| DB01268 | Sunitinib | approved, investigational | yes | inhibitor | Details |
| DB04879 | Vatalanib | investigational | unknown | | Details |
| DB05075 | TG-100801 | investigational | unknown | | Details |
| DB06080 | Linifanib | investigational | unknown | | Details |
| DB05913 | OSI-930 | investigational | unknown | | Details |
| DB06101 | IMC-1C11 | investigational | unknown | | Details |
| DB05932 | Denibulin | investigational | unknown | | Details |
| DB06589 | Pazopanib | approved | yes | inhibitor | Details |
| DB06626 | Axitinib | approved, investigational | yes | inhibitor | Details |
| DB07288 | N-(4-chlorophenyl)-2-[(pyridin-4-ylmethyl)amino]benzamide | experimental | unknown | | Details |
| DB08896 | Regorafenib | approved | yes | inhibitor | Details |
| DB00398 | Sorafenib | approved, investigational | yes | inhibitor | Details |
| DB09078 | Lenvatinib | approved, investigational | yes | inhibitor | Details |
| DB09079 | Nintedanib | approved | yes | inhibitor | Details |
| DB09221 | Polaprezinc | experimental | unknown | agonist | Details |
| DB10770 | Foreskin fibroblast (neonatal) | approved | yes | agonist | Details |
| DB12010 | Fostamatinib | approved, investigational | unknown | inhibitor | Details |
| DB15685 | Selpercatinib | approved, investigational | unknown | inhibitor | Details |
| DB11800 | Tivozanib | approved, investigational | yes | inhibitor | Details |