Nucleoside Reverse Transcriptase Inhibitors

Name
Nucleoside Reverse Transcriptase Inhibitors
Accession Number
DBCAT002755  (DBCAT001086)
Description

Not Available

Drugs
DrugDrug Description
AbacavirAn antiviral nucleoside reverse transcriptase inhibitor used in combination with other antiretrovirals for the treatment of HIV.
AdefovirNot Annotated
DexelvucitabineDexelvucitabine has been used in trials studying the treatment of HIV Infections and Human Immunodeficiency Virus.
DidanosineA reverse transcriptase inhibitor used to treat HIV.
ElvucitabineInvestigated for use/treatment in hepatitis (viral, B) and HIV infection.
EmtricitabineA nucleoside reverse transcriptase inhibitor used for the treatment and prophylaxis of HIV.
EntecavirA nucleoside analogue used in the treatment of chronic hepatitis B for patients with active viral replication, histological evidence of active disease, or persistent elevations in liver transaminases.
LamivudineA reverse transcriptase inhibitor used to treat HIV and hepatitis B infections.
StavudineA dideoxynucleoside used in the treatment of HIV infection.
TelbivudineA thymidine nucleoside analog used for the treatment of chronic hepatitis B with clinical evidence of viral replication or persistent elevations in serum aminotransferases (ALT or AST).
TenofovirA nucleotide analog indicated in the treatment of HIV infections.
ZalcitabineA dideoxynucleoside used to treat HIV.
ZidovudineA dideoxynucleoside used in the treatment of HIV infection.
Drugs & Drug Targets
DrugTargetType
AbacavirGag-Pol polyproteintarget
AbacavirAdenosine kinaseenzyme
AbacavirReverse transcriptase/RNaseHtarget
AbacavirUDP-glucuronosyltransferase 1A1enzyme
AbacavirAlcohol dehydrogenase 6enzyme
AdefovirDNA polymerase catalytic subunittarget
AdefovirProtein Ptarget
DexelvucitabineReverse transcriptase/RNaseHtarget
DidanosineGag-Pol polyproteintarget
DidanosineAlbumincarrier
DidanosineEquilibrative nucleoside transporter 2transporter
DidanosineEquilibrative nucleoside transporter 1transporter
DidanosineReverse transcriptase/RNaseHtarget
DidanosinePurine nucleoside phosphorylasetarget
DidanosineSolute carrier family 22 member 6transporter
ElvucitabineGag-Pol polyproteintarget
ElvucitabineReverse transcriptase/RNaseHtarget
EmtricitabineGag-Pol polyproteintarget
EmtricitabineMultidrug and toxin extrusion protein 1transporter
EmtricitabineAlbumincarrier
EmtricitabineDeoxycytidine kinaseenzyme
EmtricitabineReverse transcriptase/RNaseHtarget
EntecavirReverse transcriptasetarget
LamivudineSolute carrier family 22 member 1transporter
LamivudineATP-binding cassette sub-family C member 3transporter
LamivudineGag-Pol polyproteintarget
LamivudineAlbumincarrier
Lamivudine5'(3')-deoxyribonucleotidase, cytosolic typeenzyme
LamivudineATP-binding cassette sub-family C member 2transporter
LamivudineATP-binding cassette sub-family C member 4transporter
LamivudineATP-dependent translocase ABCB1transporter
LamivudineEthanolamine-phosphate cytidylyltransferaseenzyme
LamivudineCholine-phosphate cytidylyltransferase Aenzyme
LamivudineNucleoside diphosphate kinase Benzyme
LamivudineNucleoside diphosphate kinase Aenzyme
LamivudinePhosphoglycerate kinase 1enzyme
LamivudineUMP-CMP kinaseenzyme
LamivudineDeoxycytidine kinaseenzyme
LamivudineSolute carrier family 22 member 3transporter
LamivudineSolute carrier family 22 member 2transporter
LamivudineReverse transcriptase/RNaseHtarget
LamivudineBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
LamivudineDNAtarget
LamivudineProtein Ptarget
LamivudineMultidrug resistance-associated protein 1transporter
LamivudineSolute carrier family 22 member 6transporter
StavudineGag-Pol polyproteintarget
StavudineAlbumincarrier
StavudineSodium/nucleoside cotransporter 1transporter
StavudineReverse transcriptase/RNaseHtarget
StavudineSolute carrier family 22 member 6transporter
TelbivudineDNAtarget
TelbivudineProtein Ptarget
TenofovirReverse transcriptase/RNaseHtarget
TenofovirAdenylate kinase 2, mitochondrialenzyme
TenofovirReverse transcriptasetarget
TenofovirDNA polymerasetarget
TenofovirAlbumincarrier
TenofovirGag-Pol polyproteintarget
TenofovirAdenylate kinase isoenzyme 1enzyme
TenofovirNucleoside diphosphate kinase Benzyme
TenofovirNucleoside diphosphate kinase Aenzyme
TenofovirATP-binding cassette sub-family C member 4transporter
TenofovirOrganic anion transporter 3transporter
TenofovirSolute carrier family 22 member 6transporter
TenofovirATP-dependent translocase ABCB1transporter
ZalcitabineGag-Pol polyproteintarget
ZalcitabineAlbumincarrier
ZalcitabineEquilibrative nucleoside transporter 2transporter
ZalcitabineEquilibrative nucleoside transporter 1transporter
ZalcitabineReverse transcriptase/RNaseHtarget
ZalcitabineSolute carrier family 22 member 7transporter
ZalcitabineSolute carrier family 22 member 6transporter
ZalcitabineDeoxycytidine kinaseenzyme
ZidovudineSolute carrier family 22 member 6transporter
ZidovudineSolute carrier family 22 member 2transporter
ZidovudineSolute carrier family 22 member 7transporter
ZidovudineOrganic anion transporter 3transporter
ZidovudineReverse transcriptase/RNaseHtarget
ZidovudineCytochrome P450 3A4enzyme
ZidovudineSolute carrier family 22 member 11transporter
ZidovudineSodium/nucleoside cotransporter 1transporter
ZidovudineEquilibrative nucleoside transporter 2transporter
ZidovudineATP-dependent translocase ABCB1transporter
ZidovudineATP-binding cassette sub-family C member 4transporter
ZidovudineATP-binding cassette sub-family C member 5transporter
ZidovudineBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
ZidovudineGag-Pol polyproteintarget
ZidovudineReceptor-type tyrosine-protein kinase FLT3target
ZidovudineTelomerase reverse transcriptasetarget
ZidovudineThymidine kinase, cytosolicenzyme
ZidovudineUDP-glucuronosyltransferase 2B7enzyme
ZidovudineUDP-glucuronosyltransferase 1A1enzyme
ZidovudineCytochrome P450 2C9enzyme
ZidovudineCytochrome P450 2A6enzyme
ZidovudineAlbumincarrier