Hypnotics and Sedatives

Name
Hypnotics and Sedatives
Accession Number
DBCAT000452
Description

Drugs used to induce drowsiness or sleep or to reduce psychological excitement or anxiety.

Drugs
DrugDrug Description
AcecarbromalAcecarbromal is a small molecule drug. Acecarbromal has a monoisotopic molecular weight of 278.03 Da.
Acetylglycinamide chloral hydrateNot Annotated
AllobarbitalNot Annotated
AlprazolamA triazolobenzodiazepine with intermediate onset commonly used to treat panic disorders and generalized anxiety in addition to anxiety associated with depression.
AmobarbitalA barbiturate derivative used for the induction of sedation during procedures, short-term management of insomnia, and acute management of refractory tonic-clonic seizures.
AprobarbitalAprobarbital is a barbiturate derivative synthesized in the 1920s by Ernst Preiswerk. It was determined that the substance was capable of demonstrating sedative, hypnotic, and anticonvulsant effects. A primary treatment...
ApronalideApronalide is approved in Japan. Apronalide has been withdrawn from the market in many other countries due to patient development of thrombocytopenic purpura .
AzaperoneAzaperone is a pyridinylpiperazine and butyrophenone agent that is capable of eliciting neuroleptic sedative and antiemetic effects. It is subsequently employed predominantly as a veterinary tranquilizer and mainly for pigs...
AZD-3043AZD3043 has been used in trials studying the treatment and basic science of Safety, Sedation, Tolerability, and Pharmacokinetics.
BarbitalA long-acting barbiturate that depresses most metabolic processes at high doses. It is used as a hypnotic and sedative and may induce dependence. Barbital is also used in veterinary practice...
BentazepamNot Annotated
BromazepamA short-acting benzodiazepine with intermediate onset commonly used to treat panic disorders and severe anxiety.
BromisovalNot Annotated
BrotizolamA benzodiazepine analogue with sedative-hypnotic properties used for short-term treatment of severe or debilitating insomnia.
ButabarbitalA barbiturate drug used as a sedative and hypnotic.
ButalbitalA barbiturate drug used for symptomatic treatment of tension-type headache in various combinations with acetaminophen, aspirin, caffeine, and codeine.
ButobarbitalFor the treatment of insomnia.
CarbromalNot Annotated
Chloral hydrateA mild hypnotic used for experimental purposes that was previously used for the treatment of insomnia.
ChloraloseChloralose is a small molecule drug. Chloralose has a monoisotopic molecular weight of 307.96 Da.
ChlordiazepoxideA benzodiazepine used to treat the withdrawal symptoms of acute alcoholism, to treat preoperative anxiety, and to treat anxiety over a short term period.
ChlorhexadolChlorhexadol is a sedative and hypnotic which is regulated in the United States as a Schedule III controlled substance. It is a derivative of chloral hydrate.
CinolazepamA benzodiazepine used to manage severe and debilitating forms of sleep disorders of various origins in adults.
CipepofolAn alkylphenol GABA-A positive allosteric modulator used for induction of general anesthesia in adults undergoing surgery.
ClomethiazoleInvestigated for use/treatment in strokes.
CP-96345Not Annotated
CyclobarbitalNot Annotated
DaridorexantA dual orexin receptor antagonist used to treat insomnia in adults.
DetomidineUsed as a large animal sedative, primarily in horses.
DexmedetomidineAn alpha-2 agonist used for sedation during various procedures.
DiazepamA long-acting benzodiazepine with rapid onset commonly used to treat panic disorders, severe anxiety, alcohol withdrawal, and seizures.
DichloralphenazoneDichloralphenazone is a sedative composed of chloral hydrate and phenazone. It is typically found in combination products Nodolor and Midrin containing isometheptene and acetaminophen used for the relief of tension...
DiphenhydramineA H1 receptor antihistamine used in the treatment of seasonal allergies, and various allergic reactions including sneezing, runny nose, itchy/watery eyes, itching of nose or throat, pruritus, urticaria, insect bites/stings, and allergic rashes.
DoxefazepamNot Annotated
DoxepinA psychotropic agent used for the treatment of depression, anxiety, manic-depressive disorder, and insomnia.
EmeproniumNot Annotated
EstazolamA benzodiazepine used for the short-term management of insomnia.
EszopicloneA sedative-hypnotic used in the treatment of insomnia, improving both the latency phase and the maintenance phase of sleep.
EthchlorvynolA sedative hypnotic agent used for the short-term management of insomnia.
EtizolamA thienodiazepine derivative used to treat anxiety and insomnia.
EtomidateA short-acting intravenous anesthetic indicated for the induction of anesthesia and supplementation of subpotent anesthesia during short operative procedures.
FluanisoneNot Annotated
FlunitrazepamA benzodiazepine used to manage anxiety disorders and insomnia.
FlurazepamA long-acting benzodiazepine with a rapid onset of action that is commonly used to treat insomnia.
FospropofolA sedative-­hypnotic agent indicated for monitored anesthesia care (MAC) sedation in adult patients undergoing diagnostic or therapeutic procedures.
GedocarnilNot Annotated
GlutethimideFor the treatment of insomnia.
HeptabarbitalUsed mainly for sedation and hypnosis.
HexapropymateNot Annotated
HexobarbitalFor the induction of anesthesia prior to the use of other general anesthetic agents and for induction of anesthesia for short surgical, diagnostic, or therapeutic procedures associated with minimal painful...
IndiplonIndiplon has been used in trials studying the treatment of Insomnia and Depression.
LemborexantA dual orexin antagonist indicated for the treatment of sleep-onset and/or sleep maintenance insomnia.
LoprazolamLoprazolam is an imidazobenzodiazepine with anxiolytic, anticonvulsant, hypnotic, sedative and skeletal muscle relaxant properties. It is indicated for the short-term treatment of insomnia including difficulty in falling asleep and/or frequent...
LorazepamA short-acting benzodiazepine commonly used to treat panic disorders, severe anxiety, and seizures.
LormetazepamA benzodiazepine indicated in the treatment of anxiety and the induction of anesthesia.
MedazepamA long-acting benzodiazepine used for its sedative and anxiolytic properties.
MedetomidineMedetomidine is a synthetic compound used as a surgical anesthetic and analgesic. It is normally found as its hydrochloride salt, medetomidine hydrochloride. Medetomidine is an intravenously available alpha-2 adrenergic agonist....
MelatoninAn endogenous hormone produced by the pineal gland that regulates sleep-wake cycles and when provided exogenously has beneficial effects on sleep-onset latency; available as an over-the-counter supplement.
MeprobamateAn anxiolytic drug used for the short-term management of anxiety symptoms.
MepyramineAn antihistamine agent used for the symptomatic treatment of allergy, hypersensitivity reactions, and pruritic skin disorders.
MethapyrileneMethapyrilene, formerly marketed in many drug products, was shown to be a potent carcinogen. Manufacturers voluntarily withdrew methapyriline drug products from the market in May and June 1979.
MethaqualoneFor the treatment of insomnia, and as a sedative and muscle relaxant.
MethohexitalAn anesthetic used to induce deep sedation.
MethylpentynolNot Annotated
MethylphenobarbitalFor the relief of anxiety, tension, and apprehension, also used as an anticonvulsant for the treatment of epilepsy.
MethyprylonFor the treatment of insomnia.
MidazolamA short-acting benzodiazepine with rapid onset that is commonly used in seizures, anesthesia and anxiety disorders.
NiaprazineNiaprazine is a selective brain catecholamine depletor.
NitrazepamA long-acting benzodiazepine with intermediate onset commonly used to treat panic disorders, severe anxiety, insomnia, and seizures.
OcinaplonInvestigated for use/treatment in anxiety disorders.
OxazepamAn intermediate-acting benzodiazepine with slow onset commonly used to treat panic disorders, severe anxiety, alcohol withdrawals, and insomnia.
PagocloneFor the potential treatment of panic and anxiety disorders.
ParaldehydeA central nervous system depressant previously used to control convulsions due to various clinical causes, including tetanus, status epilepticus, and convulsive drugs.
Passiflora incarnata flowerA herbal product indicated in the treatment of stress, nervousness, anxiety, irritability, and trouble sleeping.
PentobarbitalA barbiturate drug used to induce sleep, cause sedation, and control certain types of seizures.
PhenibutNot Annotated
PhenobarbitalA long-lasting barbiturate and anticonvulsant used in the treatment of all types of seizures, except for absent seizures.
PhetharbitalPhetharbital is a small molecule drug. Phetharbital has a monoisotopic molecular weight of 260.12 Da.
PrimidoneAn antiepileptic used to treat grand mal, psychomotor, and focal epileptic seizures.
PropiomazinePropiomazine is largely used for its antihistamininc sleep inducing effects in treating insomnia.
PropofolA medication used in general anesthesia and for sedation.
ProxibarbalProxibarbal is a derivative of barbiturates, which has been used to treat migraines. Proxibarbal was approved in France but was withdrawn from the market due to the risk of inducing...
PyrazolamNot Annotated
PyrithyldioneNot Annotated
QuazepamA long-acting benzodiazepine used to manage insomnia.
RamelteonA melatonin receptor agonist used to treat insomnia.
RemifentanilAn opioid analgesic used in anesthesia.
RemimazolamAn ultra short-acting benzodiazepine used for the induction and maintenence of procedural sedation during short procedures.
ReposalReposal is a barbiturate derivative invented in the 1960s in Denmark that has sedative, hypnotic and anticonvulsant properties. It was used primarily in the treatment of insomnia.
RilmazafoneRilmazafone is a small molecule drug. The usage of the INN stem '-zafone' in the name indicates that Rilmazafone is a alozafone derivative. Rilmazafone has a monoisotopic molecular weight of...
RomifidineRomifidine is a veterinary drug utilized as a sedative primarily in large animals, most frequently horses. It is also used less commonly in a wide variety of other animal species....
S-EthylisothioureaS-Ethylisothiourea is a nitric oxide synthase inhibitor.
ScopolamineA belladonna alkaloid with anticholinergic effects indicated for the treatment of nausea and vomiting associated with motion sickness and postoperative nausea and vomiting (PONV).
SecobarbitalA barbiturate used for the short-term treatment of insomnia.
SuvorexantA orexin receptor antagonist used to treat insomnia that is characterized by difficulties with sleep onset and/or sleep maintenance.
TalbutalFor use as a sedative and hypnotic.
TasimelteonA melatonin receptor agonist used to treat Non- 24-Hour Sleep-Wake Disorder.
TemazepamA short-acting benzodiazepine commonly used to treat panic disorders, severe anxiety, and insomnia.
ThiamylalUsed for the production of complete anaesthesia of short duration, for the induction of general anaesthesia, and for inducing a hypnotic state.
ThiopentalA barbiturate used to induce general anesthesia, treat convulsions, and reduce intracranial pressure.
TriazolamA benzodiazepine used for short term treatment of insomnia.
TriclofosNot Annotated
ValerianA plant used in some non-prescription natural health products.
ValnoctamideValnoctamide has been used in trials studying the treatment of Mania and Schizoaffective Disorder, Manic Type.
VinbarbitalNot Annotated
VinylbitalNot Annotated
XylazineA non-opioid and clonidine analog with analgesic and muscle relaxant properties used as a tranquilizer used in veterinary medicine.
ZaleplonA sedative used for short term treatment of insomnia in adults.
ZolpidemA sedative hypnotic used for the short-term treatment of insomnia to improve sleep latency.
ZopicloneA nonbenzodiazepine hypnotic used for the short-term management of insomnia.