Cytochrome P-450 CYP2C8 Inhibitors (strength unknown)

Name
Cytochrome P-450 CYP2C8 Inhibitors (strength unknown)
Accession Number
DBCAT004479
Description

Not Available

Drugs
DrugDrug Description
CerivastatinA statin (or HMG CoA reductase inhibitor) used with dietary changes to decrease lipid levels and reduce the risk of cardiovascular events.
LapatinibAn antineoplastic agent and tyrosine kinase inhibitor used for the treatment of advanced or metastatic HER-positive breast cancer in patients who received prior chemotherapeutic treatments.
RaloxifeneA selective estrogen receptor modulator that is used to prevent and treat osteoporosis and reduce the risk of invasive breast cancer in high-risk postmenopausal women.
QuercetinA natural flavonoid found in foods and natural supplement products.
EthinylestradiolAn estradiol used as a contraceptive.
ColchicineAn alkaloid used to treat gout and Familial Mediterranean Fever as well as prevent major cardiovascular events.
IsoniazidAn antibiotic used to treat mycobacterial infections; most commonly use in combination with other antimycobacterial agents for the treatment of active or latent tuberculosis.
MetronidazoleA nitroimidazole used to treat trichomoniasis, amebiasis, inflammatory lesions of rosacea, and bacterial infections, as well as prevent postoperative infections.
NilutamideAn antineoplastic hormone used to treat prostate cancer.
PhenelzineA monoamine oxidase inhibitor used to treat atypical, nonendogenous, or neurotic depression.
SulfaphenazoleFor the treatment bacterial infections.
TerfenadineAn antihistamine for the treatment of allergy symptoms.
TriazolamA benzodiazepine used for short term treatment of insomnia.
DiethylstilbestrolUsed in the treatment of prostate cancer. Previously used in the prevention of miscarriage or premature delivery in pregnant women prone to miscarriage or premature delivery.
VismodegibA hedgehog pathway inhibitor used to treat patients with locally advanced or metastatic basal cell carcinoma.
RegorafenibA kinase inhibitor used to treat patients with metastatic colorectal cancer, unresectable, locally advanced, or metastatic gastrointestinal stromal tumors, and hepatocellular carcinoma.
LumacaftorA protein chaperone used in combination with ivacaftor for the treatment of cystic fibrosis in patients who are homozygous for the F508del mutation in the CFTR gene.
MidostaurinAn antineoplastic agent used to treat high-risk acute myeloid leukemia (AML) with specific mutations, aggressive systemic mastocytosis (ASM), systemic mastocytosis with associated hematologic neoplasm (SM-AHN), or mast cell leukemia (MCL).
EnasidenibAn isocitrate dehydrogenase-2 inhibitor used to treat relapsed or refractory acute myeloid leukemia with an isocitrate dehydrogenase-2 mutation.
LetermovirAn antiviral medication used for prophylaxis in adult transplant recipients at risk of cytomegalovirus (CMV) infection and disease.
BosutinibAn antineoplastic agent used for the treatment of chronic, accelerated, or blast phase Philadelphia chromosome-positive (Ph+) chronic myelogenous leukemia (CML) in adults with inadequate clinical response to other treatments.
DeferasiroxAn iron chelator used to treat chronic iron overload caused by blood transfusions. Also used in patients with non-transfusion-dependent thalassemia syndromes, and in patients with elevated liver iron concentration and serum ferritin.
RifampicinAn antibiotic used to treat several types of mycobacterial infections including Mycobacterium avium complex, leprosy, and in combination with other antibacterials to treat latent or active tuberculosis.
VerapamilA non-dihydropyridine calcium channel blocker used in the treatment of angina, arrhythmia, and hypertension.
SimvastatinAn HMG-CoA reductase inhibitor used to lower lipid levels and reduce the risk of cardiovascular events including myocardial infarction and stroke.
SulfinpyrazoneA platelet inhibitory and uricosuric agent used to inhibit thrombotic and embolic processes and to manage the chronic phases of gout .
MontelukastA leukotriene receptor antagonist used as part of an asthma therapy regimen, to prevent exercise induced bronchoconstriction, and to treat seasonal allergic rhinitis.
NilvadipineA calcium channel blocker used to manage arterial hypertension.
LiotrixMay be used to treat primary, secondary or tertiary hypothyroidism. May also be used to suppress thyroid stimulating hormone (TSH) secretion in patients with simple (nontoxic) goiter, subacute or chronic...
MometasoneA corticosteroid with no indications.
MifepristoneA cortisol receptor blocker used to treat Cushing's syndrome, and to terminate pregnancies up to 70 days gestation.
VemurafenibA kinase inhibitor used to treat patients with Erdheim-Chester Disease who have the BRAF V600 mutation, and melanoma in patients who have the BRAF V600E mutation.
SorafenibA kinase inhibitor used to treat unresectable liver carcinoma, advanced renal carcinoma, and differentiated thyroid carcinoma.
EltrombopagA thrombopoietin receptor agonist used to treat thrombocytopenia or aplastic anemia associated with various etiologies.
LicofeloneFor the management of osteoarthritis.
BezafibrateA lipid-lowering fibrate used in the management of primary and secondary hyperlipidaemia, when there is a lack of clinical improvement following lifestyle modifications or correction of the underlying disorder.
IdelalisibAn antineoplastic kinase inhibitor used to treat chronic lymphocytic leukemia (CLL), relapsed follicular B-cell non-Hodgkin lymphoma (FL), and relapsed small lymphocytic lymphoma (SLL).
CandesartanAn angiotensin-receptor blocker indicated in the treatment of hypertension.
IsavuconazoleIndicated for patients 18 years of age and older for the treatment of invasive aspergillosis [FDA Label]. Indicated for patients 18 years of age and older for the treatment of...
OpicaponeA catechol-O-methyltransferase inhibitor used as an adjunct treatment for Parkinson's Disease in adults currently receiving levodopa and a dopa decarboxylase inhibitor.
RifamycinAn antibacterial used to treat traveler's diarrhea.
TriclabendazoleAn anthelmintic drug used to treat fascioliasis.
AlpelisibAlpelisib is indicated in combination with fulvestrant to treat postmenopausal women, and men, with advanced or metastatic breast cancer. This cancer must be hormone receptor (HR)-positive, human epidermal growth factor...
BalaglitazoneBalaglitazone has been used in trials studying the treatment of Diabetes Mellitus, Type 2.
CiglitazoneDeveloped by Takeda Pharmaceuticals in the early 1980s, it is considered the prototypical compound for the thiazolidinedione class. Ciglitazone was never used as a medication, but it sparked interest in...
LobeglitazoneLobeglitazone was approved by the Ministry of Food and Drug Safety (South Korea) in 2013, and is being monitored by postmarketing surveillance until 2019. Lobeglitazone is not approved for use...
NetoglitazoneNetoglitazone (MCC-555) is a hypoglycemic agent.
RivoglitazoneRivoglitazone (INN) is a thiazolidinedione undergoing research for use in the treatment of type 2 diabetes. It is being developed by Daiichi Sankyo Co.
Mometasone furoateA corticosteroid used to treat asthma, allergic rhinitis, nasal congestion, nasal polyps, dermatitis, and pruritus.
TolbutamideA sulfonylurea used to treat hyperglycemia in patients with type 2 diabetes mellitus.
NifedipineA dihydropyridine calcium channel blocker indicated for the management of several subtypes of angina pectoris, and hypertension.
CholecalciferolA form of Vitamin D used in the treatment of specific medical conditions such as refractory rickets, hypoparathyroidism, and familial hypophosphatemia, as well as osteoporosis and chronic kidney disease.
AtorvastatinAn HMG-CoA reductase inhibitor used to lower lipid levels and reduce the risk of cardiovascular disease including myocardial infarction and stroke.
LosartanAn angiotensin receptor blocker used to treat hypertension and diabetic nephropathy, and is used to reduce the risk of stroke.
Mefenamic acidAn NSAID used to treat mild to moderate pain for no more than a week, and primary dysmenorrhea.
TroleandomycinFor the treatment of bacterial infection.
EzetimibeA cholesterol absorption inhibitor used to lower total cholesterol, LDL-C, Apo-B, and non-HDL-C in primary hyperlipidemia and familial cholesterolemia.
AnastrozoleA competitive, selective, non-steroidal aromatase inhibitor used as adjuvant therapy for the treatment of hormone receptor-positive breast cancer in postmenopausal women.
AbemaciclibA medication used to treat HR+ HER2- advanced or metastatic breast cancer.
AmlodipineA calcium channel blocker used to treat hypertension and angina.
ElexacaftorA small molecule CFTR corrector used in combination with tezacaftor and ivacaftor for the treatment of cystic fibrosis patients with one F508del-CFTR mutation.
FavipiravirAn antiviral used to manage influenza, and that has the potential to target other viral infections.
Methylene blueAn oxidation-reduction agent used for the treatment of pediatric and adult patients with acquired methemoglobinemia.
SelpercatinibA RET receptor tyrosine kinase inhibitor for the treatment of RET-driven non-small cell lung cancer, medullary thyroid cancer, and thyroid cancer in appropriate patient populations.
RipretinibA kinase inhibitor used to treat advanced gastrointestinal stromal tumor (GIST).
ClofazimineA riminophenazine antimycobacterial used to treat leprosy.
SaquinavirAn HIV protease inhibitor used in combination with other antiretroviral agents for the treatment of HIV-1 with advanced immunodeficiency.
MiconazoleAn azole antifungal with broad-spectrum activity used to treat fungal infections affecting the vagina, mouth and skin, including candidiasis.
PralsetinibA RET receptor tyrosine kinase inhibitor for the treatment of metastatic RET-driven non-small cell lung cancer.
LonafarnibA potent farnesyl transferase inhibitor used to reduce mortality associated with Hutchinson-Gilford progeria syndrome (HGPS) and other progeroid laminopathies.
ZafirlukastA leukotriene receptor antagonist used for prophylaxis and chronic treatment of asthma.
MenadioneThe primary known function of vitamin K is to assist in the normal clotting of blood, but it may also play a role in normal bone calcification.
RilpivirineA non-nucleoside reverse transcriptase inhibitor (NNRTI) used in combination with other antiretrovirals to specifically treat human immunodeficiency virus type 1 (HIV-1).
IbrexafungerpA triterpene antifungal indicated in the treatment of vulvovaginal candidiasis and prevention of recurrent vulvovaginal candidiasis in post-menarchal patients.
BrincidofovirAn oral lipid prodrug of cidofovir used in the treatment of human smallpox disease.
LevoketoconazoleOne of two enantiomeric forms of racemic ketoconazole that strongly inhibits multiple steroidogenic enzymes and is used for the symptomatic treatment of endogenous Cushing's syndrome.
CannabidiolAn active cannabinoid used as an adjunctive treatment for the management of seizures associated with Lennox-Gastaut syndrome or Dravet syndrome and symptomatic relief of moderate to severe neuropathic pain or other painful conditions, like cancer.
NabiloneA synthetic delta-9-THC used in the treatment of anorexia and weight loss in HIV patients as well as nausea and vomiting in cancer chemotherapy.
Medical CannabisThe use of the plant species Cannabis sativa and Cannabis indica, popularly known as marijuana, has gained popularity in recent years for the management of a wide variety of medical...
Birch bark extractA herbal medicinal product used to treat partial thickness wounds.
StiripentolAn antiepileptic agent used in combination with other anticonvulsants to treat seizures associated with Dravet syndrome.
Telotristat ethylA tryptophan hydroxylase inhibitor that is used to treat carcinoid syndrome diarrhea.
LinzagolixA selective gonadotropin-releasing hormone (GnRH) receptor antagonist used for the symptomatic treatment of uterine fibroids.
AnacaulaseA mix of proteolytic enzymes indicated for eschar removal in adults with deep partial thickness and/or full-thickness thermal burns.
DaprodustatA small-molecule hypoxia-inducible factor prolyl hydroxylase inhibitor used for the treatment of anemia in patients with chronic kidney disease.
TezacaftorA medication used to treat homozygous or heterozygous F508del mutation cystic fibrosis.
VadadustatAn oral hypoxia-inducible factor prolyl-hydroxylase inhibitor used to treat symptomatic anemia associated with chronic kidney disease in adults on chronic maintenance dialysis.
EncorafenibA kinase inhibitor used to treat unresectable or metastatic melanoma with specific mutations.
IsavuconazoniumA triazole antifungal used for the treatment of invasive aspergillosis and mucormycosis.
Drugs & Drug Targets
DrugTargetType
Cerivastatin3-hydroxy-3-methylglutaryl-coenzyme A reductasetarget
CerivastatinCytochrome P450 2C8enzyme
CerivastatinCytochrome P450 3A4enzyme
CerivastatinCytochrome P450 2D6enzyme
CerivastatinCytochrome P450 2C9enzyme
CerivastatinCytochrome P450 3A5enzyme
CerivastatinCytochrome P450 3A7enzyme
CerivastatinP-glycoprotein 1transporter
CerivastatinCanalicular multispecific organic anion transporter 1transporter
CerivastatinATP-binding cassette sub-family G member 2transporter
CerivastatinSolute carrier organic anion transporter family member 1B1transporter
CerivastatinCytochrome P450 2B6enzyme
CerivastatinUDP-glucuronosyltransferase 1-1enzyme
CerivastatinBile salt export pumptransporter
LapatinibEpidermal growth factor receptortarget
LapatinibReceptor tyrosine-protein kinase erbB-2target
LapatinibCytochrome P450 3A4enzyme
LapatinibCytochrome P450 2C8enzyme
LapatinibP-glycoprotein 1transporter
LapatinibAntigen peptide transporter 1transporter
LapatinibCytochrome P450 3A5enzyme
LapatinibCytochrome P450 2C19enzyme
RaloxifeneEstrogen receptor alphatarget
RaloxifeneEstrogen receptor betatarget
RaloxifeneAldehyde oxidaseenzyme
RaloxifeneCytochrome P450 2C8enzyme
RaloxifeneCytochrome P450 2B6enzyme
RaloxifeneCytochrome P450 19A1enzyme
RaloxifeneCytochrome P450 3A4enzyme
RaloxifeneSerpin B9target
RaloxifeneTrefoil factor 1target
RaloxifeneUDP-glucuronosyltransferase 1-1enzyme
RaloxifeneSerum albumincarrier
RaloxifeneAlpha-1-acid glycoprotein 1carrier
RaloxifeneSolute carrier organic anion transporter family member 1B1transporter
RaloxifeneSolute carrier organic anion transporter family member 1B3transporter
RaloxifeneP-glycoprotein 1transporter
RaloxifeneATP-binding cassette sub-family G member 2transporter
RaloxifeneCanalicular multispecific organic anion transporter 1transporter
RaloxifeneCanalicular multispecific organic anion transporter 2transporter
RaloxifeneMultidrug resistance-associated protein 4transporter
RaloxifeneUDP-glucuronosyltransferase 1-10enzyme
RaloxifeneUDP-glucuronosyltransferase 1-8enzyme
QuercetinTyrosine-protein kinase HCKtarget
QuercetinCytochrome P450 2C8enzyme
QuercetinMultidrug resistance-associated protein 1transporter
QuercetinCanalicular multispecific organic anion transporter 1transporter
QuercetinMonocarboxylate transporter 2transporter
QuercetinSolute carrier organic anion transporter family member 2B1transporter
QuercetinP-glycoprotein 1transporter
QuercetinMonocarboxylate transporter 1transporter
QuercetinATP-binding cassette sub-family G member 2transporter
QuercetinPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoformtarget
QuercetinUDP-glucuronosyltransferase 3A1target
QuercetinATP synthase subunit alpha, mitochondrialtarget
QuercetinATP synthase subunit beta, mitochondrialtarget
QuercetinATP synthase subunit gamma, mitochondrialtarget
QuercetinSerine/threonine-protein kinase pim-1target
QuercetinHTH-type transcriptional regulator TtgRtarget
Quercetin3-hydroxyisobutyryl-CoA hydrolase, mitochondrialtarget
Quercetin3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZtarget
QuercetinSerine/threonine-protein kinase 17Btarget
QuercetinEstrogen receptor alphatarget
QuercetinEstrogen receptor betatarget
QuercetinRibosyldihydronicotinamide dehydrogenase [quinone]target
QuercetinSerum albumincarrier
QuercetinAryl hydrocarbon receptortarget
QuercetinCytochrome P450 1B1target
QuercetinActin, cytoplasmic 1target
QuercetinCasein kinase II subunit alphatarget
QuercetinCasein kinase II subunit betatarget
QuercetinEukaryotic translation initiation factor 3 subunit Ftarget
QuercetinHeat shock protein HSP 90-alphatarget
QuercetinHeat shock-related 70 kDa protein 2target
QuercetinRuvB-like 2target
QuercetinSplicing factor 3B subunit 3target
QuercetinUbiquitin-like modifier-activating enzyme 1target
QuercetinSex hormone-binding globulintarget
QuercetinCarbonyl reductase [NADPH] 1target
QuercetinCCAAT/enhancer-binding protein betatarget
QuercetinNuclear receptor subfamily 1 group I member 2target
QuercetinSolute carrier organic anion transporter family member 1B1transporter
QuercetinCytochrome P450 2C9enzyme
QuercetinCytochrome P450 1A2enzyme
QuercetinCytochrome P450 2E1enzyme
QuercetinCytochrome P450 2C19enzyme
QuercetinCytochrome P450 3A Subfamilyenzyme
QuercetinCytochrome P450 2D6enzyme
EthinylestradiolEstrogen receptor alphatarget
EthinylestradiolNuclear receptor subfamily 1 group I member 2target
EthinylestradiolCytochrome P450 3A4enzyme
EthinylestradiolCytochrome P450 2C8enzyme
EthinylestradiolBile salt export pumptransporter
EthinylestradiolSodium/bile acid cotransportertransporter
EthinylestradiolCanalicular multispecific organic anion transporter 1transporter
EthinylestradiolP-glycoprotein 1transporter
EthinylestradiolUDP-glucuronosyltransferase 1-1enzyme
EthinylestradiolCytochrome P450 2C19enzyme
EthinylestradiolUDP-glucuronosyltransferase 1-4enzyme
EthinylestradiolUDP-glucuronosyltransferase 1-9enzyme
EthinylestradiolCytochrome P450 2C9enzyme
EthinylestradiolCytochrome P450 1A2enzyme
EthinylestradiolEstrogen sulfotransferaseenzyme
EthinylestradiolSulfotransferase 1A3/1A4enzyme
EthinylestradiolCytochrome P450 3A5enzyme
EthinylestradiolUDP-glucuronosyltransferase 2B7enzyme
EthinylestradiolUDP-glucuronosyltransferase 1-3enzyme
EthinylestradiolCatechol O-methyltransferaseenzyme
EthinylestradiolSolute carrier organic anion transporter family member 1A2transporter
EthinylestradiolSerum albumincarrier
EthinylestradiolSex hormone-binding globulincarrier
ColchicineTubulin beta chaintarget
ColchicineCytochrome P450 3A4enzyme
ColchicineP-glycoprotein 1transporter
ColchicineCytochrome P450 2B6enzyme
ColchicineCytochrome P450 2C8enzyme
ColchicineCytochrome P450 2E1enzyme
ColchicineSerum albumincarrier
IsoniazidCatalase-peroxidasetarget
IsoniazidEnoyl-[acyl-carrier-protein] reductase [NADH]target
IsoniazidCytochrome P450 2E1enzyme
IsoniazidCytochrome P450 1A2enzyme
IsoniazidCytochrome P450 2C9enzyme
IsoniazidCytochrome P450 2D6enzyme
IsoniazidCytochrome P450 2C19enzyme
IsoniazidArylamine N-acetyltransferase 2enzyme
IsoniazidArylamine N-acetyltransferaseenzyme
IsoniazidCytochrome P450 2A6enzyme
IsoniazidCytochrome P450 2C8enzyme
IsoniazidCytochrome P450 2C8target
IsoniazidCytochrome P450 1A2target
IsoniazidCytochrome P450 3A4target
IsoniazidCytochrome P450 2C19target
IsoniazidDihydrofolate reductasetarget
IsoniazidSerum albumincarrier
IsoniazidCytochrome P450 3A4enzyme
MetronidazoleOxygen-insensitive NADPH nitroreductasetarget
MetronidazoleCytochrome P450 2C9enzyme
MetronidazoleCytochrome P450 3A4enzyme
MetronidazoleCytochrome P450 2C8enzyme
MetronidazoleUDP-glucuronosyltransferase 1-1enzyme
MetronidazoleAnaerobic bacterial DNAtarget
MetronidazoleProtozoal DNAtarget
MetronidazoleP-glycoprotein 1transporter
MetronidazoleCytochrome P450 2A6enzyme
MetronidazoleCytochrome P450 3A5enzyme
MetronidazoleCytochrome P450 3A7enzyme
NilutamideAndrogen receptortarget
NilutamideCytochrome P450 2C19enzyme
NilutamideNADPH--cytochrome P450 reductaseenzyme
PhenelzineMembrane primary amine oxidasetarget
PhenelzineAmine oxidase [flavin-containing] Btarget
PhenelzineAmine oxidase [flavin-containing] Atarget
PhenelzineAmine oxidase [flavin-containing] Aenzyme
PhenelzineAmine oxidase [flavin-containing] Benzyme
PhenelzineCytochrome P450 2E1enzyme
Phenelzine4-aminobutyrate aminotransferase, mitochondrialtarget
PhenelzineGlutamic acid decarboxylasetarget
PhenelzineAlanine aminotransferase 1target
PhenelzineAlanine aminotransferase 2target
PhenelzineCytochrome P450 2C19enzyme
PhenelzineCytochrome P450 2C8enzyme
PhenelzineCytochrome P450 3A4enzyme
PhenelzineCytochrome P450 3A5enzyme
PhenelzineCytochrome P450 3A7enzyme
PhenelzineCytochrome P450 2D6enzyme
PhenelzineCytochrome P450 3A Subfamilyenzyme
SulfaphenazoleCytochrome P450 2C9enzyme
SulfaphenazoleCytochrome P450 2B6enzyme
SulfaphenazoleCytochrome P450 2C8enzyme
SulfaphenazoleCytochrome P450 2D6enzyme
SulfaphenazoleDihydropteroate synthasetarget
TerfenadineHistamine H1 receptortarget
TerfenadinePotassium voltage-gated channel subfamily H member 2target
TerfenadineCytochrome P450 3A4enzyme
TerfenadineCytochrome P450 2D6enzyme
TerfenadineMuscarinic acetylcholine receptor M3target
TerfenadineCytochrome P450 3A5enzyme
TerfenadineCytochrome P450 3A7enzyme
TerfenadineP-glycoprotein 1transporter
TerfenadineCytochrome P450 2C8enzyme
TerfenadineCytochrome P450 2J2enzyme
TerfenadineMuscarinic acetylcholine receptor M1target
TerfenadineMuscarinic acetylcholine receptor M5target
TerfenadineMuscarinic acetylcholine receptor M4target
TerfenadineMuscarinic acetylcholine receptor M2target
TerfenadineBile salt export pumptransporter
Terfenadinealpha1-acid glycoproteincarrier
TerfenadineSerum albumincarrier
TriazolamCytochrome P450 3A4enzyme
TriazolamCytochrome P450 3A5enzyme
TriazolamCytochrome P450 3A7enzyme
TriazolamCytochrome P450 2C8enzyme
TriazolamGABA(A) Receptor Benzodiazepine Binding Sitetarget
TriazolamGABA(A) Receptortarget
DiethylstilbestrolEstrogen receptor alphatarget
DiethylstilbestrolEstrogen-related receptor gammatarget
DiethylstilbestrolTransthyretincarrier
DiethylstilbestrolCatechol O-methyltransferaseenzyme
DiethylstilbestrolCytochrome P450 19A1enzyme
DiethylstilbestrolATP-binding cassette sub-family G member 2transporter
DiethylstilbestrolP-glycoprotein 1transporter
DiethylstilbestrolEstrogen receptor betatarget
DiethylstilbestrolCytochrome P450 3A4enzyme
DiethylstilbestrolCytochrome P450 2C8enzyme
DiethylstilbestrolCytochrome P450 2C9enzyme
DiethylstilbestrolCytochrome P450 2E1enzyme
DiethylstilbestrolSteroid hormone receptor ERR1target
DiethylstilbestrolSteroid hormone receptor ERR2target
DiethylstilbestrolNuclear receptor coactivator 2target
DiethylstilbestrolNuclear receptor subfamily 1 group I member 2target
DiethylstilbestrolAndrogen receptortarget
DiethylstilbestrolSex hormone-binding globulintarget
DiethylstilbestrolSolute carrier organic anion transporter family member 1B1transporter
DiethylstilbestrolSolute carrier organic anion transporter family member 2B1transporter
DiethylstilbestrolBile salt export pumptransporter
VismodegibSmoothened homologtarget
VismodegibCytochrome P450 2C9enzyme
VismodegibCytochrome P450 3A4enzyme
VismodegibP-glycoprotein 1transporter
VismodegibCytochrome P450 2C8enzyme
VismodegibCytochrome P450 2C19enzyme
VismodegibATP-binding cassette sub-family G member 2transporter
VismodegibSerum albumincarrier
VismodegibAlpha-1-acid glycoprotein 1carrier
RegorafenibCytochrome P450 3A4enzyme
RegorafenibUDP-glucuronosyltransferase 1-9enzyme
RegorafenibProto-oncogene tyrosine-protein kinase receptor Rettarget
RegorafenibVascular endothelial growth factor receptor 1target
RegorafenibVascular endothelial growth factor receptor 2target
RegorafenibVascular endothelial growth factor receptor 3target
RegorafenibMast/stem cell growth factor receptor Kittarget
RegorafenibPlatelet-derived growth factor receptor alphatarget
RegorafenibPlatelet-derived growth factor receptor betatarget
RegorafenibFibroblast growth factor receptor 1target
RegorafenibFibroblast growth factor receptor 2target
RegorafenibAngiopoietin-1 receptortarget
RegorafenibDiscoidin domain-containing receptor 2target
RegorafenibHigh affinity nerve growth factor receptortarget
RegorafenibEphrin type-A receptor 2target
RegorafenibRAF proto-oncogene serine/threonine-protein kinasetarget
RegorafenibSerine/threonine-protein kinase B-raftarget
RegorafenibCytochrome P450 2C8enzyme
RegorafenibCytochrome P450 2C9enzyme
RegorafenibCytochrome P450 2B6enzyme
RegorafenibMitogen-activated protein kinase 11target
RegorafenibTyrosine-protein kinase FRKtarget
RegorafenibTyrosine-protein kinase ABL1target
RegorafenibP-glycoprotein 1transporter
RegorafenibATP-binding cassette sub-family G member 2transporter
RegorafenibUDP-glucuronosyltransferase 1-1enzyme
RegorafenibCytochrome P450 2C19enzyme
LumacaftorCytochrome P450 2B6enzyme
LumacaftorCytochrome P450 2C8enzyme
LumacaftorCytochrome P450 2C9enzyme
LumacaftorCytochrome P450 2C19enzyme
LumacaftorSerum albumincarrier
LumacaftorCystic fibrosis transmembrane conductance regulatortarget
LumacaftorCytochrome P450 3A4enzyme
LumacaftorP-glycoprotein 1transporter
MidostaurinProtein kinase C alpha typetarget
MidostaurinVascular endothelial growth factor receptor 2target
MidostaurinMast/stem cell growth factor receptor Kittarget
MidostaurinPlatelet-derived growth factor receptor alphatarget
MidostaurinPlatelet-derived growth factor receptor betatarget
MidostaurinReceptor-type tyrosine-protein kinase FLT3target
MidostaurinCytochrome P450 3A Subfamilyenzyme
MidostaurinCytochrome P450 1A2enzyme
MidostaurinCytochrome P450 2B6enzyme
MidostaurinCytochrome P450 2C8enzyme
MidostaurinCytochrome P450 2C9enzyme
MidostaurinCytochrome P450 2C19enzyme
MidostaurinCytochrome P450 2D6enzyme
MidostaurinCytochrome P450 2E1enzyme
MidostaurinCytochrome P450 3A4enzyme
MidostaurinCytochrome P450 3A5enzyme
MidostaurinCytochrome P450 3A7enzyme
MidostaurinCytochrome P450 3A43enzyme
EnasidenibCytochrome P450 1A2enzyme
EnasidenibCytochrome P450 2B6enzyme
EnasidenibIsocitrate dehydrogenase [NADP], mitochondrialtarget
EnasidenibCytochrome P450 2C8enzyme
EnasidenibCytochrome P450 2C9enzyme
EnasidenibCytochrome P450 2C19enzyme
EnasidenibCytochrome P450 2D6enzyme
EnasidenibCytochrome P450 3A4enzyme
EnasidenibUDP-glucuronosyltransferase 1-1enzyme
EnasidenibUDP-glucuronosyltransferase 1-3enzyme
EnasidenibUDP-glucuronosyltransferase 1-4enzyme
EnasidenibUDP-glucuronosyltransferase 1-9enzyme
EnasidenibUDP-glucuronosyltransferase 2B7enzyme
EnasidenibUDP-glucuronosyltransferase 2B15enzyme
EnasidenibP-glycoprotein 1transporter
EnasidenibATP-binding cassette sub-family G member 2transporter
EnasidenibSolute carrier family 22 member 6transporter
EnasidenibSolute carrier organic anion transporter family member 1B1transporter
EnasidenibSolute carrier family 22 member 2transporter
EnasidenibSolute carrier organic anion transporter family member 1B3transporter
EnasidenibSolute carrier family 22 member 8transporter
EnasidenibSerum albumincarrier
LetermovirUDP-glucuronosyltransferase 1-1enzyme
LetermovirUDP-glucuronosyltransferase 1-3enzyme
LetermovirSolute carrier organic anion transporter family member 1B1transporter
LetermovirSolute carrier organic anion transporter family member 1B3transporter
LetermovirCytochrome P450 2D6enzyme
LetermovirCytochrome P450 2C8enzyme
LetermovirCytochrome P450 2C19enzyme
LetermovirCytochrome P450 2C9enzyme
LetermovirCytochrome P450 2B6enzyme
LetermovirP-glycoprotein 1transporter
LetermovirATP-binding cassette sub-family G member 2transporter
LetermovirBile salt export pumptransporter
LetermovirSolute carrier family 22 member 8transporter
LetermovirCanalicular multispecific organic anion transporter 1transporter
LetermovirCMV DNA Terminase Complextarget
LetermovirCytochrome P450 3A Subfamilyenzyme
BosutinibTyrosine-protein kinase ABL1target
BosutinibTyrosine-protein kinase Lyntarget
BosutinibProto-oncogene tyrosine-protein kinase Srctarget
BosutinibP-glycoprotein 1transporter
BosutinibCytochrome P450 3A4enzyme
BosutinibDual specificity mitogen-activated protein kinase kinase 1target
BosutinibDual specificity mitogen-activated protein kinase kinase 2target
BosutinibMitogen-activated protein kinase kinase kinase 2target
BosutinibCalcium/calmodulin-dependent protein kinase type II subunit gammatarget
BosutinibCytochrome P450 2C8enzyme
BosutinibTyrosine-protein kinase Fgrtarget
BosutinibTyrosine-protein kinase HCKtarget
BosutinibTyrosine-protein kinase Tectarget
BosutinibSTE20-like serine/threonine-protein kinasetarget
DeferasiroxIrontarget
DeferasiroxCytochrome P450 3A4enzyme
DeferasiroxUDP-glucuronosyltransferase 1-1enzyme
DeferasiroxUDP-glucuronosyltransferase 1-3enzyme
DeferasiroxUDP-glucuronosyltransferase 1-9enzyme
DeferasiroxCytochrome P450 2C8enzyme
DeferasiroxCytochrome P450 1A2enzyme
RifampicinDNA-directed RNA polymerase subunit betatarget
RifampicinNuclear receptor subfamily 1 group I member 2target
RifampicinCytochrome P450 3A4enzyme
RifampicinCytochrome P450 1A2enzyme
RifampicinCytochrome P450 2C8enzyme
RifampicinUDP-glucuronosyltransferase 1-1enzyme
RifampicinCytochrome P450 2C9enzyme
RifampicinCytochrome P450 2B6enzyme
RifampicinCytochrome P450 2C19enzyme
RifampicinCanalicular multispecific organic anion transporter 2transporter
RifampicinMultidrug resistance-associated protein 5transporter
RifampicinP-glycoprotein 1transporter
RifampicinCanalicular multispecific organic anion transporter 1transporter
RifampicinSolute carrier organic anion transporter family member 2B1transporter
RifampicinBile salt export pumptransporter
RifampicinMultidrug resistance-associated protein 1transporter
RifampicinSolute carrier organic anion transporter family member 1A2transporter
RifampicinSolute carrier organic anion transporter family member 1B3transporter
RifampicinSolute carrier family 22 member 7transporter
RifampicinSolute carrier organic anion transporter family member 1B1transporter
RifampicinCytochrome P450 2A6enzyme
RifampicinCytochrome P450 2E1enzyme
RifampicinCytochrome P450 3A43enzyme
RifampicinCytochrome P450 3A7enzyme
RifampicinSolute carrier family 22 member 6transporter
RifampicinSolute carrier family 22 member 8transporter
RifampicinUDP-glucuronosyltransferase 1-9enzyme
RifampicinCytochrome P450 3A5enzyme
RifampicinSerum albumincarrier
Rifampicinalpha1-acid glycoproteincarrier
VerapamilATP-sensitive inward rectifier potassium channel 11target
VerapamilVoltage-dependent T-type calcium channel subunit alpha-1Gtarget
VerapamilPotassium voltage-gated channel subfamily H member 2target
VerapamilVoltage-dependent L-type calcium channel subunit alpha-1Ctarget
VerapamilCytochrome P450 1A2enzyme
VerapamilCytochrome P450 3A5enzyme
VerapamilVoltage-dependent N-type calcium channel subunit alpha-1Btarget
VerapamilVoltage-dependent P/Q-type calcium channel subunit alpha-1Atarget
VerapamilSodium-dependent serotonin transportertarget
VerapamilCytochrome P450 3A4enzyme
VerapamilP-glycoprotein 1transporter
VerapamilSolute carrier family 22 member 1transporter
VerapamilCanalicular multispecific organic anion transporter 2transporter
VerapamilMultidrug resistance-associated protein 4transporter
VerapamilSolute carrier family 22 member 5transporter
VerapamilSolute carrier organic anion transporter family member 1A2transporter
VerapamilMultidrug resistance-associated protein 7transporter
VerapamilSolute carrier family 22 member 4transporter
VerapamilSolute carrier organic anion transporter family member 1B1transporter
VerapamilCytochrome P450 2C8enzyme
VerapamilCytochrome P450 2C9enzyme
VerapamilCytochrome P450 2B6enzyme
VerapamilCytochrome P450 2C19enzyme
VerapamilCytochrome P450 2D6enzyme
VerapamilAlpha-1A adrenergic receptortarget
VerapamilAlpha-1B adrenergic receptortarget
VerapamilAlpha-1D adrenergic receptortarget
VerapamilSerum albumincarrier
VerapamilAlpha-1-acid glycoprotein 1carrier
VerapamilCytochrome P450 2C18enzyme
VerapamilCytochrome P450 2E1enzyme
VerapamilMultidrug resistance-associated protein 1transporter
VerapamilMultidrug and toxin extrusion protein 1transporter
VerapamilMultidrug and toxin extrusion protein 2transporter
VerapamilVoltage-dependent T-type calcium channel subunit alpha-1Htarget
VerapamilVoltage-dependent calcium channeltarget
VerapamilP-glycoprotein 1target
Simvastatin3-hydroxy-3-methylglutaryl-coenzyme A reductasetarget
SimvastatinCytochrome P450 3A4enzyme
SimvastatinCytochrome P450 2C8enzyme
SimvastatinCytochrome P450 2C9enzyme
SimvastatinCytochrome P450 3A5enzyme
SimvastatinP-glycoprotein 1transporter
SimvastatinSolute carrier organic anion transporter family member 1A2transporter
SimvastatinSolute carrier organic anion transporter family member 1B1transporter
SimvastatinCytochrome P450 2B6enzyme
SimvastatinCytochrome P450 2D6enzyme
SimvastatinUDP-glucuronosyltransferase 1-1enzyme
SimvastatinUDP-glucuronosyltransferase 1-3enzyme
SimvastatinUDP-glucuronosyltransferase 2B7enzyme
SimvastatinCanalicular multispecific organic anion transporter 1transporter
SimvastatinIntegrin alpha-Ltarget
SimvastatinBile salt export pumptransporter
SimvastatinCytochrome P450 2C19enzyme
SimvastatinSolute carrier organic anion transporter family member 2B1transporter
SimvastatinSolute carrier organic anion transporter family member 1B3transporter
SimvastatinHistone deacetylase 2target
SimvastatinCocaine esteraseenzyme
SimvastatinLiver carboxylesterase 1enzyme
SulfinpyrazoneMultidrug resistance-associated protein 1target
SulfinpyrazoneCanalicular multispecific organic anion transporter 1target
SulfinpyrazoneFatty acid-binding protein, intestinalcarrier
SulfinpyrazoneCytochrome P450 2C9enzyme
SulfinpyrazoneCanalicular multispecific organic anion transporter 2transporter
SulfinpyrazoneMultidrug resistance-associated protein 4transporter
SulfinpyrazoneMultidrug resistance-associated protein 5transporter
SulfinpyrazoneMultidrug resistance-associated protein 6transporter
SulfinpyrazoneMultidrug resistance-associated protein 1transporter
SulfinpyrazoneCanalicular multispecific organic anion transporter 1transporter
SulfinpyrazoneCytochrome P450 3A4enzyme
SulfinpyrazoneCytochrome P450 2B6enzyme
SulfinpyrazoneCytochrome P450 2C8enzyme
SulfinpyrazoneSolute carrier family 22 member 12target
SulfinpyrazoneNuclear receptor subfamily 1 group I member 2target
SulfinpyrazoneBile salt export pumptransporter
MontelukastCysteinyl leukotriene receptor 1target
MontelukastArachidonate 5-lipoxygenasetarget
MontelukastCytochrome P450 3A4enzyme
MontelukastCytochrome P450 2C9enzyme
MontelukastCytochrome P450 2C8enzyme
MontelukastSolute carrier organic anion transporter family member 2B1transporter
MontelukastProstaglandin G/H synthase 1enzyme
MontelukastCytochrome P450 2A6enzyme
NilvadipineCytochrome P450 3A4enzyme
NilvadipineCytochrome P450 2A6enzyme
NilvadipineCytochrome P450 2C19enzyme
NilvadipineCytochrome P450 2C8enzyme
NilvadipineCytochrome P450 2E1enzyme
NilvadipineVoltage-dependent L-type calcium channel subunit alpha-1Ctarget
NilvadipineVoltage-dependent calcium channel subunit alpha-2/delta-1target
NilvadipineVoltage-dependent L-type calcium channel subunit beta-2target
NilvadipineVoltage-dependent L-type calcium channel subunit alpha-1Dtarget
NilvadipineVoltage-dependent L-type calcium channel subunit alpha-1Starget
NilvadipineVoltage-dependent calcium channel subunit alpha-2/delta-3target
NilvadipineVoltage-dependent T-type calcium channel subunit alpha-1Htarget
NilvadipineVoltage-dependent T-type calcium channel subunit alpha-1Itarget
NilvadipineVoltage gated L-type calcium channeltarget
NilvadipineVoltage-dependent T-type calcium channeltarget
LiotrixThyroid hormone receptor alphatarget
LiotrixThyroid hormone receptor betatarget
LiotrixCytochrome P450 2C8enzyme
LiotrixSolute carrier organic anion transporter family member 1A2transporter
LiotrixSolute carrier organic anion transporter family member 1B1transporter
LiotrixSolute carrier organic anion transporter family member 1B3transporter
LiotrixSolute carrier organic anion transporter family member 4C1transporter
LiotrixSodium/bile acid cotransportertransporter
LiotrixSolute carrier organic anion transporter family member 1C1transporter
LiotrixSolute carrier organic anion transporter family member 4A1transporter
LiotrixSolute carrier family 22 member 8transporter
LiotrixMonocarboxylate transporter 8transporter
LiotrixMonocarboxylate transporter 10transporter
LiotrixP-glycoprotein 1transporter
LiotrixTransthyretincarrier
LiotrixThyroxine-binding globulincarrier
LiotrixSerum albumincarrier
LiotrixCytochrome P450 3A4enzyme
MometasoneGlucocorticoid receptortarget
MometasoneCytochrome P450 2C8enzyme
MometasoneProgesterone receptortarget
MometasoneCytochrome P450 3A4enzyme
MometasoneCytochrome P450 3A5enzyme
MifepristoneProgesterone receptortarget
MifepristoneGlucocorticoid receptortarget
MifepristoneCytochrome P450 3A4enzyme
MifepristoneCytochrome P450 3A5enzyme
MifepristoneP-glycoprotein 1transporter
MifepristoneMultidrug resistance-associated protein 1transporter
MifepristoneCytochrome P450 2D6enzyme
MifepristoneProstate-specific antigentarget
MifepristoneNuclear receptor subfamily 1 group I member 2target
MifepristoneBile salt export pumptransporter
MifepristoneCytochrome P450 2C8enzyme
MifepristoneCytochrome P450 2C9enzyme
MifepristoneSolute carrier organic anion transporter family member 1B1transporter
MifepristoneSolute carrier organic anion transporter family member 1B3transporter
VemurafenibSerum albumincarrier
VemurafenibAlpha-1-acid glycoprotein 1carrier
VemurafenibCytochrome P450 1A2enzyme
VemurafenibCytochrome P450 2D6enzyme
VemurafenibCytochrome P450 3A4enzyme
VemurafenibSerine/threonine-protein kinase B-raftarget
VemurafenibMultidrug resistance-associated protein 1transporter
VemurafenibATP-binding cassette sub-family G member 2transporter
VemurafenibCytochrome P450 2C9enzyme
VemurafenibCytochrome P450 2C8enzyme
VemurafenibCytochrome P450 2B6enzyme
VemurafenibP-glycoprotein 1transporter
SorafenibSerine/threonine-protein kinase B-raftarget
SorafenibReceptor-type tyrosine-protein kinase FLT3target
SorafenibRAF proto-oncogene serine/threonine-protein kinasetarget
SorafenibVascular endothelial growth factor receptor 3target
SorafenibPlatelet-derived growth factor receptor betatarget
SorafenibMast/stem cell growth factor receptor Kittarget
SorafenibVascular endothelial growth factor receptor 2target
SorafenibCytochrome P450 3A4enzyme
SorafenibUDP-glucuronosyltransferase 1-9enzyme
SorafenibCytochrome P450 2B6enzyme
SorafenibCytochrome P450 2C8enzyme
SorafenibCytochrome P450 3A5enzyme
SorafenibCytochrome P450 3A7enzyme
SorafenibCytochrome P450 2C9enzyme
SorafenibMultidrug resistance-associated protein 4transporter
SorafenibP-glycoprotein 1transporter
SorafenibCanalicular multispecific organic anion transporter 1transporter
SorafenibATP-binding cassette sub-family G member 2transporter
SorafenibCytochrome P450 1A2enzyme
SorafenibCytochrome P450 2C19enzyme
SorafenibCytochrome P450 2D6enzyme
SorafenibUDP-glucuronosyltransferase 1-1enzyme
SorafenibRalA-binding protein 1transporter
SorafenibFibroblast growth factor receptor 1target
SorafenibProto-oncogene tyrosine-protein kinase receptor Rettarget
SorafenibVascular endothelial growth factor receptor 1target
SorafenibSolute carrier organic anion transporter family member 1B1transporter
EltrombopagThrombopoietin receptortarget
EltrombopagCytochrome P450 2C8enzyme
EltrombopagCytochrome P450 1A2enzyme
EltrombopagUDP-glucuronosyltransferase 1-1enzyme
EltrombopagUDP-glucuronosyltransferase 1-3enzyme
EltrombopagSolute carrier organic anion transporter family member 1B1transporter
EltrombopagATP-binding cassette sub-family G member 2transporter
EltrombopagUDP-glucuronosyltransferase 1-9enzyme
LicofeloneArachidonate 5-lipoxygenasetarget
LicofeloneProstaglandin G/H synthase 2target
LicofeloneGroup IIE secretory phospholipase A2target
LicofeloneCytochrome P450 2C9enzyme
LicofeloneCytochrome P450 2C8enzyme
LicofeloneCytochrome P450 2J2enzyme
LicofeloneUDP-glucuronosyltransferase 1-3enzyme
BezafibratePeroxisome proliferator-activated receptor alphatarget
BezafibrateSolute carrier organic anion transporter family member 1B1transporter
BezafibratePeroxisome proliferator-activated receptor deltatarget
BezafibratePeroxisome proliferator-activated receptor gammatarget
BezafibrateCytochrome P450 1A1enzyme
BezafibrateCytochrome P450 2C8enzyme
BezafibrateCytochrome P450 3A4enzyme
BezafibrateNuclear receptor subfamily 1 group I member 2target
BezafibrateRetinoic acid receptor RXR-alphatarget
BezafibrateRetinoic acid receptor RXR-betatarget
BezafibrateRetinoic acid receptor RXR-gammatarget
IdelalisibPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoformtarget
IdelalisibATP-binding cassette sub-family G member 2transporter
IdelalisibP-glycoprotein 1transporter
IdelalisibAldehyde oxidaseenzyme
IdelalisibCytochrome P450 2C8enzyme
IdelalisibCytochrome P450 2C19enzyme
IdelalisibCytochrome P450 2B6enzyme
IdelalisibCytochrome P450 3A4enzyme
IdelalisibSolute carrier organic anion transporter family member 1B1transporter
IdelalisibSolute carrier organic anion transporter family member 1B3transporter
IdelalisibCytochrome P450 3A5enzyme
IdelalisibCytochrome P450 3A43enzyme
IdelalisibCytochrome P450 3A7enzyme
IdelalisibUDP-glucuronosyltransferase 1-4enzyme
CandesartanType-1 angiotensin II receptortarget
CandesartanCytochrome P450 2C8enzyme
CandesartanCytochrome P450 2C9enzyme
CandesartanP-glycoprotein 1transporter
CandesartanUDP-glucuronosyltransferase 1-3enzyme
CandesartanProstaglandin G/H synthase 1enzyme
CandesartanSolute carrier organic anion transporter family member 1B1transporter
IsavuconazoleCytochrome P450 3A4enzyme
IsavuconazoleCytochrome P450 3A5enzyme
IsavuconazoleCytochrome P450 2C8enzyme
IsavuconazoleCytochrome P450 2C9enzyme
IsavuconazoleCytochrome P450 2C19enzyme
IsavuconazoleCytochrome P450 2D6enzyme
IsavuconazoleCytochrome P450 2B6enzyme
IsavuconazoleUDP-glucuronosyltransferase 1-9enzyme
IsavuconazoleUDP-glucuronosyltransferase 1-8enzyme
IsavuconazoleP-glycoprotein 1transporter
IsavuconazoleATP-binding cassette sub-family G member 2transporter
IsavuconazoleSolute carrier family 22 member 2transporter
IsavuconazoleLanosterol 14-alpha demethylasetarget
IsavuconazolePotassium voltage-gated channel subfamily H member 2target
IsavuconazoleVoltage-dependent L-type calcium channel subunit alpha-1Ctarget
IsavuconazoleG protein-activated inward rectifier potassium channel 2target
IsavuconazoleG protein-activated inward rectifier potassium channel 3target
IsavuconazoleATP-sensitive inward rectifier potassium channel 11target
IsavuconazolePotassium voltage-gated channel subfamily A member 5target
IsavuconazolePotassium voltage-gated channel subfamily D member 3target
IsavuconazolePotassium voltage-gated channel subfamily KQT member 1target
IsavuconazoleSodium channel protein type 5 subunit alphatarget
OpicaponeCytochrome P450 2C19enzyme
OpicaponeCytochrome P450 2C8enzyme
OpicaponeCatechol O-methyltransferasetarget
OpicaponeSolute carrier organic anion transporter family member 1B1transporter
OpicaponeP-glycoprotein 1transporter
OpicaponeATP-binding cassette sub-family G member 2transporter
OpicaponeSolute carrier organic anion transporter family member 1B3transporter
OpicaponeSolute carrier organic anion transporter family member 2B1transporter
OpicaponeCytochrome P450 2C9enzyme
OpicaponeCytochrome P450 1A2enzyme
OpicaponeCytochrome P450 2B6enzyme
RifamycinCytochrome P450 3A4enzyme
RifamycinCytochrome P450 2C19enzyme
RifamycinCytochrome P450 2B6enzyme
RifamycinCytochrome P450 2C8enzyme
RifamycinCytochrome P450 2C9enzyme
RifamycinSolute carrier organic anion transporter family member 1A2transporter
RifamycinSolute carrier organic anion transporter family member 1B1transporter
RifamycinSolute carrier organic anion transporter family member 1B3transporter
RifamycinSolute carrier organic anion transporter family member 2A1transporter
RifamycinSolute carrier organic anion transporter family member 2B1transporter
RifamycinSerum albumincarrier
RifamycinDNA-directed RNA polymerase subunit betatarget
RifamycinDNA-directed RNA polymerase subunit alphatarget
RifamycinDNA-directed RNA polymerase subunit beta'target
RifamycinMultidrug and toxin extrusion protein 1transporter
RifamycinCytochrome P450 1A2enzyme
RifamycinP-glycoprotein 1transporter
RifamycinCytochrome P450 2D6enzyme
TriclabendazoleCytochrome P450 1A2enzyme
TriclabendazoleCytochrome P450 2C9enzyme
TriclabendazoleExcretory Secretory (ES) proteinstarget
TriclabendazoleCytochrome P450 3A4enzyme
TriclabendazoleCytochrome P450 1A1enzyme
TriclabendazoleCytochrome P450 1B1enzyme
TriclabendazoleCytochrome P450 2C19enzyme
TriclabendazoleCytochrome P450 2D6enzyme
TriclabendazoleCytochrome P450 2A6enzyme
TriclabendazoleCytochrome P450 2C8enzyme
TriclabendazoleCytochrome P450 2B6enzyme
AlpelisibPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoformtarget
AlpelisibCytochrome P450 3A4enzyme
AlpelisibCytochrome P450 2C9enzyme
AlpelisibCytochrome P450 2C8enzyme
AlpelisibCytochrome P450 2C19enzyme
AlpelisibATP-binding cassette sub-family G member 2transporter
AlpelisibP-glycoprotein 1transporter
BalaglitazoneCytochrome P450 3A4enzyme
BalaglitazoneCytochrome P450 2C8enzyme
CiglitazonePeroxisome proliferator-activated receptor gammatarget
CiglitazoneCytochrome P450 3A4enzyme
CiglitazoneCytochrome P450 2C8enzyme
LobeglitazoneSolute carrier organic anion transporter family member 1B1transporter
LobeglitazoneSolute carrier organic anion transporter family member 3A1transporter
LobeglitazoneP-glycoprotein 1transporter
LobeglitazoneCytochrome P450 1A2enzyme
LobeglitazoneCytochrome P450 2C9enzyme
LobeglitazoneCytochrome P450 2C19enzyme
LobeglitazonePeroxisome proliferator-activated receptor gammatarget
LobeglitazoneCytochrome P450 3A4enzyme
LobeglitazoneCytochrome P450 2C8enzyme
NetoglitazoneCytochrome P450 3A4enzyme
NetoglitazoneCytochrome P450 2C8enzyme
RivoglitazoneCytochrome P450 3A4enzyme
RivoglitazoneCytochrome P450 2C8enzyme
Mometasone furoateGlucocorticoid receptortarget
Mometasone furoateCytochrome P450 2C8enzyme
Mometasone furoateProgesterone receptortarget
Mometasone furoateCytochrome P450 3A4enzyme
Mometasone furoateCytochrome P450 3A5enzyme
TolbutamideATP-sensitive inward rectifier potassium channel 1target
TolbutamideCytochrome P450 2C19enzyme
TolbutamideCytochrome P450 2C9enzyme
TolbutamideCytochrome P450 2C8enzyme
TolbutamideATP-binding cassette sub-family C member 8target
TolbutamideSolute carrier family 15 member 1transporter
TolbutamideSolute carrier organic anion transporter family member 1A2transporter
TolbutamideSolute carrier family 15 member 2transporter
TolbutamideSolute carrier family 22 member 6transporter
TolbutamideSolute carrier organic anion transporter family member 2B1transporter
TolbutamideCytochrome P450 2C18enzyme
TolbutamideSerum albumincarrier
NifedipineCytochrome P450 3A4enzyme
NifedipineCytochrome P450 2E1enzyme
NifedipineCytochrome P450 2D6enzyme
NifedipineCalmodulintarget
NifedipineVoltage-dependent L-type calcium channel subunit alpha-1Dtarget
NifedipineVoltage-dependent L-type calcium channel subunit alpha-1Starget
NifedipineVoltage-dependent L-type calcium channel subunit alpha-1Ctarget
NifedipineVoltage-dependent L-type calcium channel subunit beta-2target
NifedipinePotassium voltage-gated channel subfamily D member 3target
NifedipineVoltage-dependent T-type calcium channeltarget
NifedipineCytochrome P450 1A2enzyme
NifedipineCytochrome P450 2A6enzyme
NifedipineCytochrome P450 2C8enzyme
NifedipineCanalicular multispecific organic anion transporter 2transporter
NifedipineP-glycoprotein 1transporter
NifedipineCanalicular multispecific organic anion transporter 1transporter
NifedipineCytochrome P450 1A1enzyme
NifedipineCytochrome P450 2B6enzyme
NifedipineNuclear receptor subfamily 1 group I member 2target
NifedipineSolute carrier organic anion transporter family member 1B1transporter
NifedipineBile salt export pumptransporter
NifedipineCytochrome P450 2C9enzyme
NifedipineSerum albumincarrier
Nifedipinealpha1-acid glycoproteincarrier
NifedipineCytochrome P450 3A5enzyme
CholecalciferolVitamin D-binding proteincarrier
CholecalciferolCholesterol side-chain cleavage enzyme, mitochondrialenzyme
CholecalciferolVitamin D 25-hydroxylaseenzyme
CholecalciferolSterol 26-hydroxylase, mitochondrialenzyme
CholecalciferolCytochrome P450 2J2enzyme
CholecalciferolCytochrome P450 3A4enzyme
CholecalciferolVitamin D3 receptortarget
CholecalciferolCytochrome P450 1A1enzyme
CholecalciferolCytochrome P450 2C8enzyme
Atorvastatin3-hydroxy-3-methylglutaryl-coenzyme A reductasetarget
AtorvastatinCytochrome P450 3A4enzyme
AtorvastatinDipeptidyl peptidase 4target
AtorvastatinCytochrome P450 2D6enzyme
AtorvastatinCytochrome P450 2C9enzyme
AtorvastatinCytochrome P450 2C19enzyme
AtorvastatinCytochrome P450 3A5enzyme
AtorvastatinCytochrome P450 3A7enzyme
AtorvastatinP-glycoprotein 1transporter
AtorvastatinSolute carrier organic anion transporter family member 1A2transporter
AtorvastatinSolute carrier organic anion transporter family member 1B1transporter
AtorvastatinMultidrug resistance-associated protein 4transporter
AtorvastatinMultidrug resistance-associated protein 5transporter
AtorvastatinMultidrug resistance-associated protein 1transporter
AtorvastatinCytochrome P450 2B6enzyme
AtorvastatinCytochrome P450 2C8enzyme
AtorvastatinAryl hydrocarbon receptortarget
AtorvastatinSolute carrier organic anion transporter family member 2B1transporter
AtorvastatinSolute carrier organic anion transporter family member 1B3transporter
AtorvastatinUDP-glucuronosyltransferase 1-1enzyme
AtorvastatinUDP-glucuronosyltransferase 1-3enzyme
AtorvastatinCanalicular multispecific organic anion transporter 1transporter
AtorvastatinBile salt export pumptransporter
AtorvastatinSerum albumincarrier
AtorvastatinHistone deacetylase 2target
AtorvastatinNuclear receptor subfamily 1 group I member 3target
LosartanType-1 angiotensin II receptortarget
LosartanCytochrome P450 3A4enzyme
LosartanCytochrome P450 2C9enzyme
LosartanP-glycoprotein 1transporter
LosartanSolute carrier family 22 member 6transporter
LosartanUDP-glucuronosyltransferase 1-1enzyme
LosartanUDP-glucuronosyltransferase 1-3enzyme
LosartanUDP-glucuronosyltransferase 1-10enzyme
LosartanUDP-glucuronosyltransferase 2B7enzyme
LosartanUDP-glucuronosyltransferase 2B17enzyme
LosartanCytochrome P450 2C19enzyme
LosartanSerum albumincarrier
LosartanSolute carrier family 22 member 12transporter
LosartanSolute carrier family 2, facilitated glucose transporter member 9transporter
LosartanBile salt export pumptransporter
LosartanCytochrome P450 2C8enzyme
Mefenamic acidProstaglandin G/H synthase 2target
Mefenamic acidProstaglandin G/H synthase 1target
Mefenamic acidCytochrome P450 2C9enzyme
Mefenamic acidCytochrome P450 2C8enzyme
Mefenamic acidSerum albumincarrier
Mefenamic acidUDP-glucuronosyltransferase 1-9enzyme
Mefenamic acidCytochrome P450 1A2enzyme
Mefenamic acidUDP-glucuronosyltransferase 2B7enzyme
TroleandomycinCytochrome P450 3A5enzyme
TroleandomycinCytochrome P450 3A43enzyme
Troleandomycin50S ribosomal protein L4target
Troleandomycin50S ribosomal protein L32target
TroleandomycinP-glycoprotein 1transporter
TroleandomycinCytochrome P450 2C8enzyme
TroleandomycinCytochrome P450 3A4enzyme
TroleandomycinNuclear receptor subfamily 1 group I member 2target
TroleandomycinCytochrome P450 3A7enzyme
EzetimibeNiemann-Pick C1-like protein 1target
EzetimibeAminopeptidase Ntarget
EzetimibeSterol O-acyltransferase 1target
EzetimibeUDP-glucuronosyltransferase 1-1enzyme
EzetimibeUDP-glucuronosyltransferase 1-3enzyme
EzetimibeP-glycoprotein 1transporter
EzetimibeCanalicular multispecific organic anion transporter 1transporter
EzetimibeSolute carrier organic anion transporter family member 1B1transporter
EzetimibeUDP-glucuronosyltransferase 2B15enzyme
EzetimibeUDP-glucuronosyltransferase 2B7enzyme
EzetimibeCytochrome P450 3A4enzyme
EzetimibeCanalicular multispecific organic anion transporter 2transporter
EzetimibeATP-binding cassette sub-family G member 2transporter
EzetimibeCytochrome P450 2C8enzyme
EzetimibeBile salt export pumptransporter
AnastrozoleCytochrome P450 19A1target
AnastrozoleP-glycoprotein 1transporter
AnastrozoleCytochrome P450 3A4enzyme
AnastrozoleCytochrome P450 3A5enzyme
AnastrozoleCytochrome P450 2C8enzyme
AnastrozoleUDP-glucuronosyltransferase 1-4enzyme
AnastrozoleUDP-glucuronosyltransferase 1-3enzyme
AnastrozoleUDP-glucuronosyltransferase 2B7enzyme
AnastrozoleCytochrome P450 1A2enzyme
AnastrozoleCytochrome P450 2C9enzyme
AbemaciclibMultidrug and toxin extrusion protein 1transporter
AbemaciclibMultidrug and toxin extrusion protein 2transporter
AbemaciclibCyclin-dependent kinase 4target
AbemaciclibCyclin-dependent kinase 6target
AbemaciclibSerum albumincarrier
Abemaciclibalpha1-acid glycoproteincarrier
AbemaciclibCytochrome P450 3A4enzyme
AbemaciclibP-glycoprotein 1transporter
AbemaciclibATP-binding cassette sub-family G member 2transporter
AbemaciclibSolute carrier family 22 member 2transporter
AbemaciclibCytochrome P450 1A2enzyme
AbemaciclibCytochrome P450 2B6enzyme
AbemaciclibCytochrome P450 2C8enzyme
AbemaciclibCytochrome P450 2C9enzyme
AbemaciclibCytochrome P450 2D6enzyme
AmlodipineCarbonic anhydrase 1target
AmlodipineCytochrome P450 3A4enzyme
AmlodipineVoltage-dependent L-type calcium channel subunit alpha-1Ctarget
AmlodipineCytochrome P450 1A1enzyme
AmlodipineCytochrome P450 2B6enzyme
AmlodipineVoltage-dependent N-type calcium channel subunit alpha-1Btarget
AmlodipineVoltage-dependent L-type calcium channel subunit beta-1target
AmlodipineVoltage-dependent calcium channel subunit alpha-2/delta-3target
AmlodipineCytochrome P450 3A5enzyme
AmlodipineP-glycoprotein 1transporter
AmlodipineCytochrome P450 2C8enzyme
AmlodipineCytochrome P450 2D6enzyme
AmlodipineSphingomyelin phosphodiesterasetarget
AmlodipineVoltage-dependent T-type calcium channel subunit alpha-1Itarget
AmlodipineVoltage-dependent N-type calcium channeltarget
AmlodipineCytochrome P450 2C19enzyme
AmlodipineCytochrome P450 2C9enzyme
ElexacaftorSolute carrier organic anion transporter family member 1B1transporter
ElexacaftorSolute carrier organic anion transporter family member 1B3transporter
ElexacaftorP-glycoprotein 1transporter
ElexacaftorSerum albumincarrier
ElexacaftorCytochrome P450 3A4enzyme
ElexacaftorCytochrome P450 3A5enzyme
ElexacaftorCytochrome P450 1A2enzyme
ElexacaftorCytochrome P450 2B6enzyme
ElexacaftorCytochrome P450 2C8enzyme
ElexacaftorCytochrome P450 2C9enzyme
ElexacaftorCytochrome P450 2C19enzyme
ElexacaftorCytochrome P450 2D6enzyme
ElexacaftorCystic fibrosis transmembrane conductance regulatortarget
FavipiravirRNA-directed RNA polymerase catalytic subunittarget
FavipiravirAldehyde oxidaseenzyme
FavipiravirXanthine dehydrogenase/oxidaseenzyme
FavipiravirCytochrome P450 2C8enzyme
FavipiravirSerum albumincarrier
Favipiraviralpha1-acid glycoproteincarrier
FavipiravirP-glycoprotein 1transporter
FavipiravirSolute carrier family 22 member 6transporter
FavipiravirSolute carrier family 22 member 8transporter
FavipiravirSolute carrier family 22 member 12transporter
FavipiravirCytochrome P450 2E1enzyme
Methylene blueGuanylate cyclase soluble subunit alpha-2target
Methylene blueNitric oxide synthase, braintarget
Methylene blueUDP-glucuronosyltransferase 1-4enzyme
Methylene blueUDP-glucuronosyltransferase 1-9enzyme
Methylene blueCytochrome P450 1A2enzyme
Methylene blueCytochrome P450 2B6enzyme
Methylene blueCytochrome P450 2C8enzyme
Methylene blueCytochrome P450 2C9enzyme
Methylene blueCytochrome P450 2C19enzyme
Methylene blueCytochrome P450 3A4enzyme
Methylene blueCytochrome P450 3A5enzyme
Methylene blueSerum albumincarrier
Methylene blueP-glycoprotein 1transporter
Methylene blueSolute carrier family 22 member 2transporter
Methylene blueMultidrug and toxin extrusion protein 2transporter
Methylene blueMultidrug and toxin extrusion protein 1transporter
Methylene blueFlavin reductase (NADPH)enzyme
Methylene blueCytochrome P450 2D6enzyme
SelpercatinibProto-oncogene tyrosine-protein kinase receptor Rettarget
SelpercatinibVascular endothelial growth factor receptor 1target
SelpercatinibVascular endothelial growth factor receptor 3target
SelpercatinibFibroblast growth factor receptor 1target
SelpercatinibFibroblast growth factor receptor 2target
SelpercatinibFibroblast growth factor receptor 3target
SelpercatinibCytochrome P450 3A4enzyme
SelpercatinibCytochrome P450 2C8enzyme
SelpercatinibCytochrome P450 3A Subfamilyenzyme
SelpercatinibP-glycoprotein 1transporter
SelpercatinibATP-binding cassette sub-family G member 2transporter
SelpercatinibMultidrug and toxin extrusion protein 1transporter
RipretinibMast/stem cell growth factor receptor Kittarget
RipretinibPlatelet-derived growth factor receptor betatarget
RipretinibAngiopoietin-1 receptortarget
RipretinibVascular endothelial growth factor receptor 2target
RipretinibSerine/threonine-protein kinase B-raftarget
RipretinibPlatelet-derived growth factor receptor alphatarget
RipretinibCytochrome P450 2C8enzyme
RipretinibPlatelet-derived growth factor receptor alphaenzyme
RipretinibSerum albumincarrier
Ripretinibalpha1-acid glycoproteincarrier
RipretinibP-glycoprotein 1transporter
RipretinibATP-binding cassette sub-family G member 2transporter
RipretinibMultidrug and toxin extrusion protein 1transporter
RipretinibCytochrome P450 3A4enzyme
RipretinibCytochrome P450 2D6enzyme
RipretinibCytochrome P450 2E1enzyme
ClofazimineCytochrome P450 3A4enzyme
ClofaziminePeroxisome proliferator-activated receptor gammatarget
ClofazimineCytochrome P450 2C8enzyme
ClofazimineCytochrome P450 2D6enzyme
ClofazimineCytochrome P450 3A5enzyme
ClofaziminePotassium voltage-gated channel subfamily A member 3target
ClofazimineSerum albumincarrier
ClofazimineP-glycoprotein 1transporter
ClofazimineATP-binding cassette sub-family G member 2transporter
ClofazimineMultidrug resistance-associated protein 1transporter
SaquinavirHuman immunodeficiency virus type 1 proteasetarget
SaquinavirCytochrome P450 3A4enzyme
SaquinavirCytochrome P450 3A5enzyme
SaquinavirAlpha-1-acid glycoprotein 1carrier
SaquinavirSerum albumincarrier
SaquinavirCytochrome P450 3A7enzyme
SaquinavirP-glycoprotein 1transporter
SaquinavirSolute carrier family 22 member 1transporter
SaquinavirSolute carrier organic anion transporter family member 1A2transporter
SaquinavirATP-binding cassette sub-family G member 2transporter
SaquinavirSolute carrier organic anion transporter family member 1B1transporter
SaquinavirMultidrug resistance-associated protein 1transporter
SaquinavirCanalicular multispecific organic anion transporter 1transporter
SaquinavirCytochrome P450 2C8enzyme
SaquinavirCytochrome P450 2D6enzyme
SaquinavirSolute carrier organic anion transporter family member 2B1transporter
SaquinavirBile salt export pumptransporter
MiconazoleCytochrome P450 2C9enzyme
MiconazoleCytochrome P450 2D6enzyme
MiconazoleCytochrome P450 3A4enzyme
MiconazoleP-glycoprotein 1transporter
MiconazoleCytochrome P450 51target
MiconazoleNitric oxide synthase, endothelialtarget
MiconazoleNitric oxide synthase, inducibletarget
MiconazoleCytochrome P450 11B1, mitochondrialenzyme
MiconazoleCytochrome P450 2A6enzyme
MiconazoleCytochrome P450 2B6enzyme
MiconazoleCytochrome P450 2C19enzyme
MiconazoleCytochrome P450 2E1enzyme
MiconazoleNuclear receptor subfamily 1 group I member 2target
MiconazoleLanosterol 14-alpha demethylaseenzyme
MiconazoleCytochrome P450 19A1enzyme
MiconazoleCalcium-activated potassium channeltarget
MiconazoleVoltage-gated Potassium Channelstarget
MiconazoleInward rectifier potassium channeltarget
MiconazoleVoltage gated L-type calcium channeltarget
MiconazoleSerum albumincarrier
MiconazoleCytochrome P450 2C8enzyme
PralsetinibProto-oncogene tyrosine-protein kinase receptor Rettarget
PralsetinibEpithelial discoidin domain-containing receptor 1target
PralsetinibNT-3 growth factor receptortarget
PralsetinibReceptor-type tyrosine-protein kinase FLT3target
PralsetinibTyrosine-protein kinase JAK1target
PralsetinibTyrosine-protein kinase JAK2target
PralsetinibHigh affinity nerve growth factor receptortarget
PralsetinibVascular endothelial growth factor receptor 2target
PralsetinibPlatelet-derived growth factor receptor betatarget
PralsetinibFibroblast growth factor receptor 1target
PralsetinibFibroblast growth factor receptor 2target
PralsetinibCytochrome P450 3A4enzyme
PralsetinibCytochrome P450 3A5enzyme
PralsetinibCytochrome P450 2D6enzyme
PralsetinibCytochrome P450 1A2enzyme
PralsetinibCytochrome P450 2C8enzyme
PralsetinibCytochrome P450 2C9enzyme
PralsetinibP-glycoprotein 1transporter
PralsetinibATP-binding cassette sub-family G member 2transporter
PralsetinibSolute carrier organic anion transporter family member 1B1transporter
PralsetinibSolute carrier organic anion transporter family member 1B3transporter
PralsetinibSolute carrier family 22 member 6transporter
PralsetinibMultidrug and toxin extrusion protein 1transporter
PralsetinibMultidrug and toxin extrusion protein 2transporter
PralsetinibBile salt export pumptransporter
LonafarnibProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alphatarget
LonafarnibP-glycoprotein 1transporter
LonafarnibProtein farnesyltransferase subunit betatarget
LonafarnibCytochrome P450 3A Subfamilyenzyme
LonafarnibCytochrome P450 2C8enzyme
LonafarnibCytochrome P450 2C19enzyme
LonafarnibCytochrome P450 1A2enzyme
LonafarnibCytochrome P450 2A6enzyme
LonafarnibCytochrome P450 2C9enzyme
LonafarnibCytochrome P450 2E1enzyme
LonafarnibSolute carrier organic anion transporter family member 1B1transporter
LonafarnibSolute carrier organic anion transporter family member 1B3transporter
LonafarnibATP-binding cassette sub-family G member 2transporter
LonafarnibCytochrome P450 3A4enzyme
LonafarnibCytochrome P450 3A5enzyme
LonafarnibCanalicular multispecific organic anion transporter 1transporter
ZafirlukastCysteinyl leukotriene receptor 1target
ZafirlukastCytochrome P450 2C9enzyme
ZafirlukastCytochrome P450 2C8enzyme
ZafirlukastProstaglandin G/H synthase 1enzyme
ZafirlukastCytochrome P450 3A4enzyme
ZafirlukastCytochrome P450 1A2enzyme
ZafirlukastCytochrome P450 2C19enzyme
ZafirlukastATP-binding cassette sub-family G member 2transporter
ZafirlukastCytochrome P450 2D6enzyme
ZafirlukastSodium/bile acid cotransportertransporter
MenadioneProthrombintarget
MenadioneVitamin K epoxide reductase complex subunit 1target
MenadioneCoagulation factor IXtarget
MenadioneVitamin K-dependent gamma-carboxylasetarget
MenadioneVitamin K-dependent protein Ctarget
MenadioneVitamin K-dependent protein Starget
MenadioneNAD(P)H dehydrogenase [quinone] 1target
MenadioneRibosyldihydronicotinamide dehydrogenase [quinone]target
MenadioneVitamin K epoxide reductase complex subunit 1-like protein 1target
MenadioneXanthine dehydrogenase/oxidaseenzyme
MenadioneAldehyde oxidaseenzyme
MenadioneMethylenetetrahydrofolate reductaseenzyme
MenadioneCytochrome P450 1A1enzyme
MenadioneOsteocalcintarget
MenadioneCytochrome P450 1A2enzyme
MenadioneCytochrome P450 2A6enzyme
MenadioneCytochrome P450 1B1enzyme
MenadioneCytochrome P450 2B6enzyme
MenadioneCytochrome P450 2C8enzyme
MenadioneCytochrome P450 2C9enzyme
MenadioneCytochrome P450 2C19enzyme
MenadioneCytochrome P450 2D6enzyme
MenadioneCytochrome P450 2E1enzyme
MenadioneCytochrome P450 3A4enzyme
MenadioneCytochrome P450 3A5enzyme
MenadioneCytochrome P450 3A7enzyme
RilpivirineCytochrome P450 3A4enzyme
RilpivirineReverse transcriptase/RNaseHtarget
RilpivirineNuclear receptor subfamily 1 group I member 2target
RilpivirineCytochrome P450 2C19enzyme
RilpivirineCytochrome P450 2B6enzyme
RilpivirineP-glycoprotein 1transporter
RilpivirineATP-binding cassette sub-family G member 2transporter
RilpivirineSolute carrier organic anion transporter family member 1B1transporter
RilpivirineSolute carrier organic anion transporter family member 1B3transporter
RilpivirineSerum albumincarrier
RilpivirineCytochrome P450 2D6enzyme
RilpivirineCytochrome P450 2C9enzyme
RilpivirineCytochrome P450 2C8enzyme
RilpivirineCytochrome P450 2E1enzyme
IbrexafungerpCytochrome P450 3A4enzyme
IbrexafungerpUDP-glucuronosyltransferases (UGTs)enzyme
IbrexafungerpSulfotransferaseenzyme
IbrexafungerpCytochrome P450 2C8enzyme
IbrexafungerpP-glycoprotein 1transporter
IbrexafungerpSolute carrier organic anion transporter family member 1B3transporter
IbrexafungerpSerum albumincarrier
Ibrexafungerp1,3-beta-glucan synthase component GSC2target
IbrexafungerpGTP-binding protein RHO1target
BrincidofovirLeukotriene-B(4) omega-hydroxylase 1enzyme
BrincidofovirSphingomyelin phosphodiesteraseenzyme
BrincidofovirDNA polymerasetarget
BrincidofovirCytochrome P450 1A2enzyme
BrincidofovirCytochrome P450 2B6enzyme
BrincidofovirCytochrome P450 2C8enzyme
BrincidofovirCytochrome P450 2C9enzyme
BrincidofovirCytochrome P450 2C19enzyme
BrincidofovirCytochrome P450 2D6enzyme
BrincidofovirATP-binding cassette sub-family G member 2transporter
BrincidofovirCanalicular multispecific organic anion transporter 1transporter
BrincidofovirBile salt export pumptransporter
BrincidofovirSolute carrier organic anion transporter family member 1B1transporter
BrincidofovirSolute carrier family 22 member 6transporter
BrincidofovirSolute carrier family 22 member 8transporter
BrincidofovirSolute carrier organic anion transporter family member 1B3transporter
BrincidofovirVariola virus DNAtarget
LevoketoconazoleCytochrome P450 11B1, mitochondrialtarget
LevoketoconazoleLanosterol 14-alpha demethylasetarget
LevoketoconazoleCytochrome P450 3A4enzyme
LevoketoconazoleCytochrome P450 3A5enzyme
LevoketoconazoleSteroid 21-hydroxylaseenzyme
LevoketoconazoleP-glycoprotein 1transporter
LevoketoconazoleSteroid 17-alpha-hydroxylase/17,20 lyasetarget
LevoketoconazoleCytochrome P450 11B2, mitochondrialtarget
LevoketoconazoleCholesterol side-chain cleavage enzyme, mitochondrialtarget
LevoketoconazoleSolute carrier family 22 member 2transporter
LevoketoconazoleMultidrug and toxin extrusion protein 1transporter
LevoketoconazoleCytochrome P450 2B6enzyme
LevoketoconazoleCytochrome P450 2C8enzyme
LevoketoconazoleCytochrome P450 1A2enzyme
LevoketoconazoleCytochrome P450 7A1enzyme
LevoketoconazoleCytochrome P450 19A1enzyme
CannabidiolCytochrome P450 2C9enzyme
CannabidiolCytochrome P450 2C19enzyme
CannabidiolCytochrome P450 2D6enzyme
CannabidiolCytochrome P450 3A4enzyme
CannabidiolCannabinoid receptor 1target
CannabidiolCannabinoid receptor 2target
CannabidiolG-protein coupled receptor 12target
CannabidiolGlycine receptor subunit alpha-1target
CannabidiolGlycine receptor (alpha-1/beta)target
CannabidiolGlycine receptor subunit alpha-3target
CannabidiolN-arachidonyl glycine receptortarget
CannabidiolG-protein coupled receptor 55target
Cannabidiol5-hydroxytryptamine receptor 1Atarget
Cannabidiol5-hydroxytryptamine receptor 2Atarget
CannabidiolNeuronal acetylcholine receptor subunit alpha-7target
CannabidiolDelta-type opioid receptortarget
CannabidiolMu-type opioid receptortarget
CannabidiolPeroxisome proliferator-activated receptor gammatarget
CannabidiolCytochrome P450 3A5enzyme
CannabidiolSerotonin N-acetyltransferaseenzyme
CannabidiolCytochrome P450 1A1enzyme
CannabidiolFatty-acid amide hydrolase 1enzyme
CannabidiolArachidonate 5-lipoxygenaseenzyme
CannabidiolArachidonate 15-lipoxygenaseenzyme
CannabidiolQuinone oxidoreductaseenzyme
CannabidiolMultidrug resistance-associated protein 1transporter
CannabidiolATP-binding cassette sub-family G member 2transporter
CannabidiolEquilibrative nucleoside transporter 1transporter
CannabidiolTransient receptor potential cation channel subfamily V member 1target
CannabidiolVoltage-dependent T-type calcium channel subunit alpha-1Gtarget
CannabidiolVoltage-dependent T-type calcium channel subunit alpha-1Htarget
CannabidiolVoltage-dependent T-type calcium channel subunit alpha-1Itarget
CannabidiolTransient receptor potential cation channel subfamily A member 1target
CannabidiolTransient receptor potential cation channel subfamily M member 8target
CannabidiolTransient receptor potential cation channel subfamily V member 2target
CannabidiolTransient receptor potential cation channel subfamily V member 3target
CannabidiolTransient receptor potential cation channel subfamily V member 4target
CannabidiolVoltage-dependent anion-selective channel protein 1target
Cannabidiol5-hydroxytryptamine receptor 3Atarget
CannabidiolAdenosine receptor A1target
CannabidiolProstaglandin G/H synthase 1target
CannabidiolProstaglandin G/H synthase 2target
CannabidiolAcetyl-CoA acetyltransferase, mitochondrialtarget
CannabidiolSteroid 17-alpha-hydroxylase/17,20 lyasetarget
Cannabidiol3-hydroxy-3-methylglutaryl-coenzyme A reductasetarget
CannabidiolGlutathione reductase, mitochondrialtarget
CannabidiolGlutathione peroxidase 1target
CannabidiolIndoleamine 2,3-dioxygenase 1target
CannabidiolCytochrome P450 1B1target
CannabidiolNAD(P)H dehydrogenase [quinone] 1target
CannabidiolCatalasetarget
CannabidiolCytochrome P450 3A5target
CannabidiolCytochrome P450 2D6target
CannabidiolSuperoxide dismutase [Cu-Zn]target
CannabidiolCytochrome P450 1A2target
CannabidiolCytochrome P450 3A7target
CannabidiolSerotonin N-acetyltransferasetarget
CannabidiolN-acylethanolamine-hydrolyzing acid amidasetarget
CannabidiolCytochrome P450 1A2enzyme
CannabidiolCytochrome P450 1B1enzyme
CannabidiolCytochrome P450 2A6enzyme
CannabidiolCytochrome P450 2B6enzyme
CannabidiolCytochrome P450 2C8enzyme
CannabidiolCytochrome P450 2E1enzyme
CannabidiolCytochrome P450 3A7enzyme
CannabidiolUDP-glucuronosyltransferase 1-7enzyme
CannabidiolUDP-glucuronosyltransferase 1-9enzyme
CannabidiolUDP-glucuronosyltransferase 2B7enzyme
CannabidiolUDP-glucuronosyltransferase 2B17enzyme
CannabidiolP-glycoprotein 1transporter
CannabidiolCytochrome P450 2J2enzyme
CannabidiolLiver carboxylesterase 1enzyme
NabiloneCannabinoid receptor 2target
NabiloneCannabinoid receptor 1target
NabiloneCytochrome P450 2E1enzyme
NabiloneCytochrome P450 2C8enzyme
NabiloneCytochrome P450 2C9enzyme
NabiloneCytochrome P450 3A4enzyme
NabiloneCytochrome P450 2J2enzyme
Medical CannabisCannabinoid receptor 1target
Medical CannabisCannabinoid receptor 2target
Medical CannabisCytochrome P450 2C9enzyme
Medical CannabisCytochrome P450 2C19enzyme
Medical CannabisCytochrome P450 2D6enzyme
Medical CannabisCytochrome P450 3A4enzyme
Medical CannabisG-protein coupled receptor 12target
Medical CannabisGlycine receptor subunit alpha-1target
Medical CannabisGlycine receptor (alpha-1/beta)target
Medical CannabisGlycine receptor subunit alpha-3target
Medical CannabisN-arachidonyl glycine receptortarget
Medical CannabisG-protein coupled receptor 55target
Medical Cannabis5-hydroxytryptamine receptor 1Atarget
Medical Cannabis5-hydroxytryptamine receptor 2Atarget
Medical CannabisNeuronal acetylcholine receptor subunit alpha-7target
Medical CannabisDelta-type opioid receptortarget
Medical CannabisMu-type opioid receptortarget
Medical CannabisPeroxisome proliferator-activated receptor gammatarget
Medical CannabisCytochrome P450 3A5enzyme
Medical CannabisCytochrome P450 3A7enzyme
Medical CannabisCytochrome P450 1A1enzyme
Medical CannabisCytochrome P450 1A2enzyme
Medical CannabisCytochrome P450 1B1enzyme
Medical CannabisArachidonate 5-lipoxygenaseenzyme
Medical CannabisArachidonate 15-lipoxygenaseenzyme
Medical CannabisSuperoxide dismutase [Cu-Zn]enzyme
Medical CannabisMultidrug resistance-associated protein 1transporter
Medical CannabisATP-binding cassette sub-family G member 2transporter
Medical CannabisEquilibrative nucleoside transporter 1transporter
Medical CannabisTransient receptor potential cation channel subfamily V member 1target
Medical CannabisVoltage-dependent T-type calcium channel subunit alpha-1Gtarget
Medical CannabisVoltage-dependent T-type calcium channel subunit alpha-1Htarget
Medical CannabisVoltage-dependent T-type calcium channel subunit alpha-1Itarget
Medical CannabisTransient receptor potential cation channel subfamily A member 1target
Medical CannabisTransient receptor potential cation channel subfamily M member 8target
Medical CannabisTransient receptor potential cation channel subfamily V member 2target
Medical CannabisTransient receptor potential cation channel subfamily V member 3target
Medical CannabisTransient receptor potential cation channel subfamily V member 4target
Medical CannabisVoltage-dependent anion-selective channel protein 1target
Medical CannabisN-acyl-phosphatidylethanolamine-hydrolyzing phospholipase Dtarget
Medical CannabisN-acylethanolamine-hydrolyzing acid amidasetarget
Medical CannabisSerotonin N-acetyltransferasetarget
Medical CannabisPhospholipase A2target
Medical CannabisSuperoxide dismutase [Cu-Zn]target
Medical CannabisFatty-acid amide hydrolase 1target
Medical CannabisCatalasetarget
Medical CannabisQuinone oxidoreductasetarget
Medical CannabisSphingomyelin phosphodiesterasetarget
Medical CannabisGlutathione peroxidase 1target
Medical CannabisGlutathione reductase, mitochondrialtarget
Medical Cannabis3-hydroxy-3-methylglutaryl-coenzyme A reductasetarget
Medical CannabisIndoleamine 2,3-dioxygenase 1target
Medical CannabisProstaglandin G/H synthase 1target
Medical CannabisProstaglandin G/H synthase 2target
Medical CannabisSteroid 17-alpha-hydroxylase/17,20 lyasetarget
Medical CannabisAcetyl-CoA acetyltransferase, mitochondrialtarget
Medical CannabisCytochrome P450 2A6enzyme
Medical CannabisCytochrome P450 2B6enzyme
Medical CannabisCytochrome P450 2C8enzyme
Medical CannabisCytochrome P450 2E1enzyme
Medical CannabisCytochrome P450 2J2enzyme
Medical CannabisUDP-glucuronosyltransferase 1-7enzyme
Medical CannabisUDP-glucuronosyltransferase 1-8enzyme
Medical CannabisUDP-glucuronosyltransferase 1-9enzyme
Medical CannabisUDP-glucuronosyltransferase 1-10enzyme
Medical CannabisUDP-glucuronosyltransferase 2B17enzyme
Medical CannabisLiver carboxylesterase 1enzyme
Medical CannabisP-glycoprotein 1transporter
Medical CannabisUDP-glucuronosyltransferase 2B7enzyme
Birch bark extractCytochrome P450 2C8enzyme
Birch bark extractCytochrome P450 3A Subfamilyenzyme
StiripentolCytochrome P450 2C19enzyme
StiripentolCytochrome P450 2D6enzyme
StiripentolCytochrome P450 3A4enzyme
StiripentolCytochrome P450 1A2enzyme
StiripentolCytochrome P450 2C9enzyme
StiripentolGABA(A) Receptortarget
StiripentolL-lactate dehydrogenase A chaintarget
StiripentolL-lactate dehydrogenase B chaintarget
StiripentolCytochrome P450 2B6enzyme
StiripentolCytochrome P450 2C8enzyme
StiripentolP-glycoprotein 1transporter
StiripentolATP-binding cassette sub-family G member 2transporter
Telotristat ethylTryptophan 5-hydroxylase 2target
Telotristat ethylTryptophan 5-hydroxylase 1target
Telotristat ethylP-glycoprotein 1transporter
Telotristat ethylCytochrome P450 3A4enzyme
Telotristat ethylCytochrome P450 2B6enzyme
Telotristat ethylLiver carboxylesterase 1enzyme
Telotristat ethylATP-binding cassette sub-family G member 2carrier
Telotristat ethylCocaine esteraseenzyme
Telotristat ethylUDP-glucuronosyltransferase 2B4enzyme
Telotristat ethylUDP-glucuronosyltransferase 2B7enzyme
Telotristat ethylCytochrome P450 2C9enzyme
Telotristat ethylCytochrome P450 2C19enzyme
Telotristat ethylCytochrome P450 2D6enzyme
Telotristat ethylCytochrome P450 2C8enzyme
LinzagolixCytochrome P450 2C8enzyme
LinzagolixGonadotropin-releasing hormone receptortarget
LinzagolixSerum albumincarrier
LinzagolixCytochrome P450 2C9enzyme
LinzagolixCytochrome P450 3A4enzyme
LinzagolixSolute carrier organic anion transporter family member 1B1transporter
LinzagolixSolute carrier organic anion transporter family member 1B3transporter
LinzagolixSolute carrier family 22 member 8transporter
LinzagolixATP-binding cassette sub-family G member 2transporter
LinzagolixSolute carrier family 22 member 6transporter
AnacaulaseCytochrome P450 2C8enzyme
AnacaulaseCytochrome P450 2C9enzyme
AnacaulaseAlpha-1-antichymotrypsintarget
AnacaulaseAlpha-2-macroglobulintarget
DaprodustatEgl nine homolog 1target
DaprodustatEgl nine homolog 2target
DaprodustatEgl nine homolog 3target
DaprodustatCytochrome P450 2C8enzyme
DaprodustatCytochrome P450 3A4enzyme
DaprodustatSolute carrier organic anion transporter family member 1B1transporter
DaprodustatSolute carrier organic anion transporter family member 1B3transporter
DaprodustatSolute carrier family 22 member 6transporter
DaprodustatSolute carrier family 22 member 8transporter
DaprodustatATP-binding cassette sub-family G member 2transporter
TezacaftorCytochrome P450 3A4enzyme
TezacaftorCytochrome P450 3A5enzyme
TezacaftorCystic fibrosis transmembrane conductance regulatortarget
TezacaftorP-glycoprotein 1transporter
TezacaftorATP-binding cassette sub-family G member 2transporter
TezacaftorSolute carrier family 22 member 2transporter
TezacaftorSolute carrier family 22 member 6transporter
TezacaftorSolute carrier family 22 member 8transporter
TezacaftorSolute carrier organic anion transporter family member 1B1transporter
TezacaftorCytochrome P450 1A2enzyme
TezacaftorCytochrome P450 2B6enzyme
TezacaftorCytochrome P450 2C8enzyme
TezacaftorCytochrome P450 2C9enzyme
TezacaftorCytochrome P450 2C19enzyme
TezacaftorCytochrome P450 2D6enzyme
TezacaftorSolute carrier organic anion transporter family member 1B3transporter
VadadustatEgl nine homolog 2target
VadadustatEgl nine homolog 3target
VadadustatEgl nine homolog 1target
VadadustatHypoxia-inducible factor 1-alphatarget
VadadustatEndothelial PAS domain-containing protein 1target
VadadustatUDP-glucuronosyltransferase 1-1enzyme
VadadustatUDP-glucuronosyltransferase 1-7enzyme
VadadustatUDP-glucuronosyltransferase 1-8enzyme
VadadustatUDP-glucuronosyltransferase 1-9enzyme
VadadustatUDP-glucuronosyltransferase 2B7enzyme
VadadustatCytochrome P450 2B6enzyme
VadadustatCytochrome P450 2C8enzyme
VadadustatCytochrome P450 3A4enzyme
VadadustatATP-binding cassette sub-family G member 2transporter
VadadustatSolute carrier family 22 member 8transporter
VadadustatSolute carrier family 22 member 6transporter
VadadustatSerum albumincarrier
VadadustatCytochrome P450 2C9enzyme
EncorafenibCytochrome P450 3A4enzyme
EncorafenibCytochrome P450 2C19enzyme
EncorafenibCytochrome P450 2D6enzyme
EncorafenibSerine/threonine-protein kinase B-raftarget
EncorafenibG1/S-specific cyclin-D1target
EncorafenibUDP-glucuronosyltransferase 1-1enzyme
EncorafenibSerum albumincarrier
EncorafenibCytochrome P450 1A2enzyme
EncorafenibCytochrome P450 2B6enzyme
EncorafenibCytochrome P450 2C8enzyme
EncorafenibCytochrome P450 2C9enzyme
EncorafenibCytochrome P450 3A5enzyme
EncorafenibCytochrome P450 3A7enzyme
EncorafenibP-glycoprotein 1transporter
EncorafenibSolute carrier family 22 member 2transporter
EncorafenibATP-binding cassette sub-family G member 2transporter
EncorafenibSolute carrier family 22 member 6transporter
EncorafenibSolute carrier family 22 member 8transporter
EncorafenibSolute carrier organic anion transporter family member 1B1transporter
EncorafenibSolute carrier organic anion transporter family member 1B3transporter
EncorafenibRAF proto-oncogene serine/threonine-protein kinasetarget
EncorafenibMitogen-activated protein kinase 8target
EncorafenibMitogen-activated protein kinase 9target
EncorafenibMitogen-activated protein kinase 10target
EncorafenibLIM domain kinase 1target
EncorafenibLIM domain kinase 2target
EncorafenibDual specificity mitogen-activated protein kinase kinase 4target
EncorafenibSerine/threonine-protein kinase 36target
IsavuconazoniumCytochrome P450 3A4enzyme
IsavuconazoniumP-glycoprotein 1transporter
IsavuconazoniumCytochrome P450 3A5enzyme
IsavuconazoniumCholinesteraseenzyme
IsavuconazoniumCytochrome P450 2C8enzyme
IsavuconazoniumCytochrome P450 2C9enzyme
IsavuconazoniumCytochrome P450 2C19enzyme
IsavuconazoniumCytochrome P450 2D6enzyme
IsavuconazoniumCytochrome P450 2B6enzyme
IsavuconazoniumATP-binding cassette sub-family G member 2transporter
IsavuconazoniumSolute carrier family 22 member 2transporter
IsavuconazoniumLanosterol 14-alpha demethylasetarget
IsavuconazoniumSerum albumincarrier