| DB00218 | Moxifloxacin | approved, investigational | yes | inhibitor | Details |
| DB00365 | Grepafloxacin | approved, investigational, withdrawn | yes | inhibitor | Details |
| DB00467 | Enoxacin | approved, investigational | yes | inhibitor | Details |
| DB00487 | Pefloxacin | approved | yes | inhibitor | Details |
| DB00537 | Ciprofloxacin | approved, investigational | yes | inhibitor | Details |
| DB00685 | Trovafloxacin | approved, investigational, withdrawn | yes | inhibitor | Details |
| DB00978 | Lomefloxacin | approved, investigational | yes | inhibitor | Details |
| DB01059 | Norfloxacin | approved | yes | inhibitor | Details |
| DB01137 | Levofloxacin | approved, investigational | yes | inhibitor | Details |
| DB01155 | Gemifloxacin | approved, investigational | yes | inhibitor | Details |
| DB01165 | Ofloxacin | approved | yes | inhibitor | Details |
| DB01208 | Sparfloxacin | approved, investigational, withdrawn | yes | inhibitor | Details |
| DB01405 | Temafloxacin | withdrawn | yes | inhibitor | Details |
| DB00827 | Cinoxacin | approved, investigational, withdrawn | yes | inhibitor | Details |
| DB04576 | Fleroxacin | experimental | yes | inhibitor | Details |
| DB06771 | Besifloxacin | approved | yes | antagonist | Details |
| DB09047 | Finafloxacin | approved, investigational | yes | inhibitor | Details |
| DB12924 | Ozenoxacin | approved, investigational | yes | inhibitor | Details |