Acid Reducers

Name
Acid Reducers
Accession Number
DBCAT003864
Description

Drugs which actively reduce the hydronium concentration of the gastric system. Includes proton pump inhibitors and H2 antagonist drugs.

Drugs
DrugDrug Description
AsenapineAn atypical antipsychotic used to treat patients with bipolar I disorder and patients with schizophrenia.
CimetidineA histamine H2 receptor antagonist used to manage GERD, peptic ulcer disease, and indigestion.
DexlansoprazoleA proton pump inhibitor used to treat erosive esophagitis, heartburn, and gastroesophageal reflux disease (GERD).
DexrabeprazoleA proton pump inhibitor indicated in the treatment of gastroesophageal reflux disease and gastrointestinal ulcers.
DoxepinA psychotropic agent used for the treatment of depression, anxiety, manic-depressive disorder, and insomnia.
EpinastineAn H1 receptor antagonist used to prevent itching in allergic conjunctivitis.
EsomeprazoleA proton pump inhibitor used to treat GERD, reduce the risk of NSAID associated gastric ulcers, eradicate H. pylori, and to treat conditions causing gastric acid hypersecretion.
FamotidineA histamine H2 receptor antagonist used to treat duodenal ulcers, benign gastric ulcers, GERD, and Zollinger-Ellison syndrome.
LansoprazoleA proton pump inhibitor used to help gastrointestinal ulcers heal, to treat symptoms of gastroesophageal reflux disease (GERD), to eradicate Helicobacter pylori, and to treat hypersecretory conditions such as Zollinger-Ellison Syndrome.
MethanthelineFor the treatment of peptic ulcer disease, irritable bowel syndrome, pancreatitis, gastritis, biliary dyskinesia, pylorosplasm, and reflex neurogenic bladder in children.
MetiamidePotential in the treatment and the management of acid-reflux disorders (GERD), peptic ulcer disease, heartburn, and acid indigestion.
NizatidineAn H2 receptor antagonist used to treat GERD and a variety of ulcers.
OmeprazoleA proton pump inhibitor used to treat GERD associated conditions such as heartburn and gastric acid hypersecretion, and to promote healing of tissue damage and ulcers caused by gastric acid and H. pylori infection.
PantoprazoleA proton pump inhibitor used to treat erosive esophagitis, gastric acid hypersecretion, and to promote healing of tissue damage caused by gastric acid.
PromethazineA first-generation antihistamine used for the treatment of allergic conditions, nausea and vomiting, and motion sickness.
RabeprazoleA proton pump inhibitor used to help gastrointestinal ulcers heal, to treat symptoms of gastroesophageal reflux disease (GERD), to eradicate Helicobacter pylori, and to treat hypersecretory conditions such as Zollinger-Ellison Syndrome.
RanitidineA histamine H2 antagonist used to treat duodenal ulcers, Zollinger-Ellison syndrome, gastric ulcers, GERD, and erosive esophagitis.
Roxatidine acetateFor the treatment of disorders of the upper gastro-intestinal region that are due to an excess of hydrochloric acid in the gastric juice, i.e. duodenal ulcers, benign gastric ulcers. Also...
Drugs & Drug Targets
DrugTargetType
Asenapine5-hydroxytryptamine receptor 2Btarget
Asenapine5-hydroxytryptamine receptor 2Ctarget
Asenapine5-hydroxytryptamine receptor 6target
Asenapine5-hydroxytryptamine receptor 7target
AsenapineAlpha-2A adrenergic receptortarget
AsenapineAlpha-2B adrenergic receptortarget
AsenapineAlpha-2C adrenergic receptortarget
AsenapineAlpha-1A adrenergic receptortarget
AsenapineDopamine receptor D1target
AsenapineDopamine receptor D2target
AsenapineDopamine receptor D3target
AsenapineDopamine receptor D4target
AsenapineHistamine H1 receptortarget
AsenapineHistamine H2 receptortarget
AsenapineCytochrome P450 1A2enzyme
AsenapineCytochrome P450 2D6enzyme
Asenapine5-hydroxytryptamine receptor 5Atarget
AsenapineUDP-glucuronosyltransferase 1A4enzyme
AsenapineCytochrome P450 3A4enzyme
AsenapineBeta-1 adrenergic receptortarget
AsenapineBeta-2 adrenergic receptortarget
AsenapineAlbumincarrier
Asenapinealpha1-acid glycoproteincarrier
Asenapine5-hydroxytryptamine receptor 2Atarget
Asenapine5-hydroxytryptamine receptor 1Btarget
Asenapine5-hydroxytryptamine receptor 1Atarget
CimetidineSolute carrier family 22 member 6transporter
CimetidineMultidrug and toxin extrusion protein 1transporter
CimetidineAlbumincarrier
CimetidineMultidrug and toxin extrusion protein 2transporter
CimetidineBile salt export pumptransporter
CimetidineFlavin-containing monooxygenase 1enzyme
CimetidineFlavin-containing monooxygenase 3enzyme
CimetidineCytochrome P450 2E1enzyme
CimetidineCytochrome P450 2C9enzyme
CimetidineCytochrome P450 2C8enzyme
CimetidineCytochrome P450 11B1, mitochondrialenzyme
CimetidineSolute carrier family 22 member 7transporter
CimetidineSolute carrier family 22 member 11transporter
CimetidineSolute carrier family 22 member 4transporter
CimetidineOrganic anion transporter 3transporter
CimetidineOrganic cation/carnitine transporter 2transporter
CimetidineSolute carrier family 22 member 3transporter
CimetidineSolute carrier family 22 member 1transporter
CimetidineSolute carrier family 22 member 2transporter
CimetidineATP-dependent translocase ABCB1transporter
CimetidineCytochrome P450 3A5enzyme
CimetidineCytochrome P450 3A4enzyme
CimetidineCytochrome P450 2C19enzyme
CimetidineCytochrome P450 2D6enzyme
CimetidineCytochrome P450 1A2enzyme
CimetidineHistamine H2 receptortarget
DexlansoprazoleN(G),N(G)-dimethylarginine dimethylaminohydrolase 1target
DexlansoprazolePotassium-transporting ATPase subunit betatarget
DexlansoprazoleCytochrome P450 3A4enzyme
DexlansoprazoleCytochrome P450 2C19enzyme
DexlansoprazolePotassium-transporting ATPase alpha chain 1target
DexrabeprazolePotassium-transporting ATPase alpha chain 1target
DexrabeprazoleHydrogen potassium ATPasetarget
DexrabeprazoleCytochrome P450 2C19enzyme
DoxepinAlpha-1A adrenergic receptortarget
DoxepinMuscarinic acetylcholine receptor M5target
Doxepin5-hydroxytryptamine receptor 6target
DoxepinCytochrome P450 3A4enzyme
DoxepinAlpha-1D adrenergic receptortarget
DoxepinAlpha-1B adrenergic receptortarget
Doxepin5-hydroxytryptamine receptor 2Ctarget
Doxepin5-hydroxytryptamine receptor 2Btarget
DoxepinATP-dependent translocase ABCB1transporter
DoxepinHistamine H4 receptortarget
DoxepinCytochrome P450 1A2enzyme
DoxepinVoltage-gated inwardly rectifying potassium channel KCNH2target
DoxepinCytochrome P450 2C9enzyme
DoxepinCytochrome P450 2C19enzyme
DoxepinSodium-dependent serotonin transportertarget
DoxepinSodium-dependent noradrenaline transportertarget
DoxepinAlpha-1-acid glycoprotein 1carrier
DoxepinAlbumincarrier
DoxepinMuscarinic acetylcholine receptor M4target
DoxepinMuscarinic acetylcholine receptor M3target
DoxepinMuscarinic acetylcholine receptor M2target
DoxepinMuscarinic acetylcholine receptor M1target
DoxepinCytochrome P450 2D6enzyme
Doxepin5-hydroxytryptamine receptor 1Atarget
Doxepin5-hydroxytryptamine receptor 2Atarget
DoxepinHistamine H2 receptortarget
DoxepinHistamine H1 receptortarget
EpinastineHistamine H1 receptortarget
EpinastineHistamine H2 receptortarget
EpinastineAlpha-1A adrenergic receptortarget
EpinastineAlpha-2A adrenergic receptortarget
Epinastine5-hydroxytryptamine receptor 2Atarget
Epinastine5-hydroxytryptamine receptor 7target
EpinastineATP-dependent translocase ABCB1transporter
EpinastineCytochrome P450 3A4enzyme
EpinastineCytochrome P450 2D6enzyme
EpinastineCytochrome P450 2B6enzyme
EsomeprazolePotassium-transporting ATPase subunit betatarget
EsomeprazoleOrganic anion transporter 3transporter
EsomeprazoleATP-dependent translocase ABCB1transporter
EsomeprazoleN(G),N(G)-dimethylarginine dimethylaminohydrolase 1target
EsomeprazoleCytochrome P450 3A4enzyme
EsomeprazoleCytochrome P450 2C19enzyme
EsomeprazolePotassium-transporting ATPase alpha chain 1target
FamotidineSolute carrier family 22 member 6transporter
FamotidineCytochrome P450 1A2enzyme
FamotidineMultidrug and toxin extrusion protein 1transporter
FamotidineOrganic anion transporter 3transporter
FamotidineSolute carrier family 22 member 2transporter
FamotidineHistamine H2 receptortarget
LansoprazoleOrganic anion transporter 3transporter
LansoprazoleSolute carrier family 22 member 1transporter
LansoprazoleSolute carrier family 22 member 2transporter
LansoprazoleSolute carrier family 22 member 3transporter
LansoprazoleCytochrome P450 2D6enzyme
LansoprazoleCytochrome P450 2C8enzyme
LansoprazoleCytochrome P450 2C18enzyme
LansoprazoleCytochrome P450 1B1enzyme
LansoprazoleCytochrome P450 1A1enzyme
LansoprazoleMicrotubule-associated protein tautarget
LansoprazoleBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
LansoprazoleATP-dependent translocase ABCB1transporter
LansoprazoleCytochrome P450 3A4enzyme
LansoprazoleCytochrome P450 2C9enzyme
LansoprazoleCytochrome P450 2C19enzyme
LansoprazolePotassium-transporting ATPase alpha chain 1target
MethanthelineMuscarinic acetylcholine receptor M1target
MethanthelineHistamine H2 receptortarget
MethanthelineMuscarinic acetylcholine receptor M2target
MethanthelineMuscarinic acetylcholine receptor M3target
MethanthelineMuscarinic acetylcholine receptor M4target
MethanthelineMuscarinic acetylcholine receptor M5target
MethanthelineAcetylcholinesteraseenzyme
MetiamideHistamine H2 receptortarget
NizatidineHistamine H2 receptortarget
NizatidineATP-dependent translocase ABCB1transporter
NizatidineCholinesteraseenzyme
OmeprazolePotassium-transporting ATPase subunit betatarget
OmeprazoleAryl hydrocarbon receptortarget
OmeprazoleCytochrome P450 2D6enzyme
OmeprazoleCytochrome P450 2C8enzyme
OmeprazoleCytochrome P450 2C18enzyme
OmeprazoleCytochrome P450 1B1enzyme
OmeprazoleCytochrome P450 1A1enzyme
OmeprazolePotassium-transporting ATPase alpha chain 1target
OmeprazoleATP-dependent translocase ABCB1transporter
OmeprazoleATP-binding cassette sub-family C member 3transporter
OmeprazoleCytochrome P450 1A2enzyme
OmeprazoleCytochrome P450 2C9enzyme
OmeprazoleCytochrome P450 3A4enzyme
OmeprazoleCytochrome P450 2C19enzyme
OmeprazoleBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
PantoprazoleBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
PantoprazoleATP-dependent translocase ABCB1transporter
PantoprazolePotassium-transporting ATPase subunit betatarget
PantoprazoleN(G),N(G)-dimethylarginine dimethylaminohydrolase 1target
PantoprazoleOrganic anion transporter 3transporter
PantoprazoleCytochrome P450 3A4enzyme
PantoprazoleCytochrome P450 2C19enzyme
PantoprazolePotassium-transporting ATPase alpha chain 1target
PromethazineDopamine receptor D2target
PromethazineHistamine H1 receptortarget
PromethazineMuscarinic acetylcholine receptor M4target
PromethazineMuscarinic acetylcholine receptor M1target
PromethazineMuscarinic acetylcholine receptor M5target
PromethazineMuscarinic acetylcholine receptor M2target
PromethazineMuscarinic acetylcholine receptor M3target
PromethazineCytochrome P450 2D6enzyme
PromethazineCytochrome P450 2B6enzyme
PromethazineATP-dependent translocase ABCB1transporter
PromethazineCytochrome P450 2C9enzyme
PromethazineHistamine H2 receptortarget
PromethazineAlpha adrenergic receptortarget
PromethazineP2 Purinoceptorstarget
PromethazineVoltage-gated sodium channel alpha subunittarget
PromethazineVoltage-gated Potassium Channelstarget
PromethazineATP-binding cassette sub-family C member 3transporter
PromethazineATP-binding cassette sub-family C member 4transporter
PromethazineAlbumincarrier
PromethazineCalmodulintarget
PromethazineNMDA receptortarget
RabeprazoleCytochrome P450 2C8enzyme
RabeprazoleCytochrome P450 2D6enzyme
RabeprazoleCytochrome P450 2C9enzyme
RabeprazoleCytochrome P450 1A2enzyme
RabeprazoleCytochrome P450 1A1enzyme
RabeprazoleBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
RabeprazoleCytochrome P450 2C19enzyme
RabeprazoleCytochrome P450 3A4enzyme
RabeprazolePotassium-transporting ATPase alpha chain 1target
RanitidineSolute carrier family 22 member 2transporter
RanitidineAcetylcholinesterasetarget
RanitidineCytochrome P450 3A4enzyme
RanitidineOrganic anion transporter 3transporter
RanitidineATP-dependent translocase ABCB1transporter
RanitidineSolute carrier family 22 member 1transporter
RanitidineCytochrome P450 2D6enzyme
RanitidineCytochrome P450 1A2enzyme
RanitidineHistamine H2 receptortarget
RanitidineAcetylcholinesteraseenzyme
Roxatidine acetateHistamine H2 receptortarget