| DB00302 | Tranexamic acid | approved | yes | inhibitor | Details |
| DB00513 | Aminocaproic acid | approved, investigational | yes | inhibitor | Details |
| DB00013 | Urokinase | approved, investigational, withdrawn | yes | activator | Details |
| DB03709 | Bicine | experimental | unknown | | Details |
| DB00086 | Streptokinase | approved, investigational | yes | activator | Details |
| DB04925 | Desmoteplase | investigational | unknown | | Details |
| DB06692 | Aprotinin | approved, investigational, withdrawn | unknown | | Details |
| DB00031 | Tenecteplase | approved | yes | activator | Details |
| DB00009 | Alteplase | approved, investigational | yes | activator | Details |
| DB00029 | Anistreplase | approved | yes | activator | Details |
| DB00015 | Reteplase | approved, investigational | yes | activator | Details |
| DB12831 | Gabexate | investigational | yes | inhibitor | Details |
| DB09130 | Copper | approved, investigational | unknown | | Details |