| Acemetacin | Human Cyclooxygenases | target |
| Acemetacin | ATP-binding cassette sub-family C member 1 | transporter |
| Acemetacin | UDP-glucuronosyltransferase 2B7 | enzyme |
| Acemetacin | Prostaglandin G/H synthase 2 | target |
| Acemetacin | Prostaglandin G/H synthase 1 | target |
| Acoramidis | Broad substrate specificity ATP-binding cassette transporter ABCG2 | transporter |
| Acoramidis | Organic anion transporter 3 | transporter |
| Acoramidis | Solute carrier family 22 member 6 | transporter |
| Acoramidis | UDP-glucuronosyltransferase 2B7 | enzyme |
| Acoramidis | UDP-glucuronosyltransferase 1A1 | enzyme |
| Acoramidis | UDP-glucuronosyltransferase 1A9 | enzyme |
| Acoramidis | Cytochrome P450 2C9 | enzyme |
| Acoramidis | Transthyretin | target |
| Ambrisentan | Solute carrier organic anion transporter family member 1B3 | transporter |
| Ambrisentan | Cytochrome P450 3A5 | enzyme |
| Ambrisentan | Solute carrier organic anion transporter family member 1B1 | transporter |
| Ambrisentan | ATP-dependent translocase ABCB1 | transporter |
| Ambrisentan | UDP-glucuronosyltransferase 2B7 | enzyme |
| Ambrisentan | UDP-glucuronosyltransferase 1A3 | enzyme |
| Ambrisentan | UDP-glucuronosyltransferase 1A9 | enzyme |
| Ambrisentan | Cytochrome P450 3A4 | enzyme |
| Ambrisentan | Cytochrome P450 2C19 | enzyme |
| Ambrisentan | Endothelin-1 receptor | target |
| Ambrisentan | Endothelin receptor type B | target |
| Anastrozole | Cytochrome P450 2C9 | enzyme |
| Anastrozole | Cytochrome P450 1A2 | enzyme |
| Anastrozole | UDP-glucuronosyltransferase 2B7 | enzyme |
| Anastrozole | UDP-glucuronosyltransferase 1A3 | enzyme |
| Anastrozole | UDP-glucuronosyltransferase 1A4 | enzyme |
| Anastrozole | Cytochrome P450 2C8 | enzyme |
| Anastrozole | Cytochrome P450 3A5 | enzyme |
| Anastrozole | Cytochrome P450 3A4 | enzyme |
| Anastrozole | ATP-dependent translocase ABCB1 | transporter |
| Anastrozole | Aromatase | target |
| Aprocitentan | Endothelin-1 receptor | target |
| Aprocitentan | Endothelin receptor type B | target |
| Aprocitentan | UDP-glucuronosyltransferase 1A1 | enzyme |
| Aprocitentan | UDP-glucuronosyltransferase 2B7 | enzyme |
| Aprocitentan | Albumin | carrier |
| Aprocitentan | Cytochrome P450 3A4 | enzyme |
| Aprocitentan | Cytochrome P450 2C8 | enzyme |
| Aprocitentan | Cytochrome P450 2C9 | enzyme |
| Aprocitentan | Cytochrome P450 2C18 | enzyme |
| Aprocitentan | Cytochrome P450 2C19 | enzyme |
| Aprocitentan | ATP-dependent translocase ABCB1 | transporter |
| Aprocitentan | Broad substrate specificity ATP-binding cassette transporter ABCG2 | transporter |
| Aprocitentan | Bile salt export pump | transporter |
| Aprocitentan | Hepatic sodium/bile acid cotransporter | transporter |
| Artenimol | Plasmepsin IV | target |
| Artenimol | Heat shock protein beta-1 | target |
| Artenimol | Acyl-CoA synthetase | target |
| Artenimol | 60S ribosomal protein L2 | target |
| Artenimol | V-type proton ATPase catalytic subunit A | target |
| Artenimol | Calcium-transporting ATPase | target |
| Artenimol | Glycophorin-binding protein 130 | target |
| Artenimol | 40S ribosomal protein S19 | target |
| Artenimol | Serine repeat antigen 5 | target |
| Artenimol | High molecular weight rhoptry protein 2 | target |
| Artenimol | 60S ribosomal protein L3 | target |
| Artenimol | Protein ARV | target |
| Artenimol | Small ribosomal subunit protein eS1 | target |
| Artenimol | Phosphoethanolamine N-methyltransferase | target |
| Artenimol | Large ribosomal subunit protein uL4 | target |
| Artenimol | Enolase | target |
| Artenimol | Hypoxanthine-guanine-xanthine phosphoribosyltransferase | target |
| Artenimol | Endoplasmin, putative | target |
| Artenimol | Glutamate dehydrogenase | target |
| Artenimol | Probable ATP-dependent 6-phosphofructokinase | target |
| Artenimol | Spermidine synthase | target |
| Artenimol | Thioredoxin-related protein, putative | target |
| Artenimol | Protein disulfide-isomerase | target |
| Artenimol | L-lactate dehydrogenase | target |
| Artenimol | Pyruvate kinase | target |
| Artenimol | RNA helicase | target |
| Artenimol | Heat shock protein 90 | target |
| Artenimol | Cell division cycle protein 48 homologue, putative | target |
| Artenimol | Fructose-bisphosphate aldolase | target |
| Artenimol | Glyceraldehyde-3-phosphate dehydrogenase | target |
| Artenimol | Actin-1 | target |
| Artenimol | Elongation factor 2 | target |
| Artenimol | Multidrug resistance protein 1 | target |
| Artenimol | Elongation factor 1-alpha | target |
| Artenimol | Ornithine aminotransferase | target |
| Artenimol | P-type Ca(2+) transporter | target |
| Artenimol | Translationally-controlled tumor protein homolog | target |
| Artenimol | Nucleophosmin | target |
| Artenimol | Spliceosome RNA helicase DDX39B | target |
| Artenimol | Serine hydroxymethyltransferase, mitochondrial | target |
| Artenimol | Probable ATP-dependent RNA helicase DDX5 | target |
| Artenimol | Protein disulfide-isomerase | target |
| Artenimol | Myosin-9 | target |
| Artenimol | Phosphoglycerate mutase 1 | target |
| Artenimol | Cytochrome c | target |
| Artenimol | Glyceraldehyde-3-phosphate dehydrogenase | target |
| Artenimol | Fructose-bisphosphate aldolase A | target |
| Artenimol | Tubulin beta chain | target |
| Artenimol | Tubulin beta-4A chain | target |
| Artenimol | Tubulin beta-6 chain | target |
| Artenimol | Heat shock cognate 71 kDa protein | target |
| Artenimol | Zyxin | target |
| Artenimol | Vimentin | target |
| Artenimol | Tubulin alpha-1A chain | target |
| Artenimol | Tropomyosin alpha-1 chain | target |
| Artenimol | Triosephosphate isomerase | target |
| Artenimol | Transgelin-2 | target |
| Artenimol | Transgelin | target |
| Artenimol | Serine/arginine-rich splicing factor 4 | target |
| Artenimol | Signal recognition particle 14 kDa protein | target |
| Artenimol | H(+)-exporting diphosphatase | target |
| Artenimol | S-adenosylmethionine synthase | target |
| Artenimol | Knob-associated histidine-rich protein | target |
| Artenimol | Tubulin alpha chain | target |
| Artenimol | Heterogeneous nuclear ribonucleoprotein D0 | target |
| Artenimol | Small nuclear ribonucleoprotein Sm D2 | target |
| Artenimol | Splicing factor, proline- and glutamine-rich | target |
| Artenimol | Splicing factor 1 | target |
| Artenimol | Small ribosomal subunit protein uS4 | target |
| Artenimol | Small ribosomal subunit protein eS8 | target |
| Artenimol | Small ribosomal subunit protein eS6 | target |
| Artenimol | Small ribosomal subunit protein uS7 | target |
| Artenimol | Small ribosomal subunit protein eS28 | target |
| Artenimol | Actin, cytoplasmic 2 | target |
| Artenimol | Alpha-aminoadipic semialdehyde dehydrogenase | target |
| Artenimol | Annexin A2 | target |
| Artenimol | ATP synthase F(1) complex subunit alpha, mitochondrial | target |
| Artenimol | ATP synthase F(0) complex subunit g, mitochondrial | target |
| Artenimol | ATP synthase peripheral stalk subunit OSCP, mitochondrial | target |
| Artenimol | Calpastatin | target |
| Artenimol | T-complex protein 1 subunit gamma | target |
| Artenimol | Cofilin-1 | target |
| Artenimol | Chloride intracellular channel protein 1 | target |
| Artenimol | Cysteine and glycine-rich protein 1 | target |
| Artenimol | Dihydropyrimidinase-related protein 2 | target |
| Artenimol | Desmoplakin | target |
| Artenimol | Elongation factor 1-alpha 1 | target |
| Artenimol | Alpha-enolase | target |
| Artenimol | Filamin-A | target |
| Artenimol | Alpha-ketoglutarate-dependent dioxygenase FTO | target |
| Artenimol | Glucose-6-phosphate 1-dehydrogenase | target |
| Artenimol | Glyceraldehyde-3-phosphate dehydrogenase, testis-specific | target |
| Artenimol | Glucose-6-phosphate isomerase | target |
| Artenimol | Heterogeneous nuclear ribonucleoproteins A2/B1 | target |
| Artenimol | P-type sodium-transporting ATPase4 | target |
| Artenimol | Heterogeneous nuclear ribonucleoprotein K | target |
| Artenimol | Heterochromatin protein 1-binding protein 3 | target |
| Artenimol | 40S ribosomal protein S3 | target |
| Artenimol | Ras GTPase-activating-like protein IQGAP1 | target |
| Artenimol | Far upstream element-binding protein 2 | target |
| Artenimol | L-lactate dehydrogenase A chain | target |
| Artenimol | L-lactate dehydrogenase B chain | target |
| Artenimol | Galectin-1 | target |
| Artenimol | Microtubule-associated protein 4 | target |
| Artenimol | Malate dehydrogenase, cytoplasmic | target |
| Artenimol | Puromycin-sensitive aminopeptidase | target |
| Artenimol | Profilin-1 | target |
| Artenimol | Phosphoglycerate kinase 1 | target |
| Artenimol | Pyruvate kinase PKM | target |
| Artenimol | Peptidyl-prolyl cis-trans isomerase A | target |
| Artenimol | Peroxiredoxin-1 | target |
| Artenimol | Large ribosomal subunit protein uL16 | target |
| Artenimol | Large ribosomal subunit protein eL14 | target |
| Artenimol | Large ribosomal subunit protein eL18 | target |
| Artenimol | Large ribosomal subunit protein uL23 | target |
| Artenimol | Large ribosomal subunit protein uL29 | target |
| Artenimol | Large ribosomal subunit protein uL4 | target |
| Artenimol | Small ribosomal subunit protein uS15 | target |
| Artenimol | Small ribosomal subunit protein eS17 | target |
| Artenimol | Small ribosomal subunit protein uS13 | target |
| Artenimol | Small ribosomal subunit protein eS19 | target |
| Artenimol | Plasmepsin I | target |
| Artenimol | Chloroquine resistance transporter | target |
| Artenimol | 14-3-3 protein I | target |
| Artenimol | Isoleucine--tRNA ligase, putative | target |
| Artenimol | Plasmodium RESA N-terminal domain-containing protein | target |
| Artenimol | Tubulin beta chain | target |
| Artenimol | 60S ribosomal protein L27 | target |
| Artenimol | Translocation protein SEC62 | target |
| Artenimol | Autophagy-related protein 18 | target |
| Artenimol | Mature parasite-infected erythrocyte surface antigen | target |
| Artenimol | Importin-7, putative | target |
| Artenimol | Importin subunit alpha | target |
| Artenimol | Peptidyl-prolyl cis-trans isomerase | target |
| Artenimol | DnaJ protein, putative | target |
| Artenimol | Merozoite surface protein 1 | target |
| Artenimol | Glutamate--tRNA ligase | target |
| Artenimol | T-complex protein 1 subunit eta | target |
| Artenimol | Plasmepsin II | target |
| Artenimol | Chaperone, putative | target |
| Artenimol | Rhoptry neck protein 3 | target |
| Artenimol | 40S ribosomal protein S5, putative | target |
| Artenimol | Skeleton-binding protein 1 | target |
| Artenimol | Purine nucleoside phosphorylase | target |
| Artenimol | Adenosylhomocysteinase | target |
| Artenimol | Adenosine deaminase | target |
| Artenimol | Methionine--tRNA ligase | target |
| Artenimol | carbamoyl-phosphate synthase (ammonia) | target |
| Artenimol | Signal recognition particle receptor subunit beta | target |
| Artenimol | TVN-junction protein 1 | target |
| Artenimol | Coatomer alpha subunit, putative | target |
| Artenimol | Hexokinase | target |
| Artenimol | Proteasome subunit alpha type | target |
| Artenimol | Haloacid dehalogenase-like hydrolase | target |
| Artenimol | Insulinase, putative | target |
| Artenimol | 40S ribosomal protein S21 | target |
| Artenimol | Ubiquitin-conjugating enzyme E2 | target |
| Artenimol | Eukaryotic translation initiation factor 3 subunit C | target |
| Artenimol | 60S ribosomal protein L24, putative | target |
| Artenimol | 60S ribosomal protein L23 | target |
| Artenimol | Large ribosomal subunit protein uL22 | target |
| Artenimol | Plasmepsin III | target |
| Artenimol | Endoplasmic reticulum chaperone GRP170 | target |
| Artenimol | 60S ribosomal protein L10, putative | target |
| Artenimol | Esterase, putative | target |
| Artenimol | Polyadenylate-binding protein | target |
| Artenimol | Ubiquitin-60S ribosomal protein L40 | target |
| Artenimol | ribose-phosphate diphosphokinase | target |
| Artenimol | 2-Cys peroxiredoxin | target |
| Artenimol | Protein transport protein SEC31 | target |
| Artenimol | Dipeptidyl aminopeptidase 1 | target |
| Artenimol | Ring-infected erythrocyte surface antigen | target |
| Artenimol | RNA helicase | target |
| Artenimol | Calcium-dependent protein kinase 4 | target |
| Artenimol | GTP-binding nuclear protein Ran | target |
| Artenimol | Nucleoside transporter 2 | target |
| Artenimol | Anamorsin homolog | target |
| Artenimol | Glutamine synthetase, putative | target |
| Artenimol | 60S ribosomal protein L30e, putative | target |
| Artenimol | Serine/threonine-protein | target |
| Artenimol | Threonine--tRNA ligase | target |
| Artenimol | cAMP-dependent protein kinase regulatory subunit | target |
| Artenimol | Thioredoxin-like protein 1 | target |
| Artenimol | 60S ribosomal protein L21 | target |
| Artenimol | 60S ribosomal protein L14, putative | target |
| Artenimol | Inner membrane complex sub-compartment protein 3 | target |
| Artenimol | HSP40, subfamily A | target |
| Artenimol | Pyridoxal 5'-phosphate synthase subunit Pdx1 | target |
| Artenimol | UDP-glucuronosyltransferase 1A9 | enzyme |
| Artenimol | UDP-glucuronosyltransferase 2B7 | enzyme |
| Artenimol | Albumin | target |
| Artenimol | Cytochrome P450 2D6 | enzyme |
| Artenimol | Cytochrome P450 2C19 | enzyme |
| Artesunate | Albumin | carrier |
| Artesunate | Organic anion transporter 3 | transporter |
| Artesunate | Solute carrier organic anion transporter family member 1B1 | transporter |
| Artesunate | ATP-dependent translocase ABCB1 | transporter |
| Artesunate | Broad substrate specificity ATP-binding cassette transporter ABCG2 | transporter |
| Artesunate | UDP-glucuronosyltransferase 1A9 | enzyme |
| Artesunate | UDP-glucuronosyltransferase 2B7 | enzyme |
| Artesunate | Cytochrome P450 2A6 | enzyme |
| Artesunate | Malaria protein EXP-1 | target |
| Asciminib | Cytochrome P450 2C9 | enzyme |
| Asciminib | Solute carrier family 22 member 1 | transporter |
| Asciminib | Solute carrier organic anion transporter family member 1B3 | transporter |
| Asciminib | Solute carrier organic anion transporter family member 1B1 | transporter |
| Asciminib | ATP-dependent translocase ABCB1 | transporter |
| Asciminib | Cytochrome P450 2C19 | enzyme |
| Asciminib | UDP-glucuronosyltransferase 1A1 | enzyme |
| Asciminib | Broad substrate specificity ATP-binding cassette transporter ABCG2 | transporter |
| Asciminib | Tyrosine-protein kinase ABL1 | target |
| Asciminib | UDP-glucuronosyltransferase 2B17 | enzyme |
| Asciminib | UDP-glucuronosyltransferase 2B7 | enzyme |
| Asciminib | Cytochrome P450 3A4 | enzyme |
| Bempedoic acid | ATP-binding cassette sub-family C member 3 | transporter |
| Bempedoic acid | ATP-citrate synthase | target |
| Bempedoic acid | Long-chain fatty acid transport protein 2 | enzyme |
| Bempedoic acid | Solute carrier organic anion transporter family member 1B1 | transporter |
| Bempedoic acid | NUAK family SNF1-like kinase 2 | enzyme |
| Bempedoic acid | UDP-glucuronosyltransferase 2B7 | enzyme |
| Bempedoic acid | Solute carrier organic anion transporter family member 1B3 | transporter |
| Cannabidiol | Glycine receptor subunit alpha-3 | target |
| Cannabidiol | Glycine receptor (alpha-1/beta) | target |
| Cannabidiol | Glycine receptor subunit alpha-1 | target |
| Cannabidiol | G protein-coupled receptor 12 | target |
| Cannabidiol | Cannabinoid receptor 2 | target |
| Cannabidiol | Cannabinoid receptor 1 | target |
| Cannabidiol | Cytochrome P450 3A4 | enzyme |
| Cannabidiol | Cytochrome P450 2D6 | enzyme |
| Cannabidiol | Cytochrome P450 2C19 | enzyme |
| Cannabidiol | Cytochrome P450 2C9 | enzyme |
| Cannabidiol | N-arachidonyl glycine receptor | target |
| Cannabidiol | G protein-coupled receptor 55 | target |
| Cannabidiol | 5-hydroxytryptamine receptor 1A | target |
| Cannabidiol | 5-hydroxytryptamine receptor 2A | target |
| Cannabidiol | Neuronal acetylcholine receptor subunit alpha-7 | target |
| Cannabidiol | Delta-type opioid receptor | target |
| Cannabidiol | Mu-type opioid receptor | target |
| Cannabidiol | Peroxisome proliferator-activated receptor gamma | target |
| Cannabidiol | Cytochrome P450 3A5 | enzyme |
| Cannabidiol | Serotonin N-acetyltransferase | enzyme |
| Cannabidiol | Cytochrome P450 1A1 | enzyme |
| Cannabidiol | Fatty-acid amide hydrolase 1 | enzyme |
| Cannabidiol | Polyunsaturated fatty acid 5-lipoxygenase | enzyme |
| Cannabidiol | Polyunsaturated fatty acid lipoxygenase ALOX15 | enzyme |
| Cannabidiol | Zeta-crystallin | enzyme |
| Cannabidiol | ATP-binding cassette sub-family C member 1 | transporter |
| Cannabidiol | Broad substrate specificity ATP-binding cassette transporter ABCG2 | transporter |
| Cannabidiol | Equilibrative nucleoside transporter 1 | transporter |
| Cannabidiol | Transient receptor potential cation channel subfamily V member 1 | target |
| Cannabidiol | Voltage-dependent T-type calcium channel subunit alpha-1G | target |
| Cannabidiol | Voltage-dependent T-type calcium channel subunit alpha-1H | target |
| Cannabidiol | Voltage-dependent T-type calcium channel subunit alpha-1I | target |
| Cannabidiol | Transient receptor potential cation channel subfamily A member 1 | target |
| Cannabidiol | Transient receptor potential cation channel subfamily M member 8 | target |
| Cannabidiol | Transient receptor potential cation channel subfamily V member 2 | target |
| Cannabidiol | Transient receptor potential cation channel subfamily V member 3 | target |
| Cannabidiol | Transient receptor potential cation channel subfamily V member 4 | target |
| Cannabidiol | Non-selective voltage-gated ion channel VDAC1 | target |
| Cannabidiol | 5-hydroxytryptamine receptor 3A | target |
| Cannabidiol | Adenosine receptor A1 | target |
| Cannabidiol | Prostaglandin G/H synthase 1 | target |
| Cannabidiol | Prostaglandin G/H synthase 2 | target |
| Cannabidiol | Acetyl-CoA acetyltransferase, mitochondrial | target |
| Cannabidiol | Steroid 17-alpha-hydroxylase/17,20 lyase | target |
| Cannabidiol | 3-hydroxy-3-methylglutaryl-coenzyme A reductase | target |
| Cannabidiol | Glutathione reductase, mitochondrial | target |
| Cannabidiol | Glutathione peroxidase 1 | target |
| Cannabidiol | Indoleamine 2,3-dioxygenase 1 | target |
| Cannabidiol | NAD(P)H dehydrogenase [quinone] 1 | target |
| Cannabidiol | Catalase | target |
| Cannabidiol | Superoxide dismutase [Cu-Zn] | target |
| Cannabidiol | Serotonin N-acetyltransferase | target |
| Cannabidiol | N-acylethanolamine-hydrolyzing acid amidase | target |
| Cannabidiol | Cytochrome P450 1A2 | enzyme |
| Cannabidiol | Cytochrome P450 1B1 | enzyme |
| Cannabidiol | Cytochrome P450 2A6 | enzyme |
| Cannabidiol | Cytochrome P450 2B6 | enzyme |
| Cannabidiol | Cytochrome P450 2C8 | enzyme |
| Cannabidiol | Cytochrome P450 2E1 | enzyme |
| Cannabidiol | Cytochrome P450 3A7 | enzyme |
| Cannabidiol | UDP-glucuronosyltransferase 1A7 | enzyme |
| Cannabidiol | UDP-glucuronosyltransferase 1A9 | enzyme |
| Cannabidiol | UDP-glucuronosyltransferase 2B7 | enzyme |
| Cannabidiol | UDP-glucuronosyltransferase 2B17 | enzyme |
| Cannabidiol | ATP-dependent translocase ABCB1 | transporter |
| Cannabidiol | Cytochrome P450 2J2 | enzyme |
| Cannabidiol | Liver carboxylesterase 1 | enzyme |
| Cannabinol | Cytochrome P450 3A4 | enzyme |
| Cannabinol | Cytochrome P450 2C19 | enzyme |
| Cannabinol | Cytochrome P450 1A1 | enzyme |
| Cannabinol | Cytochrome P450 1A2 | enzyme |
| Cannabinol | Cytochrome P450 1B1 | enzyme |
| Cannabinol | Cytochrome P450 2A6 | enzyme |
| Cannabinol | Cytochrome P450 2B6 | enzyme |
| Cannabinol | Cytochrome P450 2C9 | enzyme |
| Cannabinol | Cytochrome P450 2D6 | enzyme |
| Cannabinol | Cytochrome P450 3A5 | enzyme |
| Cannabinol | Cytochrome P450 3A7 | enzyme |
| Cannabinol | UDP-glucuronosyltransferase 1A7 | enzyme |
| Cannabinol | UDP-glucuronosyltransferase 1A8 | enzyme |
| Cannabinol | UDP-glucuronosyltransferase 1A9 | enzyme |
| Cannabinol | UDP-glucuronosyltransferase 1A10 | enzyme |
| Cannabinol | UDP-glucuronosyltransferase 2B7 | enzyme |
| Cannabinol | ATP-dependent translocase ABCB1 | transporter |
| Cannabinol | Broad substrate specificity ATP-binding cassette transporter ABCG2 | transporter |
| Cannabinol | ATP-binding cassette sub-family C member 1 | transporter |
| Cannabinol | Cytochrome P450 2E1 | enzyme |
| Cannabinol | Cytochrome P450 2J2 | enzyme |
| Cannabinol | Liver carboxylesterase 1 | enzyme |
| Cannabinol | Cannabinoid receptor 1 | target |
| Capivasertib | UDP-glucuronosyltransferase 2B7 | enzyme |
| Capivasertib | RAC-alpha serine/threonine-protein kinase | target |
| Capivasertib | RAC-beta serine/threonine-protein kinase | target |
| Capivasertib | RAC-gamma serine/threonine-protein kinase | target |
| Capivasertib | Broad substrate specificity ATP-binding cassette transporter ABCG2 | transporter |
| Capivasertib | Solute carrier organic anion transporter family member 1B1 | transporter |
| Capivasertib | Solute carrier organic anion transporter family member 1B3 | transporter |
| Capivasertib | Organic anion transporter 3 | transporter |
| Capivasertib | Multidrug and toxin extrusion protein 1 | transporter |
| Capivasertib | Cytochrome P450 3A4 | enzyme |
| Capivasertib | Solute carrier family 22 member 2 | transporter |
| Capivasertib | Multidrug and toxin extrusion protein 2 | transporter |
| Carbamazepine | UDP-glucuronosyltransferase 1A1 | enzyme |
| Carbamazepine | ATP-dependent translocase ABCB1 | transporter |
| Carbamazepine | Cytochrome P450 2C9 | enzyme |
| Carbamazepine | Cytochrome P450 2C19 | enzyme |
| Carbamazepine | Cytochrome P450 1A2 | enzyme |
| Carbamazepine | Cytochrome P450 3A4 | enzyme |
| Carbamazepine | Cytochrome P450 2B6 | enzyme |
| Carbamazepine | Cytochrome P450 2C8 | enzyme |
| Carbamazepine | Voltage-gated sodium channel alpha subunit | target |
| Carbamazepine | UDP-glucuronosyltransferase 2B7 | enzyme |
| Carbamazepine | RalA-binding protein 1 | transporter |
| Carbamazepine | ATP-binding cassette sub-family C member 2 | transporter |
| Carbamazepine | Neuronal acetylcholine receptor subunit alpha-4 | target |
| Carbamazepine | Nuclear receptor subfamily 1 group I member 2 | target |
| Carbamazepine | UDP-glucuronosyltransferase 1A6 | enzyme |
| Carbamazepine | UDP-glucuronosyltransferase 1A7 | enzyme |
| Carbamazepine | Cytochrome P450 3A5 | enzyme |
| Carvedilol | Alpha-2B adrenergic receptor | target |
| Carvedilol | Beta-1 adrenergic receptor | target |
| Carvedilol | NADH dehydrogenase [ubiquinone] 1 subunit C2 | target |
| Carvedilol | Beta-2 adrenergic receptor | target |
| Carvedilol | Vascular endothelial growth factor A, long form | target |
| Carvedilol | Natriuretic peptides B | target |
| Carvedilol | Gap junction alpha-1 protein | target |
| Carvedilol | Voltage-gated inwardly rectifying potassium channel KCNH2 | target |
| Carvedilol | Vascular cell adhesion protein 1 | target |
| Carvedilol | Alpha-1 adrenergic receptors | target |
| Carvedilol | Beta adrenergic receptor | target |
| Carvedilol | Inward rectifier potassium channel 2 | target |
| Carvedilol | UDP-glucuronosyltransferase 2B7 | enzyme |
| Carvedilol | UDP-glucuronosyltransferase 2B4 | enzyme |
| Carvedilol | Albumin | carrier |
| Carvedilol | UDP-glucuronosyltransferase 1A1 | enzyme |
| Carvedilol | Inward rectifier potassium channel 4 | target |
| Carvedilol | Hypoxia-inducible factor 1-alpha | target |
| Carvedilol | E-selectin | target |
| Carvedilol | Alpha-2A adrenergic receptor | target |
| Carvedilol | Alpha-1A adrenergic receptor | target |
| Carvedilol | Alpha-2C adrenergic receptor | target |
| Carvedilol | Alpha-1B adrenergic receptor | target |
| Carvedilol | Alpha-1D adrenergic receptor | target |
| Carvedilol | Cytochrome P450 2E1 | enzyme |
| Carvedilol | Cytochrome P450 1A1 | enzyme |
| Carvedilol | Cytochrome P450 3A4 | enzyme |
| Carvedilol | Cytochrome P450 1A2 | enzyme |
| Carvedilol | ATP-dependent translocase ABCB1 | transporter |
| Carvedilol | Xanthine dehydrogenase/oxidase | enzyme |
| Carvedilol | Cytochrome P450 2D6 | enzyme |
| Carvedilol | Cytochrome P450 2C9 | enzyme |
| Cenobamate | Cytochrome P450 2A6 | enzyme |
| Cenobamate | Gamma-aminobutyric acid receptor subunit alpha-1 | target |
| Cenobamate | Voltage-gated sodium channel alpha subunit | target |
| Cenobamate | Cytochrome P450 2C8 | enzyme |
| Cenobamate | Albumin | carrier |
| Cenobamate | Cytochrome P450 3A5 | enzyme |
| Cenobamate | Cytochrome P450 3A4 | enzyme |
| Cenobamate | Cytochrome P450 2C19 | enzyme |
| Cenobamate | Cytochrome P450 2B6 | enzyme |
| Cenobamate | UDP-glucuronosyltransferase 2B7 | enzyme |
| Cenobamate | UDP-glucuronosyltransferase 2B4 | enzyme |
| Cenobamate | Cytochrome P450 2E1 | enzyme |
| Cobimetinib | Dual specificity mitogen-activated protein kinase kinase 1 | target |
| Cobimetinib | Cytochrome P450 3A4 | enzyme |
| Cobimetinib | Solute carrier organic anion transporter family member 1B1 | transporter |
| Cobimetinib | Solute carrier organic anion transporter family member 1B3 | transporter |
| Cobimetinib | Broad substrate specificity ATP-binding cassette transporter ABCG2 | transporter |
| Cobimetinib | ATP-dependent translocase ABCB1 | transporter |
| Cobimetinib | UDP-glucuronosyltransferase 2B7 | enzyme |
| Cobimetinib | Cytochrome P450 2D6 | enzyme |
| Cobimetinib | Dual specificity mitogen-activated protein kinase kinase 2 | target |
| Cobimetinib | Alpha-1-acid glycoprotein 1 | carrier |
| Cobimetinib | Cytochrome P450 3A5 | enzyme |
| Codeine | UDP-glucuronosyltransferase 2B4 | enzyme |
| Codeine | UDP-glucuronosyltransferase 2B7 | enzyme |
| Codeine | Cytochrome P450 3A4 | enzyme |
| Codeine | Cytochrome P450 2D6 | enzyme |
| Codeine | Kappa-type opioid receptor | target |
| Codeine | Delta-type opioid receptor | target |
| Codeine | Mu-type opioid receptor | target |
| Codeine | Solute carrier family 22 member 1 | transporter |
| Dabigatran etexilate | Prothrombin | target |
| Dabigatran etexilate | ATP-dependent translocase ABCB1 | transporter |
| Dabigatran etexilate | Liver carboxylesterase 1 | enzyme |
| Dabigatran etexilate | Cocaine esterase | enzyme |
| Dabigatran etexilate | UDP-glucuronosyltransferase 1A9 | enzyme |
| Dabigatran etexilate | UDP-glucuronosyltransferase 2B7 | enzyme |
| Dabigatran etexilate | UDP-glucuronosyltransferase 2B15 | enzyme |
| Dabigatran etexilate | Ribosyldihydronicotinamide dehydrogenase [quinone] | enzyme |
| Dabigatran etexilate | Albumin | carrier |
| Dapagliflozin | Sodium/glucose cotransporter 2 | target |
| Dapagliflozin | Cytochrome P450 1A1 | enzyme |
| Dapagliflozin | Cytochrome P450 1A2 | enzyme |
| Dapagliflozin | Cytochrome P450 2A6 | enzyme |
| Dapagliflozin | Cytochrome P450 2C9 | enzyme |
| Dapagliflozin | Cytochrome P450 2D6 | enzyme |
| Dapagliflozin | Cytochrome P450 3A4 | enzyme |
| Dapagliflozin | UDP-glucuronosyltransferase 1A9 | enzyme |
| Dapagliflozin | UDP-glucuronosyltransferase 2B4 | enzyme |
| Dapagliflozin | UDP-glucuronosyltransferase 2B7 | enzyme |
| Dapagliflozin | ATP-dependent translocase ABCB1 | transporter |
| Desomorphine | UDP-glucuronosyltransferase 2B7 | enzyme |
| Desomorphine | UDP-glucuronosyltransferase 2B4 | enzyme |
| Desomorphine | UDP-glucuronosyltransferase 1A10 | enzyme |
| Desomorphine | UDP-glucuronosyltransferase 1A9 | enzyme |
| Desomorphine | UDP-glucuronosyltransferase 1A8 | enzyme |
| Desomorphine | UDP-glucuronosyltransferase 1A3 | enzyme |
| Desomorphine | UDP-glucuronosyltransferase 1A1 | enzyme |
| Desomorphine | Cytochrome P450 3A4 | enzyme |
| Desomorphine | Cytochrome P450 2D6 | enzyme |
| Desomorphine | Cytochrome P450 2C19 | enzyme |
| Desomorphine | Cytochrome P450 2C18 | enzyme |
| Desomorphine | Cytochrome P450 2C9 | enzyme |
| Desomorphine | Cytochrome P450 2C8 | enzyme |
| Desomorphine | Cytochrome P450 2B6 | enzyme |
| Desomorphine | UDP-glucuronosyltransferase 2B15 | enzyme |
| Desomorphine | UDP-glucuronosyltransferase 2B17 | enzyme |
| Dexibuprofen | Solute carrier organic anion transporter family member 2B1 | transporter |
| Dexibuprofen | Solute carrier family 22 member 11 | transporter |
| Dexibuprofen | Organic anion transporter 3 | transporter |
| Dexibuprofen | Solute carrier family 22 member 6 | transporter |
| Dexibuprofen | Solute carrier organic anion transporter family member 1A2 | transporter |
| Dexibuprofen | ATP-binding cassette sub-family C member 1 | transporter |
| Dexibuprofen | ATP-binding cassette sub-family C member 4 | transporter |
| Dexibuprofen | Albumin | carrier |
| Dexibuprofen | Cytochrome P450 2C9 | enzyme |
| Dexibuprofen | Cystic fibrosis transmembrane conductance regulator | target |
| Dexibuprofen | Peroxisome proliferator-activated receptor gamma | target |
| Dexibuprofen | Fatty acid-binding protein, intestinal | target |
| Dexibuprofen | Tissue-type plasminogen activator | target |
| Dexibuprofen | Thrombomodulin | target |
| Dexibuprofen | Apoptosis regulator Bcl-2 | target |
| Dexibuprofen | Prostaglandin G/H synthase 2 | target |
| Dexibuprofen | Prostaglandin G/H synthase 1 | target |
| Dexibuprofen | Human Cyclooxygenases | target |
| Dexibuprofen | Alpha-methylacyl-CoA racemase | enzyme |
| Dexibuprofen | Protein S100-A7 | target |
| Dexibuprofen | Platelet glycoprotein Ib alpha chain | target |
| Dexibuprofen | Peroxisome proliferator-activated receptor alpha | target |
| Dexibuprofen | Solute carrier family 15 member 1 | target |
| Dexibuprofen | Cytochrome P450 2C19 | enzyme |
| Dexibuprofen | Cytochrome P450 2C8 | enzyme |
| Dexibuprofen | UDP-glucuronosyltransferase 2B7 | enzyme |
| Dexibuprofen | UDP-glucuronosyltransferase 2B4 | enzyme |
| Dexibuprofen | UDP-glucuronosyltransferase 1A9 | enzyme |
| Dexibuprofen | UDP-glucuronosyltransferase 1A3 | enzyme |
| Dexibuprofen | UDP-glucuronosyltransferase 1A1 | enzyme |
| Dexibuprofen | ATP-dependent translocase ABCB1 | transporter |
| Dextromethorphan | Neuronal acetylcholine receptor subunit alpha-3 | target |
| Dextromethorphan | Membrane-associated progesterone receptor component 1 | target |
| Dextromethorphan | Cytochrome P450 2C19 | enzyme |
| Dextromethorphan | Cytochrome P450 2B6 | enzyme |
| Dextromethorphan | Cytochrome P450 2C9 | enzyme |
| Dextromethorphan | Sigma non-opioid intracellular receptor 1 | target |
| Dextromethorphan | Neuronal acetylcholine receptor subunit alpha-2 | target |
| Dextromethorphan | Sodium-dependent serotonin transporter | target |
| Dextromethorphan | Glutamate receptor ionotropic, NMDA 3A | target |
| Dextromethorphan | Cytochrome P450 2D6 | enzyme |
| Dextromethorphan | Cytochrome P450 3A4 | enzyme |
| Dextromethorphan | Cytochrome P450 3A7 | enzyme |
| Dextromethorphan | Neuronal acetylcholine receptor subunit alpha-4 | target |
| Dextromethorphan | Neuronal acetylcholine receptor subunit beta-4 | target |
| Dextromethorphan | Neuronal acetylcholine receptor subunit beta-2 | target |
| Dextromethorphan | Neuronal acetylcholine receptor subunit alpha-7 | target |
| Dextromethorphan | Mu-type opioid receptor | target |
| Dextromethorphan | Delta-type opioid receptor | target |
| Dextromethorphan | Kappa-type opioid receptor | target |
| Dextromethorphan | NADPH oxidase | target |
| Dextromethorphan | Sodium-dependent noradrenaline transporter | target |
| Dextromethorphan | UDP-glucuronosyltransferase 2B4 | enzyme |
| Dextromethorphan | UDP-glucuronosyltransferase 2B7 | enzyme |
| Dextromethorphan | UDP-glucuronosyltransferase 2B15 | enzyme |
| Dextromethorphan | UDP-glucuronosyltransferase 2B17 | enzyme |
| Dextromethorphan | Aromatase | target |
| Dextromethorphan | Glutamate receptor ionotropic, NMDA 2A | target |
| Diclofenac | Albumin | carrier |
| Diclofenac | Solute carrier organic anion transporter family member 1C1 | transporter |
| Diclofenac | Human Cyclooxygenases | target |
| Diclofenac | ATP-dependent translocase ABCB1 | transporter |
| Diclofenac | Phospholipase A2, membrane associated | enzyme |
| Diclofenac | Potassium voltage-gated channel subfamily KQT member 3 | transporter |
| Diclofenac | Potassium voltage-gated channel subfamily KQT member 2 | transporter |
| Diclofenac | Acid-sensing ion channel 1 | transporter |
| Diclofenac | Sodium channel protein type 4 subunit alpha | transporter |
| Diclofenac | Polyunsaturated fatty acid 5-lipoxygenase | enzyme |
| Diclofenac | UDP-glucuronosyltransferase 2B4 | enzyme |
| Diclofenac | UDP-glucuronosyltransferase 1A9 | enzyme |
| Diclofenac | UDP-glucuronosyltransferase 1A3 | enzyme |
| Diclofenac | Bile salt export pump | transporter |
| Diclofenac | Solute carrier organic anion transporter family member 1B1 | transporter |
| Diclofenac | Prostaglandin G/H synthase 1 | target |
| Diclofenac | Prostaglandin G/H synthase 2 | target |
| Diclofenac | Transthyretin | carrier |
| Diclofenac | Cytochrome P450 2C9 | enzyme |
| Diclofenac | Cytochrome P450 2C19 | enzyme |
| Diclofenac | Cytochrome P450 1A2 | enzyme |
| Diclofenac | Cytochrome P450 2C8 | enzyme |
| Diclofenac | Cytochrome P450 2E1 | enzyme |
| Diclofenac | ATP-binding cassette sub-family C member 4 | transporter |
| Diclofenac | ATP-binding cassette sub-family C member 1 | transporter |
| Diclofenac | Solute carrier family 22 member 6 | transporter |
| Diclofenac | Organic anion transporter 3 | transporter |
| Diclofenac | Cytochrome P450 2C18 | enzyme |
| Diclofenac | Solute carrier family 22 member 11 | transporter |
| Diclofenac | UDP-glucuronosyltransferase 2B7 | enzyme |
| Diclofenac | Cytochrome P450 3A4 | enzyme |
| Diclofenac | Cytochrome P450 2B6 | enzyme |
| Edaravone | Apoptosis regulator Bcl-2 | target |
| Edaravone | Solute carrier family 22 member 6 | transporter |
| Edaravone | Organic anion transporter 3 | transporter |
| Edaravone | UDP-glucuronosyltransferase 1A1 | enzyme |
| Edaravone | UDP-glucuronosyltransferase 1A6 | enzyme |
| Edaravone | UDP-glucuronosyltransferase 1A7 | enzyme |
| Edaravone | UDP-glucuronosyltransferase 1A8 | enzyme |
| Edaravone | UDP-glucuronosyltransferase 1A9 | enzyme |
| Edaravone | UDP-glucuronosyltransferase 1A10 | enzyme |
| Edaravone | UDP-glucuronosyltransferase 2B7 | enzyme |
| Edaravone | UDP-glucuronosyltransferase 2B17 | enzyme |
| Edaravone | Sulfotransferase | enzyme |
| Edaravone | Albumin | carrier |
| Elafibranor | Bile salt export pump | transporter |
| Elafibranor | Peroxisome proliferator-activated receptor gamma | target |
| Elafibranor | Prostaglandin reductase 1 | enzyme |
| Elafibranor | Cytochrome P450 2J2 | enzyme |
| Elafibranor | UDP-glucuronosyltransferase 1A3 | enzyme |
| Elafibranor | UDP-glucuronosyltransferase 1A4 | enzyme |
| Elafibranor | UDP-glucuronosyltransferase 2B7 | enzyme |
| Elafibranor | Cytochrome P450 2C8 | enzyme |
| Elafibranor | UDP-glucuronosyltransferase 1A6 | enzyme |
| Elafibranor | Peroxisome proliferator-activated receptor delta | target |
| Elafibranor | Broad substrate specificity ATP-binding cassette transporter ABCG2 | transporter |
| Elafibranor | ATP-binding cassette sub-family C member 2 | transporter |
| Elafibranor | ATP-binding cassette sub-family C member 3 | transporter |
| Elafibranor | Albumin | carrier |
| Elafibranor | Cytochrome P450 3A4 | enzyme |
| Elafibranor | Peroxisome proliferator-activated receptor alpha | target |
| Empagliflozin | ATP-dependent translocase ABCB1 | transporter |
| Empagliflozin | UDP-glucuronosyltransferase 1A9 | enzyme |
| Empagliflozin | UDP-glucuronosyltransferase 1A8 | enzyme |
| Empagliflozin | UDP-glucuronosyltransferase 1A3 | enzyme |
| Empagliflozin | UDP-glucuronosyltransferase 2B7 | enzyme |
| Empagliflozin | Sodium/glucose cotransporter 2 | target |
| Empagliflozin | Broad substrate specificity ATP-binding cassette transporter ABCG2 | transporter |
| Empagliflozin | Organic anion transporter 3 | transporter |
| Empagliflozin | Solute carrier organic anion transporter family member 1B1 | transporter |
| Empagliflozin | Solute carrier organic anion transporter family member 1B3 | transporter |
| Enasidenib | Broad substrate specificity ATP-binding cassette transporter ABCG2 | transporter |
| Enasidenib | UDP-glucuronosyltransferase 1A3 | enzyme |
| Enasidenib | Cytochrome P450 1A2 | enzyme |
| Enasidenib | Cytochrome P450 2B6 | enzyme |
| Enasidenib | Isocitrate dehydrogenase [NADP], mitochondrial | target |
| Enasidenib | Isocitrate dehydrogenase [NAD] subunit gamma, mitochondrial | target |
| Enasidenib | Isocitrate dehydrogenase [NAD] subunit beta, mitochondrial | target |
| Enasidenib | Isocitrate dehydrogenase [NAD] subunit alpha, mitochondrial | target |
| Enasidenib | Isocitrate dehydrogenase [NADP] cytoplasmic | target |
| Enasidenib | Albumin | carrier |
| Enasidenib | Organic anion transporter 3 | transporter |
| Enasidenib | Solute carrier organic anion transporter family member 1B3 | transporter |
| Enasidenib | Solute carrier family 22 member 2 | transporter |
| Enasidenib | Solute carrier organic anion transporter family member 1B1 | transporter |
| Enasidenib | Solute carrier family 22 member 6 | transporter |
| Enasidenib | Cytochrome P450 2C8 | enzyme |
| Enasidenib | ATP-dependent translocase ABCB1 | transporter |
| Enasidenib | UDP-glucuronosyltransferase 2B15 | enzyme |
| Enasidenib | UDP-glucuronosyltransferase 2B7 | enzyme |
| Enasidenib | UDP-glucuronosyltransferase 1A9 | enzyme |
| Enasidenib | UDP-glucuronosyltransferase 1A4 | enzyme |
| Enasidenib | Cytochrome P450 2C9 | enzyme |
| Enasidenib | UDP-glucuronosyltransferase 1A1 | enzyme |
| Enasidenib | Cytochrome P450 3A4 | enzyme |
| Enasidenib | Cytochrome P450 2D6 | enzyme |
| Enasidenib | Cytochrome P450 2C19 | enzyme |
| Enavogliflozin | Cytochrome P450 3A4 | enzyme |
| Enavogliflozin | Cytochrome P450 2C19 | enzyme |
| Enavogliflozin | UDP-glucuronosyltransferase 1A4 | enzyme |
| Enavogliflozin | UDP-glucuronosyltransferase 1A9 | enzyme |
| Enavogliflozin | UDP-glucuronosyltransferase 2B7 | enzyme |
| Enavogliflozin | Sodium/glucose cotransporter 2 | target |
| Epirubicin | DNA topoisomerase 2-beta | target |
| Epirubicin | Cytosolic phospholipase A2 | enzyme |
| Epirubicin | UDP-glucuronosyltransferase 2B7 | enzyme |
| Epirubicin | ATP-binding cassette sub-family C member 1 | transporter |
| Epirubicin | DNA | target |
| Epirubicin | DNA topoisomerase 2-alpha | target |
| Ertugliflozin | UDP-glucuronosyltransferase 1A4 | enzyme |
| Ertugliflozin | UDP-glucuronosyltransferase 1A9 | enzyme |
| Ertugliflozin | UDP-glucuronosyltransferase 2B7 | enzyme |
| Ertugliflozin | Sodium/glucose cotransporter 2 | target |
| Ertugliflozin | ATP-dependent translocase ABCB1 | transporter |
| Ertugliflozin | Broad substrate specificity ATP-binding cassette transporter ABCG2 | transporter |
| Ertugliflozin | Albumin | carrier |
| Ertugliflozin | UDP-glucuronosyltransferase 1A1 | enzyme |
| Estetrol | Estrogen receptor beta | target |
| Estetrol | Estrogen receptor | target |
| Estetrol | Alpha-1-acid glycoprotein 1 | carrier |
| Estetrol | Estrogen receptor | target |
| Estetrol | UDP-glucuronosyltransferase 2B7 | enzyme |
| Estetrol | Cytochrome P450 3A4 | enzyme |
| Estetrol | Albumin | carrier |
| Ethinylestradiol | UDP-glucuronosyltransferase 1A9 | enzyme |
| Ethinylestradiol | Sex hormone-binding globulin | carrier |
| Ethinylestradiol | Albumin | carrier |
| Ethinylestradiol | Solute carrier organic anion transporter family member 1A2 | transporter |
| Ethinylestradiol | Catechol O-methyltransferase | enzyme |
| Ethinylestradiol | UDP-glucuronosyltransferase 1A3 | enzyme |
| Ethinylestradiol | UDP-glucuronosyltransferase 2B7 | enzyme |
| Ethinylestradiol | Cytochrome P450 3A5 | enzyme |
| Ethinylestradiol | Sulfotransferase 1A3 | enzyme |
| Ethinylestradiol | Sulfotransferase 1E1 | enzyme |
| Ethinylestradiol | Cytochrome P450 1A2 | enzyme |
| Ethinylestradiol | Estrogen receptor | target |
| Ethinylestradiol | Nuclear receptor subfamily 1 group I member 2 | target |
| Ethinylestradiol | Cytochrome P450 3A4 | enzyme |
| Ethinylestradiol | Cytochrome P450 2C8 | enzyme |
| Ethinylestradiol | Bile salt export pump | transporter |
| Ethinylestradiol | Hepatic sodium/bile acid cotransporter | transporter |
| Ethinylestradiol | ATP-binding cassette sub-family C member 2 | transporter |
| Ethinylestradiol | ATP-dependent translocase ABCB1 | transporter |
| Ethinylestradiol | UDP-glucuronosyltransferase 1A1 | enzyme |
| Ethinylestradiol | Cytochrome P450 2C19 | enzyme |
| Ethinylestradiol | UDP-glucuronosyltransferase 1A4 | enzyme |
| Ethinylestradiol | Cytochrome P450 2C9 | enzyme |
| Etodolac | Solute carrier family 22 member 6 | transporter |
| Etodolac | UDP-glucuronosyltransferase 1A3 | enzyme |
| Etodolac | UDP-glucuronosyltransferase 1A10 | enzyme |
| Etodolac | UDP-glucuronosyltransferase 2B7 | enzyme |
| Etodolac | Prostaglandin G/H synthase 1 | target |
| Etodolac | Prostaglandin G/H synthase 2 | target |
| Etodolac | Cytochrome P450 2C9 | enzyme |
| Etodolac | UDP-glucuronosyltransferase 1A9 | enzyme |
| Etodolac | Retinoic acid receptor RXR-alpha | target |
| Etodolac | Albumin | carrier |
| Ezetimibe | Broad substrate specificity ATP-binding cassette transporter ABCG2 | transporter |
| Ezetimibe | Cytochrome P450 2C8 | enzyme |
| Ezetimibe | Bile salt export pump | transporter |
| Ezetimibe | ATP-binding cassette sub-family C member 3 | transporter |
| Ezetimibe | Cytochrome P450 3A4 | enzyme |
| Ezetimibe | UDP-glucuronosyltransferase 2B7 | enzyme |
| Ezetimibe | UDP-glucuronosyltransferase 2B15 | enzyme |
| Ezetimibe | Solute carrier organic anion transporter family member 1B1 | transporter |
| Ezetimibe | ATP-binding cassette sub-family C member 2 | transporter |
| Ezetimibe | ATP-dependent translocase ABCB1 | transporter |
| Ezetimibe | UDP-glucuronosyltransferase 1A3 | enzyme |
| Ezetimibe | UDP-glucuronosyltransferase 1A1 | enzyme |
| Ezetimibe | Sterol O-acyltransferase 1 | target |
| Ezetimibe | Aminopeptidase N | target |
| Ezetimibe | NPC1-like intracellular cholesterol transporter 1 | target |
| Febuxostat | Cytochrome P450 2C9 | enzyme |
| Febuxostat | UDP-glucuronosyltransferase 1A1 | enzyme |
| Febuxostat | Broad substrate specificity ATP-binding cassette transporter ABCG2 | transporter |
| Febuxostat | Albumin | carrier |
| Febuxostat | Xanthine dehydrogenase/oxidase | target |
| Febuxostat | UDP-glucuronosyltransferase 1A3 | enzyme |
| Febuxostat | UDP-glucuronosyltransferase 1A9 | enzyme |
| Febuxostat | UDP-glucuronosyltransferase 2B7 | enzyme |
| Febuxostat | Cytochrome P450 2C8 | enzyme |
| Febuxostat | Cytochrome P450 1A2 | enzyme |
| Flurbiprofen | Human Cyclooxygenases | target |
| Flurbiprofen | Prostaglandin G/H synthase 2 | target |
| Flurbiprofen | Prostaglandin G/H synthase 1 | target |
| Flurbiprofen | Cytochrome P450 2C9 | enzyme |
| Flurbiprofen | Albumin | carrier |
| Flurbiprofen | ATP-binding cassette sub-family C member 4 | transporter |
| Flurbiprofen | Solute carrier family 22 member 6 | transporter |
| Flurbiprofen | UDP-glucuronosyltransferase 2B7 | enzyme |
| Flurbiprofen | UDP-glucuronosyltransferase 1A1 | enzyme |
| Flurbiprofen | UDP-glucuronosyltransferase 1A3 | enzyme |
| Flurbiprofen | UDP-glucuronosyltransferase 1A9 | enzyme |
| Flurbiprofen | UDP-glucuronosyltransferase 2B4 | enzyme |
| Fluvastatin | Cytochrome P450 2C9 | enzyme |
| Fluvastatin | 3-hydroxy-3-methylglutaryl-coenzyme A reductase | target |
| Fluvastatin | Cytochrome P450 3A4 | enzyme |
| Fluvastatin | Cytochrome P450 2C8 | enzyme |
| Fluvastatin | Cytochrome P450 2D6 | enzyme |
| Fluvastatin | Cytochrome P450 2C19 | enzyme |
| Fluvastatin | Cytochrome P450 1A1 | enzyme |
| Fluvastatin | Solute carrier organic anion transporter family member 1B1 | transporter |
| Fluvastatin | Solute carrier organic anion transporter family member 1B3 | transporter |
| Fluvastatin | Solute carrier organic anion transporter family member 2B1 | transporter |
| Fluvastatin | Solute carrier family 15 member 1 | transporter |
| Fluvastatin | Cytochrome P450 3A5 | enzyme |
| Fluvastatin | UDP-glucuronosyltransferase 1A1 | enzyme |
| Fluvastatin | UDP-glucuronosyltransferase 1A3 | enzyme |
| Fluvastatin | UDP-glucuronosyltransferase 2B7 | enzyme |
| Fluvastatin | ATP-binding cassette sub-family C member 2 | transporter |
| Fluvastatin | Cytochrome P450 2B6 | enzyme |
| Fluvastatin | Histone deacetylase 2 | target |
| Formoterol | Solute carrier family 22 member 3 | transporter |
| Formoterol | Cytochrome P450 2D6 | enzyme |
| Formoterol | Cytochrome P450 2C19 | enzyme |
| Formoterol | Organic cation/carnitine transporter 2 | transporter |
| Formoterol | Cytochrome P450 2C9 | enzyme |
| Formoterol | Beta-2 adrenergic receptor | target |
| Formoterol | Beta-1 adrenergic receptor | target |
| Formoterol | Beta-3 adrenergic receptor | target |
| Formoterol | Cytochrome P450 2A6 | enzyme |
| Formoterol | UDP-glucuronosyltransferase 1A1 | enzyme |
| Formoterol | Albumin | carrier |
| Formoterol | Solute carrier family 22 member 4 | transporter |
| Formoterol | Solute carrier family 22 member 1 | transporter |
| Formoterol | UDP-glucuronosyltransferase 2B15 | enzyme |
| Formoterol | UDP-glucuronosyltransferase 2B7 | enzyme |
| Formoterol | UDP-glucuronosyltransferase 1A9 | enzyme |
| Formoterol | UDP-glucuronosyltransferase 1A8 | enzyme |
| Gemfibrozil | Peroxisome proliferator-activated receptor alpha | target |
| Gemfibrozil | Cytochrome P450 2C9 | enzyme |
| Gemfibrozil | Cytochrome P450 2C8 | enzyme |
| Gemfibrozil | Cytochrome P450 1A2 | enzyme |
| Gemfibrozil | Cytochrome P450 2C19 | enzyme |
| Gemfibrozil | UDP-glucuronosyltransferase 1A9 | enzyme |
| Gemfibrozil | Cytochrome P450 3A4 | enzyme |
| Gemfibrozil | UDP-glucuronosyltransferase 1A3 | enzyme |
| Gemfibrozil | Solute carrier organic anion transporter family member 1B1 | target |
| Gemfibrozil | UDP-glucuronosyltransferase 2B7 | enzyme |
| Gemfibrozil | Solute carrier organic anion transporter family member 1B3 | target |
| Gemfibrozil | Lipoprotein lipase | target |
| Gemfibrozil | UDP-glucuronosyltransferase 1A1 | enzyme |
| Gemfibrozil | Solute carrier organic anion transporter family member 2B1 | target |
| Gemfibrozil | Organic anion transporter 3 | target |
| Gemfibrozil | Albumin | carrier |
| Gemfibrozil | UDP-glucuronosyltransferase 2B17 | enzyme |
| Gemfibrozil | UDP-glucuronosyltransferase 2B4 | enzyme |
| Hydromorphone | Mu-type opioid receptor | target |
| Hydromorphone | Albumin | carrier |
| Hydromorphone | Delta-type opioid receptor | target |
| Hydromorphone | Kappa-type opioid receptor | target |
| Hydromorphone | Cytochrome P450 2C9 | enzyme |
| Hydromorphone | UDP-glucuronosyltransferase 1A3 | enzyme |
| Hydromorphone | UDP-glucuronosyltransferase 2B7 | enzyme |
| Ibuprofen | Prostaglandin G/H synthase 2 | target |
| Ibuprofen | Human Cyclooxygenases | target |
| Ibuprofen | Interleukin-8 | target |
| Ibuprofen | C-X-C chemokine receptor type 2 | target |
| Ibuprofen | C-X-C chemokine receptor type 1 | target |
| Ibuprofen | Cytochrome P450 3A4 | enzyme |
| Ibuprofen | Alpha-methylacyl-CoA racemase | enzyme |
| Ibuprofen | Protein S100-A7 | target |
| Ibuprofen | Prostaglandin G/H synthase 1 | target |
| Ibuprofen | Platelet glycoprotein Ib alpha chain | target |
| Ibuprofen | Cytochrome P450 2C9 | enzyme |
| Ibuprofen | Albumin | carrier |
| Ibuprofen | ATP-binding cassette sub-family C member 4 | transporter |
| Ibuprofen | ATP-binding cassette sub-family C member 1 | transporter |
| Ibuprofen | Solute carrier organic anion transporter family member 1A2 | transporter |
| Ibuprofen | Solute carrier family 22 member 6 | transporter |
| Ibuprofen | Organic anion transporter 3 | transporter |
| Ibuprofen | Solute carrier family 22 member 11 | transporter |
| Ibuprofen | Solute carrier organic anion transporter family member 2B1 | transporter |
| Ibuprofen | ATP-dependent translocase ABCB1 | transporter |
| Ibuprofen | UDP-glucuronosyltransferase 1A3 | enzyme |
| Ibuprofen | UDP-glucuronosyltransferase 1A9 | enzyme |
| Ibuprofen | UDP-glucuronosyltransferase 2B4 | enzyme |
| Ibuprofen | UDP-glucuronosyltransferase 2B7 | enzyme |
| Ibuprofen | Cytochrome P450 2C8 | enzyme |
| Ibuprofen | Cytochrome P450 2C19 | enzyme |
| Ibuprofen | Apoptosis regulator Bcl-2 | target |
| Ibuprofen | Thrombomodulin | target |
| Ibuprofen | Fatty acid-binding protein, intestinal | target |
| Ibuprofen | Peroxisome proliferator-activated receptor gamma | target |
| Ibuprofen | Cystic fibrosis transmembrane conductance regulator | target |
| Ibuprofen | Peroxisome proliferator-activated receptor alpha | target |
| Indomethacin | ATP-binding cassette sub-family C member 3 | transporter |
| Indomethacin | ATP-binding cassette sub-family C member 2 | transporter |
| Indomethacin | ATP-binding cassette sub-family C member 6 | transporter |
| Indomethacin | Human Cyclooxygenases | target |
| Indomethacin | Interferon-induced, double-stranded RNA-activated protein kinase | target |
| Indomethacin | Bile salt export pump | transporter |
| Indomethacin | Solute carrier organic anion transporter family member 1B1 | transporter |
| Indomethacin | Aldo-keto reductase family 1 member C3 | target |
| Indomethacin | Peroxisome proliferator-activated receptor alpha | target |
| Indomethacin | UDP-glucuronosyltransferase 2B7 | enzyme |
| Indomethacin | Liver carboxylesterase 1 | enzyme |
| Indomethacin | UDP-glucuronosyltransferase 1A1 | enzyme |
| Indomethacin | Cytochrome P450 2C9 | enzyme |
| Indomethacin | Solute carrier family 22 member 7 | transporter |
| Indomethacin | Hepatic sodium/bile acid cotransporter | transporter |
| Indomethacin | Solute carrier family 22 member 11 | transporter |
| Indomethacin | ATP-binding cassette sub-family C member 11 | transporter |
| Indomethacin | Organic anion transporter 3 | transporter |
| Indomethacin | Solute carrier family 22 member 6 | transporter |
| Indomethacin | Solute carrier organic anion transporter family member 1A2 | transporter |
| Indomethacin | ATP-binding cassette sub-family C member 1 | transporter |
| Indomethacin | ATP-dependent translocase ABCB1 | transporter |
| Indomethacin | ATP-binding cassette sub-family C member 4 | transporter |
| Indomethacin | Albumin | carrier |
| Indomethacin | Peroxisome proliferator-activated receptor gamma | target |
| Indomethacin | Prostaglandin D2 receptor 2 | target |
| Indomethacin | Lactoylglutathione lyase | target |
| Indomethacin | Prostaglandin reductase 2 | target |
| Indomethacin | Phospholipase A2, membrane associated | target |
| Indomethacin | UDP-glucuronosyltransferase 1A9 | enzyme |
| Indomethacin | Cytochrome P450 2C19 | enzyme |
| Indomethacin | Prostaglandin G/H synthase 2 | target |
| Indomethacin | Prostaglandin G/H synthase 1 | target |
| Ketorolac | Prostaglandin G/H synthase 1 | target |
| Ketorolac | Prostaglandin G/H synthase 2 | target |
| Ketorolac | UDP-glucuronosyltransferase 2B7 | enzyme |
| Ketorolac | Cytochrome P450 2C8 | enzyme |
| Ketorolac | Cytochrome P450 2C9 | enzyme |
| Ketorolac | Human Cyclooxygenases | target |
| Labetalol | alpha1-acid glycoprotein | carrier |
| Labetalol | ATP-binding cassette sub-family B member 5 | transporter |
| Labetalol | UDP-glucuronosyltransferase 1A1 | enzyme |
| Labetalol | Albumin | carrier |
| Labetalol | Cytochrome P450 2C19 | enzyme |
| Labetalol | Cytochrome P450 2D6 | enzyme |
| Labetalol | Beta-2 adrenergic receptor | target |
| Labetalol | Beta-1 adrenergic receptor | target |
| Labetalol | Alpha-1 adrenergic receptors | target |
| Labetalol | UDP-glucuronosyltransferase 2B7 | enzyme |
| Labetalol | UDP-glucuronosyltransferase 1A9 | enzyme |
| Letrozole | ATP-dependent translocase ABCB1 | transporter |
| Letrozole | Aromatase | target |
| Letrozole | Cytochrome P450 3A4 | enzyme |
| Letrozole | Cytochrome P450 2A6 | enzyme |
| Letrozole | Aromatase | enzyme |
| Letrozole | Cytochrome P450 2C19 | enzyme |
| Letrozole | Albumin | carrier |
| Letrozole | UDP-glucuronosyltransferase 2B7 | enzyme |
| Losartan | Erythropoietin receptor | target |
| Losartan | Cytochrome P450 2C9 | enzyme |
| Losartan | ATP-dependent translocase ABCB1 | transporter |
| Losartan | Solute carrier family 22 member 6 | transporter |
| Losartan | UDP-glucuronosyltransferase 1A1 | enzyme |
| Losartan | UDP-glucuronosyltransferase 1A3 | enzyme |
| Losartan | UDP-glucuronosyltransferase 1A10 | enzyme |
| Losartan | UDP-glucuronosyltransferase 2B7 | enzyme |
| Losartan | Bile salt export pump | transporter |
| Losartan | Cytochrome P450 2C8 | enzyme |
| Losartan | Solute carrier family 2, facilitated glucose transporter member 9 | transporter |
| Losartan | Solute carrier family 22 member 12 | transporter |
| Losartan | Albumin | carrier |
| Losartan | Cytochrome P450 2C19 | enzyme |
| Losartan | UDP-glucuronosyltransferase 2B17 | enzyme |
| Losartan | Type-1 angiotensin II receptor | target |
| Losartan | Cytochrome P450 3A4 | enzyme |
| Lovastatin | Bile salt export pump | transporter |
| Lovastatin | Albumin | carrier |
| Lovastatin | Cytochrome P450 2C19 | enzyme |
| Lovastatin | Solute carrier organic anion transporter family member 2B1 | transporter |
| Lovastatin | Solute carrier organic anion transporter family member 1B3 | transporter |
| Lovastatin | ATP-binding cassette sub-family C member 2 | transporter |
| Lovastatin | UDP-glucuronosyltransferase 2B7 | enzyme |
| Lovastatin | UDP-glucuronosyltransferase 1A3 | enzyme |
| Lovastatin | UDP-glucuronosyltransferase 1A1 | enzyme |
| Lovastatin | Solute carrier organic anion transporter family member 1B1 | transporter |
| Lovastatin | Solute carrier organic anion transporter family member 1A2 | transporter |
| Lovastatin | ATP-dependent translocase ABCB1 | transporter |
| Lovastatin | Serum paraoxonase/lactonase 3 | enzyme |
| Lovastatin | Histone deacetylase 2 | target |
| Lovastatin | Integrin alpha-L | target |
| Lovastatin | Cytochrome P450 2C8 | enzyme |
| Lovastatin | Cytochrome P450 3A4 | enzyme |
| Lovastatin | 3-hydroxy-3-methylglutaryl-coenzyme A reductase | target |
| Loxoprofen | UDP-glucuronosyltransferase 2B7 | enzyme |
| Loxoprofen | Human Cyclooxygenases | target |
| Loxoprofen | Prostaglandin G/H synthase 2 | target |
| Loxoprofen | Prostaglandin G/H synthase 1 | target |
| Loxoprofen | Carbonyl reductase [NADPH] 1 | enzyme |
| Loxoprofen | Cytochrome P450 3A Subfamily | enzyme |
| Medical Cannabis | 5-hydroxytryptamine receptor 1A | target |
| Medical Cannabis | 5-hydroxytryptamine receptor 2A | target |
| Medical Cannabis | Neuronal acetylcholine receptor subunit alpha-7 | target |
| Medical Cannabis | Delta-type opioid receptor | target |
| Medical Cannabis | Mu-type opioid receptor | target |
| Medical Cannabis | Peroxisome proliferator-activated receptor gamma | target |
| Medical Cannabis | Cytochrome P450 3A5 | enzyme |
| Medical Cannabis | Cytochrome P450 3A7 | enzyme |
| Medical Cannabis | Cytochrome P450 1A1 | enzyme |
| Medical Cannabis | Cytochrome P450 1A2 | enzyme |
| Medical Cannabis | Cytochrome P450 1B1 | enzyme |
| Medical Cannabis | Polyunsaturated fatty acid 5-lipoxygenase | enzyme |
| Medical Cannabis | Polyunsaturated fatty acid lipoxygenase ALOX15 | enzyme |
| Medical Cannabis | Superoxide dismutase [Cu-Zn] | enzyme |
| Medical Cannabis | ATP-binding cassette sub-family C member 1 | transporter |
| Medical Cannabis | Broad substrate specificity ATP-binding cassette transporter ABCG2 | transporter |
| Medical Cannabis | Equilibrative nucleoside transporter 1 | transporter |
| Medical Cannabis | Transient receptor potential cation channel subfamily V member 1 | target |
| Medical Cannabis | Voltage-dependent T-type calcium channel subunit alpha-1G | target |
| Medical Cannabis | Voltage-dependent T-type calcium channel subunit alpha-1H | target |
| Medical Cannabis | Voltage-dependent T-type calcium channel subunit alpha-1I | target |
| Medical Cannabis | Transient receptor potential cation channel subfamily A member 1 | target |
| Medical Cannabis | Transient receptor potential cation channel subfamily M member 8 | target |
| Medical Cannabis | Transient receptor potential cation channel subfamily V member 2 | target |
| Medical Cannabis | Transient receptor potential cation channel subfamily V member 3 | target |
| Medical Cannabis | Transient receptor potential cation channel subfamily V member 4 | target |
| Medical Cannabis | Non-selective voltage-gated ion channel VDAC1 | target |
| Medical Cannabis | N-acyl-phosphatidylethanolamine-hydrolyzing phospholipase D | target |
| Medical Cannabis | N-acylethanolamine-hydrolyzing acid amidase | target |
| Medical Cannabis | Serotonin N-acetyltransferase | target |
| Medical Cannabis | Phospholipase A2 | target |
| Medical Cannabis | Superoxide dismutase [Cu-Zn] | target |
| Medical Cannabis | Fatty-acid amide hydrolase 1 | target |
| Medical Cannabis | Catalase | target |
| Medical Cannabis | Zeta-crystallin | target |
| Medical Cannabis | Sphingomyelin phosphodiesterase | target |
| Medical Cannabis | Glutathione peroxidase 1 | target |
| Medical Cannabis | Glutathione reductase, mitochondrial | target |
| Medical Cannabis | 3-hydroxy-3-methylglutaryl-coenzyme A reductase | target |
| Medical Cannabis | Indoleamine 2,3-dioxygenase 1 | target |
| Medical Cannabis | Prostaglandin G/H synthase 1 | target |
| Medical Cannabis | Prostaglandin G/H synthase 2 | target |
| Medical Cannabis | Steroid 17-alpha-hydroxylase/17,20 lyase | target |
| Medical Cannabis | Cytochrome P450 2E1 | enzyme |
| Medical Cannabis | Cytochrome P450 2J2 | enzyme |
| Medical Cannabis | UDP-glucuronosyltransferase 1A7 | enzyme |
| Medical Cannabis | UDP-glucuronosyltransferase 1A8 | enzyme |
| Medical Cannabis | UDP-glucuronosyltransferase 1A9 | enzyme |
| Medical Cannabis | UDP-glucuronosyltransferase 1A10 | enzyme |
| Medical Cannabis | UDP-glucuronosyltransferase 2B17 | enzyme |
| Medical Cannabis | Cytochrome P450 2C8 | enzyme |
| Medical Cannabis | ATP-dependent translocase ABCB1 | transporter |
| Medical Cannabis | UDP-glucuronosyltransferase 2B7 | enzyme |
| Medical Cannabis | Cytochrome P450 2B6 | enzyme |
| Medical Cannabis | Cytochrome P450 2A6 | enzyme |
| Medical Cannabis | Acetyl-CoA acetyltransferase, mitochondrial | target |
| Medical Cannabis | Liver carboxylesterase 1 | enzyme |
| Medical Cannabis | Cannabinoid receptor 1 | target |
| Medical Cannabis | Cannabinoid receptor 2 | target |
| Medical Cannabis | Cytochrome P450 2C9 | enzyme |
| Medical Cannabis | Cytochrome P450 2C19 | enzyme |
| Medical Cannabis | Cytochrome P450 2D6 | enzyme |
| Medical Cannabis | Cytochrome P450 3A4 | enzyme |
| Medical Cannabis | G protein-coupled receptor 12 | target |
| Medical Cannabis | Glycine receptor subunit alpha-1 | target |
| Medical Cannabis | Glycine receptor (alpha-1/beta) | target |
| Medical Cannabis | Glycine receptor subunit alpha-3 | target |
| Medical Cannabis | N-arachidonyl glycine receptor | target |
| Medical Cannabis | G protein-coupled receptor 55 | target |
| Midazolam | Cytochrome P450 3A4 | enzyme |
| Midazolam | Cytochrome P450 3A5 | enzyme |
| Midazolam | UDP-glucuronosyltransferase 1A4 | enzyme |
| Midazolam | Cytochrome P450 3A7 | enzyme |
| Midazolam | GABA(A) Receptor | target |
| Midazolam | GABA(A) Receptor Benzodiazepine Binding Site | target |
| Midazolam | ATP-dependent translocase ABCB1 | transporter |
| Midazolam | Albumin | carrier |
| Midazolam | Alpha-1-acid glycoprotein 1 | carrier |
| Midazolam | Adenosine receptor A2a | target |
| Midazolam | Excitatory amino acid transporter 2 | transporter |
| Midazolam | UDP-glucuronosyltransferase 2B7 | enzyme |
| Midazolam | UDP-glucuronosyltransferase 2B4 | enzyme |
| Midazolam | Translocator protein | target |
| Mirabegron | Alpha-1-acid glycoprotein 1 | carrier |
| Mirabegron | ATP-dependent translocase ABCB1 | transporter |
| Mirabegron | Solute carrier family 22 member 3 | transporter |
| Mirabegron | Cytochrome P450 3A4 | enzyme |
| Mirabegron | Cytochrome P450 2D6 | enzyme |
| Mirabegron | Solute carrier organic anion transporter family member 1A2 | transporter |
| Mirabegron | Albumin | carrier |
| Mirabegron | Beta-1 adrenergic receptor | target |
| Mirabegron | UDP-glucuronosyltransferase 1A8 | enzyme |
| Mirabegron | Solute carrier family 22 member 2 | transporter |
| Mirabegron | Solute carrier family 22 member 1 | transporter |
| Mirabegron | UDP-glucuronosyltransferase 1A3 | enzyme |
| Mirabegron | UDP-glucuronosyltransferase 2B7 | enzyme |
| Mirabegron | Beta-3 adrenergic receptor | target |
| Mirabegron | Cholinesterase | enzyme |
| Mirdametinib | Dual specificity mitogen-activated protein kinase kinase 2 | target |
| Mirdametinib | Broad substrate specificity ATP-binding cassette transporter ABCG2 | transporter |
| Mirdametinib | ATP-dependent translocase ABCB1 | transporter |
| Mirdametinib | UDP-glucuronosyltransferase 2B7 | enzyme |
| Mirdametinib | UDP-glucuronosyltransferase 1A6 | enzyme |
| Mirdametinib | Carboxylesterase | enzyme |
| Mirdametinib | Dual specificity mitogen-activated protein kinase kinase 1 | target |
| Mitiglinide | ATP-sensitive inward rectifier potassium channel 10 | target |
| Mitiglinide | UDP-glucuronosyltransferase 2B7 | enzyme |
| Mitiglinide | UDP-glucuronosyltransferase 1A3 | enzyme |
| Mitiglinide | Peroxisome proliferator-activated receptor gamma | target |
| Mitiglinide | ATP-binding cassette sub-family C member 8 | target |
| Morphine | Albumin | carrier |
| Morphine | Lymphocyte antigen 96 | target |
| Morphine | UDP-glucuronosyltransferase 1A3 | enzyme |
| Morphine | UDP-glucuronosyltransferase 2B4 | enzyme |
| Morphine | UDP-glucuronosyltransferase 2B15 | enzyme |
| Morphine | UDP-glucuronosyltransferase 1A8 | enzyme |
| Morphine | UDP-glucuronosyltransferase 1A1 | enzyme |
| Morphine | UDP-glucuronosyltransferase 2B7 | enzyme |
| Morphine | Cytochrome P450 3A4 | enzyme |
| Morphine | Mu-type opioid receptor | target |
| Morphine | Cytochrome P450 2C8 | enzyme |
| Morphine | Delta-type opioid receptor | target |
| Morphine | ATP-dependent translocase ABCB1 | transporter |
| Morphine | Kappa-type opioid receptor | target |
| Mycophenolate mofetil | UDP-glucuronosyltransferase 1A9 | enzyme |
| Mycophenolate mofetil | UDP-glucuronosyltransferase 2B7 | enzyme |
| Mycophenolate mofetil | UDP-glucuronosyltransferase 1A8 | enzyme |
| Mycophenolate mofetil | UDP-glucuronosyltransferase 1A6 | enzyme |
| Mycophenolate mofetil | UDP-glucuronosyltransferase 1A10 | enzyme |
| Mycophenolate mofetil | Liver carboxylesterase 1 | enzyme |
| Mycophenolate mofetil | Cytochrome P450 3A4 | enzyme |
| Mycophenolate mofetil | Cytochrome P450 3A5 | enzyme |
| Mycophenolate mofetil | Cytochrome P450 2C8 | enzyme |
| Mycophenolate mofetil | Solute carrier organic anion transporter family member 1B1 | transporter |
| Mycophenolate mofetil | Solute carrier organic anion transporter family member 1B3 | transporter |
| Mycophenolate mofetil | Broad substrate specificity ATP-binding cassette transporter ABCG2 | transporter |
| Mycophenolate mofetil | ATP-dependent translocase ABCB1 | transporter |
| Mycophenolate mofetil | 6-pyruvoyl tetrahydrobiopterin synthase | target |
| Mycophenolate mofetil | Carboxylic ester hydrolase | enzyme |
| Mycophenolate mofetil | ATP-binding cassette sub-family C member 2 | transporter |
| Mycophenolate mofetil | Prostaglandin E2 receptor EP2 subtype | target |
| Mycophenolate mofetil | Inosine-5'-monophosphate dehydrogenase | target |
| Mycophenolate mofetil | Inosine-5'-monophosphate dehydrogenase 2 | target |
| Mycophenolate mofetil | Inosine-5'-monophosphate dehydrogenase 1 | target |
| Mycophenolate mofetil | UDP-glucuronosyltransferase 1A1 | enzyme |
| Mycophenolate mofetil | UDP-glucuronosyltransferase 1A7 | enzyme |
| Mycophenolic acid | Albumin | carrier |
| Mycophenolic acid | UDP-glucuronosyltransferase 1A8 | enzyme |
| Mycophenolic acid | UDP-glucuronosyltransferase 1A10 | enzyme |
| Mycophenolic acid | Cytochrome P450 3A4 | enzyme |
| Mycophenolic acid | Cytochrome P450 3A5 | enzyme |
| Mycophenolic acid | Cytochrome P450 2C8 | enzyme |
| Mycophenolic acid | Inosine-5'-monophosphate dehydrogenase | target |
| Mycophenolic acid | UDP-glucuronosyltransferase 1A7 | enzyme |
| Mycophenolic acid | UDP-glucuronosyltransferase 2B7 | enzyme |
| Mycophenolic acid | UDP-glucuronosyltransferase 1A9 | enzyme |
| Mycophenolic acid | UDP-glucuronosyltransferase 1A1 | enzyme |
| Mycophenolic acid | Inosine-5'-monophosphate dehydrogenase 1 | target |
| Mycophenolic acid | Inosine-5'-monophosphate dehydrogenase 2 | target |
| Mycophenolic acid | UDP-glucuronosyltransferase 1A6 | enzyme |
| Nalmefene | UDP-glucuronosyltransferase 1A3 | enzyme |
| Nalmefene | Mu-type opioid receptor | target |
| Nalmefene | Kappa-type opioid receptor | target |
| Nalmefene | Delta-type opioid receptor | target |
| Nalmefene | UDP-glucuronosyltransferase 1A8 | enzyme |
| Nalmefene | Cytochrome P450 3A4 | enzyme |
| Nalmefene | Cytochrome P450 3A5 | enzyme |
| Nalmefene | UDP-glucuronosyltransferase 2B7 | enzyme |
| Nandrolone decanoate | UDP-glucuronosyltransferase 1A10 | enzyme |
| Nandrolone decanoate | Sex hormone-binding globulin | carrier |
| Nandrolone decanoate | UDP-glucuronosyltransferase 1A1 | enzyme |
| Nandrolone decanoate | UDP-glucuronosyltransferase 1A3 | enzyme |
| Nandrolone decanoate | UDP-glucuronosyltransferase 2B4 | enzyme |
| Nandrolone decanoate | UDP-glucuronosyltransferase 1A4 | enzyme |
| Nandrolone decanoate | Dopamine receptor | target |
| Nandrolone decanoate | Insulin-like growth factor 1 receptor | target |
| Nandrolone decanoate | 5-hydroxytryptamine receptor 1B | target |
| Nandrolone decanoate | 5-hydroxytryptamine 2 receptor | target |
| Nandrolone decanoate | Protein c-Fos | target |
| Nandrolone decanoate | Androgen receptor | target |
| Nandrolone decanoate | Amine oxidase [flavin-containing] A | enzyme |
| Nandrolone decanoate | Amine oxidase [flavin-containing] B | enzyme |
| Nandrolone decanoate | Aromatase | enzyme |
| Nandrolone decanoate | UDP-glucuronosyltransferase 2B7 | enzyme |
| Naproxen | UDP-glucuronosyltransferase 1A7 | enzyme |
| Naproxen | UDP-glucuronosyltransferase 1A8 | enzyme |
| Naproxen | UDP-glucuronosyltransferase 1A9 | enzyme |
| Naproxen | UDP-glucuronosyltransferase 1A10 | enzyme |
| Naproxen | Organic anion transporter 3 | transporter |
| Naproxen | Pancreatic triacylglycerol lipase | target |
| Naproxen | Human Cyclooxygenases | target |
| Naproxen | Prostaglandin G/H synthase 2 | target |
| Naproxen | Prostaglandin G/H synthase 1 | target |
| Naproxen | Albumin | carrier |
| Naproxen | Cytochrome P450 2C9 | enzyme |
| Naproxen | Cytochrome P450 1A2 | enzyme |
| Naproxen | Solute carrier organic anion transporter family member 1A2 | transporter |
| Naproxen | Solute carrier family 22 member 6 | transporter |
| Naproxen | Cytochrome P450 2C8 | enzyme |
| Naproxen | UDP-glucuronosyltransferase 1A6 | enzyme |
| Naproxen | UDP-glucuronosyltransferase 1A3 | enzyme |
| Naproxen | ATP-dependent translocase ABCB1 | transporter |
| Naproxen | Bile salt export pump | transporter |
| Naproxen | Peptostreptococcal albumin-binding protein | target |
| Naproxen | UDP-glucuronosyltransferase 2B7 | enzyme |
| Osalmid | Ribonucleoside-diphosphate reductase subunit M2 | target |
| Osalmid | Cytochrome P450 2C9 | enzyme |
| Osalmid | UDP-glucuronosyltransferase 1A1 | enzyme |
| Osalmid | UDP-glucuronosyltransferase 1A6 | enzyme |
| Osalmid | UDP-glucuronosyltransferase 1A9 | enzyme |
| Osalmid | UDP-glucuronosyltransferase 2B7 | enzyme |
| Osalmid | UDP-glucuronosyltransferase 2B15 | enzyme |
| Osalmid | Cytochrome P450 1A2 | enzyme |
| Osilodrostat | Multidrug and toxin extrusion protein 1 | transporter |
| Osilodrostat | Organic anion transporter 3 | transporter |
| Osilodrostat | Solute carrier family 22 member 6 | transporter |
| Osilodrostat | Solute carrier family 22 member 2 | transporter |
| Osilodrostat | Solute carrier family 22 member 1 | transporter |
| Osilodrostat | Solute carrier organic anion transporter family member 1B1 | transporter |
| Osilodrostat | Cytochrome P450 2E1 | enzyme |
| Osilodrostat | Cytochrome P450 2C19 | enzyme |
| Osilodrostat | Cytochrome P450 1A2 | enzyme |
| Osilodrostat | Cytochrome P450 3A5 | enzyme |
| Osilodrostat | UDP-glucuronosyltransferase 2B10 | enzyme |
| Osilodrostat | UDP-glucuronosyltransferase 2B7 | enzyme |
| Osilodrostat | UDP-glucuronosyltransferase 1A4 | enzyme |
| Osilodrostat | Cytochrome P450 2D6 | enzyme |
| Osilodrostat | Cytochrome P450 2B6 | enzyme |
| Osilodrostat | Cytochrome P450 3A4 | enzyme |
| Osilodrostat | UDP-glucuronosyltransferase 1A1 | enzyme |
| Osilodrostat | Cytochrome P450 11B1, mitochondrial | target |
| Osilodrostat | Cytochrome P450 11B2, mitochondrial | target |
| Oxazepam | Albumin | carrier |
| Oxazepam | GABA(A) Receptor Benzodiazepine Binding Site | target |
| Oxazepam | GABA(A) Receptor | target |
| Oxazepam | UDP-glucuronosyltransferase 1A9 | enzyme |
| Oxazepam | Translocator protein | target |
| Oxazepam | UDP-glucuronosyltransferase 2B7 | enzyme |
| Oxazepam | UDP-glucuronosyltransferase 2B15 | enzyme |
| PF-06835919 | UDP-glucuronosyltransferase 2B7 | enzyme |
| PF-06835919 | Ketohexokinase | target |
| PF-06835919 | Solute carrier organic anion transporter family member 1B1 | transporter |
| PF-06835919 | Solute carrier family 22 member 7 | transporter |
| PF-06835919 | Cytochrome P450 2C8 | enzyme |
| PF-06835919 | Cytochrome P450 2C9 | enzyme |
| PF-06835919 | Cytochrome P450 3A Subfamily | enzyme |
| Pitavastatin | Integrin alpha-L | target |
| Pitavastatin | ATP-dependent translocase ABCB1 | transporter |
| Pitavastatin | Solute carrier organic anion transporter family member 1B1 | transporter |
| Pitavastatin | Solute carrier organic anion transporter family member 1B3 | transporter |
| Pitavastatin | UDP-glucuronosyltransferase 2B7 | enzyme |
| Pitavastatin | UDP-glucuronosyltransferase 1A3 | enzyme |
| Pitavastatin | Cytochrome P450 2C9 | enzyme |
| Pitavastatin | Cytochrome P450 2C8 | enzyme |
| Pitavastatin | 3-hydroxy-3-methylglutaryl-coenzyme A reductase | target |
| Pitavastatin | Solute carrier organic anion transporter family member 2B1 | transporter |
| Pitavastatin | Hepatic sodium/bile acid cotransporter | transporter |
| Pitavastatin | Broad substrate specificity ATP-binding cassette transporter ABCG2 | transporter |
| Pitavastatin | ATP-binding cassette sub-family C member 2 | transporter |
| Pitavastatin | Albumin | carrier |
| Pitavastatin | Alpha-1-acid glycoprotein 1 | carrier |
| Pitavastatin | Bile salt export pump | transporter |
| Ponesimod | UDP-glucuronosyltransferase 2B7 | enzyme |
| Ponesimod | UDP-glucuronosyltransferase 1A1 | enzyme |
| Ponesimod | Cytochrome P450 4F12 | enzyme |
| Ponesimod | Cytochrome P450 4F3 | enzyme |
| Ponesimod | Cytochrome P450 3A5 | enzyme |
| Ponesimod | Cytochrome P450 3A4 | enzyme |
| Ponesimod | Cytochrome P450 2J2 | enzyme |
| Ponesimod | Sphingosine 1-phosphate receptor 1 | target |
| Silodosin | HERG human cardiac K+ channel | target |
| Silodosin | Aldo-keto reductase family 1 member A1 | enzyme |
| Silodosin | Aldehyde dehydrogenase, mitochondrial | enzyme |
| Silodosin | UDP-glucuronosyltransferase 2B7 | enzyme |
| Silodosin | Alpha-1B adrenergic receptor | target |
| Silodosin | Alpha-1D adrenergic receptor | target |
| Silodosin | Cytochrome P450 3A4 | enzyme |
| Silodosin | ATP-dependent translocase ABCB1 | transporter |
| Silodosin | Phosphatidylcholine translocator ABCB4 | transporter |
| Silodosin | Alpha-1A adrenergic receptor | target |
| Simvastatin | Solute carrier organic anion transporter family member 2B1 | transporter |
| Simvastatin | Cytochrome P450 2C19 | enzyme |
| Simvastatin | Bile salt export pump | transporter |
| Simvastatin | Integrin alpha-L | target |
| Simvastatin | ATP-binding cassette sub-family C member 2 | transporter |
| Simvastatin | UDP-glucuronosyltransferase 2B7 | enzyme |
| Simvastatin | UDP-glucuronosyltransferase 1A3 | enzyme |
| Simvastatin | UDP-glucuronosyltransferase 1A1 | enzyme |
| Simvastatin | Cytochrome P450 2D6 | enzyme |
| Simvastatin | Cytochrome P450 2B6 | enzyme |
| Simvastatin | Solute carrier organic anion transporter family member 1B1 | transporter |
| Simvastatin | Solute carrier organic anion transporter family member 1A2 | transporter |
| Simvastatin | ATP-dependent translocase ABCB1 | transporter |
| Simvastatin | Cytochrome P450 3A5 | enzyme |
| Simvastatin | Cytochrome P450 2C9 | enzyme |
| Simvastatin | Cytochrome P450 2C8 | enzyme |
| Simvastatin | Cytochrome P450 3A4 | enzyme |
| Simvastatin | 3-hydroxy-3-methylglutaryl-coenzyme A reductase | target |
| Simvastatin | Solute carrier organic anion transporter family member 1B3 | transporter |
| Simvastatin | Histone deacetylase 2 | target |
| Simvastatin | Cocaine esterase | enzyme |
| Simvastatin | Liver carboxylesterase 1 | enzyme |
| Sotagliflozin | UDP-glucuronosyltransferase 2B7 | enzyme |
| Sotagliflozin | Cytochrome P450 3A4 | enzyme |
| Sotagliflozin | UDP-glucuronosyltransferase 1A1 | enzyme |
| Sotagliflozin | Sodium/glucose cotransporter 1 | target |
| Sotagliflozin | Cytochrome P450 2D6 | enzyme |
| Sotagliflozin | ATP-dependent translocase ABCB1 | transporter |
| Sotagliflozin | Broad substrate specificity ATP-binding cassette transporter ABCG2 | transporter |
| Sotagliflozin | Solute carrier organic anion transporter family member 1B1 | transporter |
| Sotagliflozin | Solute carrier organic anion transporter family member 1B3 | transporter |
| Sotagliflozin | ATP-binding cassette sub-family C member 2 | transporter |
| Sotagliflozin | UDP-glucuronosyltransferase 1A9 | enzyme |
| Sotagliflozin | Sodium/glucose cotransporter 2 | target |
| Suprofen | Human Cyclooxygenases | target |
| Suprofen | Albumin | carrier |
| Suprofen | UDP-glucuronosyltransferase 2B7 | enzyme |
| Suprofen | Solute carrier family 22 member 12 | transporter |
| Suprofen | UDP-glucuronosyltransferase 1A1 | enzyme |
| Suprofen | Cytochrome P450 2C9 | enzyme |
| Suprofen | Prostaglandin G/H synthase 2 | target |
| Suprofen | Prostaglandin G/H synthase 1 | target |
| Tamoxifen | Cytochrome P450 2C8 | enzyme |
| Tamoxifen | Cytochrome P450 2D6 | enzyme |
| Tamoxifen | Cytochrome P450 3A4 | enzyme |
| Tamoxifen | Cytochrome P450 2C9 | enzyme |
| Tamoxifen | Estrogen receptor beta | target |
| Tamoxifen | Estrogen receptor | target |
| Tamoxifen | Cytochrome P450 2B6 | enzyme |
| Tamoxifen | Liver carboxylesterase 1 | enzyme |
| Tamoxifen | Cytochrome P450 3A5 | enzyme |
| Tamoxifen | Cytochrome P450 1A1 | enzyme |
| Tamoxifen | Bile salt export pump | transporter |
| Tamoxifen | Cytochrome P450 2C19 | enzyme |
| Tamoxifen | Flavin-containing monooxygenase 1 | enzyme |
| Tamoxifen | Flavin-containing monooxygenase 3 | enzyme |
| Tamoxifen | Cytochrome P450 3A7 | enzyme |
| Tamoxifen | ATP-dependent translocase ABCB1 | transporter |
| Tamoxifen | Broad substrate specificity ATP-binding cassette transporter ABCG2 | transporter |
| Tamoxifen | Aromatase | enzyme |
| Tamoxifen | Cytochrome P450 2A6 | enzyme |
| Tamoxifen | Cytochrome P450 2E1 | enzyme |
| Tamoxifen | UDP-glucuronosyltransferase 1A10 | enzyme |
| Tamoxifen | Sulfotransferase 1A1 | enzyme |
| Tamoxifen | ATP-binding cassette sub-family C member 2 | transporter |
| Tamoxifen | 3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase | target |
| Tamoxifen | Protein kinase C | target |
| Tamoxifen | Androgen receptor | target |
| Tamoxifen | Voltage-gated inwardly rectifying potassium channel KCNH2 | target |
| Tamoxifen | Nuclear receptor subfamily 1 group I member 2 | target |
| Tamoxifen | Estrogen-related receptor gamma | target |
| Tamoxifen | Sex hormone-binding globulin | target |
| Tamoxifen | Albumin | carrier |
| Tamoxifen | Mitogen-activated protein kinase 8 | target |
| Tamoxifen | Phospholipid-transporting ATPase ABCA1 | transporter |
| Tamoxifen | Sulfotransferase 1E1 | enzyme |
| Tamoxifen | UDP-glucuronosyltransferase 2B17 | enzyme |
| Tamoxifen | UDP-glucuronosyltransferase 2B7 | enzyme |
| Tamoxifen | Cytochrome P450 1A2 | enzyme |
| Tamoxifen | Sulfotransferase 2A1 | enzyme |
| Tamoxifen | Thyroxine-binding globulin | carrier |
| Tamoxifen | Cytochrome P450 1B1 | enzyme |
| Tapentadol | UDP-glucuronosyltransferase 2B7 | enzyme |
| Tapentadol | UDP-glucuronosyltransferase 1A9 | enzyme |
| Tapentadol | Sodium-dependent serotonin transporter | target |
| Tapentadol | Cytochrome P450 2C19 | enzyme |
| Tapentadol | Cytochrome P450 2C9 | enzyme |
| Tapentadol | Cytochrome P450 2D6 | enzyme |
| Tapentadol | Mu-type opioid receptor | target |
| Tapentadol | Kappa-type opioid receptor | target |
| Tapentadol | Delta-type opioid receptor | target |
| Tapentadol | Sodium-dependent noradrenaline transporter | target |
| Tradipitant | ATP-dependent translocase ABCB1 | transporter |
| Tradipitant | UDP-glucuronosyltransferase 2B7 | enzyme |
| Tradipitant | UDP-glucuronosyltransferase 1A4 | enzyme |
| Tradipitant | Cytochrome P450 2C8 | enzyme |
| Tradipitant | Cytochrome P450 2C19 | enzyme |
| Tradipitant | Cytochrome P450 3A4 | enzyme |
| Tradipitant | Substance-P receptor | target |
| Tretinoin | Retinoic acid receptor gamma | target |
| Tretinoin | Retinoic acid receptor RXR-beta | target |
| Tretinoin | Aldehyde dehydrogenase 1A1 | target |
| Tretinoin | Retinoic acid-induced protein 3 | target |
| Tretinoin | Retinoic acid receptor RXR-gamma | target |
| Tretinoin | Retinal dehydrogenase 2 | target |
| Tretinoin | Retinoic acid receptor responder protein 1 | target |
| Tretinoin | Cytochrome P450 2C8 | enzyme |
| Tretinoin | Cellular retinoic acid-binding protein 1 | transporter |
| Tretinoin | Cellular retinoic acid-binding protein 2 | transporter |
| Tretinoin | Cytochrome P450 2B6 | enzyme |
| Tretinoin | Cytochrome P450 3A4 | enzyme |
| Tretinoin | Cytochrome P450 3A5 | enzyme |
| Tretinoin | Cytochrome P450 2A6 | enzyme |
| Tretinoin | Cytochrome P450 3A7 | enzyme |
| Tretinoin | Cytochrome P450 2C18 | enzyme |
| Tretinoin | Cytochrome P450 2C9 | enzyme |
| Tretinoin | Cytochrome P450 4A11 | enzyme |
| Tretinoin | Cytochrome P450 1A1 | enzyme |
| Tretinoin | Retinoic acid receptor alpha | target |
| Tretinoin | Retinoic acid receptor beta | target |
| Tretinoin | Lipocalin-1 | target |
| Tretinoin | Odorant-binding protein 2a | target |
| Tretinoin | Retinol-binding protein 4 | target |
| Tretinoin | Albumin | carrier |
| Tretinoin | [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial | target |
| Tretinoin | Retinoic acid receptor RXR-alpha | target |
| Tretinoin | Carcinoembryonic antigen | target |
| Tretinoin | UDP-glucuronosyltransferase 2B7 | enzyme |
| Tretinoin | Cytochrome P450 2E1 | enzyme |
| Tretinoin | Cytochrome P450 26A1 | enzyme |
| Tretinoin | Cellular retinoic acid-binding protein 1 | target |
| Troglitazone | Cytochrome P450 1A1 | enzyme |
| Troglitazone | Aromatase | enzyme |
| Troglitazone | Peroxisome proliferator-activated receptor gamma | target |
| Troglitazone | Glutathione S-transferase P | target |
| Troglitazone | Peroxisome proliferator-activated receptor alpha | target |
| Troglitazone | Peroxisome proliferator-activated receptor delta | target |
| Troglitazone | UDP-glucuronosyltransferase 2B15 | enzyme |
| Troglitazone | UDP-glucuronosyltransferase 2B7 | enzyme |
| Troglitazone | UDP-glucuronosyltransferase 1A10 | enzyme |
| Troglitazone | UDP-glucuronosyltransferase 1A9 | enzyme |
| Troglitazone | UDP-glucuronosyltransferase 1A8 | enzyme |
| Troglitazone | UDP-glucuronosyltransferase 1A7 | enzyme |
| Troglitazone | UDP-glucuronosyltransferase 1A6 | enzyme |
| Troglitazone | UDP-glucuronosyltransferase 1A4 | enzyme |
| Troglitazone | UDP-glucuronosyltransferase 1A3 | enzyme |
| Troglitazone | Cytochrome P450 3A7 | enzyme |
| Troglitazone | Cytochrome P450 3A5 | enzyme |
| Troglitazone | Cytochrome P450 2C9 | enzyme |
| Troglitazone | Steroid hormone receptor ERR1 | target |
| Troglitazone | Estrogen-related receptor gamma | target |
| Troglitazone | Solute carrier organic anion transporter family member 1B1 | transporter |
| Troglitazone | Bile salt export pump | transporter |
| Troglitazone | Cytochrome P450 2C8 | enzyme |
| Troglitazone | UDP-glucuronosyltransferase 1A1 | enzyme |
| Troglitazone | Cytochrome P450 2C19 | enzyme |
| Troglitazone | Cytochrome P450 3A4 | enzyme |
| Troglitazone | Equilibrative nucleoside transporter 1 | target |
| Troglitazone | Plasminogen activator inhibitor 1 | target |
| Troglitazone | Cytochrome P450 2B6 | enzyme |
| Troglitazone | Long-chain-fatty-acid--CoA ligase 4 | target |
| Vadadustat | Prolyl hydroxylase EGLN2 | target |
| Vadadustat | Prolyl hydroxylase EGLN3 | target |
| Vadadustat | Egl nine homolog 1 | target |
| Vadadustat | Hypoxia-inducible factor 1-alpha | target |
| Vadadustat | Endothelial PAS domain-containing protein 1 | target |
| Vadadustat | UDP-glucuronosyltransferase 1A1 | enzyme |
| Vadadustat | UDP-glucuronosyltransferase 1A7 | enzyme |
| Vadadustat | UDP-glucuronosyltransferase 1A8 | enzyme |
| Vadadustat | UDP-glucuronosyltransferase 1A9 | enzyme |
| Vadadustat | UDP-glucuronosyltransferase 2B7 | enzyme |
| Vadadustat | Cytochrome P450 2B6 | enzyme |
| Vadadustat | Cytochrome P450 2C8 | enzyme |
| Vadadustat | Cytochrome P450 3A4 | enzyme |
| Vadadustat | Broad substrate specificity ATP-binding cassette transporter ABCG2 | transporter |
| Vadadustat | Organic anion transporter 3 | transporter |
| Vadadustat | Solute carrier family 22 member 6 | transporter |
| Vadadustat | Albumin | carrier |
| Vadadustat | Cytochrome P450 2C9 | enzyme |
| Vadimezan | UDP-glucuronosyltransferase 1A9 | enzyme |
| Vadimezan | UDP-glucuronosyltransferase 2B7 | enzyme |
| Vadimezan | Cytochrome P450 1A2 | enzyme |
| Vadimezan | Nuclear factor NF-kappa-B p105 subunit | target |
| Vadimezan | Nuclear factor NF-kappa-B p100 subunit | target |
| Vadimezan | Transcription factor p65 | target |
| Vadimezan | Proto-oncogene c-Rel | target |
| Vadimezan | Transcription factor RelB | target |
| Valproic acid | Histone deacetylase 9 | target |
| Valproic acid | Short/branched chain specific acyl-CoA dehydrogenase, mitochondrial | target |
| Valproic acid | Cytochrome P450 2A6 | enzyme |
| Valproic acid | Cytochrome P450 2B6 | enzyme |
| Valproic acid | Cytochrome P450 2C9 | enzyme |
| Valproic acid | Organic cation/carnitine transporter 2 | transporter |
| Valproic acid | Solute carrier family 22 member 6 | transporter |
| Valproic acid | Organic anion transporter 3 | transporter |
| Valproic acid | Monocarboxylate transporter 1 | transporter |
| Valproic acid | Solute carrier family 22 member 7 | transporter |
| Valproic acid | Cytochrome P450 3A5 | enzyme |
| Valproic acid | UDP-glucuronosyltransferase 1A9 | enzyme |
| Valproic acid | Prostaglandin G/H synthase 1 | enzyme |
| Valproic acid | Cytochrome P450 1A2 | enzyme |
| Valproic acid | Cytochrome P450 2C19 | enzyme |
| Valproic acid | Cytochrome P450 3A4 | enzyme |
| Valproic acid | UDP-glucuronosyltransferase 1A4 | enzyme |
| Valproic acid | UDP-glucuronosyltransferase 1A8 | enzyme |
| Valproic acid | UDP-glucuronosyltransferase 1A10 | enzyme |
| Valproic acid | UDP-glucuronosyltransferase 1A6 | enzyme |
| Valproic acid | Histone deacetylase 2 | target |
| Valproic acid | Sodium channel protein | target |
| Valproic acid | UDP-glucuronosyltransferase 2B7 | enzyme |
| Valproic acid | UDP-glucuronosyltransferase 2B15 | enzyme |
| Valproic acid | 2-oxoglutarate dehydrogenase complex component E1 | target |
| Valproic acid | Succinate-semialdehyde dehydrogenase, mitochondrial | target |
| Valproic acid | Glycogen synthase kinase-3 alpha | target |
| Valproic acid | 4-aminobutyrate aminotransferase, mitochondrial | target |
| Valproic acid | Programmed cell death 1 ligand 1 | target |
| Valproic acid | Ornithine decarboxylase | target |
| Valproic acid | Hepatocyte growth factor | target |
| Valproic acid | Cyclin-dependent kinase inhibitor 1 | target |
| Valproic acid | Histone deacetylase | target |
| Valproic acid | Solute carrier organic anion transporter family member 2B1 | transporter |
| Valproic acid | UDP-glucuronosyltransferase 1A1 | enzyme |
| Valproic acid | Albumin | carrier |
| Valproic acid | Peroxisome proliferator-activated receptor gamma | target |
| Valproic acid | Peroxisome proliferator-activated receptor delta | target |
| Valproic acid | Peroxisome proliferator-activated receptor alpha | target |
| Valproic acid | UDP-glucuronosyltransferase 1A3 | enzyme |
| Vamorolone | Mineralocorticoid receptor | target |
| Vamorolone | UDP-glucuronosyltransferase 2B17 | enzyme |
| Vamorolone | UDP-glucuronosyltransferase 2B7 | enzyme |
| Vamorolone | UDP-glucuronosyltransferase 1A3 | enzyme |
| Vamorolone | Cytochrome P450 2C8 | enzyme |
| Vamorolone | Cytochrome P450 3A5 | enzyme |
| Vamorolone | Cytochrome P450 3A4 | enzyme |
| Vamorolone | Glucocorticoid receptor | target |
| Vicadrostat | Cytochrome P450 11B2, mitochondrial | target |
| Vicadrostat | UDP-glucuronosyltransferase 2B7 | enzyme |
| Zaltoprofen | Cytochrome P450 2C9 | enzyme |
| Zaltoprofen | Prostaglandin G/H synthase 1 | enzyme |
| Zaltoprofen | Prostaglandin G/H synthase 2 | target |
| Zaltoprofen | Prostaglandin G/H synthase 1 | target |
| Zaltoprofen | Peroxisome proliferator-activated receptor gamma | target |
| Zaltoprofen | UDP-glucuronosyltransferase 2B7 | enzyme |
| Zidovudine | ATP-binding cassette sub-family C member 4 | transporter |
| Zidovudine | ATP-binding cassette sub-family C member 5 | transporter |
| Zidovudine | Broad substrate specificity ATP-binding cassette transporter ABCG2 | transporter |
| Zidovudine | Telomerase reverse transcriptase | target |
| Zidovudine | Thymidine kinase, cytosolic | enzyme |
| Zidovudine | UDP-glucuronosyltransferase 2B7 | enzyme |
| Zidovudine | UDP-glucuronosyltransferase 1A1 | enzyme |
| Zidovudine | Gag-Pol polyprotein | target |
| Zidovudine | Receptor-type tyrosine-protein kinase FLT3 | target |
| Zidovudine | ATP-dependent translocase ABCB1 | transporter |
| Zidovudine | Equilibrative nucleoside transporter 2 | transporter |
| Zidovudine | Sodium/nucleoside cotransporter 1 | transporter |
| Zidovudine | Solute carrier family 22 member 11 | transporter |
| Zidovudine | Organic anion transporter 3 | transporter |
| Zidovudine | Solute carrier family 22 member 7 | transporter |
| Zidovudine | Solute carrier family 22 member 6 | transporter |
| Zidovudine | Solute carrier family 22 member 2 | transporter |
| Zidovudine | Reverse transcriptase/RNaseH | target |
| Zidovudine | Cytochrome P450 3A4 | enzyme |
| Zidovudine | Cytochrome P450 2A6 | enzyme |
| Zidovudine | Albumin | carrier |
| Zidovudine | Cytochrome P450 2C9 | enzyme |