| DB00477 | Chlorpromazine | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB00408 | Loxapine | approved | unknown | binder | Details |
| DB00458 | Imipramine | approved | unknown | binder | Details |
| DB00726 | Trimipramine | approved | unknown | binder | Details |
| DB00248 | Cabergoline | approved | unknown | agonist | Details |
| DB00988 | Dopamine | approved | unknown | agonist | Details |
| DB00696 | Ergotamine | approved | unknown | agonist | Details |
| DB00568 | Cinnarizine | approved, investigational | unknown | binder | Details |
| DB00334 | Olanzapine | approved, investigational | unknown | antagonist | Details |
| DB06148 | Mianserin | approved, investigational | unknown | binder | Details |
| DB09097 | Quinagolide | approved, investigational | unknown | agonist | Details |
| DB00555 | Lamotrigine | approved, investigational | unknown | inhibitor | Details |
| DB09225 | Zotepine | approved, investigational, withdrawn | yes | antagonist | Details |
| DB11584 | Pipradrol | approved | unknown | agonist | Details |
| DB11274 | Dihydro-alpha-ergocryptine | approved | yes | partial agonist | Details |
| DB00715 | Paroxetine | approved, investigational | unknown | other/unknown | Details |