Tumor Necrosis Factor Blockers

Name
Tumor Necrosis Factor Blockers
Accession Number
DBCAT003245  (DBCAT001648, DBCAT002087)
Description

Compounds or agents that bind to and inhibit the synthesis or activity of TUMOR NECROSIS FACTOR-alpha. Such agents are used to treat inflammatory bowel diseases and other inflammatory diseases.

Drugs
DrugDrug Description
(2R)-N-HYDROXY-2-[(3S)-3-METHYL-3-{4-[(2-METHYLQUINOLIN-4-YL)METHOXY]PHENYL}-2-OXOPYRROLIDIN-1-YL]PROPANAMIDENot Available
AdalimumabA monoclonal anti-tumor necrosis factor alpha antibody used in the treatment of a wide variety of inflammatory conditions such as rheumatoid arthritis, Crohn's disease, and ankylosing spondylitis.
AfelimomabInvestigated for use/treatment in sepsis and septicemia.
AmrinoneA positive inotropic agent and phosphodiesterase inhibitor used in the management of treatment of congestive heart failure.
AN0128Investigated for use/treatment in acne, atopic dermatitis, pediatric indications, and psoriasis and psoriatic disorders.
AstegolimabAstegolimab is under investigation in clinical trial NCT04386616 (A Study to Evaluate the Safety and Efficacy of MSTT1041A (Astegolimab) or UTTR1147A in Patients With Severe COVID-19 Pneumonia).
AtaciceptA TACI-Fc fusion protein and dual BAFF/APRIL inhibitor indicated to reduce proteinuria in adults with primary IgA nephropathy at risk for progression.
BaicaleinBaicalein is under investigation in clinical trial NCT03830684 (A Randomized, Double-blind, Placebo-controlled, Multicenter and Phase ⅡA Clinical Trial for the Effectiveness and Safety of Baicalein Tablets in the Treatment of...
BalinatunfibBalinatunfib is a small molecule drug. Balinatunfib has a monoisotopic molecular weight of 502.19 Da.
CamobucolCamobucol is a small molecule drug. Camobucol has a monoisotopic molecular weight of 574.32 Da.
Certolizumab pegolA tumor necrosis factor (TNF) blocker used to treat a variety of autoimmune and autoinflammatory conditions like Crohn's disease, rheumatoid arthritis, active psoriatic arthritis, ankylosing spondylitis, axial spondyloarthritis, and plaque psoriasis.
ChloroquineAn antimalarial drug used to treat susceptible infections with P. vivax, P. malariae, P. ovale, and P. falciparum. It is also used for second line treatment for rheumatoid arthritis.
CP1-1189CPI-1189 has been used in trials studying the treatment of HIV Infections and AIDS Dementia Complex.
DeupirfenidoneDeupirfenidone is under investigation in clinical trial NCT05321420 (LYT-100 in Patients With Idiopathic Pulmonary Fibrosis (IPF)).
EtanerceptA protein therapy based on the binding fragment of the tumour necrosis factor alpha receptor used to treat severe rheumatoid arthritis and moderate to severe plaque psoriasis.
GolimumabA TNFα inhibitor used in the symptomatic treatment of various active inflammatory disorders, such as rheumatoid arthritis, psoriatic arthritis, ankylosing spondylitis, and ulcerative colitis.
InfliximabA monoclonal anti tumor necrosis factor alpha antibody used in the treatment of a wide variety of inflammatory conditions such as rheumatoid arthritis, Crohn's disease, and ankylosing spondylitis.
ISIS 104838ISIS 104838 is under investigation in clinical trial NCT00048321 (ISIS 104838, an Inhibitor of Tumor Necrosis Factor, for Active Rheumatoid Arthritis).
Isopropyl alcoholAn antiseptic and disinfectant used in a variety of clinical and domestic settings.
LenabasumAjulemic acid has been used in trials studying the treatment of Cystic Fibrosis, Dermatomyositis, and Diffuse Cutaneous Systemic Sclerosis.
LenalidomideA thalidomide derivative used to treat multiple myeloma and anemia in low to intermediate risk myelodysplastic syndrome.
LenerceptNot Annotated
LicaminlimabLicaminlimab is under investigation in clinical trial NCT05896670 (Safety and Efficacy of Licaminlimab Ophthalmic Suspension for the Treatment of Dry Eye Disease).
OrtataxelOrtataxel has been used in trials studying the treatment of Lymphoma, Lung Cancer, Glioblastoma, and Kidney Cancer.
OzoralizumabOzoralizumab has been used in trials studying the treatment of Rheumatoid Arthritis and Active Rheumatoid Arthritis.
PegsunerceptInvestigated for use/treatment in rheumatoid arthritis.
PirfenidoneAn agent used for the treatment of idiopathic pulmonary fibrosis (IPF).
PlaculumabPlaculumab has been used in trials studying the treatment of Rheumatoid Arthritis.
PolaprezincPeptic ulcer disease, dyspepsia .
PomalidomideA thalidomide analogue used in combination with dexamethasone to treat patients with multiple myeloma.
PseudoephedrineAn alpha and beta adrenergic agonist used to treat nasal and sinus congestion, as well as allergic rhinitis.
RDP58Investigated for use/treatment in ulcerative colitis and crohn's disease.
RemtolumabRemtolumab is under investigation in clinical trial NCT02433340 (Phase 2, Multicenter, Open-Label Extension (OLE) Study With ABT-122 in Rheumatoid Arthritis Subjects Who Have Completed the Preceding M12-963 Study).
SenlizumabNot Annotated
SibeprenlimabA APRIL-directed monoclonal antibody used to reduce proteinuria in adults with primary immunoglobulin A nephropathy (IgAN).
TAK-715TAK-715 is under investigation in clinical trial NCT00760864 (Safety and Efficacy of TAK-715 in Subjects With Rheumatoid Arthritis).
TanfanerceptTanfanercept is under investigation in clinical trial NCT06400589 (A Study to Evaluate the Efficacy and Safety of Tanfanercept (HL036) in Dry Eye Disease).
ThalidomideA medication used to treat cancers, particularly newly diagnosed multiple myeloma, and erythema nodosum leprosum.
TiamulinTiamulin is a pleuromutilin antibiotic drug that is used in veterinary medicine particularly for pigs and poultry.
XPro1595XPro1595 is an investigational dominant-negative protein that neutralizes soluble TNF.
XTMAB-16XTMAB-16 is a monoclonal antibody directed against tumour necrosis factor-alpha (TNFα).
YisaipuNot Annotated
ZofinZofin, previously known as Organicell Flow, is a nanoparticle-based therapeutic derived from perinatal sources which is manufactured in a way that retains the naturally occurring microRNAs without the addition of...
Drugs & Drug Targets
DrugTargetType
(2R)-N-HYDROXY-2-[(3S)-3-METHYL-3-{4-[(2-METHYLQUINOLIN-4-YL)METHOXY]PHENYL}-2-OXOPYRROLIDIN-1-YL]PROPANAMIDEDisintegrin and metalloproteinase domain-containing protein 33target
(2R)-N-HYDROXY-2-[(3S)-3-METHYL-3-{4-[(2-METHYLQUINOLIN-4-YL)METHOXY]PHENYL}-2-OXOPYRROLIDIN-1-YL]PROPANAMIDECollagenase 3target
(2R)-N-HYDROXY-2-[(3S)-3-METHYL-3-{4-[(2-METHYLQUINOLIN-4-YL)METHOXY]PHENYL}-2-OXOPYRROLIDIN-1-YL]PROPANAMIDEMatrilysintarget
(2R)-N-HYDROXY-2-[(3S)-3-METHYL-3-{4-[(2-METHYLQUINOLIN-4-YL)METHOXY]PHENYL}-2-OXOPYRROLIDIN-1-YL]PROPANAMIDETumor necrosis factortarget
(2R)-N-HYDROXY-2-[(3S)-3-METHYL-3-{4-[(2-METHYLQUINOLIN-4-YL)METHOXY]PHENYL}-2-OXOPYRROLIDIN-1-YL]PROPANAMIDENeutrophil collagenasetarget
(2R)-N-HYDROXY-2-[(3S)-3-METHYL-3-{4-[(2-METHYLQUINOLIN-4-YL)METHOXY]PHENYL}-2-OXOPYRROLIDIN-1-YL]PROPANAMIDEStromelysin-1target
(2R)-N-HYDROXY-2-[(3S)-3-METHYL-3-{4-[(2-METHYLQUINOLIN-4-YL)METHOXY]PHENYL}-2-OXOPYRROLIDIN-1-YL]PROPANAMIDE72 kDa type IV collagenasetarget
(2R)-N-HYDROXY-2-[(3S)-3-METHYL-3-{4-[(2-METHYLQUINOLIN-4-YL)METHOXY]PHENYL}-2-OXOPYRROLIDIN-1-YL]PROPANAMIDEMatrix metalloproteinase-9target
(2R)-N-HYDROXY-2-[(3S)-3-METHYL-3-{4-[(2-METHYLQUINOLIN-4-YL)METHOXY]PHENYL}-2-OXOPYRROLIDIN-1-YL]PROPANAMIDEMatrix metalloproteinase-14target
(2R)-N-HYDROXY-2-[(3S)-3-METHYL-3-{4-[(2-METHYLQUINOLIN-4-YL)METHOXY]PHENYL}-2-OXOPYRROLIDIN-1-YL]PROPANAMIDEDisintegrin and metalloproteinase domain-containing protein 17target
AdalimumabTumor necrosis factortarget
AfelimomabTumor necrosis factortarget
AmrinonecAMP-specific 3',5'-cyclic phosphodiesterase 4 (PDE4)target
AmrinonecGMP-inhibited 3',5'-cyclic phosphodiesterase 3Btarget
AmrinonecGMP-inhibited 3',5'-cyclic phosphodiesterase 3Atarget
AmrinoneTumor necrosis factortarget
AN0128Tumor necrosis factortarget
AstegolimabInterleukin-1 receptor-like 1target
AtaciceptTumor necrosis factor ligand superfamily member 13target
AtaciceptTumor necrosis factor ligand superfamily member 13Btarget
BaicaleinP-selectintarget
BaicaleinLactoylglutathione lyasetarget
BaicaleinTumor necrosis factortarget
BaicaleinXanthine dehydrogenase/oxidasetarget
BaicaleinL-selectintarget
BaicaleinProlyl endopeptidasetarget
BaicaleinPolyunsaturated fatty acid 5-lipoxygenasetarget
BalinatunfibTumor necrosis factortarget
BalinatunfibTumor necrosis factor receptor superfamily member 1Atarget
CamobucolTumor necrosis factortarget
Certolizumab pegolTumor necrosis factortarget
Certolizumab pegolAldo-keto reductase family 1 member A1enzyme
ChloroquineToll-like receptor 9target
ChloroquineTumor necrosis factortarget
ChloroquineAtypical chemokine receptor 1target
ChloroquineAngiotensin-converting enzyme 2target
ChloroquineCytochrome P450 3A4enzyme
ChloroquineGlutathione S-transferase A2target
ChloroquineGlutathione S-transferase Mu 1target
ChloroquineHigh mobility group protein B1target
Chloroquinealpha1-acid glycoproteincarrier
ChloroquineCytochrome P450 1A1enzyme
ChloroquineAlbumincarrier
ChloroquineCytochrome P450 2D6enzyme
ChloroquineATP-dependent translocase ABCB1transporter
ChloroquineGlutathione S-transferasetarget
ChloroquineCytochrome P450 3A5enzyme
ChloroquineCytochrome P450 2C8enzyme
CP1-1189Tumor necrosis factortarget
EtanerceptTumor necrosis factortarget
EtanerceptLow affinity immunoglobulin gamma Fc region receptor III-Btarget
EtanerceptLow affinity immunoglobulin gamma Fc region receptor III-Atarget
EtanerceptHigh affinity immunoglobulin gamma Fc receptor Itarget
EtanerceptLow affinity immunoglobulin gamma Fc region receptor II-atarget
EtanerceptLow affinity immunoglobulin gamma Fc region receptor II-btarget
EtanerceptLow affinity immunoglobulin gamma Fc region receptor II-ctarget
EtanerceptComplement component 1q (C1q)target
EtanerceptLymphotoxin-alphatarget
GolimumabTumor necrosis factortarget
InfliximabTumor necrosis factortarget
ISIS 104838Tumor necrosis factortarget
Isopropyl alcoholTumor necrosis factortarget
Isopropyl alcoholPhospholipase A2, membrane associatedtarget
Isopropyl alcoholGTP cyclohydrolase 1target
Isopropyl alcoholHeme oxygenase 1target
Isopropyl alcoholOxysterols receptor LXR-betatarget
Isopropyl alcoholNitric oxide synthase 3target
LenabasumTumor necrosis factortarget
LenalidomideTumor necrosis factortarget
LenalidomideATP-dependent translocase ABCB1transporter
LenalidomideProtein cereblontarget
LenalidomideCadherin-5target
LenalidomideTumor necrosis factor ligand superfamily member 11target
LenalidomideProstaglandin G/H synthase 2target
LicaminlimabTumor necrosis factortarget
OrtataxelTumor necrosis factortarget
OzoralizumabTumor necrosis factortarget
PegsunerceptTumor necrosis factortarget
PirfenidoneATP-dependent translocase ABCB1transporter
PirfenidoneCytochrome P450 1A2enzyme
PirfenidoneCytochrome P450 2C9enzyme
PirfenidoneCytochrome P450 2C19enzyme
PirfenidoneCytochrome P450 2D6enzyme
PirfenidoneCytochrome P450 2E1enzyme
PirfenidoneAlbumincarrier
PirfenidoneCytochrome P450 3A4enzyme
PirfenidoneTransforming growth factor beta-1 proproteintarget
PlaculumabTumor necrosis factortarget
PolaprezincPeroxiredoxin-5, mitochondrialenzyme
PolaprezincVascular endothelial growth factor receptor 1target
PolaprezincGlutathione S-transferase theta-1enzyme
PolaprezincGlutathione peroxidase 1enzyme
PolaprezincPeroxiredoxin-1enzyme
PolaprezincBeta-nerve growth factortarget
PolaprezincPlatelet-derived growth factor receptor betatarget
PolaprezincHeat shock protein HSP 90-alphatarget
PolaprezincHeat shock protein HSP 90-betatarget
PolaprezincTumor necrosis factortarget
PolaprezincInterleukin-6target
PolaprezincSuperoxide dismutase [Mn], mitochondrialenzyme
PolaprezincHeme oxygenase 1enzyme
PolaprezincSuperoxide dismutase [Cu-Zn]enzyme
PolaprezincInterleukin-3target
PomalidomideCytochrome P450 1A2enzyme
PomalidomideCytochrome P450 3A4enzyme
PomalidomideATP-dependent translocase ABCB1transporter
PomalidomideProtein cereblontarget
PomalidomideTumor necrosis factortarget
PomalidomideProstaglandin G/H synthase 2target
Pseudoephedrineactivator protein 1target
PseudoephedrineD(2) dopamine receptortarget
PseudoephedrineSodium-dependent serotonin transportertransporter
PseudoephedrineSodium-dependent dopamine transportertransporter
PseudoephedrineSodium-dependent noradrenaline transportertransporter
PseudoephedrineAlbumincarrier
PseudoephedrineInterleukin-2target
PseudoephedrineNuclear factor NF-kappa-B p105 subunittarget
PseudoephedrineTumor necrosis factortarget
PseudoephedrineNuclear factor of activated T-cells, cytoplasmic 1target
PseudoephedrineSodium-dependent serotonin transportertarget
PseudoephedrineSodium-dependent noradrenaline transportertarget
PseudoephedrineSodium-dependent dopamine transportertarget
PseudoephedrineBeta-1 adrenergic receptortarget
PseudoephedrineAmine oxidase [flavin-containing] Aenzyme
PseudoephedrineAlpha-2A adrenergic receptortarget
PseudoephedrineAlpha-1A adrenergic receptortarget
PseudoephedrineBeta-2 adrenergic receptortarget
RDP58Tumor necrosis factortarget
RemtolumabTumor necrosis factortarget
RemtolumabInterleukin-17Atarget
SenlizumabTumor necrosis factortarget
SibeprenlimabTumor necrosis factor ligand superfamily member 13target
TAK-715Mitogen-activated protein kinase 14target
TanfanerceptTumor necrosis factortarget
ThalidomideProtein cereblontarget
ThalidomideDNAtarget
ThalidomideCytochrome P450 3A5enzyme
ThalidomideCytochrome P450 2B6enzyme
Thalidomidealpha1-acid glycoproteintarget
ThalidomideProstaglandin G/H synthase 2enzyme
ThalidomideProstaglandin G/H synthase 1enzyme
ThalidomideCytochrome P450 2C9enzyme
ThalidomideCytochrome P450 2C19enzyme
ThalidomideCytochrome P450 3A4enzyme
ThalidomideTumor necrosis factortarget
ThalidomideCytochrome P450 1A1enzyme
TiamulinCytochrome P450 3A4enzyme
TiamulinCytochrome P450 2E1enzyme
TiamulinATP-dependent translocase ABCB1transporter
TiamulinTumor necrosis factortarget
XPro1595Tumor necrosis factortarget
XTMAB-16Tumor necrosis factortarget
YisaipuTumor necrosis factortarget
ZofinTumor necrosis factortarget
ZofinInterleukin-6target
ZofinInterleukin-8target
ZofinFibroblast growth factor 2target
ZofinInterferon betatarget
ZofinInsulin-like growth factor 1target
ZofinInterleukin-36 alphatarget
ZofinInterleukin-37target
ZofinTransforming growth factor beta-2 proproteintarget
ZofinVascular endothelial growth factor A, long formtarget
ZofinC-C motif chemokine 8target
ZofinStromal cell-derived factor 1target