| DB00300 | Tenofovir disoproxil | approved, investigational | yes | inhibitor | Details |
| DB07935 | 5-[(5-fluoro-3-methyl-1H-indazol-4-yl)oxy]benzene-1,3-dicarbonitrile | experimental | unknown | | Details |
| DB01048 | Abacavir | approved, investigational | yes | inhibitor | Details |
| DB00705 | Delavirdine | approved | yes | inhibitor | Details |
| DB00900 | Didanosine | approved | yes | inhibitor | Details |
| DB00625 | Efavirenz | approved, investigational | yes | inhibitor | Details |
| DB00879 | Emtricitabine | approved, investigational | yes | inhibitor | Details |
| DB00709 | Lamivudine | approved, investigational | yes | inhibitor | Details |
| DB00238 | Nevirapine | approved | yes | inhibitor | Details |
| DB00649 | Stavudine | approved, investigational | yes | inhibitor | Details |
| DB00943 | Zalcitabine | approved, investigational | yes | inhibitor | Details |
| DB00495 | Zidovudine | approved | yes | inhibitor | Details |
| DB08864 | Rilpivirine | approved | yes | inhibitor | Details |
| DB09299 | Tenofovir alafenamide | approved | yes | inhibitor | Details |
| DB11365 | Sennosides | experimental | unknown | inhibitor | Details |
| DB11799 | Bictegravir | approved, investigational | yes | antagonist | Details |
| DB12855 | Apricitabine | investigational | unknown | inhibitor | Details |
| DB12301 | Doravirine | approved, investigational | unknown | inhibitor | Details |
| DB14126 | Tenofovir | experimental, investigational | yes | inhibitor | Details |
| DB12753 | Racivir | investigational | unknown | inhibitor | Details |
| DB12470 | Dexelvucitabine | investigational | unknown | inhibitor | Details |
| DB06236 | Elvucitabine | investigational | unknown | inhibitor | Details |
| DB06198 | Alovudine | investigational | unknown | inhibitor | Details |
| DB06619 | Amdoxovir | investigational | unknown | inhibitor | Details |
| DB08502 | Capravirine | investigational | unknown | inhibitor | Details |
| DB06414 | Etravirine | approved | unknown | inhibitor | Details |