| DB00712 | Flurbiprofen | approved, investigational | unknown | substrate | Details |
| DB01050 | Ibuprofen | approved | unknown | substrate | Details |
| DB06741 | Gavestinel | investigational | unknown | substrate | Details |
| DB00295 | Morphine | approved, investigational | no | substrate | Details |
| DB08907 | Canagliflozin | approved | unknown | substrate | Details |
| DB00318 | Codeine | approved, illicit | unknown | substrate | Details |
| DB06292 | Dapagliflozin | approved | no | substrate | Details |
| DB09213 | Dexibuprofen | approved, investigational | unknown | substrate | Details |
| DB00586 | Diclofenac | approved, vet_approved | unknown | substrate | Details |
| DB01136 | Carvedilol | approved, investigational | unknown | substrate | Details |
| DB01241 | Gemfibrozil | approved | unknown | substrate | Details |
| DB06119 | Cenobamate | approved, investigational | unknown | substrate | Details |
| DB00514 | Dextromethorphan | approved | unknown | substrate | Details |
| DB08804 | Nandrolone decanoate | approved, illicit | unknown | substrate | Details |
| DB00647 | Dextropropoxyphene | approved, illicit, investigational, withdrawn | unknown | inhibitor | Details |
| DB00333 | Methadone | approved | no | inhibitor | Details |
| DB12095 | Telotristat ethyl | approved, investigational | no | inducer | Details |
| DB00349 | Clobazam | approved, illicit | unknown | inhibitor | Details |
| DB00683 | Midazolam | approved, illicit | no | substrate | Details |