Tebipenem pivoxil is an oral carbapenem antibacterial indicated for complicated urinary tract infections, including pyelonephritis, caused by susceptible Enterobacterales and Enterococcus faecalis in adults with limited or no alternative oral treatment options. Tebipenem pivoxil is an orally administered prodrug of tebipenem, a carbapenem antibacterial that kills bacteria by binding essential penicillin-binding proteins and disrupting cell wall biosynthesis.
- Mechanism
- Curator reviewed
Pharmacologically active on Penicillin-binding protein
- Primary indication
- Tebipenem pivoxil is indicated for the treatment of complicated urinary tract infections (cUTI), including pyelonephritis, caused by Escherichia coli, Klebsiella pneumoniae, Enterobacter cloacae species complex, Klebsiella oxytoca, and Enterococcus faecalis, in adult patients who have...Curator reviewed · 2 structured indications
- Formula / weight
- C22H31N3O6S2 · 497.63 g/mol (avg)
- Code names
- L-084 · LJC-11084 · ME-1211
Resolves to
SNUDIPVBUUXCDG-QHSBEEBCSA-NSMILES[H][C@]12[C@@H](C)C(SC3CN(C3)C3=NCCS3)=C(N1C(=O)[C@]2([H])[C@@H](C)O)C(=O)OCOC(=O)C(C)(C)CWhat you can answer from here — as of September 12, 2026
Which other approved drugs treat the same conditions as Tebipenem pivoxil, and which companies have late-stage candidates in those indications?
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