| DB04725 | Licofelone | investigational | unknown | substrate | Details |
| DB00169 | Cholecalciferol | approved, nutraceutical | unknown | substrate | Details |
| DB00637 | Astemizole | approved, withdrawn | unknown | substrate | Details |
| DB00342 | Terfenadine | approved, withdrawn | unknown | inhibitor | Details |
| DB06228 | Rivaroxaban | approved | unknown | substrate | Details |
| DB06605 | Apixaban | approved | unknown | substrate | Details |
| DB08918 | Levomilnacipran | approved, investigational | unknown | substrate | Details |
| DB08931 | Riociguat | approved | unknown | substrate | Details |
| DB09148 | Florbetaben (18F) | approved | no | substrate | Details |
| DB09030 | Vorapaxar | approved | no | substrate | Details |
| DB04855 | Dronedarone | approved | unknown | inhibitor | Details |
| DB01118 | Amiodarone | approved, investigational | unknown | inhibitor | Details |
| DB15305 | Risdiplam | approved, investigational | unknown | substrate | Details |
| DB12016 | Ponesimod | approved, investigational | unknown | substrate | Details |
| DB05316 | Pimavanserin | approved, investigational | unknown | substrate | Details |
| DB00470 | Dronabinol | approved, illicit | unknown | substrateinhibitor | Details |
| DB00486 | Nabilone | approved, investigational | unknown | substrate | Details |
| DB09061 | Cannabidiol | approved, investigational | no | inhibitor | Details |
| DB14737 | Cannabinol | experimental, investigational | no | inhibitor | Details |
| DB14009 | Medical Cannabis | experimental, investigational | unknown | substrateinhibitor | Details |