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Phorbol 12-myristate 13-acetate diester
go.drugbank.com/drugs/DB17045InvestigationalPhorbol 12-myristate 13-acetate diester is an inducer of neutrophil extracellular traps (NETs).[A253087]
Synonyms: 12-o-tetradecanoylphorbol-13-acetatePI-103
go.drugbank.com/drugs/DB17046ExperimentalPI-103 is an inhibitor of p110α of class I PI3K.[A253092]
Synonyms: Phenol, 3-(4-(4-morpholinyl)pyrido(3',2':4,5)furo(3,2-d)pyrimidin-2-yl)-Categories: Heterocyclic Compounds, 1-RingPIK-75
go.drugbank.com/drugs/DB17047ExperimentalPIK-75 is a preferential p110 alpha/gamma PI3K inhibitor.[A253097]
Synonyms: Benzenesulfonic acid, 2-methyl-5-nitro-, 2-((6-bromoimidazo(1,2-a)pyridin-3-yl)methylene)-1-methylhydrazideCategories: Phosphatidylinositol 3-Kinases, antagonists & inhibitorsPlumbagin
go.drugbank.com/drugs/DB17048InvestigationalPlumbagin is a compound investigated for its anticancer activity. It has been found that it inactivates the Akt/NF-kB, MMP-9 and VEGF pathways.[A253102]
Synonyms: 5-hydroxy-2-methyl-1,4-naphthalenedioneCategories: Compounds used in a research, industrial, or household settingRS-39604
go.drugbank.com/drugs/DB17050ExperimentalRS-39604 is a selective 5-HT4 receptor antagonist.[A253112]
Synonyms: Methanesulfonamide, n-(2-(4-(3-(4-amino-5-chloro-2-((3,5-dimethoxyphenyl)methoxy)phenyl)-3-oxopropyl)-1-piperidinyl)ethyl)-Salts: RS-39604 hydrochlorideSB-218078
go.drugbank.com/drugs/DB17051ExperimentalSB-218078 is a specific inhibitor of CHK1.[A253117]
Synonyms: 9,10,11,12-tetrahydro-9,12-epoxy-1h-diindolo(1,2,3-fg:3',2',1'-kl)pyrrolo(3,4-i)(1,6)benzodiazocine-1,3(2h)-dione, 9,12-epoxy-1h-diindolo(1,2,3-fg:3',2',1'-kl)pyrrolo(3,4-i)(1,6)benzodiazocine-1,3(2h)-dione, 9,10,11,12-tetrahydro-Salts: SB-218078 hydrochlorideScriptaid
go.drugbank.com/drugs/DB17053ExperimentalScriptaid is a histone deacetylase (HDAC) inhibitor researched for its anti-tumor properties.[A253127]
Synonyms: 1h-benz(de)isoquinoline-2(3h)-hexanamide, n-hydroxy-1,3-dioxo-, N-hydroxy-1,3-dioxo-1h-benz(de)isoquinoline-2(3h)-hexan amideCategories: Heterocyclic Compounds, 2-RingSKF-96365 free base
go.drugbank.com/drugs/DB17054ExperimentalSKF-96365 is a receptor-mediated calcium entry (RMCE) inhibitor structurally different from other calcium antagonists.[A253132]
Synonyms: 1-(2-(3-(4-methoxyphenyl)propoxy)-4-methoxyphenylethyl)-1h-imidazoleCategories: Heterocyclic Compounds, 1-RingSNX-2112
go.drugbank.com/drugs/DB17055ExperimentalSNX-2112 is a heat shock protein 90 (Hsp90) inhibitor.[A253137]
Synonyms: Benzamide, 2-((trans-4-hydroxycyclohexyl)amino)-4-(4,5,6,7-tetrahydro-6,6-dimethyl-4-oxo-3-(trifluoromethyl)-1h-indazol-1-yl)-SRT-1720
go.drugbank.com/drugs/DB17057ExperimentalSRT-1720 is an activator of NAD(+)-dependent histone deacetylase SIRT1.[A253147]
Synonyms: 2-quinoxalinecarboxamide, n-(2-(3-(1-piperazinylmethyl)imidazo(2,1-b)thiazol-6-yl)phenyl)-, N-(2-(3-(1-piperazinylmethyl)imidazo(2,1-b)thiazol-6-yl)phenyl)-2-quinoxalinecarboxamide