-aminobutyric acid A (GABA(a)) receptor positive modulator indicated for the treatment of postpartum depression (PPD) in adult women [FDA Label][A176080, A176083, F4063, F4066, F4072].
ReproterolA short-acting β2 adrenoreceptor agonist used to treat various types of asthma including allergic asthma, non-allergic asthma, and exercise-induced asthma.
LevomenolLevomenol has been known to elicit a number of potentially beneficial pharmacological effects, including anti-irritant, anti-inflammatory, and anti-microbial actions. Bisabolol is also demonstrated to enhance the percutaneous absorption of certain...
PolicresulenNot Annotated
Choline salicylateThe oral gel is indicated for the relief of pain and discomfort of common mouth ulcers, cold sores, denture sore spots, infant teething and mouth ulcers, and sore spots due...
NabiximolsIn Canada, Sativex has received a Notice of Compliance (NOC) for use as an as adjunctive treatment for symptomatic relief of spasticity in patients with multiple sclerosis (MS) who have...
BromotheophyllineBromotheophylline is used as a diuretic and also, in combination with DB00316, it is used for the relief of temporary water weight gain, bloating, swelling and full feeling associated with...
Segesterone acetateSegesterone acetate in combination with ethinyl estradiol is indicated for use by females of reproductive potential to prevent pregnancy as a combination hormonal contraceptive (CHC). It induces contraception for thirteen...
Anti-SARS-CoV-2 REGN-COV2Anti-SARS-COV-2 REGN-COV2 is a combination of novel antibodies designed by Regeneron for both the prevention and treatment of SARS-COV-2, the virus that causes COVID-19. This drug is a combination of...
AZD7442AZD7442 is a combination of SARS-CoV-2 antibodies (AZD8895 + AZD1061) currently undergoing phase I clinical trials for the prevention and treatment of COVID-19. It was developed by AstraZeneca with the...
Lactobacillus acidophilusNot Annotated
PiroctonePiroctone olamine is used in combination with other substances as a part of shampoo effectively reduced the amount of dandruff and, at the same time, provided hair conditioning advantages. Recently...
MetadoxineA medication used to increase the clearance of alcohol in patients with chronic alcohol dependancy.
LatanoprostAn isopropyl ester prodrug used to treat increased intraocular pressure.
Amphotericin BAn antifungal used to treat fungal infections in neutropenic patients, cryptococcal meningitis in HIV infection, fungal infections, and leishmaniasis.
IcodextrinAn iso-osmotic solution used for continuous peritoneal dialysis or automated peritoneal dialysis.
ProbenecidA medication used to treat gouty arthritis, tophaceous gout, and hyperuricemia.
GatifloxacinA fourth generation fluoroquinolone used to treat a wide variety of infections in the body.
CarbetocinAn oxytocin agent used to control postpartum hemorrhage and bleeding after giving birth.
St. John's WortAn herbal ingredient used in non-prescription therapeutic products for the short-term treatment of minor skin irritations, insomnia, depression, and anxiety.
GinsengA herbal supplement used in many health products.
CamphorA compound used topically to help relieve pain and also as a topical antiseptic. May also be used in vaporizers to help suppress coughing. This medication should not be swallowed.
Propylene glycolA clear, colorless, viscous organic solvent and diluent used in pharmaceutical preparations.
Phenylethyl alcoholAn antimicrobial, antiseptic, and disinfectant that is used also as an aromatic essence and preservative in pharmaceutics and perfumery.
PhenolAn antiseptic and disinfectant used in a variety of settings.
TromethamineA proton acceptor used for the prevention and correction of metabolic acidosis associated with various clinical conditions, such as cardiac bypass surgery.
EucalyptolA common ingredient in mouthwash and cosmetics derived naturally from the eucalyptus plant that is frequently used to to improve symptoms of airway mucus hypersecretion.
Octylphenoxy polyethoxyethanolNot Available
BZL101Investigated for use/treatment in breast cancer.
Pradefovir mesylateInvestigated for use as a prodrug for Hepsera in treating hepatitis (viral, B).
LLL-3348Investigated for use/treatment in psoriasis and psoriatic disorders.
FerumoxytolAn intravenous iron replacement product used to treat iron deficiency anemia (IDA) in patients with chronic kidney disease (CKD), or in patients who are unable to tolerate or who have not responded adequately to oral iron supplementation.
Ethanolamine oleateA mild sclerosing agent used in the treatment of esophageal varices with recent bleeding episodes.
PolidocanolA sclerosing agent used for the treatment of uncomplicated spider veins and uncomplicated reticular veins, all less than 3 mm in diameter, in the lower extremity.
Methyl salicylateA topical counter-irritant used for the symptomatic relief of acute musculoskeletal pain in the muscles, joints, and tendons.
TragacanthAn extract from Tragacanth used in allergy testing.
CloveAn extract from Clove used in allergy testing.
PovidoneWhen in complex with iodine, indicated for inducing antisepsis for prevention of infection in minor cuts, scrapes, and burns.
Polysorbate 80It is used as a solubilizer, antimicrobial preservative and disinfectant .
BenzalkoniumAn antiseptic agent used as a preservative in medications or as a disinfectant in cleaning products.
Capsicum oleoresinA medication used to treat minor aches and pains of muscles and joints.
Silicon dioxideAn ingredient found in a variety of supplements and vitamins.
Polysorbate 20Polysorbate 20 is a polysorbate-type nonionic surfactant used in many commercial, household and pharmaceutical products. It is composed of 20 repeated units of polyethylene glycol via ethoxylation. Polysorbate 20 is...
Benzoin resinA compound used to protect small wounds or canker sores.
Poloxamer 407Poloxamer 407 is a polyoxyethylene polymer and hydrophilic non-ionic surfactant. It consists of a central hydrophobic block of polypropylene glycol that is flanked on each side by polyethylene glycol blocks,...
Poloxamer 188A medication used to clean wounds.
ChlorobutanolNo approved therapeutic indications on its own.
ThimerosalUsed as preservative in some cosmetics, topical pharmaceuticals, and biological drug products, which includes vaccines [L1671, L1672, L1673].
LifitegrastA medication used to treat dry eye disease.
TricaprylinTricaprilin has been used in trials studying the supportive care and treatment of Alzheimer's Disease.
NorfluraneNorflurane is under investigation in clinical trial NCT01673061 (Vapocoolant Spray for Numbing Small Boils Before Incision and Drainage).
Vitex agnus-castus fruit extractA herbal product used to treat an irregular menstrual period, premenstrual symptoms, and mastodynia
Horse chestnutA plant extract indicated in the treatment of venous insufficiency and other disorders caused by poor circulation.
ValerianA plant used in some non-prescription natural health products.
Black cohoshA herbal product indicated in the symptomatic treatment of menopause.
Morrhuic acidMorrhuic acid is a mixture of unsaturated fatty acids obtained from cod liver oil.
TriethylhexanoinTriethylhexanoin is an ingredient of cosmetic products as a fragrant solvent.
Microcrystalline celluloseA polysaccharide with glucose units linked as in CELLOBIOSE. It is the chief constituent of plant fibers, cotton being the purest natural form of the substance. As a raw material,...
PropylparabenPropylparaben is used in allergenic testing.
CinnamaldehydeCinnamaldehyde is approved by the FDA for use within allergenic epicutaneous patch tests which are indicated for use as an aid in the diagnosis of allergic contact dermatitis (ACD) in...
BromothalonilBromothalonil is approved for use within allergenic epicutaneous patch tests which are indicated for use as an aid in the diagnosis of allergic contact dermatitis (ACD) in persons 6 years...
MethylparabenMethylparaben is used in allergenic testing.
BilberryNot Annotated
Echinacea purpurea flowering topNot Annotated
Echinacea purpureaNot Annotated
Centella asiaticaCentella asiatica is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.
Calendula officinalis flowerCalendula officinalis flower is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.
RosemaryRosemary is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.
TurmericTurmeric is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.
Phellinus linteus myceliumPhellinus linteus mycelium is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.
Panax ginseng wholePanax ginseng whole is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.
Rehmannia glutinosa rootRehmannia glutinosa root is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.
Arnica montanaArnica montana is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.
EleutheroEleuthero is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.
Panax notoginseng rootPanax notoginseng root is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.
Tribulus terrestris fruitTribulus terrestris fruit is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.
Tangerine peelTangerine peel is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.
Chamaemelum nobile flowerChamaemelum nobile flower is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.
Nelumbo nucifera flowerNelumbo nucifera flower is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.
Angelica sinensis rootAngelica sinensis root is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.
Salvia miltiorrhiza rootSalvia miltiorrhiza root is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.
Prunus armeniaca seedPrunus armeniaca seed is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.
Arnica montana flowerArnica montana flower is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.
Forsythia suspensa fruitForsythia suspensa fruit is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.
Platycodon grandiflorus rootPlatycodon grandiflorus root is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.
ChamomileChamomile is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.
Saw palmettoSaw palmetto is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.
Scutellaria baicalensis rootScutellaria baicalensis root is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.
Milk thistleMilk thistle is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.
Sophora flavescens rootNot Annotated
Plantago ovata seedA plant extract indicated in the treatment of occasional constipation.
Sambucus nigra flowerNot Annotated
Willow barkNot Annotated
ClonazolamNot Annotated
Olea europaea leafNot Annotated
Polygala senega rootNot Annotated
Polyacrylamide (crosslinked; 2 mole percent bisacrylamide)Polyacrylamide (crosslinked; 2 mole percent bisacrylamide) is under investigation in clinical trial NCT00629083 (Bulking Agents for the Treatment of Stress Urinary Incontinence in Females).
Hydroxypropyl betadexHydroxypropyl betadex is under investigation in clinical trial NCT03471143 (Study of IV VTS-270 for Infantile Liver Disease Associated With Niemann-Pick Disease, Type C).
PradefovirPradefovir is a prodrug of adefovir.
Anise oilNot Annotated
Hawthorn leaf with flowerNot Annotated
AnetholeAn excipient added to medications for flavouring.
AcrizanibAcrizanib is under investigation in clinical trial NCT02355028 (LHA510 Proof-of-concept Study as a Maintenance Therapy for Patients With Wet Age-related Macular Degeneration).
Gentiana lutea extractA medication used to treat bloating and gas.
Pygeum africanum barkA plant extract indicated in the symptomatic treatment of prostatic hypertrophy.
Paeonia lactiflora rootNot Annotated
Vitis vinifera seedNot Annotated
Gastrodia elata wholeNot Annotated
Juniper tarNot Annotated
Drugs & Drug Targets
DrugTargetType
Sodium tetradecyl sulfateVitamin K-dependent protein Ctarget
Sodium tetradecyl sulfateVitamin K-dependent protein Starget
DimenhydrinateHistamine H1 receptortarget
TrimetrexateDihydrofolate reductasetarget
TrimetrexateFolate transporter 1transporter
TetryzolineAlpha-1 adrenergic receptorstarget
TetryzolineAlpha-2 adrenergic receptorstarget
Omega-3-acid ethyl estersSterol O-acyltransferase 1enzyme
Omega-3-acid ethyl estersSterol regulatory element-binding protein 1target
SennosidesReverse transcriptase/RNaseHtarget
SennosidesAquaporin-3target
Ferrous sulfate anhydrousNatural resistance-associated macrophage protein 2transporter
Ferrous sulfate anhydrousCeruloplasminenzyme
Ferrous sulfate anhydrousHemoglobin subunit alphatarget
Ferrous sulfate anhydrousTransferrin receptortarget
Ferrous sulfate anhydrousSolute carrier family 40 member 1transporter
Ferrous sulfate anhydrousHepcidinenzyme
Ferrous sulfate anhydrousSerotransferrinenzyme
Ferrous sulfate anhydrousHephaestinenzyme
Ferrous sulfate anhydrousCytochrome b reductase 1enzyme
Ginkgo bilobaCytochrome P450 2C9enzyme
Ginkgo bilobaPhospholipase A2, membrane associatedtarget
Ginkgo bilobaSodium-dependent noradrenaline transportertarget
Ginkgo bilobaGlycine receptor subunit alpha-1target
Ginkgo bilobaGamma-aminobutyric acid receptor subunit alpha-1target
Ginkgo bilobaGamma-aminobutyric acid receptor subunit beta-2target
Ginkgo bilobaGamma-aminobutyric acid receptor subunit gamma-2target
Ginkgo bilobaCytochrome P450 3A4enzyme
Ginkgo bilobaAmine oxidase [flavin-containing] Atarget
Ginkgo bilobaNitric oxide synthase, inducibletarget
Ginkgo bilobaCytochrome P450 1B1enzyme
Ginkgo bilobaCytochrome P450 1A1enzyme
Ginkgo bilobaCytochrome P450 1A2enzyme
D-glucoseHexokinase-1enzyme
D-glucoseGlucokinaseenzyme
D-glucoseSolute carrier family 2, facilitated glucose transporter member 1transporter
D-glucoseSolute carrier family 2, facilitated glucose transporter member 2transporter
D-glucoseSolute carrier family 2, facilitated glucose transporter member 3transporter
D-glucoseSolute carrier family 2, facilitated glucose transporter member 4transporter
D-glucoseSolute carrier family 2, facilitated glucose transporter member 5transporter
D-glucoseSolute carrier family 2, facilitated glucose transporter member 6transporter
D-glucoseSolute carrier family 2, facilitated glucose transporter member 7transporter
D-glucoseSolute carrier family 2, facilitated glucose transporter member 8transporter
D-glucoseSolute carrier family 2, facilitated glucose transporter member 9transporter
D-glucoseSolute carrier family 2, facilitated glucose transporter member 10transporter
D-glucoseSolute carrier family 2, facilitated glucose transporter member 11transporter
D-glucoseSolute carrier family 2, facilitated glucose transporter member 12transporter
D-glucoseSodium/glucose cotransporter 1transporter
D-glucoseSodium/glucose cotransporter 2transporter
D-glucoseSerum albumincarrier
FructoseMaltoporintarget
Polyethylene glycolP-glycoprotein 1transporter
Medical CannabisCannabinoid receptor 1target
Medical CannabisCannabinoid receptor 2target
Medical CannabisCytochrome P450 2C9enzyme
Medical CannabisCytochrome P450 2C19enzyme
Medical CannabisCytochrome P450 2D6enzyme
Medical CannabisCytochrome P450 3A4enzyme
Medical CannabisG-protein coupled receptor 12target
Medical CannabisGlycine receptor subunit alpha-1target
Medical CannabisGlycine receptor (alpha-1/beta)target
Medical CannabisGlycine receptor subunit alpha-3target
Medical CannabisN-arachidonyl glycine receptortarget
Medical CannabisG-protein coupled receptor 55target
Medical Cannabis5-hydroxytryptamine receptor 1Atarget
Medical Cannabis5-hydroxytryptamine receptor 2Atarget
Medical CannabisNeuronal acetylcholine receptor subunit alpha-7target
Medical CannabisDelta-type opioid receptortarget
Medical CannabisMu-type opioid receptortarget
Medical CannabisPeroxisome proliferator-activated receptor gammatarget
Medical CannabisCytochrome P450 3A5enzyme
Medical CannabisCytochrome P450 3A7enzyme
Medical CannabisCytochrome P450 1A1enzyme
Medical CannabisCytochrome P450 1A2enzyme
Medical CannabisCytochrome P450 1B1enzyme
Medical CannabisArachidonate 5-lipoxygenaseenzyme
Medical CannabisArachidonate 15-lipoxygenaseenzyme
Medical CannabisSuperoxide dismutase [Cu-Zn]enzyme
Medical CannabisMultidrug resistance-associated protein 1transporter
Medical CannabisATP-binding cassette sub-family G member 2transporter
Medical CannabisEquilibrative nucleoside transporter 1transporter
Medical CannabisTransient receptor potential cation channel subfamily V member 1target
Medical CannabisVoltage-dependent T-type calcium channel subunit alpha-1Gtarget
Medical CannabisVoltage-dependent T-type calcium channel subunit alpha-1Htarget
Medical CannabisVoltage-dependent T-type calcium channel subunit alpha-1Itarget
Medical CannabisTransient receptor potential cation channel subfamily A member 1target
Medical CannabisTransient receptor potential cation channel subfamily M member 8target
Medical CannabisTransient receptor potential cation channel subfamily V member 2target
Medical CannabisTransient receptor potential cation channel subfamily V member 3target
Medical CannabisTransient receptor potential cation channel subfamily V member 4target
Medical CannabisVoltage-dependent anion-selective channel protein 1target
Medical CannabisN-acyl-phosphatidylethanolamine-hydrolyzing phospholipase Dtarget
Medical CannabisN-acylethanolamine-hydrolyzing acid amidasetarget
Medical CannabisArylalkylamine N-acetyltransferasetarget
Medical CannabisPhospholipase A2target
Medical CannabisSuperoxide dismutase [Cu-Zn]target
Medical CannabisFatty-acid amide hydrolase 1target
Medical CannabisCatalasetarget
Medical CannabisQuinone oxidoreductasetarget
Medical CannabisSphingomyelin phosphodiesterasetarget
Medical CannabisGlutathione peroxidase 1target
Medical CannabisGlutathione reductase, mitochondrialtarget
Medical Cannabis3-hydroxy-3-methylglutaryl-coenzyme A reductasetarget
Medical CannabisIndoleamine 2,3-dioxygenase 1target
Medical CannabisProstaglandin G/H synthase 1target
Medical CannabisProstaglandin G/H synthase 2target
Medical CannabisSteroid 17-alpha-hydroxylase/17,20 lyasetarget
Medical CannabisAcetyl-CoA acetyltransferase, mitochondrialtarget
Medical CannabisCytochrome P450 2A6enzyme
Medical CannabisCytochrome P450 2B6enzyme
Medical CannabisCytochrome P450 2C8enzyme
Medical CannabisCytochrome P450 2E1enzyme
Medical CannabisCytochrome P450 2J2enzyme
Medical CannabisUDP-glucuronosyltransferase 1-7enzyme
Medical CannabisUDP-glucuronosyltransferase 1-8enzyme
Medical CannabisUDP-glucuronosyltransferase 1-9enzyme
Medical CannabisUDP-glucuronosyltransferase 1-10enzyme
Medical CannabisUDP-glucuronosyltransferase 2B17enzyme
Medical CannabisLiver carboxylesterase 1enzyme
Medical CannabisP-glycoprotein 1transporter
Medical CannabisUDP-glucuronosyltransferase 2B7enzyme
Carboprost tromethamineProstaglandin E2 receptor EP1 subtypetarget
IrinotecanDNA topoisomerase I, mitochondrialtarget
IrinotecanDNA topoisomerase 1target
IrinotecanCytochrome P450 3A4enzyme
IrinotecanCytochrome P450 3A5enzyme
IrinotecanUDP-glucuronosyltransferase 1-1enzyme
IrinotecanUDP-glucuronosyltransferase 1-9enzyme
IrinotecanLiver carboxylesterase 1enzyme
IrinotecanCytochrome P450 3A7enzyme
IrinotecanCytochrome P450 2B6enzyme
IrinotecanSolute carrier family 22 member 3transporter
IrinotecanSolute carrier organic anion transporter family member 1B1transporter
IrinotecanMultidrug resistance-associated protein 1transporter
IrinotecanATP-binding cassette sub-family G member 2transporter
IrinotecanSerum albumincarrier
IrinotecanCocaine esteraseenzyme
IrinotecanCholinesteraseenzyme
IrinotecanP-glycoprotein 1transporter
IrinotecanCanalicular multispecific organic anion transporter 1transporter
QuinidineSodium channel protein type 5 subunit alphatarget
QuinidineAlpha-1-acid glycoprotein 1carrier
QuinidinePotassium voltage-gated channel subfamily H member 2target
QuinidinePotassium channel subfamily K member 1target
QuinidinePotassium channel subfamily K member 6target
QuinidineCytochrome P450 1A2enzyme
QuinidineCytochrome P450 2E1enzyme
QuinidineCytochrome P450 1A1enzyme
QuinidineCytochrome P450 2D6enzyme
QuinidineCytochrome P450 3A4enzyme
QuinidineCytochrome P450 3A7enzyme
QuinidineSolute carrier family 22 member 2transporter
QuinidineSolute carrier family 22 member 1transporter
QuinidineSolute carrier family 22 member 5transporter
QuinidineP-glycoprotein 1transporter
QuinidineSolute carrier organic anion transporter family member 1A2transporter
QuinidineSolute carrier family 22 member 8transporter
QuinidineCanalicular multispecific organic anion transporter 1transporter
QuinidineSolute carrier family 22 member 4transporter
QuinidineSolute carrier organic anion transporter family member 1B1transporter
QuinidineCytochrome P450 2B6enzyme
QuinidineCytochrome P450 2C9enzyme
QuinidineAlpha-1A adrenergic receptortarget
QuinidineAlpha-1B adrenergic receptortarget
QuinidineAlpha-1D adrenergic receptortarget
QuinidineBile salt export pumptransporter
QuinidineCytochrome P450 2C8enzyme
QuinidineSerum albumincarrier
IbuprofenProstaglandin G/H synthase 1target
IbuprofenProstaglandin G/H synthase 2target
IbuprofenCytochrome P450 2C9enzyme
IbuprofenSerum albumincarrier
IbuprofenMultidrug resistance-associated protein 4transporter
IbuprofenMultidrug resistance-associated protein 1transporter
IbuprofenSolute carrier organic anion transporter family member 1A2transporter
IbuprofenSolute carrier family 22 member 6transporter
IbuprofenSolute carrier family 22 member 8transporter
IbuprofenSolute carrier family 22 member 11transporter
IbuprofenSolute carrier organic anion transporter family member 2B1transporter
IbuprofenP-glycoprotein 1transporter
IbuprofenUDP-glucuronosyltransferase 1-3enzyme
IbuprofenUDP-glucuronosyltransferase 1-9enzyme
IbuprofenUDP-glucuronosyltransferase 2B4enzyme
IbuprofenUDP-glucuronosyltransferase 2B7enzyme
IbuprofenCytochrome P450 2C8enzyme
IbuprofenCytochrome P450 2C19enzyme
IbuprofenApoptosis regulator Bcl-2target
IbuprofenThrombomodulintarget
IbuprofenFatty acid-binding protein, intestinaltarget
IbuprofenPeroxisome proliferator-activated receptor gammatarget
IbuprofenCystic fibrosis transmembrane conductance regulatortarget
IbuprofenPeroxisome proliferator-activated receptor alphatarget
IbuprofenPlatelet glycoprotein Ib alpha chaintarget
IbuprofenProtein S100-A7target
IbuprofenAlpha-methylacyl-CoA racemaseenzyme
IbuprofenCytochrome P450 3A4enzyme
AminophyllinecGMP-inhibited 3',5'-cyclic phosphodiesterase Atarget
AminophyllineAdenosine receptor A3target
AminophyllineAdenosine receptor A1target
AminophyllineCytochrome P450 1A2enzyme
AminophyllineCytochrome P450 2E1enzyme
AminophyllineCytochrome P450 3A4enzyme
AminophyllineHistone deacetylase 2target
AlmitrineSodium/potassium-transporting ATPase subunit alpha-1target
LiotrixThyroid hormone receptor alphatarget
LiotrixThyroid hormone receptor betatarget
LiotrixCytochrome P450 2C8enzyme
LiotrixSolute carrier organic anion transporter family member 1A2transporter
LiotrixSolute carrier organic anion transporter family member 1B1transporter
LiotrixSolute carrier organic anion transporter family member 1B3transporter
LiotrixSolute carrier organic anion transporter family member 4C1transporter
LiotrixSodium/bile acid cotransportertransporter
LiotrixSolute carrier organic anion transporter family member 1C1transporter
LiotrixSolute carrier organic anion transporter family member 4A1transporter
LiotrixSolute carrier family 22 member 8transporter
LiotrixMonocarboxylate transporter 8transporter
LiotrixMonocarboxylate transporter 10transporter
LiotrixP-glycoprotein 1transporter
LiotrixTransthyretincarrier
LiotrixThyroxine-binding globulincarrier
LiotrixSerum albumincarrier
LiotrixCytochrome P450 3A4enzyme
OMS-103HPTumor necrosis factortarget
OMS-103HPInterleukin-1 receptor type 1target
NorelgestrominSteryl-sulfataseenzyme
NorelgestrominProgesterone receptortarget
NorelgestrominSerum albumintarget
NorelgestrominAndrogen receptortarget
NorelgestrominCytochrome P450 3A4enzyme
SacubitrilNeprilysintarget
SacubitrilSolute carrier organic anion transporter family member 1B1transporter
SacubitrilSolute carrier organic anion transporter family member 1B3transporter
BrexanoloneGABA(A) Receptortarget
BrexanoloneAldose reductaseenzyme
LevomenolSolute carrier organic anion transporter family member 1B1transporter
LevomenolSolute carrier organic anion transporter family member 1B3transporter
Choline salicylateCholine-phosphate cytidylyltransferase Btarget
Choline salicylateAcetylcholinesterasetarget
Choline salicylateCholine-phosphate cytidylyltransferase Atarget
Choline salicylatePhospholipase D2target
Choline salicylateCholinesterasetarget
Choline salicylatePhospholipase D1target
Choline salicylateSolute carrier family 22 member 2transporter
Choline salicylateSolute carrier family 22 member 1transporter
Choline salicylateSolute carrier family 22 member 3transporter
Choline salicylateSolute carrier family 22 member 5transporter
Choline salicylateSolute carrier family 22 member 4transporter
Choline salicylateCholine/ethanolaminephosphotransferase 1enzyme
Choline salicylateCholine transporter-like protein 1transporter
Choline salicylateCholine transporter-like protein 4transporter
Choline salicylateCholine transporter-like protein 3transporter
Choline salicylateCholine/ethanolamine kinaseenzyme
Choline salicylateCholine O-acetyltransferaseenzyme
Choline salicylateCholine kinase alphaenzyme
Choline salicylateCholine dehydrogenase, mitochondrialenzyme
Choline salicylateHigh affinity choline transporter 1transporter
Choline salicylateNeuronal acetylcholine receptor subunit alpha-7target
NabiximolsCannabinoid receptor 1target
NabiximolsCannabinoid receptor 2target
NabiximolsG-protein coupled receptor 12target
NabiximolsCytochrome P450 2C9enzyme
NabiximolsCytochrome P450 2C19enzyme
NabiximolsCytochrome P450 2D6enzyme
NabiximolsCytochrome P450 3A4enzyme
NabiximolsGlycine receptor subunit alpha-1target
NabiximolsGlycine receptor (alpha-1/beta)target
NabiximolsGlycine receptor subunit alpha-3target
NabiximolsN-arachidonyl glycine receptortarget
NabiximolsG-protein coupled receptor 55target
Nabiximols5-hydroxytryptamine receptor 1Atarget
Nabiximols5-hydroxytryptamine receptor 2Atarget
NabiximolsNeuronal acetylcholine receptor subunit alpha-7target
NabiximolsDelta-type opioid receptortarget
NabiximolsMu-type opioid receptortarget
NabiximolsPeroxisome proliferator-activated receptor gammatarget
NabiximolsCytochrome P450 3A5enzyme
NabiximolsArachidonate 5-lipoxygenaseenzyme
NabiximolsArachidonate 15-lipoxygenaseenzyme
NabiximolsMultidrug resistance-associated protein 1transporter
NabiximolsATP-binding cassette sub-family G member 2transporter
NabiximolsEquilibrative nucleoside transporter 1transporter
NabiximolsTransient receptor potential cation channel subfamily V member 1target
NabiximolsVoltage-dependent T-type calcium channel subunit alpha-1Gtarget
NabiximolsVoltage-dependent T-type calcium channel subunit alpha-1Htarget
NabiximolsVoltage-dependent T-type calcium channel subunit alpha-1Itarget
NabiximolsTransient receptor potential cation channel subfamily A member 1target
NabiximolsTransient receptor potential cation channel subfamily M member 8target
NabiximolsTransient receptor potential cation channel subfamily V member 2target
NabiximolsTransient receptor potential cation channel subfamily V member 3target
NabiximolsTransient receptor potential cation channel subfamily V member 4target
NabiximolsVoltage-dependent anion-selective channel protein 1target
NabiximolsProstaglandin G/H synthase 1target
NabiximolsProstaglandin G/H synthase 2target
NabiximolsAcetyl-CoA acetyltransferase, mitochondrialtarget
NabiximolsSteroid 17-alpha-hydroxylase/17,20 lyasetarget
Nabiximols3-hydroxy-3-methylglutaryl-coenzyme A reductasetarget
NabiximolsGlutathione reductase, mitochondrialtarget
NabiximolsGlutathione peroxidase 1target
NabiximolsIndoleamine 2,3-dioxygenase 1target
NabiximolsArylalkylamine N-acetyltransferasetarget
NabiximolsCytochrome P450 1B1target
NabiximolsCytochrome P450 3A5target
NabiximolsCytochrome P450 2D6target
NabiximolsCytochrome P450 1A2target
NabiximolsCytochrome P450 1A1target
NabiximolsCytochrome P450 3A7target
NabiximolsQuinone oxidoreductasetarget
NabiximolsCatalasetarget
NabiximolsFatty-acid amide hydrolase 1target
NabiximolsSuperoxide dismutase [Cu-Zn]target
NabiximolsN-acylethanolamine-hydrolyzing acid amidasetarget
BromotheophyllineCytochrome P450 1A2enzyme
Segesterone acetateGlucocorticoid receptortarget
Segesterone acetateProgesterone receptortarget
Segesterone acetateAndrogen receptortarget
Segesterone acetateCytochrome P450 3A4enzyme
Anti-SARS-CoV-2 REGN-COV2Spike glycoproteintarget
LatanoprostProstaglandin F2-alpha receptortarget
LatanoprostSolute carrier organic anion transporter family member 2A1transporter
LatanoprostSolute carrier family 22 member 6transporter
LatanoprostSolute carrier family 22 member 8transporter
LatanoprostCorneal esterasesenzyme
Amphotericin BErgosteroltarget
IcodextrinPancreatic alpha-amylaseenzyme
ProbenecidSolute carrier family 22 member 8target
ProbenecidSolute carrier family 22 member 11target
ProbenecidSerum albumincarrier
ProbenecidSolute carrier family 22 member 2transporter
ProbenecidSolute carrier family 22 member 1transporter
ProbenecidCanalicular multispecific organic anion transporter 2transporter
ProbenecidMultidrug resistance-associated protein 4transporter
ProbenecidMultidrug resistance-associated protein 5transporter
ProbenecidMonocarboxylate transporter 2transporter
ProbenecidSolute carrier family 22 member 5transporter
ProbenecidMultidrug resistance-associated protein 6transporter
ProbenecidMultidrug resistance-associated protein 1transporter
ProbenecidSolute carrier organic anion transporter family member 1A2transporter
ProbenecidMonocarboxylate transporter 1transporter
ProbenecidSodium/bile acid cotransportertransporter
ProbenecidSolute carrier family 22 member 6transporter
ProbenecidSolute carrier family 22 member 10transporter
ProbenecidSolute carrier family 22 member 8transporter
ProbenecidCanalicular multispecific organic anion transporter 1transporter
ProbenecidATP-binding cassette sub-family C member 11transporter
ProbenecidSolute carrier family 22 member 11transporter
ProbenecidSolute carrier organic anion transporter family member 1C1transporter
ProbenecidSolute carrier family 22 member 7transporter
ProbenecidSolute carrier family 22 member 6target
ProbenecidPannexin-1target
ProbenecidCytochrome P450 2C8enzyme
ProbenecidCytochrome P450 3A4enzyme
ProbenecidSolute carrier family 22 member 12transporter
ProbenecidSolute carrier family 2, facilitated glucose transporter member 9transporter
ProbenecidTaste receptor type 2 member 16target
ProbenecidUDP-glucuronosyltransferase 1-1enzyme
ProbenecidCytochrome P450 2C9enzyme
GatifloxacinSerum albumincarrier
GatifloxacinDNA gyrase subunit Atarget
GatifloxacinDNA gyrase subunit Btarget
GatifloxacinDNA topoisomerase 4 subunit Atarget
GatifloxacinDNA topoisomerase 4 subunit Btarget
GatifloxacinCytochrome P450 1A2enzyme
CarbetocinOxytocin receptortarget
St. John's WortP-glycoprotein 1transporter
St. John's WortCytochrome P450 3A4enzyme
St. John's WortCytochrome P450 2D6enzyme
St. John's WortCytochrome P450 2C19enzyme
GinsengInterleukin-6target
GinsengProstaglandin G/H synthase 2target
GinsengAryl hydrocarbon receptortarget
CamphorCamphor 5-monooxygenasetarget
CamphorTransient receptor potential cation channel subfamily V member 1target
CamphorTransient receptor potential cation channel subfamily V member 3target
CamphorTransient receptor potential cation channel subfamily A member 1target
CamphorTransient receptor potential cation channel subfamily M member 8target
Propylene glycolB12-independent glycerol dehydratasetarget
Phenylethyl alcoholParathion hydrolasetarget
PhenolThermolysintarget
PhenolSerum albumintarget
TromethamineAmyloid beta A4 proteintarget
Octylphenoxy polyethoxyethanolTroponin C, skeletal muscletarget
Pradefovir mesylateCytochrome P450 3A4target
LLL-3348Interleukin-10target
FerumoxytolSerotransferrincarrier
Ethanolamine oleateCalcium ionstarget
Ethanolamine oleateCoagulation factor XIItarget
Capsicum oleoresinTransient receptor potential cation channel subfamily V member 1target
Silicon dioxideMacrophage receptor MARCOtarget
ChlorobutanolPotassium voltage-gated channel subfamily H member 2target
ThimerosalSerum albumincarrier
ThimerosalInositol 1,4,5-trisphosphate receptor type 1transporter
ThimerosalMethionine synthasetarget
ThimerosalCystine/glutamate transportertarget
ThimerosalSodium/potassium-transporting ATPase subunit gammatarget
ThimerosalGlutathione reductase, mitochondrialenzyme
ThimerosalGlutathione peroxidase 1enzyme
ThimerosalSuperoxide dismutase [Mn], mitochondrialenzyme
LifitegrastIntegrin alpha-Ltarget
LifitegrastCytochrome P450 2C9enzyme
LifitegrastSolute carrier organic anion transporter family member 1A2transporter
LifitegrastSolute carrier organic anion transporter family member 2B1transporter
Black cohoshCytochrome P450 3A4enzyme
Black cohoshCytochrome P450 3A2enzyme
Black cohoshCytochrome P450 1A2enzyme
Black cohoshCytochrome P450 2C9enzyme
Black cohoshCytochrome P450 2D6enzyme