| Lorcaserin | Organic compounds | Organoheterocyclic compounds | Benzazepines | Not Available | Details |
| Osanetant | Organic compounds | Benzenoids | Benzene and substituted derivatives | Benzoyl derivatives | Details |
| Piboserod | Organic compounds | Organoheterocyclic compounds | Indoles and derivatives | Indolecarboxylic acids and derivatives | Details |
| Pralnacasan | Organic compounds | Organic acids and derivatives | Carboxylic acids and derivatives | Amino acids, peptides, and analogues | Details |
| Vildagliptin | Organic compounds | Organic acids and derivatives | Carboxylic acids and derivatives | Amino acids, peptides, and analogues | Details |
| Voacamine | Organic compounds | Alkaloids and derivatives | Ibogan-type alkaloids | Not Available | Details |
| Voglibose | Organic compounds | Organic oxygen compounds | Organooxygen compounds | Alcohols and polyols | Details |
| Vatalanib | Organic compounds | Organoheterocyclic compounds | Diazanaphthalenes | Benzodiazines | Details |
| Enoximone | Organic compounds | Organic oxygen compounds | Organooxygen compounds | Carbonyl compounds | Details |
| Elacridar | Organic compounds | Organoheterocyclic compounds | Quinolines and derivatives | Benzoquinolines | Details |
| Edotecarin | Organic compounds | Organoheterocyclic compounds | Indoles and derivatives | Carbazoles | Details |
| Darusentan | Organic compounds | Benzenoids | Benzene and substituted derivatives | Diphenylmethanes | Details |
| Dapoxetine | Organic compounds | Benzenoids | Naphthalenes | Not Available | Details |
| Cilansetron | Organic compounds | Organoheterocyclic compounds | Indoles and derivatives | Carbazoles | Details |
| Calanolide A | Organic compounds | Phenylpropanoids and polyketides | Coumarins and derivatives | Pyranocoumarins | Details |
| Brecanavir | Organic compounds | Benzenoids | Benzene and substituted derivatives | Phenylbutylamines | Details |
| Bifeprunox | Organic compounds | Benzenoids | Benzene and substituted derivatives | Biphenyls and derivatives | Details |
| Bicifadine | Organic compounds | Organoheterocyclic compounds | Piperidines | Phenylpiperidines | Details |
| Bepotastine | Organic compounds | Benzenoids | Benzene and substituted derivatives | Benzylethers | Details |
| Becocalcidiol | Organic compounds | Lipids and lipid-like molecules | Steroids and steroid derivatives | Vitamin D and derivatives | Details |
| Phenserine | Organic compounds | Organoheterocyclic compounds | Indoles and derivatives | Pyrroloindoles | Details |
| Vapreotide | Organic Compounds | Organic Acids | Carboxylic Acids and Derivatives | Amino Acids, Peptides, and Analogues | Details |
| Lucinactant | Organic Compounds | Organic Acids | Carboxylic Acids and Derivatives | Amino Acids, Peptides, and Analogues | Details |
| Ximelagatran | Organic compounds | Organic acids and derivatives | Carboxylic acids and derivatives | Amino acids, peptides, and analogues | Details |
| Nesiritide | Organic Compounds | Organic Acids | Carboxylic Acids and Derivatives | Amino Acids, Peptides, and Analogues | Details |
| Thymalfasin | Organic Compounds | Organic Acids | Carboxylic Acids and Derivatives | Amino Acids, Peptides, and Analogues | Details |
| Galiximab | Organic Compounds | Organic Acids | Carboxylic Acids and Derivatives | Amino Acids, Peptides, and Analogues | Details |
| Pagoclone | Organic compounds | Organoheterocyclic compounds | Diazanaphthalenes | Naphthyridines | Details |
| Amolimogene | Organic Compounds | Organic Acids | Carboxylic Acids and Derivatives | Amino Acids, Peptides, and Analogues | Details |
| Tesmilifene | Organic compounds | Benzenoids | Benzene and substituted derivatives | Diphenylmethanes | Details |