Purine Nucleosides

Name
Purine Nucleosides
Accession Number
DBCAT000252
Description

Purines with a RIBOSE attached that can be phosphorylated to PURINE NUCLEOTIDES.

Drugs
DrugDrug Description
2-FluoroadenosineNot Available
2'-deoxythioguanosineNot Annotated
3-DeazaadenosineNot Available
5-iodotubercidinNot Available
5'-Fluoro-5'-DeoxyadenosineNot Available
5'-O-(N-(Alanyl)sulfamoyl)adenosineNot Available
5'-S-methyl-5'-thioadenosineNot Available
7-MethylguanosineNot Available
8-Chloroadenosine8-Chloroadenosine is under investigation in clinical trial NCT02509546 (8-chloroadenosine in Treating Patients With Relapsed or Refractory Acute Myeloid Leukemia).
8-hydroxy-2'-deoxyguanosineNot Available
9-deazainosineNot Available
AbacavirAn antiviral nucleoside reverse transcriptase inhibitor used in combination with other antiretrovirals for the treatment of HIV.
Abacavir hydroxyacetatePrurisol is under investigation for the treatment of Chronic Stable Plaque Psoriasis. Prurisol has been investigated for the treatment of Plaque Psoriasis.
AdemetionineS-Adenosylmethionine (SAMe) is used as a drug in Europe for the treatment of depression, liver disorders, fibromyalgia, and osteoarthritis. It has also been introduced into the United States market as...
AdenosineA medication used in myocardial perfusion scintigraphy and to treat supraventricular tachycardia.
AMG-319Not Annotated
AZD-8848AZD-8848 is under investigation in clinical trial NCT01818869 (To Assess the Safety, Tolerability, Pharmacokinetics and Pharmacodynamics of Multiple Doses AZD8848 in Healthy Subjects).
BentracimabBentracimab is under investigation in clinical trial NCT04286438 (Bentracimab (PB2452) in Ticagrelor-treated Patients With Uncontrolled Major or Life-threatening Bleeding or Requiring Urgent Surgery or Invasive Procedure).
BinodenosonFor cardiac pharmacologic stress SPECT imaging, which is used to diagnose coronary artery disease.
CladribineA purine antimetabolite used to treat Multiple Sclerosis (MS) and hairy cell leukemia.
CordycepinCordycepin has been used in trials studying the treatment of Leukemia.
Deoxycytidylyl-3',5'-guanosineNot Available
DeoxyinosineNot Available
DeuremidevirDeuremidevir is a small molecule drug. Deuremidevir is under investigation in clinical trial NCT06328400 (A Study to Evaluate the Safety, Tolerability, and Pharmacokinetics of Oral Deuremidevir Hydrobromide for Suspension).
DidanosineA reverse transcriptase inhibitor used to treat HIV.
DideoxyadenosineNot Annotated
FadraciclibCYC-065 is under investigation in clinical trial NCT03739554 (CYC065 CDK Inhibitor and Venetoclax Study in Relapsed/Refractory CLL).
FludarabineA purine analog antimetabolite that inhibits DNA synthesis.
GalidesivirGalidesivir is an adenosine analogue that has been investigated for use against Zaire Ebolavirus. In animal studies, galidesivir was effective in increasing the survival rates from infections caused by various...
GS-441524An experimental nucleoside analog antiviral investigated for its use in the treatment of Ebola and SARS-CoV-2 infections.
GS-6620GS-6620 is under investigation in clinical trial NCT01316237 (A Study Evaluating the Safety, Tolerability, Pharmacokinetics and Antiviral Activity of GS-6620 in Treatment Naïve Subjects With Chronic Hepatitis C Virus Infection).
GS-9667Not Annotated
GuanosineGuanosine is a nucleoside comprising guanine attached to a ribose (ribofuranose) ring via a β-N9-glycosidic bond. Guanosine can be phosphorylated to become GMP (guanosine monophosphate), cGMP (cyclic guanosine monophosphate), GDP...
InosineA nutritional supplement touted to improve athletic performance and a drug used in vitro as a red blood cell rejuvenator for a unit of red blood cells that will be used in a clinical setting.
Inosine pranobexA medication used to treat subacute sclerosing panencephalitis.
IsatoribineFor the treatment of Hepatitis C.
IslatravirA nucleoside analog reverse transcriptase inhibitor (NRTI) indicated in combination with doravirine for the treatment of HIV-1 infection in virologically-suppressed adults on a stable antiretroviral regimen.
LodenosineLodenosine is a small molecule drug. The usage of the INN stem '-nosine' in the name indicates that Lodenosine is a purine nucleoside analogue. Lodenosine has a monoisotopic molecular weight...
LoxoribineNot Available
MethylthioinosineAn analog of inosine with a methylthio group replacing the hydroxyl group in the 6-position.
MetrifudilMetrifudil is a small molecule drug. The usage of the INN stem '-dil' in the name indicates that Metrifudil is a vasodilator. Metrifudil has a monoisotopic molecular weight of 371.16...
N(6)-dimethylallyladenineNot Available
NamodenosonNamodenoson has been used in trials studying the treatment of Chronic Hepatitis C and Hepatocellular Carcinoma.
NebularineNot Available
PiclidenosonInvestigated for use/treatment in cancer/tumors (unspecified), eye disorders/infections, psoriasis and psoriatic disorders, and rheumatoid arthritis. Can-Fite BioPharma has reported that by targeting the adenosine A3-receptor, CF101 may also be used...
PuromycinPuromycin is an antibiotic that prevents bacterial protein translation. It is utilized as a selective agent in laboratory cell cultures. Puromycin is toxic to both prokaryotic and eukaryotic cells, resulting...
S-Adenosyl-1,8-Diamino-3-ThiooctaneNot Available
S-adenosyl-L-homocysteine5'-S-(3-Amino-3-carboxypropyl)-5'-thioadenosine. Formed from S-adenosylmethionine after transmethylation reactions.
SelodenosonSelodenoson is under investigation in clinical trial NCT00040001 (Safety and Efficacy Study of an A1-adenosine Receptor Agonist to Slow Heart Rate in Atrial Fibrillation).
SinefunginSinefungin is a solid. This compound belongs to the purine nucleosides and analogues. These are compounds comprising a purine base attached to a sugar. The proteins that adenosyl-ornithine target include...
SonedenosonSonedenoson has been used in trials studying the treatment of Foot Ulcer, Diabetic and Diabetes Complications.
TecadenosonInvestigated for use/treatment in arrhythmia and atrial fibrillation.
TicagrelorA P2Y12 platelet inhibitor used in patients with a history of myocardial infarction or with acute coronary syndrome (ACS) to prevent future myocardial infarction, stroke and cardiovascular death.
TrabodenosonTrabodenoson has been used in trials studying the treatment of Ocular Hypertension (OHT) and Primary Open-Angle Glaucoma (POAG).
TubercidinAn antibiotic purine ribonucleoside that readily substitutes for adenosine in the biological system, but its incorporation into DNA and RNA has an inhibitory effect on the metabolism of these nucleic...
UK-432097UK-432,097 has been used in trials studying the treatment of Pulmonary Disease, Chronic Obstructive.
VidarabineAn antiviral agent used to treat various viral infections.
Drugs & Drug Targets
DrugTargetType
2-FluoroadenosinePurine nucleoside phosphorylase DeoD-typetarget
3-DeazaadenosineIAG-nucleoside hydrolasetarget
5-iodotubercidinCasein kinase I isoform gamma-2target
5-iodotubercidinSerine/threonine-protein kinase haspintarget
5-iodotubercidinMitogen-activated protein kinase 3target
5'-Fluoro-5'-DeoxyadenosineFluorinasetarget
5'-O-(N-(Alanyl)sulfamoyl)adenosineBifunctional glutamate/proline--tRNA ligasetarget
5'-S-methyl-5'-thioadenosineAdenosine receptor A1target
5'-S-methyl-5'-thioadenosineAdenosine receptor A2btarget
5'-S-methyl-5'-thioadenosineAdenosine receptor A2atarget
5'-S-methyl-5'-thioadenosineAdenosine receptor A3target
5'-S-methyl-5'-thioadenosineS-methyl-5'-thioadenosine phosphorylasetarget
5'-S-methyl-5'-thioadenosineType II methyltransferase M.RsrItarget
7-MethylguanosineCap-specific mRNA (nucleoside-2'-O-)-methyltransferasetarget
8-ChloroadenosineAdenosine deaminaseenzyme
8-ChloroadenosineMitochondrial ATP synthase F1 domaintarget
8-hydroxy-2'-deoxyguanosineRas-related C3 botulinum toxin substrate 1target
8-hydroxy-2'-deoxyguanosineN-glycosylase/DNA lyaseenzyme
9-deazainosinePurine nucleoside phosphorylasetarget
AbacavirAlcohol dehydrogenase 6enzyme
AbacavirUDP-glucuronosyltransferase 1A1enzyme
AbacavirReverse transcriptase/RNaseHtarget
AbacavirAdenosine kinaseenzyme
AbacavirGag-Pol polyproteintarget
AdemetionineCytochrome P450 2E1enzyme
AdemetionineArsenite methyltransferasetarget
AdemetionineCap-specific mRNA (nucleoside-2'-O-)-methyltransferase 1target
AdemetionineSpermidine synthaseenzyme
AdemetionineCatechol O-methyltransferasetarget
AdemetionineS-adenosylmethionine synthase isoform type-1target
AdemetionineCystathionine beta-synthasetarget
AdemetionineS-adenosylmethionine synthase isoform type-2target
AdemetionineS-adenosylmethionine decarboxylase proenzymetarget
AdemetionineGlycine N-methyltransferasetarget
AdenosineAdenosine kinaseenzyme
AdenosineAdenosine receptor A1target
AdenosineAdenosine receptor A2atarget
AdenosineAdenosine receptor A2btarget
AdenosineSolute carrier family 28 member 3transporter
AdenosineEquilibrative nucleoside transporter 1transporter
AdenosineEquilibrative nucleoside transporter 2transporter
AdenosineEquilibrative nucleoside transporter 3transporter
AdenosineEquilibrative nucleoside transporter 4transporter
AdenosineSodium/nucleoside cotransporter 1transporter
AdenosineSodium/nucleoside cotransporter 2transporter
AdenosineGap junction alpha-1 proteintransporter
AdenosineAdenylate kinase isoenzyme 1enzyme
AdenosineNucleoside diphosphate kinase Aenzyme
AdenosineNucleoside diphosphate kinase Benzyme
AdenosinePurine nucleoside phosphorylaseenzyme
AdenosineXanthine dehydrogenase/oxidaseenzyme
AdenosineAlbumincarrier
AdenosineAdenosine receptortarget
AdenosineAdenosine deaminaseenzyme
AdenosineAdenosine receptor A3target
AMG-319Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoformtarget
AZD-8848Toll-like receptor 7target
BinodenosonAdenosine receptor A2atarget
CladribineATP-dependent translocase ABCB1transporter
CladribineAdenosine deaminasetarget
CladribinePoly [ADP-ribose] polymerase 1target
CladribineDeoxyguanosine kinase, mitochondrialenzyme
CladribineEquilibrative nucleoside transporter 1transporter
CladribinePurine nucleoside phosphorylasetarget
CladribineDNAtarget
CladribineRibonucleoside-diphosphate reductase large subunittarget
CladribineRibonucleoside-diphosphate reductase subunit M2target
CladribineRibonucleoside-diphosphate reductase subunit M2 Btarget
CladribineDNA polymerase alpha catalytic subunittarget
CladribineDNA polymerase epsilon catalytic subunit Atarget
CladribineDNA polymerase epsilon subunit 2target
CladribineDNA polymerase epsilon subunit 3target
CladribineDNA polymerase epsilon subunit 4target
CladribineBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
CladribineDeoxycytidine kinaseenzyme
CladribineSolute carrier family 28 member 3transporter
CordycepinPoly(A) polymerase alphatarget
CordycepinAdenosine kinaseenzyme
Cordycepin5'-AMP-activated protein kinasetarget
CordycepinAdenosine deaminaseenzyme
Deoxycytidylyl-3',5'-guanosineRibonuclease pancreatictarget
DeoxyinosineEndonuclease Vtarget
DeoxyinosineAdenosine deaminase 2enzyme
DeoxyinosineDNA-3-methyladenine glycosylaseenzyme
DeoxyinosineDeoxyguanosine kinase, mitochondrialenzyme
DeoxyinosineEndonuclease Venzyme
DeoxyinosinePurine nucleoside phosphorylaseenzyme
DeoxyinosineAdenosine deaminaseenzyme
DeoxyinosineDNA-3-methyladenine glycosylasetarget
DeuremidevirReplicase polyprotein 1abtarget
DidanosineGag-Pol polyproteintarget
DidanosineAlbumincarrier
DidanosineEquilibrative nucleoside transporter 2transporter
DidanosineEquilibrative nucleoside transporter 1transporter
DidanosineReverse transcriptase/RNaseHtarget
DidanosinePurine nucleoside phosphorylasetarget
DidanosineSolute carrier family 22 member 6transporter
DideoxyadenosineAdenosine deaminaseenzyme
DideoxyadenosineAdenylate cyclasetarget
FadraciclibCyclin-dependent kinase 2target
FadraciclibCyclin-dependent kinase 9target
FludarabineAdenosine deaminasetarget
FludarabineSolute carrier family 28 member 3transporter
FludarabineDeoxycytidine kinasetarget
FludarabineDNAtarget
FludarabineDNA polymerase alpha catalytic subunittarget
FludarabineRibonucleoside-diphosphate reductase large subunittarget
FludarabineEquilibrative nucleoside transporter 1transporter
GalidesivirReplicase polyprotein 1abtarget
GalidesivirRNA-directed RNA polymerase Ltarget
GS-441524RNA-directed RNA polymerase Ltarget
GS-441524Replicase polyprotein 1abtarget
GS-6620Genome polyproteintarget
GuanosinePurine nucleoside phosphorylasetarget
GuanosineDNA polymerase catalytic subunittarget
GuanosineUridine phosphorylasetarget
GuanosineDNA polymerase catalytic subunittarget
GuanosineDNA-directed DNA polymerasetarget
InosinePurine nucleoside phosphorylase DeoD-typetarget
InosineXanthine dehydrogenase/oxidaseenzyme
InosineSolute carrier family 28 member 3transporter
InosineIAG-nucleoside hydrolasetarget
InosinePurine nucleoside phosphorylasetarget
Inosine pranobexCyclic nucleotide phosphodiesterasetarget
IsatoribineToll-like receptor 7target
IslatravirReverse transcriptase/RNaseHtarget
IslatravirBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
LodenosineGag-Pol polyproteintarget
LoxoribineToll-like receptor 7target
MethylthioinosinePurine nucleoside phosphorylase DeoD-typetarget
MetrifudilAdenosine receptor A3target
MetrifudilAdenosine receptor A2atarget
MetrifudilAdenosine receptor A1target
N(6)-dimethylallyladenineCyclin-dependent kinase 2target
NamodenosonAdenosine receptor A3target
NebularineAdenosine deaminasetarget
PiclidenosonAdenosine receptor A3target
PuromycinRibosomal protein uL16-liketarget
PuromycinLarge ribosomal subunit protein uL13target
PuromycinLarge ribosomal subunit protein uL14target
PuromycinLarge ribosomal subunit protein eL15target
PuromycinLarge ribosomal subunit protein eL19target
PuromycinLarge ribosomal subunit protein uL23target
PuromycinProbable ribosome biogenesis protein RLP24target
PuromycinRibosomal protein uL24-liketarget
PuromycinLarge ribosomal subunit protein uL2target
PuromycinLarge ribosomal subunit protein eL37target
PuromycinLarge ribosomal subunit protein uL3target
PuromycinLarge ribosomal subunit protein uL5target
PuromycinLeucyl/phenylalanyl-tRNA--protein transferasetarget
S-Adenosyl-1,8-Diamino-3-ThiooctanePolyamine aminopropyltransferasetarget
S-adenosyl-L-homocysteinetRNA (cytidine(34)-2'-O)-methyltransferasetarget
S-adenosyl-L-homocysteineDNA adenine methylasetarget
S-adenosyl-L-homocysteinePhenylethanolamine N-methyltransferasetarget
S-adenosyl-L-homocysteineCyclopropane mycolic acid synthase 2target
S-adenosyl-L-homocysteineDNA (cytosine-5)-methyltransferase 3Btarget
S-adenosyl-L-homocysteineHistamine N-methyltransferaseenzyme
S-adenosyl-L-homocysteineProtein-L-isoaspartate O-methyltransferasetarget
S-adenosyl-L-homocysteineType II methyltransferase M.TaqItarget
S-adenosyl-L-homocysteineCap-specific mRNA (nucleoside-2'-O-)-methyltransferasetarget
S-adenosyl-L-homocysteineChemotaxis protein methyltransferasetarget
S-adenosyl-L-homocysteineuroporphyrinogen-III C-methyltransferasetarget
S-adenosyl-L-homocysteineUroporphyrinogen-III C-methyltransferasetarget
S-adenosyl-L-homocysteinetRNA (guanine-N(1)-)-methyltransferasetarget
S-adenosyl-L-homocysteineAclacinomycin 10-hydroxylase RdmBtarget
S-adenosyl-L-homocysteineDiphthine methyl ester synthasetarget
S-adenosyl-L-homocysteineCyclopropane mycolic acid synthase MmaA2target
S-adenosyl-L-homocysteinetRNA (guanine-N(1)-)-methyltransferasetarget
S-adenosyl-L-homocysteineHistone-lysine N-methyltransferase SETD7target
S-adenosyl-L-homocysteineType II methyltransferase M.HhaItarget
S-adenosyl-L-homocysteineSiroheme synthasetarget
S-adenosyl-L-homocysteineProtein arginine N-methyltransferase 1target
S-adenosyl-L-homocysteineCyclopropane mycolic acid synthase 3target
S-adenosyl-L-homocysteineGenome polyproteintarget
S-adenosyl-L-homocysteineType II methyltransferase M.PvuIItarget
S-adenosyl-L-homocysteineType II methyltransferase M.RsrItarget
S-adenosyl-L-homocysteineGlycine N-methyltransferasetarget
S-adenosyl-L-homocysteinetRNA (cytosine(38)-C(5))-methyltransferasetarget
S-adenosyl-L-homocysteinerRNA adenine N-6-methyltransferasetarget
S-adenosyl-L-homocysteineRibosomal RNA small subunit methyltransferase Htarget
S-adenosyl-L-homocysteineHistamine N-methyltransferasetarget
S-adenosyl-L-homocysteineCobalt-precorrin-4 C(11)-methyltransferasetarget
S-adenosyl-L-homocysteineCatechol O-methyltransferase domain-containing protein 1target
S-adenosyl-L-homocysteineProtein-L-isoaspartate(D-aspartate) O-methyltransferasetarget
S-adenosyl-L-homocysteineProtein arginine N-methyltransferase 3target
S-adenosyl-L-homocysteineRelease factor glutamine methyltransferasetarget
S-adenosyl-L-homocysteineRelease factor glutamine methyltransferasetarget
S-adenosyl-L-homocysteineGuanidinoacetate N-methyltransferasetarget
S-adenosyl-L-homocysteineCarminomycin 4-O-methyltransferase DnrKtarget
SelodenosonAdenosine receptor A1target
SinefunginType II methyltransferase M.TaqItarget
SinefunginType II methyltransferase M.RsrItarget
SinefunginAclacinomycin 10-hydroxylase RdmBtarget
SinefunginrRNA adenine N-6-methyltransferasetarget
SonedenosonAdenosine receptor A2atarget
TecadenosonAdenosine receptor A1target
TicagrelorCytochrome P450 2B6enzyme
TicagrelorCytochrome P450 3A5enzyme
TicagrelorAlbumincarrier
TicagrelorCytochrome P450 2C9enzyme
TicagrelorATP-dependent translocase ABCB1transporter
TicagrelorP2Y purinoceptor 12target
TicagrelorCytochrome P450 3A4enzyme
TrabodenosonAdenosine receptor A1target
TubercidinPurine nucleoside phosphorylase DeoD-typetarget
UK-432097Adenosine receptor A2atarget
VidarabineAdenosine receptor A2btarget
VidarabineAdenosine deaminaseenzyme
VidarabineThymidine kinasetarget
VidarabineThymidine kinasetarget
VidarabineDNA polymerase catalytic subunittarget