| DB00426 | Famciclovir | approved, investigational | unknown | substrate | Details |
| DB00484 | Brimonidine | approved | unknown | substrate | Details |
| DB00563 | Methotrexate | approved | unknown | substrate | Details |
| DB00157 | NADH | approved, nutraceutical | unknown | substrate | Details |
| DB00170 | Menadione | approved, nutraceutical | unknown | inhibitor | Details |
| DB00481 | Raloxifene | approved, investigational | unknown | inhibitor | Details |
| DB00909 | Zonisamide | approved, investigational | unknown | substrate | Details |
| DB00962 | Zaleplon | approved, illicit, investigational | unknown | substrate | Details |
| DB00437 | Allopurinol | approved | unknown | substrate | Details |
| DB00339 | Pyrazinamide | approved, investigational | unknown | substrate | Details |
| DB03516 | Eniluracil | investigational | unknown | | Details |
| DB04827 | Urethane | approved, withdrawn | unknown | substrate | Details |
| DB00513 | Aminocaproic acid | approved, investigational | unknown | substrate | Details |
| DB01033 | Mercaptopurine | approved | unknown | substrate | Details |
| DB08840 | N-methylnicotinamide | experimental | unknown | substrate | Details |
| DB09078 | Lenvatinib | approved, investigational | no | substrate | Details |
| DB09054 | Idelalisib | approved | no | substrate | Details |
| DB00246 | Ziprasidone | approved | yes | substrate | Details |
| DB00924 | Cyclobenzaprine | approved | unknown | inhibitor | Details |
| DB12466 | Favipiravir | approved, investigational | yes | substrateinhibitor | Details |
| DB11791 | Capmatinib | approved, investigational | unknown | substrate | Details |