Serotonin Modulators

Name
Serotonin Modulators
Accession Number
DBCAT002706
Description

Not Available

Drugs
DrugDrug Description
AlaproclateAlaproclate was developed as one of the first selective serotonin reuptake inhibitor (SSRI) antidepressants by Astra AB (now AstraZeneca) in the 1970s. Development was discontinued due to concerns over hepatotoxicity...
AlmotriptanA 5-HT1B/1D receptor agonist used to treat migraines.
AmitriptylineA tricyclic antidepressant indicated in the treatment of depressive illness, either endogenous or psychotic, and to relieve depression associated anxiety.
AmoxapineA tricyclic antidepressant used in the treatment of neurotic or reactive depressive disorders and endogenous or psychotic depression.
BromocriptineA dopamine D2 receptor agonist used for the treatment of galactorrhea due to hyperprolactinemia and other prolactin-related conditions, as well as in early Parkinsonian Syndrome.
CabergolineA dopamine receptor agonist used for the treatment of hyperprolactinemic conditions due to various causes.
ChlorpheniramineA histamine-H1 receptor antagonist indicated for the management of symptoms associated with upper respiratory allergies.
CitalopramA selective serotonin reuptake inhibitor (SSRI) used in the treatment of depression.
ClomipramineA tricyclic antidepressant used in the treatment of obsessive-compulsive disorder and disorders with an obsessive-compulsive component, such as depression, schizophrenia, and Tourette’s disorder.
DA-8031DA-8031 is under investigation in clinical trial NCT01798667 (Clinical Trial to Evaluate the Efficacy and Safety of DA-8031 in Male Patients With Premature Ejaculation).
DapoxetineA selective serotonin reuptake inhibitor used in the treatment of premature ejaculation.
DesipramineA tricyclic antidepressant used in the treatment of depression.
DesvenlafaxineAn antidepressant agent and SNRI used for the treatment of major depressive disorders in adults.
DexmethylphenidateA norepinephrine-dopamine reuptake inhibitor used in the treatment of ADHD in conjunction with other therapies.
DextromethorphanAn NMDA receptor antagonist used to treat cases of dry cough.
DihydroergotamineAn ergot alkaloid used in the acute treatment of migraine headache and cluster headache.
DosulepinA tricyclic antidepressant commonly used only in patients for whom alternative therapies are ineffective due to its toxicity potential.
DoxepinA psychotropic agent used for the treatment of depression, anxiety, manic-depressive disorder, and insomnia.
DuloxetineA serotonin norepinephrine reuptake inhibitor used to treat generalized anxiety disorder, neuropathic pain, osteoarthritis, and stress incontinence.
EletriptanA triptan used for the treatment of migraines.
Ergoloid mesylateA nootropic with an unknown mechanism of action indicated in individuals over sixty who manifest signs and symptoms of an idiopathic decline in mental capacity.
ErgometrineAn ergot alkaloid used for the treatment of postpartum haemorrhage and post abortion hemorrhage in patients with uterine atony.
ErgotamineAn alpha-1 selective adrenergic agonist vasoconstrictor used to treat migraines with or without aura and cluster headaches.
EscitalopramA selective serotonin re-uptake inhibitor used in the treatment of major depressive disorder (MDD), generalized anxiety disorder (GAD), and other select psychiatric disorders such as obsessive-compulsive disorder (OCD).
EtoperidoneEtoperidone has been studied for the treatment of depression , tremors in Parkinson, extrapyramidal symptoms and male impotence . It is not certain if it was ever approved and marketed...
FemoxetineFemoxetine is a small molecule drug. Femoxetine has a monoisotopic molecular weight of 311.19 Da.
FentanylAn opioid analgesic used in anesthesia, for breakthrough cancer pain, or round the clock pain management.
FlibanserinA 5-HT receptor modulator used for the treatment of selected premenopausal women with acquired, generalized hypoactive sexual desire disorder (HSDD).
FluoxetineA selective serotonin reuptake inhibitor used to treat major depressive disorder, bulimia, OCD, premenstrual dysphoric disorder, panic disorder, and bipolar I.
FluvoxamineA selective serotonin-reuptake inhibitor used to treat obsessive-compulsive disorder.
FrovatriptanA 5-HT1B/1D receptor agonist used to treat migraines.
ImipramineA tricyclic antidepressant indicated for the treatment of depression and to reduce childhood enuresis.
IndalpineIndalpine was one of the first selective serotonin reuptake inhibitors to reach the American market. It was initially marketed by Pharmuka. However, after the emergence of widespread concern regarding adverse...
IsocarboxazidA monoamine oxidase inhibitor used to treat enduring and debilitating symptoms of depression following inadequate clinical response to other antidepressant drugs.
LevomilnacipranA selective serotonin and norepinephrine reuptake inhibitor (SNRI) used to treat major depressive disorder (MDD) in adults.
LinezolidAn oxazolidinone antibiotic used to treat infections by susceptible strains of aerobic Gram-positive bacteria.
Lithium carbonateA medication used to treat manic episodes of bipolar disorder.
Lithium cationA drug used for the management of bipolar disorder and other psychiatric conditions.
Lithium citrateLithium is used as a mood stabilizer, and is used for treatment of depression and mania. It is often used in bipolar disorder treatment.
LorcaserinA serotonin 2C receptor agonist used in conjunction with physical activity and calorie restriction for weight loss in obese patients with a body mass index (BMI) of 30 and above, and in overweight patients with weight-related comorbidities.
LorpiprazoleIn 2016, lorpiprazole was classified in the "Chemical structure-related drug-like criteria of global approved drugs" as an antipsychotic and anxiolytic. An antipsychotic is a medication used to treat a state...
LumateperoneA novel 2nd generation atypical antipsychotic used to manage schizophrenia, bipolar depression, and major depressive disorder.
MaprotilineA tetracyclic antidepressant used to treat depressive illness, major depressive disorder, bipolar disorder, and anxiety associated with depression.
MazindolA sympathomimetic used to treat obesity in combination with lifestyle modifications.
MeperidineAn opioid agonist with analgesic and sedative properties used to manage severe pain.
MethadoneAn opioid analgesic indicated for management of severe pain that is not responsive to alternative treatments. Also used to aid in detoxification and maintenance treatment of opioid addiction.
MianserinA tetracyclic antidepressant with therapeutic activity similar to amitriptyline used to treat depression and anxiety.
MilnacipranA selective serotonin and norepinephrine reuptake inhibitor (SNRI) used for the treatment of fibromyalgia and a short-term treatment of major depressive disorder.
MirtazapineA tetracyclic antidepressant used in the treatment of major depression and is used off-label as a drug for insomnia and to increase appetite.
MoclobemideA monoamine oxidase inhibitor used in the treatment of major depressive disorder and bipolar disorder.
NaratriptanA 5-HT1B/1D receptor agonist used to treat migraines.
NefazodoneAn antidepressant used in the treatment of depression.
NortriptylineA tricyclic antidepressant used in the treatment of depression.
ParoxetineA selective serotonin reuptake inhibitor used to treat major depressive disorder, panic disorder, OCD, social phobia, generalized anxiety disorder, the vasomotor symptoms of menopause, and premenstrual dysphoric disorder.
PhenelzineA monoamine oxidase inhibitor used to treat atypical, nonendogenous, or neurotic depression.
ProcarbazineAn antineoplastic agent indicated for the treatment of stage III and stage IV Hodgkin's disease in combination with other chemotherapeutic agents.
PromethazineA first-generation antihistamine used for the treatment of allergic conditions, nausea and vomiting, and motion sickness.
ProtriptylineA tricyclic antidepressant that is indicated in the treatment of depression only under close clinical supervision.
RasagilineAn irreversible inhibitor of monoamine oxidase used for the symptomatic management of idiopathic Parkinson's disease as initial monotherapy and as adjunct therapy to levodopa.
RitanserinRitanserin has been used in trials studying the treatment of Cocaine-Related Disorders.
RizatriptanA triptan used to treat migraines with or without aura.
SelegilineA monoamine oxidase inhibitor used to treat major depressive disorder and Parkinson's.
SeproxetineSeproxetine is also known as (S)-norfluoxetine. It is a selective serotonin reuptake inhibitor (SSRI). It is an active metabolite of fluoxetine. Seproxetine was being investigated by Eli Lilly as an...
SertralineA selective serotonin reuptake inhibitor (SSRI) indicated to treat major depressive disorder, social anxiety disorder and many other psychiatric conditions.
SibutramineA norepinephrine, serotonin and dopamine reuptake inhibitor indicated to assist with weight loss in obesity.
SumatriptanA serotonin receptor agonist used to treat migraines and cluster headaches.
TapentadolAn opioid used to manage severe pain that has not responded to non-opioid medications, and for which opioid analgesic therapy is appropriate.
Tedizolid phosphateAn oxazolidinone class antibiotic that inhibits bacterial protein synthesis and is proven to be effective in the treatment of certain Gram-positive bacterial infections.
TenamfetamineAn amphetamine derivative that inhibits uptake of catecholamine neurotransmitters. It is a hallucinogen. It is less toxic than its methylated derivative but in sufficient doses may still destroy serotonergic neurons...
TianeptineAn atypical tricyclic antidepressant with antidepressant and anxiolytic effects primarily used to treat major depressive disorder.
TramadolA centrally-acting opioid agonist and SNRI (serotonin/norepinephrine reuptake inhibitor) used for the management of moderate to severe pain in adults.
TranylcypromineA monoamine oxidase inhibitor used to treat major depressive disorder.
TrazodoneA serotonin uptake inhibitor used to treat major depressive disorder.
TrimipramineA tricyclic antidepressant used to treat depression.
VenlafaxineA selective serotonin and norepinephrine reuptake inhibitor (SNRI) used for the treatment of major depression, generalized or social anxiety disorder, and panic disorder.
VilazodoneAn antidepressant agent used for the treatment of major depressive disorder that targets the 5-HT transporter and 5-HT1A receptors.
VortioxetineA serotonin modulating antidepressant indicated for the treatment of major depressive disorder (MDD).
ZimelidineFor the treatment of depression.
ZolmitriptanA member of the triptan class of 5-HT(1B/1D/1F) receptor agonist drugs used for the acute treatment of migraine with or without aura in adults.
Drugs & Drug Targets
DrugTargetType
AlaproclateSodium-dependent serotonin transportertarget
AlaproclatePotassium voltage-gated channel subfamily A member 2target
AlaproclateSigma intracellular receptor 2target
AlmotriptanCytochrome P450 2D6enzyme
AlmotriptanAmine oxidase [flavin-containing] Aenzyme
AlmotriptanFlavin-containing monooxygenase 3enzyme
AlmotriptanCytochrome P450 2C19enzyme
AlmotriptanCytochrome P450 2E1enzyme
AlmotriptanCytochrome P450 2C8enzyme
Almotriptan5-hydroxytryptamine receptor 1Ftarget
AlmotriptanCytochrome P450 3A4enzyme
Almotriptan5-hydroxytryptamine receptor 1Btarget
Almotriptan5-hydroxytryptamine receptor 1Dtarget
AmitriptylineAlpha-1A adrenergic receptortarget
AmitriptylineCytochrome P450 3A4enzyme
AmitriptylineCytochrome P450 3A5enzyme
AmitriptylinePotassium voltage-gated channel subfamily A member 1target
AmitriptylineAlpha-1D adrenergic receptortarget
AmitriptylineDelta-type opioid receptortarget
AmitriptylineKappa-type opioid receptortarget
AmitriptylineHigh affinity nerve growth factor receptortarget
AmitriptylineBDNF/NT-3 growth factors receptortarget
AmitriptylineCytochrome P450 2C9enzyme
AmitriptylineCytochrome P450 2B6enzyme
AmitriptylineCytochrome P450 2C8enzyme
AmitriptylineHistamine H2 receptortarget
AmitriptylineHistamine H4 receptortarget
AmitriptylineSigma non-opioid intracellular receptor 1target
Amitriptyline5-hydroxytryptamine receptor 2Ctarget
AmitriptylineAlpha-1B adrenergic receptortarget
Amitriptyline5-hydroxytryptamine receptor 7target
Amitriptyline5-hydroxytryptamine receptor 1Dtarget
AmitriptylineMu-type opioid receptortarget
Amitriptyline5-hydroxytryptamine receptor 1Btarget
Amitriptyline5-hydroxytryptamine receptor 6target
AmitriptylinePotassium voltage-gated channel subfamily KQT member 3target
AmitriptylineUDP-glucuronosyltransferase 2B10enzyme
Amitriptyline5-hydroxytryptamine receptor 2Ctarget
AmitriptylineMuscarinic acetylcholine receptortarget
AmitriptylineHERG human cardiac K+ channeltarget
AmitriptylineATP-dependent translocase ABCB1transporter
AmitriptylineUDP-glucuronosyltransferase 1A4enzyme
AmitriptylineGlutathione S-transferases (Cytosolic)enzyme
Amitriptyline5-hydroxytryptamine receptor 1Atarget
Amitriptyline5-hydroxytryptamine receptor 2Atarget
AmitriptylineHistamine H1 receptortarget
AmitriptylineAlpha-1-acid glycoprotein 1carrier
AmitriptylineAlbumincarrier
AmitriptylineCytochrome P450 2D6enzyme
AmitriptylineCytochrome P450 2C19enzyme
AmitriptylineCytochrome P450 1A2enzyme
AmitriptylineAlpha-2A adrenergic receptortarget
AmitriptylinePotassium voltage-gated channel subfamily KQT member 2target
AmitriptylineSodium-dependent noradrenaline transportertarget
AmitriptylineSodium-dependent serotonin transportertarget
AmoxapineGABA(A) Receptortarget
AmoxapineHistamine H4 receptortarget
AmoxapineAlpha-2 adrenergic receptorstarget
Amoxapine5-hydroxytryptamine receptor 1Btarget
Amoxapine5-hydroxytryptamine receptor 1Atarget
Amoxapine5-hydroxytryptamine receptor 3Atarget
Amoxapine5-hydroxytryptamine receptor 2Btarget
AmoxapineMuscarinic acetylcholine receptortarget
AmoxapineAlpha-1 adrenergic receptorstarget
AmoxapineHistamine H1 receptortarget
AmoxapineD(4) dopamine receptortarget
AmoxapineD(3) dopamine receptortarget
Amoxapine5-hydroxytryptamine receptor 7target
Amoxapine5-hydroxytryptamine receptor 6target
Amoxapine5-hydroxytryptamine receptor 2Ctarget
Amoxapine5-hydroxytryptamine receptor 2Atarget
AmoxapineCytochrome P450 2D6enzyme
AmoxapineAlpha-1-acid glycoprotein 1carrier
AmoxapineGamma-aminobutyric acid receptor subunit alpha-1target
AmoxapineMuscarinic acetylcholine receptor M1target
AmoxapineD(1A) dopamine receptortarget
AmoxapineAlpha-1A adrenergic receptortarget
AmoxapineD(2) dopamine receptortarget
AmoxapineAlpha-2A adrenergic receptortarget
AmoxapineSodium-dependent noradrenaline transportertarget
AmoxapineSodium-dependent serotonin transportertarget
AmoxapineSodium-dependent dopamine transportertarget
AmoxapineDopamine receptortarget
BromocriptineD(4) dopamine receptortarget
Bromocriptine5-hydroxytryptamine receptor 2Btarget
BromocriptineAlpha-2B adrenergic receptortarget
BromocriptineAlpha-2C adrenergic receptortarget
Bromocriptine5-hydroxytryptamine receptor 1Atarget
BromocriptineD(3) dopamine receptortarget
BromocriptineAlpha-2A adrenergic receptortarget
Bromocriptine5-hydroxytryptamine receptor 1Dtarget
BromocriptineCytochrome P450 3A4enzyme
BromocriptineD(2) dopamine receptortarget
Bromocriptine5-hydroxytryptamine receptor 2Atarget
Bromocriptine5-hydroxytryptamine receptor 1Btarget
Bromocriptine5-hydroxytryptamine receptor 2Ctarget
BromocriptineD(1B) dopamine receptortarget
BromocriptineD(1A) dopamine receptortarget
BromocriptineAlpha-1A adrenergic receptortarget
BromocriptineAlpha-1B adrenergic receptortarget
BromocriptineAlpha-1D adrenergic receptortarget
BromocriptineATP-dependent translocase ABCB1transporter
Bromocriptine5-hydroxytryptamine receptor 7target
CabergolineATP-dependent translocase ABCB1transporter
CabergolineD(1) dopamine receptortarget
CabergolineBeta-2 adrenergic receptortarget
CabergolineBeta-1 adrenergic receptortarget
CabergolineAlpha-1D adrenergic receptortarget
CabergolineAlpha-1B adrenergic receptortarget
CabergolineAlpha-1A adrenergic receptortarget
Cabergoline5-hydroxytryptamine receptor 7target
CabergolineCytochrome P450 3A4enzyme
Cabergoline5-hydroxytryptamine receptor 2Ctarget
Cabergoline5-hydroxytryptamine receptor 1Btarget
CabergolineD(1A) dopamine receptortarget
CabergolineD(1B) dopamine receptortarget
CabergolineAlpha-2C adrenergic receptortarget
Cabergoline5-hydroxytryptamine receptor 1Atarget
CabergolineAlpha-2A adrenergic receptortarget
CabergolineD(4) dopamine receptortarget
Cabergoline5-hydroxytryptamine receptor 1Dtarget
CabergolineAlpha-2B adrenergic receptortarget
Cabergoline5-hydroxytryptamine receptor 2Atarget
CabergolineD(3) dopamine receptortarget
Cabergoline5-hydroxytryptamine receptor 2Btarget
CabergolineD(2) dopamine receptortarget
ChlorpheniramineCytochrome P450 3A4enzyme
ChlorpheniramineHistamine H1 receptortarget
ChlorpheniramineCytochrome P450 2D6enzyme
ChlorpheniramineSodium-dependent serotonin transportertarget
ChlorpheniramineSodium-dependent noradrenaline transportertarget
ChlorpheniramineSodium-dependent dopamine transportertarget
ChlorpheniramineCytochrome P450 3A5enzyme
ChlorpheniramineCytochrome P450 3A7enzyme
ChlorpheniramineSolute carrier family 22 member 2transporter
ChlorpheniramineSolute carrier family 22 member 1transporter
CitalopramATP-dependent translocase ABCB1transporter
CitalopramCytochrome P450 2C19enzyme
CitalopramAldehyde oxidaseenzyme
CitalopramAmine oxidase [flavin-containing] Benzyme
CitalopramAmine oxidase [flavin-containing] Aenzyme
CitalopramHistamine H1 receptortarget
CitalopramCytochrome P450 1A2enzyme
CitalopramCytochrome P450 3A4enzyme
CitalopramCytochrome P450 2D6enzyme
CitalopramSodium-dependent serotonin transportertarget
Clomipramine5-hydroxytryptamine receptor 2Btarget
ClomipramineCytochrome P450 3A4enzyme
ClomipramineATP-dependent translocase ABCB1transporter
ClomipramineCytochrome P450 2C19enzyme
ClomipramineCytochrome P450 2D6enzyme
ClomipramineCytochrome P450 1A2enzyme
Clomipramine5-hydroxytryptamine receptor 2Atarget
ClomipramineGlutathione S-transferase Ptarget
ClomipramineSodium-dependent noradrenaline transportertarget
Clomipramine5-hydroxytryptamine receptor 2Ctarget
ClomipramineAlbumincarrier
ClomipramineSodium-dependent serotonin transportertarget
DA-8031Sodium-dependent serotonin transportertarget
DapoxetineSodium-dependent serotonin transportertarget
DapoxetineCytochrome P450 2D6enzyme
DapoxetineCytochrome P450 3A4enzyme
Dapoxetine5-hydroxytryptamine receptor 2Ctarget
Dapoxetine5-hydroxytryptamine receptor 1Btarget
Dapoxetine5-hydroxytryptamine receptor 1Atarget
DesipramineMuscarinic acetylcholine receptor M2target
DesipramineSodium-dependent serotonin transportertarget
DesipramineHistamine H1 receptortarget
DesipramineBeta-1 adrenergic receptortarget
DesipramineCytochrome P450 2D6enzyme
DesipramineMuscarinic acetylcholine receptor M3target
DesipramineMuscarinic acetylcholine receptor M4target
DesipramineMuscarinic acetylcholine receptor M5target
DesipramineAlpha-1 adrenergic receptorstarget
Desipramine5-hydroxytryptamine receptor 2Atarget
DesipramineAlpha-1-acid glycoprotein 1carrier
DesipramineCytochrome P450 2B6enzyme
DesipramineCytochrome P450 3A4enzyme
DesipramineSolute carrier family 22 member 2transporter
DesipramineSolute carrier family 22 member 1transporter
DesipramineSolute carrier family 22 member 3transporter
DesipramineOrganic cation/carnitine transporter 2transporter
DesipramineATP-dependent translocase ABCB1transporter
DesipramineSolute carrier family 22 member 4transporter
DesipramineCytochrome P450 1A2enzyme
DesipramineCytochrome P450 2E1enzyme
DesipramineSphingomyelin phosphodiesterasetarget
Desipramine5-hydroxytryptamine receptor 1Atarget
Desipramine5-hydroxytryptamine receptor 2Ctarget
DesipramineD(2) dopamine receptortarget
DesipramineAlpha-2 adrenergic receptorstarget
DesipramineBeta-2 adrenergic receptortarget
DesipramineSodium-dependent noradrenaline transportertarget
DesipramineMuscarinic acetylcholine receptor M1target
DesvenlafaxineCytochrome P450 2C19enzyme
DesvenlafaxineUDP-glucuronosyltransferase 2B17enzyme
DesvenlafaxineUDP-glucuronosyltransferase 2B15enzyme
DesvenlafaxineUDP-glucuronosyltransferase 2B4enzyme
DesvenlafaxineCytochrome P450 3A4enzyme
DesvenlafaxineSodium-dependent serotonin transportertarget
DesvenlafaxineSodium-dependent noradrenaline transportertarget
DesvenlafaxineCytochrome P450 2D6enzyme
DesvenlafaxineSodium-dependent dopamine transportertarget
DesvenlafaxineUDP-glucuronosyltransferase 1A1enzyme
DesvenlafaxineUDP-glucuronosyltransferase 1A3enzyme
DexmethylphenidateSodium-dependent dopamine transportertarget
DexmethylphenidateSodium-dependent noradrenaline transportertarget
DexmethylphenidateSodium-dependent serotonin transportertarget
DexmethylphenidateCarboxylesteraseenzyme
DextromethorphanDelta-type opioid receptortarget
DextromethorphanNeuronal acetylcholine receptor subunit beta-4target
DextromethorphanGlutamate receptor ionotropic, NMDA 2Atarget
DextromethorphanUDP-glucuronosyltransferase 2B15enzyme
DextromethorphanUDP-glucuronosyltransferase 2B7enzyme
DextromethorphanUDP-glucuronosyltransferase 2B4enzyme
DextromethorphanSodium-dependent noradrenaline transportertarget
DextromethorphanNADPH oxidasetarget
DextromethorphanKappa-type opioid receptortarget
DextromethorphanUDP-glucuronosyltransferase 2B17enzyme
DextromethorphanMu-type opioid receptortarget
DextromethorphanNeuronal acetylcholine receptor subunit alpha-7target
DextromethorphanNeuronal acetylcholine receptor subunit beta-2target
DextromethorphanAromatasetarget
DextromethorphanNeuronal acetylcholine receptor subunit alpha-4target
DextromethorphanSigma non-opioid intracellular receptor 1target
DextromethorphanNeuronal acetylcholine receptor subunit alpha-2target
DextromethorphanSodium-dependent serotonin transportertarget
DextromethorphanGlutamate receptor ionotropic, NMDA 3Atarget
DextromethorphanCytochrome P450 2D6enzyme
DextromethorphanCytochrome P450 3A4enzyme
DextromethorphanCytochrome P450 3A7enzyme
DextromethorphanCytochrome P450 2C9enzyme
DextromethorphanCytochrome P450 2B6enzyme
DextromethorphanCytochrome P450 2C19enzyme
DextromethorphanMembrane-associated progesterone receptor component 1target
DextromethorphanNeuronal acetylcholine receptor subunit alpha-3target
Dihydroergotamine5-hydroxytryptamine receptor 1Dtarget
Dihydroergotamine5-hydroxytryptamine receptor 1Btarget
DihydroergotamineCytochrome P450 3A4enzyme
DihydroergotamineAlpha-2A adrenergic receptortarget
Dihydroergotamine5-hydroxytryptamine receptor 2Btarget
DihydroergotamineATP-dependent translocase ABCB1transporter
Dihydroergotamine5-hydroxytryptamine receptor 1Atarget
Dihydroergotamine5-hydroxytryptamine receptor 1Etarget
Dihydroergotamine5-hydroxytryptamine receptor 2Atarget
Dihydroergotamine5-hydroxytryptamine receptor 2Ctarget
DihydroergotamineAlpha-1 adrenergic receptorstarget
DihydroergotamineAlpha-2 adrenergic receptorstarget
DihydroergotamineD(2) dopamine receptortarget
DihydroergotamineD(3) dopamine receptortarget
DihydroergotamineD(4) dopamine receptortarget
Dihydroergotamine5-hydroxytryptamine receptor 1Ftarget
Dihydroergotamine5-hydroxytryptamine receptor 4target
DihydroergotamineBeta-3 adrenergic receptortarget
DosulepinCytochrome P450 1A2enzyme
Dosulepin5-hydroxytryptamine receptor 1Atarget
DosulepinCytochrome P450 2C19enzyme
DosulepinCytochrome P450 2C9enzyme
DosulepinCytochrome P450 3A4enzyme
Dosulepin5-hydroxytryptamine receptor 2Atarget
DosulepinAlpha-2 adrenergic receptorstarget
DosulepinAlpha-1 adrenergic receptorstarget
DosulepinSodium-dependent serotonin transportertarget
DosulepinSodium-dependent noradrenaline transportertarget
DosulepinMuscarinic acetylcholine receptor M5target
DosulepinMuscarinic acetylcholine receptor M4target
DosulepinMuscarinic acetylcholine receptor M3target
DosulepinMuscarinic acetylcholine receptor M2target
DosulepinMuscarinic acetylcholine receptor M1target
DosulepinHistamine H1 receptortarget
DosulepinCytochrome P450 2D6enzyme
DoxepinMuscarinic acetylcholine receptor M1target
DoxepinCytochrome P450 2D6enzyme
DoxepinHistamine H2 receptortarget
DoxepinHistamine H1 receptortarget
DoxepinSodium-dependent noradrenaline transportertarget
DoxepinCytochrome P450 1A2enzyme
DoxepinMuscarinic acetylcholine receptor M2target
DoxepinMuscarinic acetylcholine receptor M3target
DoxepinMuscarinic acetylcholine receptor M4target
DoxepinMuscarinic acetylcholine receptor M5target
DoxepinAlpha-1A adrenergic receptortarget
Doxepin5-hydroxytryptamine receptor 1Atarget
Doxepin5-hydroxytryptamine receptor 2Atarget
DoxepinCytochrome P450 2C19enzyme
DoxepinCytochrome P450 2C9enzyme
DoxepinSodium-dependent serotonin transportertarget
DoxepinATP-dependent translocase ABCB1transporter
Doxepin5-hydroxytryptamine receptor 2Btarget
Doxepin5-hydroxytryptamine receptor 2Ctarget
DoxepinAlpha-1-acid glycoprotein 1carrier
DoxepinAlpha-1B adrenergic receptortarget
DoxepinAlpha-1D adrenergic receptortarget
DoxepinCytochrome P450 3A4enzyme
Doxepin5-hydroxytryptamine receptor 6target
DoxepinHistamine H4 receptortarget
DoxepinVoltage-gated inwardly rectifying potassium channel KCNH2target
DoxepinAlbumincarrier
DuloxetineCytochrome P450 2C19enzyme
DuloxetineCytochrome P450 2B6enzyme
DuloxetineCytochrome P450 3A4enzyme
DuloxetineATP-dependent translocase ABCB1transporter
Duloxetinealpha1-acid glycoproteincarrier
DuloxetineAlbumincarrier
DuloxetineCytochrome P450 2C9enzyme
DuloxetineCytochrome P450 2D6enzyme
DuloxetineCytochrome P450 1A2enzyme
DuloxetineSodium-dependent noradrenaline transportertarget
DuloxetineSodium-dependent dopamine transportertarget
DuloxetineSodium-dependent serotonin transportertarget
Eletriptan5-hydroxytryptamine receptor 1Atarget
Eletriptan5-hydroxytryptamine receptor 7target
Eletriptan5-hydroxytryptamine receptor 2Btarget
Eletriptan5-hydroxytryptamine receptor 1Etarget
EletriptanATP-dependent translocase ABCB1transporter
EletriptanCytochrome P450 2A6enzyme
EletriptanProstaglandin G/H synthase 1enzyme
EletriptanCytochrome P450 2C19enzyme
EletriptanCytochrome P450 2C9enzyme
EletriptanCytochrome P450 2D6enzyme
EletriptanCytochrome P450 3A4enzyme
Eletriptan5-hydroxytryptamine receptor 1Btarget
Eletriptan5-hydroxytryptamine receptor 1Ftarget
Eletriptan5-hydroxytryptamine receptor 1Dtarget
Ergoloid mesylateCytochrome P450 3A4enzyme
Ergoloid mesylateSerotonin Receptorstarget
Ergoloid mesylateBeta adrenergic receptortarget
Ergoloid mesylateAlpha adrenergic receptortarget
Ergoloid mesylateDopamine receptortarget
ErgometrineATP-dependent translocase ABCB1transporter
ErgometrineCytochrome P450 3A4enzyme
ErgometrineAlpha-1A adrenergic receptortarget
ErgometrineD(2) dopamine receptortarget
Ergotamine5-hydroxytryptamine receptor 1Dtarget
Ergotamine5-hydroxytryptamine receptor 1Atarget
ErgotamineAlpha-1A adrenergic receptortarget
ErgotamineAlpha adrenergic receptortarget
ErgotamineAlpha-2C adrenergic receptortarget
Ergotamine5-hydroxytryptamine receptor 2Btarget
Ergotamine5-hydroxytryptamine receptor 2Ctarget
Ergotamine5-hydroxytryptamine receptor 1Ftarget
Ergotamine5-hydroxytryptamine receptor 1Btarget
ErgotamineD(1) dopamine receptortarget
ErgotamineATP-dependent translocase ABCB1transporter
ErgotamineAlpha-1D adrenergic receptortarget
ErgotamineAlpha-1B adrenergic receptortarget
ErgotamineCytochrome P450 3A4enzyme
ErgotamineD(2) dopamine receptortarget
ErgotamineAlpha-2A adrenergic receptortarget
Ergotamine5-hydroxytryptamine receptor 2Atarget
EscitalopramCytochrome P450 2C19enzyme
EscitalopramATP-dependent translocase ABCB1transporter
Escitalopram5-hydroxytryptamine receptor 1Atarget
Escitalopram5-hydroxytryptamine receptor 2Atarget
Escitalopram5-hydroxytryptamine receptor 2Ctarget
EscitalopramAlpha-1 adrenergic receptorstarget
EscitalopramAlpha-2 adrenergic receptorstarget
EscitalopramD(2) dopamine receptortarget
EscitalopramAmine oxidase [flavin-containing] Aenzyme
EscitalopramAmine oxidase [flavin-containing] Benzyme
EscitalopramAldehyde oxidaseenzyme
EscitalopramHistamine H1 receptortarget
EscitalopramMuscarinic acetylcholine receptor M1target
EscitalopramSodium-dependent noradrenaline transportertarget
EscitalopramSodium-dependent dopamine transportertarget
EscitalopramCytochrome P450 2D6enzyme
EscitalopramCytochrome P450 3A4enzyme
EscitalopramSodium-dependent serotonin transportertarget
Etoperidone5-hydroxytryptamine receptor 2Atarget
EtoperidoneAlpha-1 adrenergic receptorstarget
Etoperidone5-hydroxytryptamine receptor 2Ctarget
EtoperidoneAlpha-2 adrenergic receptorstarget
EtoperidoneSodium-dependent serotonin transportertransporter
EtoperidoneD(2) dopamine receptortarget
EtoperidoneMuscarinic acetylcholine receptortarget
EtoperidoneSodium-dependent dopamine transportertransporter
EtoperidoneSodium-dependent noradrenaline transportertransporter
FemoxetineSodium-dependent serotonin transportertarget
FemoxetineSerotonin Receptorstarget
FentanylMu-type opioid receptortarget
Fentanylalpha1-acid glycoproteincarrier
FentanylAlbumincarrier
FentanylATP-dependent translocase ABCB1target
FentanylKappa-type opioid receptortarget
FentanylATP-dependent translocase ABCB1transporter
FentanylCytochrome P450 3A7enzyme
FentanylCytochrome P450 3A4enzyme
FentanylDelta-type opioid receptortarget
Flibanserin5-hydroxytryptamine receptor 1Atarget
Flibanserin5-hydroxytryptamine receptor 2Atarget
FlibanserinD(4) dopamine receptortarget
FlibanserinCytochrome P450 3A4enzyme
FlibanserinATP-dependent translocase ABCB1transporter
FluoxetineNeuronal acetylcholine receptor subunit alpha-3target
FluoxetineNeuronal acetylcholine receptor subunit alpha-2target
FluoxetineNeuronal acetylcholine receptor subunit beta-4target
FluoxetineSodium-dependent serotonin transportertarget
FluoxetineCytochrome P450 2C9enzyme
FluoxetineCytochrome P450 2D6enzyme
FluoxetineCytochrome P450enzyme
FluoxetineCytochrome P450 1A2enzyme
FluoxetineCytochrome P450 3A4enzyme
FluoxetineCyclin-dependent kinases regulatory subunit 1target
Fluoxetine5-hydroxytryptamine receptor 2Ctarget
FluoxetineVoltage-gated inwardly rectifying potassium channel KCNH2target
FluoxetineAlpha-1-acid glycoprotein 1carrier
FluoxetineAlbumincarrier
FluoxetineCytochrome P450 3A5enzyme
FluoxetineCytochrome P450 2B6enzyme
FluoxetineATP-dependent translocase ABCB1transporter
FluoxetineCytochrome P450 2C19enzyme
FluvoxamineCytochrome P450 2C9enzyme
FluvoxamineBile salt export pumptransporter
FluvoxamineVoltage-gated inwardly rectifying potassium channel KCNH2target
FluvoxamineCytochrome P450 2B6enzyme
FluvoxamineCytochrome P450 2D6enzyme
FluvoxamineATP-dependent translocase ABCB1transporter
FluvoxamineCytochrome P450 3A4enzyme
FluvoxamineCytochrome P450 1A1enzyme
FluvoxamineCytochrome P450 2C19enzyme
FluvoxamineCytochrome P450 1A2enzyme
FluvoxamineSodium-dependent serotonin transportertarget
FluvoxamineCytochrome P450 3A Subfamilyenzyme
Frovatriptan5-hydroxytryptamine receptor 1Btarget
Frovatriptan5-hydroxytryptamine receptor 1Dtarget
FrovatriptanCytochrome P450 1A2enzyme
ImipramineAlbumincarrier
ImipramineVoltage-gated delayed rectifier potassium channel KCNH1target
Imipramine5-hydroxytryptamine receptor 6target
Imipramine5-hydroxytryptamine receptor 1Atarget
ImipramineSodium-dependent dopamine transportertarget
ImipramineVoltage-gated inwardly rectifying potassium channel KCNH2target
ImipramineD(2) dopamine receptortarget
ImipramineD(1) dopamine receptortarget
Imipramine5-hydroxytryptamine receptor 7target
ImipramineAlpha-1B adrenergic receptortarget
Imipramine5-hydroxytryptamine receptor 2Ctarget
ImipramineCytochrome P450 3A7enzyme
ImipramineCytochrome P450 2E1enzyme
ImipramineCytochrome P450 2C18enzyme
ImipramineCytochrome P450 1A2enzyme
ImipramineCytochrome P450 2B6enzyme
ImipramineCytochrome P450 3A4enzyme
ImipramineSolute carrier family 22 member 4transporter
ImipramineATP-dependent translocase ABCB1transporter
ImipramineSolute carrier family 22 member 3transporter
ImipramineSolute carrier family 22 member 2transporter
ImipramineAlpha-1-acid glycoprotein 1carrier
ImipramineAlpha-1D adrenergic receptortarget
ImipramineA-type voltage-gated potassium channel KCND3target
ImipramineA-type voltage-gated potassium channel KCND2target
ImipramineMuscarinic acetylcholine receptor M5target
ImipramineMuscarinic acetylcholine receptor M4target
ImipramineMuscarinic acetylcholine receptor M3target
ImipramineMuscarinic acetylcholine receptor M2target
ImipramineMuscarinic acetylcholine receptor M1target
Imipramine5-hydroxytryptamine receptor 2Atarget
ImipramineAlpha-1A adrenergic receptortarget
ImipramineHistamine H1 receptortarget
ImipramineCytochrome P450 2D6enzyme
ImipramineCytochrome P450 2C19enzyme
ImipramineSodium-dependent noradrenaline transportertarget
ImipramineSodium-dependent serotonin transportertarget
IndalpineSodium-dependent serotonin transportertarget
IndalpineCytochrome P450 3A4enzyme
IsocarboxazidAmine oxidase [flavin-containing] Atarget
IsocarboxazidMonoamine oxidasetarget
IsocarboxazidAmine oxidase [flavin-containing] Btarget
LevomilnacipranATP-dependent translocase ABCB1transporter
LevomilnacipranSodium-dependent noradrenaline transportertarget
LevomilnacipranSodium-dependent serotonin transportertarget
LevomilnacipranCytochrome P450 2J2enzyme
LevomilnacipranCytochrome P450 2D6enzyme
LevomilnacipranCytochrome P450 2C19enzyme
LevomilnacipranCytochrome P450 2C8enzyme
LevomilnacipranCytochrome P450 3A4enzyme
Linezolid23S ribosomal RNAtarget
LinezolidAmine oxidase [flavin-containing] Aenzyme
LinezolidAmine oxidase [flavin-containing] Benzyme
LinezolidAlbumincarrier
LinezolidSolute carrier family 22 member 6transporter
LinezolidOrganic anion transporter 3transporter
Lithium carbonateInositol monophosphatase 2target
Lithium carbonateInositol monophosphatase 1target
Lithium carbonateGlycogen synthase kinase-3 betatarget
Lithium carbonateGlutamate receptor 3target
Lithium carbonateEpithelial sodium channel subunit alphatransporter
Lithium carbonateEpithelial sodium channel subunit betatransporter
Lithium carbonateEpithelial sodium channel subunit gammatransporter
Lithium carbonateGlycogen synthase kinase-3 alphatarget
Lithium cationGlutamate receptor 3target
Lithium cationGlycogen synthase kinase-3 betatarget
Lithium cationInositol monophosphatase 1target
Lithium cationInositol monophosphatase 2target
Lithium citrateGlutamate receptor 3target
Lithium citrateGlycogen synthase kinase-3 betatarget
Lithium citrateInositol monophosphatase 1target
Lithium citrateInositol monophosphatase 2target
LorcaserinCytochrome P450 1A1enzyme
LorcaserinFlavin-containing monooxygenase 1enzyme
LorcaserinCytochrome P450 3A4enzyme
LorcaserinCytochrome P450 2D6enzyme
LorcaserinCytochrome P450 2C19enzyme
LorcaserinCytochrome P450 2B6enzyme
LorcaserinCytochrome P450 2A6enzyme
LorcaserinCytochrome P450 1A2enzyme
Lorcaserin5-hydroxytryptamine receptor 2Ctarget
LorpiprazoleAlpha-2 adrenergic receptorstarget
Lorpiprazole5-hydroxytryptamine receptor 2Ctarget
LorpiprazoleAlpha-1 adrenergic receptorstarget
Lorpiprazole5-hydroxytryptamine receptor 2Atarget
LorpiprazoleHistamine H1 receptortarget
LorpiprazoleSodium-dependent serotonin transportertarget
LorpiprazoleCytochrome P450 2D6enzyme
LorpiprazoleCytochrome P450 3A4enzyme
LorpiprazoleAlbumincarrier
Lumateperone5-hydroxytryptamine receptor 2Atarget
LumateperoneD(2) dopamine receptortarget
LumateperoneD(1A) dopamine receptortarget
LumateperoneSodium-dependent serotonin transportertarget
LumateperoneAldo-keto reductase familyenzyme
LumateperoneCytochrome P450 3A4enzyme
LumateperoneCytochrome P450 2C8enzyme
LumateperoneCytochrome P450 1A2enzyme
LumateperoneUDP-glucuronosyltransferase 1A1enzyme
LumateperoneUDP-glucuronosyltransferase 1A4enzyme
LumateperoneUDP-glucuronosyltransferase 2B15enzyme
LumateperoneAldo-keto reductase family 1 member C1enzyme
LumateperoneAldo-keto reductase family 1 member B10enzyme
LumateperoneAldo-keto reductase family 1 member C4enzyme
MaprotilineMuscarinic acetylcholine receptor M5target
MaprotilineAlpha-2 adrenergic receptorstarget
MaprotilineD(2) dopamine receptortarget
Maprotiline5-hydroxytryptamine receptor 7target
Maprotiline5-hydroxytryptamine receptor 2Ctarget
Maprotiline5-hydroxytryptamine receptor 2Atarget
MaprotilineCytochrome P450 1A2enzyme
MaprotilineMuscarinic acetylcholine receptor M4target
MaprotilineMuscarinic acetylcholine receptor M3target
MaprotilineMuscarinic acetylcholine receptor M2target
MaprotilineMuscarinic acetylcholine receptor M1target
MaprotilineAlpha-1-acid glycoprotein 1carrier
MaprotilineCytochrome P450 2D6enzyme
MaprotilineAlpha-1 adrenergic receptorstarget
MaprotilineSodium-dependent noradrenaline transportertarget
MaprotilineHistamine H1 receptortarget
MazindolSynaptic vesicular amine transportertarget
MazindolSodium-dependent serotonin transportertarget
MazindolSodium-dependent dopamine transportertarget
MazindolSodium-dependent noradrenaline transportertarget
MeperidineGlutamate receptor ionotropic, NMDA 1target
MeperidineATP-dependent translocase ABCB1transporter
MeperidineCytochrome P450 1A2enzyme
MeperidineLiver carboxylesterase 1target
MeperidineSodium-dependent serotonin transportertarget
MeperidineSodium-dependent noradrenaline transportertarget
MeperidineSodium-dependent dopamine transportertarget
MeperidineMu-type opioid receptortarget
MeperidineMuscarinic acetylcholine receptortarget
MeperidineAlpha-1-acid glycoprotein 1carrier
MeperidineAlbumincarrier
MeperidineCytochrome P450 3A4enzyme
MeperidineCytochrome P450 2C19enzyme
MeperidineGlutamate receptor ionotropic, NMDA 2Dtarget
MeperidineKappa-type opioid receptortarget
MeperidineCytochrome P450 2D6enzyme
MeperidineCytochrome P450 2B6enzyme
MeperidineGlutamate receptor ionotropic, NMDA 2Ctarget
MeperidineGlutamate receptor ionotropic, NMDA 2Btarget
MeperidineGlutamate receptor ionotropic, NMDA 2Atarget
MethadoneMu-type opioid receptortarget
MethadoneNeuronal acetylcholine receptor subunit alpha-4target
MethadoneCytochrome P450 2B6enzyme
MethadoneCytochrome P450 3A4enzyme
MethadoneCytochrome P450 2C19enzyme
MethadoneDelta-type opioid receptortarget
MethadoneCytochrome P450 3A7enzyme
MethadoneCytochrome P450 2D6enzyme
MethadoneATP-dependent translocase ABCB1transporter
MethadoneCytochrome P450 2C8enzyme
MethadoneAromataseenzyme
MethadoneCytochrome P450 1A2enzyme
MethadoneNMDA receptortarget
MethadoneCytochrome P450 2C18enzyme
MethadoneCytochrome P450 2C9enzyme
Methadone5-hydroxytryptamine receptor 3Atarget
MethadoneUDP-glucuronosyltransferase 2B4enzyme
MethadoneCytochrome P450 3A Subfamilyenzyme
MethadoneNeuronal acetylcholine receptor subunit beta-2target
MethadoneAlpha-1-acid glycoprotein 1carrier
MethadoneNeuronal acetylcholine receptor subunit alpha-3target
MethadoneNeuronal acetylcholine receptor subunit alpha-7target
MethadoneAlbumincarrier
MianserinSodium-dependent serotonin transportertarget
MianserinCytochrome P450 3A4enzyme
MianserinCytochrome P450 1A2enzyme
MianserinCytochrome P450 2B6enzyme
MianserinSodium-dependent noradrenaline transportertarget
MianserinHistamine H4 receptortarget
Mianserin5-hydroxytryptamine receptor 1Atarget
MianserinAlpha-2C adrenergic receptortarget
Mianserin5-hydroxytryptamine receptor 2Btarget
Mianserin5-hydroxytryptamine receptor 1Ftarget
Mianserin5-hydroxytryptamine receptor 7target
MianserinD(3) dopamine receptortarget
MianserinKappa-type opioid receptortarget
MianserinSodium-dependent dopamine transportertarget
MianserinD(2) dopamine receptortarget
Mianserin5-hydroxytryptamine receptor 6target
MianserinAlpha-1 adrenergic receptorstarget
MianserinD(1) dopamine receptortarget
MianserinCytochrome P450 2D6enzyme
Mianserin5-hydroxytryptamine receptor 2Ctarget
Mianserin5-hydroxytryptamine receptor 2Atarget
MianserinAlpha-2A adrenergic receptortarget
MianserinHistamine H1 receptortarget
MianserinAlpha-2B adrenergic receptortarget
MilnacipranSodium-dependent noradrenaline transportertarget
MilnacipranNMDA receptortarget
MilnacipranCytochrome P450 3A4enzyme
MilnacipranSodium-dependent serotonin transportertarget
MirtazapineAlpha-2 adrenergic receptorstarget
Mirtazapine5HT3 serotonin receptortarget
MirtazapineAlpha-2A adrenergic receptortarget
Mirtazapine5-hydroxytryptamine receptor 2Ctarget
MirtazapineKappa-type opioid receptortarget
MirtazapineHistamine H1 receptortarget
MirtazapineCytochrome P450 1A2enzyme
MirtazapineCytochrome P450 3A4enzyme
MirtazapineCytochrome P450 2D6enzyme
MirtazapineAlpha-1 adrenergic receptorstarget
MirtazapineSodium-dependent serotonin transportertransporter
Mirtazapine5-hydroxytryptamine receptor 2Atarget
MoclobemideAmine oxidase [flavin-containing] Benzyme
MoclobemideAmine oxidase [flavin-containing] Btarget
MoclobemideCytochrome P450 2D6enzyme
MoclobemideCytochrome P450 2C19enzyme
MoclobemideAmine oxidase [flavin-containing] Atarget
MoclobemideAmine oxidase [flavin-containing] Aenzyme
MoclobemideCytochrome P450 2C9enzyme
MoclobemideMonoamine oxidasetarget
NaratriptanAmine oxidase [flavin-containing] Aenzyme
Naratriptan5-hydroxytryptamine receptor 1Atarget
Naratriptan5-hydroxytryptamine receptor 1Ftarget
Naratriptan5-hydroxytryptamine receptor 1Btarget
Naratriptan5-hydroxytryptamine receptor 1Dtarget
NefazodoneBile salt export pumptransporter
NefazodoneSolute carrier organic anion transporter family member 2B1transporter
NefazodoneSolute carrier organic anion transporter family member 1B3transporter
NefazodoneCytochrome P450 3A Subfamilyenzyme
NefazodoneVoltage-gated inwardly rectifying potassium channel KCNH2target
NefazodoneATP-dependent translocase ABCB1transporter
NefazodoneCytochrome P450enzyme
Nefazodone5-hydroxytryptamine receptor 1Atarget
NefazodoneAlpha-2A adrenergic receptortarget
NefazodoneSodium-dependent dopamine transportertarget
NefazodoneCytochrome P450 2D6enzyme
NefazodoneCytochrome P450 3A4enzyme
NefazodoneAlpha-1B adrenergic receptortarget
NefazodoneAlpha-1A adrenergic receptortarget
NefazodoneSodium-dependent noradrenaline transportertarget
NefazodoneSodium-dependent serotonin transportertarget
Nefazodone5-hydroxytryptamine receptor 2Atarget
Nefazodone5-hydroxytryptamine receptor 2Ctarget
NortriptylineATP-dependent translocase ABCB1transporter
NortriptylineMuscarinic acetylcholine receptortarget
NortriptylineSodium-dependent noradrenaline transportertransporter
Nortriptyline5-hydroxytryptamine receptor 2Ctarget
NortriptylineSigma receptortarget
NortriptylineD(2) dopamine receptortarget
NortriptylineBeta adrenergic receptortarget
NortriptylineAlpha-2 adrenergic receptorstarget
NortriptylineSodium-dependent serotonin transportertarget
NortriptylineSodium-dependent noradrenaline transportertarget
NortriptylineCytochrome P450 1A2enzyme
NortriptylineCytochrome P450 2D6enzyme
NortriptylineAlbumincarrier
NortriptylineAlpha-1-acid glycoprotein 1carrier
NortriptylineHistamine H1 receptortarget
Nortriptyline5-hydroxytryptamine receptor 2Atarget
NortriptylineAlpha-1A adrenergic receptortarget
NortriptylineAlpha-1B adrenergic receptortarget
Nortriptyline5-hydroxytryptamine receptor 2Ctarget
NortriptylineCytochrome P450 2E1enzyme
NortriptylineCytochrome P450 2C19enzyme
NortriptylineAlpha-1D adrenergic receptortarget
NortriptylineCytochrome P450 3A5enzyme
NortriptylineCytochrome P450 3A4enzyme
Nortriptyline5-hydroxytryptamine receptor 1Atarget
ParoxetineSodium-dependent serotonin transportertarget
ParoxetineSodium-dependent noradrenaline transportertarget
Paroxetine5-hydroxytryptamine receptor 2Atarget
ParoxetineCytochrome P450 2D6enzyme
ParoxetineCytochrome P450 2B6enzyme
ParoxetineCytochrome P450 1A2enzyme
ParoxetineCytochrome P450 3A4enzyme
ParoxetineAlpha-1 adrenergic receptorstarget
ParoxetineAlpha-2 adrenergic receptorstarget
ParoxetineBeta adrenergic receptortarget
ParoxetineD(2) dopamine receptortarget
ParoxetineHistamine H1 receptortarget
ParoxetineMuscarinic acetylcholine receptortarget
Paroxetine5-hydroxytryptamine receptor 2Btarget
ParoxetineD(1) dopamine receptortarget
ParoxetineCytochrome P450 2C19enzyme
ParoxetineATP-dependent translocase ABCB1transporter
ParoxetineCytochrome P450 2C9enzyme
PhenelzineAmine oxidase [flavin-containing] Btarget
PhenelzineAmine oxidase [flavin-containing] Atarget
PhenelzineAmine oxidase [flavin-containing] Aenzyme
PhenelzineAmine oxidase [copper-containing] 3target
PhenelzineAmine oxidase [flavin-containing] Benzyme
PhenelzineMonoamine oxidasetarget
PhenelzineCytochrome P450 3A Subfamilyenzyme
PhenelzineCytochrome P450 2D6enzyme
PhenelzineCytochrome P450 3A7enzyme
PhenelzineCytochrome P450 3A5enzyme
PhenelzineCytochrome P450 3A4enzyme
PhenelzineCytochrome P450 2C8enzyme
PhenelzineCytochrome P450 2C19enzyme
PhenelzineAlanine aminotransferase 2target
PhenelzineCytochrome P450 2E1enzyme
PhenelzineAlanine aminotransferase 1target
PhenelzineGlutamate decarboxylase 2target
Phenelzine4-aminobutyrate aminotransferase, mitochondrialtarget
ProcarbazineMonoamine oxidasetarget
ProcarbazineXanthine dehydrogenase/oxidaseenzyme
ProcarbazineDNAtarget
PromethazineNMDA receptortarget
PromethazineCalmodulintarget
PromethazineAlbumincarrier
PromethazineATP-binding cassette sub-family C member 4transporter
PromethazineATP-binding cassette sub-family C member 3transporter
PromethazineVoltage-gated Potassium Channelstarget
PromethazineVoltage-gated sodium channel alpha subunittarget
PromethazineP2 Purinoceptorstarget
PromethazineAlpha adrenergic receptortarget
PromethazineHistamine H2 receptortarget
PromethazineCytochrome P450 2C9enzyme
PromethazineATP-dependent translocase ABCB1transporter
PromethazineCytochrome P450 2B6enzyme
PromethazineCytochrome P450 2D6enzyme
PromethazineMuscarinic acetylcholine receptor M3target
PromethazineMuscarinic acetylcholine receptor M2target
PromethazineMuscarinic acetylcholine receptor M5target
PromethazineMuscarinic acetylcholine receptor M1target
PromethazineMuscarinic acetylcholine receptor M4target
PromethazineHistamine H1 receptortarget
PromethazineD(2) dopamine receptortarget
ProtriptylineSodium-dependent noradrenaline transportertarget
ProtriptylineSodium-dependent serotonin transportertarget
ProtriptylineATP-dependent translocase ABCB1transporter
RasagilineCytochrome P450 1A2enzyme
RasagilineApoptosis regulator Bcl-2target
RasagilineAmine oxidase [flavin-containing] Btarget
Ritanserin5-hydroxytryptamine receptor 2Atarget
RitanserinCytochrome P450 2D6enzyme
Ritanserin5-hydroxytryptamine receptor 2Btarget
RitanserinVoltage-dependent N-type calcium channel subunit alpha-1Btarget
Ritanserin5-hydroxytryptamine receptor 2Ctarget
Rizatriptan5-hydroxytryptamine receptor 1Atarget
Rizatriptan5-hydroxytryptamine receptor 1Dtarget
Rizatriptan5-hydroxytryptamine receptor 1Btarget
Rizatriptan5-hydroxytryptamine receptor 1Ftarget
RizatriptanAmine oxidase [flavin-containing] Aenzyme
RizatriptanCytochrome P450 2D6enzyme
Rizatriptan5-hydroxytryptamine receptor 1Etarget
Rizatriptan5-hydroxytryptamine receptor 7target
SelegilineCytochrome P450 2D6enzyme
SelegilineSubstance-P receptortarget
SelegilineCytochrome P450 2C9enzyme
SelegilineCytochrome P450 2C8enzyme
SelegilineCytochrome P450 2C19enzyme
SelegilineCytochrome P450 1A2enzyme
SelegilineATP-dependent translocase ABCB1transporter
SelegilineCytochrome P450 3A4enzyme
SelegilineCytochrome P450 2A6enzyme
SelegilineAmine oxidase [flavin-containing] Atarget
SelegilineCytochrome P450 2B6enzyme
SelegilineAmine oxidase [flavin-containing] Btarget
SeproxetineSodium-dependent serotonin transportertarget
SeproxetineSodium-dependent noradrenaline transportertarget
SeproxetineCytochrome P450 3A4enzyme
SeproxetineCytochrome P450 2C19enzyme
SeproxetineCytochrome P450 2C9enzyme
SeproxetineCytochrome P450 3A7enzyme
SeproxetineCytochrome P450 3A5enzyme
SeproxetineSodium-dependent dopamine transportertarget
SertralineCytochrome P450 2D6enzyme
SertralineCytochrome P450 2C9enzyme
SertralineCytochrome P450 2C19enzyme
SertralineCytochrome P450 2B6enzyme
SertralineSodium-dependent serotonin transportertarget
SertralineSodium-dependent dopamine transportertarget
SertralineCytochrome P450enzyme
SertralineCytochrome P450 3A4enzyme
SertralineAmine oxidase [flavin-containing] Benzyme
SertralineCytochrome P450 2E1enzyme
SertralineEquilibrative nucleoside transporter 4target
SertralineSodium-dependent noradrenaline transportertarget
SertralineSigma receptortarget
SertralineAlbumincarrier
SertralineATP-dependent translocase ABCB1transporter
SertralineAmine oxidase [flavin-containing] Aenzyme
SibutramineSodium-dependent dopamine transportertarget
SibutramineSodium-dependent serotonin transportertarget
SibutramineCytochrome P450 3A4enzyme
SibutramineSodium-dependent noradrenaline transportertarget
SumatriptanSolute carrier organic anion transporter family member 1B1transporter
SumatriptanBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
SumatriptanATP-dependent translocase ABCB1transporter
SumatriptanSolute carrier organic anion transporter family member 1A2transporter
Sumatriptan5-hydroxytryptamine receptor 1Atarget
SumatriptanAmine oxidase [flavin-containing] Aenzyme
Sumatriptan5-hydroxytryptamine receptor 1Ftarget
Sumatriptan5-hydroxytryptamine receptor 1Btarget
Sumatriptan5-hydroxytryptamine receptor 1Dtarget
TapentadolSodium-dependent noradrenaline transportertarget
TapentadolUDP-glucuronosyltransferase 1A9enzyme
TapentadolSodium-dependent serotonin transportertarget
TapentadolCytochrome P450 2C19enzyme
TapentadolCytochrome P450 2C9enzyme
TapentadolCytochrome P450 2D6enzyme
TapentadolUDP-glucuronosyltransferase 2B7enzyme
TapentadolDelta-type opioid receptortarget
TapentadolKappa-type opioid receptortarget
TapentadolMu-type opioid receptortarget
Tedizolid phosphateAmine oxidase [flavin-containing] Benzyme
Tedizolid phosphateAmine oxidase [flavin-containing] Aenzyme
Tedizolid phosphate23S ribosomal RNAtarget
TenamfetamineSodium-dependent dopamine transportertarget
TenamfetamineSodium-dependent serotonin transportertarget
TenamfetamineSodium-dependent noradrenaline transportertarget
TianeptineSodium-dependent serotonin transportertarget
TianeptineCytochrome P450 3A4enzyme
TianeptineD(3) dopamine receptortarget
Tianeptine5-hydroxytryptamine receptor 1Atarget
TianeptineGlutamate receptor 1target
TianeptineMu-type opioid receptortarget
TramadolMu-type opioid receptortarget
TramadolAlpha-2 adrenergic receptorstarget
TramadolAdenosine receptor A1target
TramadolNMDA receptortarget
TramadolTransient receptor potential cation channel subfamily V member 1target
TramadolSodium channel protein type 2 subunit alphatarget
TramadolSubstance-P receptortarget
TramadolUDP-glucuronosyltransferase 1A1enzyme
TramadolMuscarinic acetylcholine receptor M1target
TramadolMuscarinic acetylcholine receptor M3target
TramadolNeuronal acetylcholine receptor subunit alpha-7target
TramadolCytochrome P450 2B6enzyme
TramadolCytochrome P450 3A4enzyme
TramadolDelta-type opioid receptortarget
TramadolCytochrome P450 2D6enzyme
TramadolSodium-dependent serotonin transportertarget
TramadolKappa-type opioid receptortarget
Tramadol5-hydroxytryptamine receptor 2Ctarget
TramadolSodium-dependent noradrenaline transportertarget
TranylcypromineCytochrome P450 3A4enzyme
TranylcypromineMonoamine oxidasetarget
TranylcypromineCytochrome P450 1A2enzyme
TranylcypromineCytochrome P450 2D6enzyme
TranylcypromineCytochrome P450 2A6enzyme
TranylcypromineCytochrome P450 2C19enzyme
TranylcypromineAmine oxidase [flavin-containing] Atarget
TranylcypromineAmine oxidase [flavin-containing] Btarget
TranylcypromineCytochrome P450 2C9enzyme
Trazodone5-hydroxytryptamine receptor 2Atarget
Trazodone5-hydroxytryptamine receptor 2Ctarget
TrazodoneSodium-dependent serotonin transportertarget
TrazodoneAlpha-1A adrenergic receptortarget
TrazodoneAlpha-2A adrenergic receptortarget
TrazodoneHistamine H1 receptortarget
Trazodone5-hydroxytryptamine receptor 1Atarget
TrazodoneCytochrome P450 2D6enzyme
TrazodoneCytochrome P450 3A4enzyme
Trazodone5-hydroxytryptamine receptor 2Ctarget
TrazodoneCytochrome P450 3A5enzyme
TrazodoneCytochrome P450 3A7enzyme
TrazodoneATP-dependent translocase ABCB1transporter
TrimipramineHistamine H1 receptortarget
TrimipramineCytochrome P450 2C19enzyme
TrimipramineATP-dependent translocase ABCB1transporter
TrimipramineCytochrome P450 2C9enzyme
Trimipramine5-hydroxytryptamine receptor 2Ctarget
Trimipramine5-hydroxytryptamine receptor 3Atarget
Trimipramine5-hydroxytryptamine receptor 1Dtarget
TrimipramineSodium-dependent noradrenaline transportertarget
TrimipramineSodium-dependent serotonin transportertarget
TrimipramineAlpha-2A adrenergic receptortarget
TrimipramineD(1) dopamine receptortarget
TrimipramineBeta adrenergic receptortarget
TrimipramineMuscarinic acetylcholine receptortarget
Trimipramine5-hydroxytryptamine receptor 2Ctarget
TrimipramineAlpha-1 adrenergic receptorstarget
TrimipramineAlpha-2B adrenergic receptortarget
TrimipramineD(2) dopamine receptortarget
TrimipramineCytochrome P450 2D6enzyme
TrimipramineAlpha-1A adrenergic receptortarget
Trimipramine5-hydroxytryptamine receptor 1Atarget
Trimipramine5-hydroxytryptamine receptor 2Atarget
TrimipramineSodium-dependent dopamine transportertarget
TrimipramineAlpha-1B adrenergic receptortarget
VenlafaxineSodium-dependent serotonin transportertarget
VenlafaxineSodium-dependent noradrenaline transportertarget
VenlafaxineCytochrome P450 2D6enzyme
VenlafaxineCytochrome P450 3A4enzyme
VenlafaxineSodium-dependent dopamine transportertarget
VenlafaxineATP-dependent translocase ABCB1transporter
VenlafaxineBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
VenlafaxineCytochrome P450 2C9enzyme
VenlafaxineCytochrome P450 2C19enzyme
Vilazodone5-hydroxytryptamine receptor 1Atarget
VilazodoneCytochrome P450 2D6enzyme
VilazodoneSodium-dependent serotonin transportertarget
VilazodoneCytochrome P450 2C19enzyme
VilazodoneCytochrome P450 3A4enzyme
VortioxetineCytochrome P450 2A6enzyme
VortioxetineCytochrome P450 2C8enzyme
VortioxetineCytochrome P450 2B6enzyme
VortioxetineCytochrome P450 2C9enzyme
VortioxetineCytochrome P450 2C19enzyme
VortioxetineCytochrome P450 3A5enzyme
VortioxetineCytochrome P450 3A4enzyme
VortioxetineCytochrome P450 2D6enzyme
VortioxetineSodium-dependent noradrenaline transportertarget
VortioxetineBeta-1 adrenergic receptortarget
Vortioxetine5-hydroxytryptamine receptor 1Btarget
Vortioxetine5-hydroxytryptamine receptor 7target
Vortioxetine5-hydroxytryptamine receptor 3Atarget
VortioxetineSodium-dependent serotonin transportertarget
Vortioxetine5-hydroxytryptamine receptor 1Atarget
ZimelidineSerotonin Receptorstarget
ZimelidineSodium-dependent serotonin transportertarget
ZimelidineATP-dependent translocase ABCB1transporter
ZimelidineAmine oxidase [flavin-containing] Btarget
ZimelidineAmine oxidase [flavin-containing] Atarget
ZimelidineCytochrome P450 3A4enzyme
Zolmitriptan5-hydroxytryptamine receptor 1Btarget
Zolmitriptan5-hydroxytryptamine receptor 1Ftarget
ZolmitriptanCytochrome P450 1A2enzyme
ZolmitriptanAmine oxidase [flavin-containing] Aenzyme
Zolmitriptan5-hydroxytryptamine receptor 1Dtarget
ZolmitriptanATP-dependent translocase ABCB1transporter
Zolmitriptan5-hydroxytryptamine receptor 7target
Zolmitriptan5-hydroxytryptamine receptor 2Atarget
Zolmitriptan5-hydroxytryptamine receptor 2Btarget
Zolmitriptan5-hydroxytryptamine receptor 1Etarget
Zolmitriptan5-hydroxytryptamine receptor 1Atarget