UGT2B7 substrates

Name
UGT2B7 substrates
Accession Number
DBCAT004610
Description

Not Available

Drugs
DrugDrug Description
HydromorphoneAn opioid analgesic used to treat moderate to severe pain when the use of an opioid is indicated.
LosartanAn angiotensin receptor blocker used to treat hypertension and diabetic nephropathy, and is used to reduce the risk of stroke.
DiclofenacAn NSAID used to treat the signs and symptoms of osteoarthritis and rheumatoid arthritis.
EtodolacAn NSAID used to treat osteoarthritis and rheumatoid arthritis, as well as acute pain.
FlurbiprofenAn NSAID used to treat the signs and symptoms of osteoarthritis and rheumatoid arthritis.
IbuprofenAn NSAID and non-selective COX inhibitor used to treat mild-moderate pain, fever, and inflammation.
NaproxenAn NSAID used to treat rheumatoid arthritis, osteoarthritis, ankylosing spondylitis, polyarticular juvenile idiopathic arthritis, tendinitis, bursitis, acute gout, primary dysmenorrhea, and mild to moderate pain.
SuprofenAn NSAID used to prevent pupil constriction in ocular surgery.
MitiglinideFor the treatment of type 2 diabetes.
ZaltoprofenA non-steroidal anti-inflammatory drug approved for use in Japan in 1993.
AmbrisentanA selective type A endothelin receptor antagonist used to treat primary pulmonary arterial hypertension and pulmonary arterial hypertension based on diagnostic classifications.
TroglitazoneFor the treatment of Type II diabetes mellitus. It is used alone or in combination with a sulfonylurea, metformin, or insulin as an adjunct to diet and exercise.
MorphineAn opioid agonist used for the relief of moderate to severe acute and chronic pain.
IndomethacinA nonsteroidal anti-inflammatory (NSAID) used for symptomatic management of chronic musculoskeletal pain conditions and to induce closure of a hemodynamically significant patent ductus arteriosus in premature infants.
Mycophenolate mofetilAn inosine monophosphate dehydrogenase inhibitor used to prevent the rejection of kidney, heart, or liver transplants.
EzetimibeA cholesterol absorption inhibitor used to lower total cholesterol, LDL-C, Apo-B, and non-HDL-C in primary hyperlipidemia and familial cholesterolemia.
Mycophenolic acidAn immunosuppressant used to prevent organ transplant rejections.
VadimezanInvestigated for use/treatment in solid tumors, lung cancer, ovarian cancer, and prostate cancer.
EpirubicinAn anthracycline topoisomerase II inhibitor used as an adjuvant to treating axillary node metastases in patients who have undergone surgical resection of primary breast cancer.
TapentadolAn opioid used to manage severe pain that has not responded to non-opioid medications, and for which opioid analgesic therapy is appropriate.
PitavastatinAn HMG-CoA reductase inhibitor used to lower lipid levels and reduce the risk of cardiovascular disease including myocardial infarction and stroke.
SilodosinAn alpha-1 adrenergic receptor antagonist used to treat symptoms associated with benign prostatic hyperplasia (BPH).
ZidovudineA dideoxynucleoside used in the treatment of HIV infection.
LovastatinAn HMG-CoA reductase inhibitor used to lower LDL cholesterol and reduce the risk of cardiovascular disease and associated conditions, including myocardial infarction and stroke.
SimvastatinAn HMG-CoA reductase inhibitor used to lower lipid levels and reduce the risk of cardiovascular events including myocardial infarction and stroke.
OxazepamAn intermediate-acting benzodiazepine with slow onset commonly used to treat panic disorders, severe anxiety, alcohol withdrawals, and insomnia.
CarbamazepineAn anticonvulsant used to treat various types of seizures and pain resulting from trigeminal neuralgia.
CodeineAn opioid analgesic used to treat moderate to severe pain when the use of an opioid is indicated.
FluvastatinAn HMG-CoA reductase inhibitor used to lower lipid levels and reduce the risk of cardiovascular disease including myocardial infarction and stroke.
Valproic acidAn anticonvulsant used to control complex partial seizures and both simple and complex absence seizures.
DapagliflozinA sodium-glucose cotransporter 2 inhibitor used in the management of type 2 diabetes mellitus.
EnasidenibAn isocitrate dehydrogenase-2 inhibitor used to treat relapsed or refractory acute myeloid leukemia with an isocitrate dehydrogenase-2 mutation.
NalmefeneAn opioid antagonist used to reduce alcohol consumption in adults with alcohol dependence and treat and prevent opioid overdose.
AcemetacinA NSAID indicated in the treatment of pain and inflammation.
ErtugliflozinAn SGLT2 inhibitor used to treat type 2 diabetes mellitus alone or in combination with other antidiabetic drugs.
ArtenimolFor the treatment of uncomplicated Plasmodium falciparum infection in adults, children, and infants aged 6 months and up weighing over 5 kg [FDA Label]. Used in combination with DB13941.
LabetalolAn alpha and beta adrenergic antagonist used to treat hypertension, angina, and sympathetic overactivity syndrome.
TamoxifenA selective estrogen receptor modulator used to treat estrogen receptor positive breast cancer, reduce the risk of invasive breast cancer following surgery, or reduce the risk of breast cancer in high risk women.
CarvedilolA non selective beta-adrenergic antagonist used to treat mild to severe chronic heart failure, hypertension, and left ventricular dysfunction following myocardial infarction in clinically stable patients.
KetorolacAn NSAID used to treat moderate to severe pain, rheumatoid arthritis, osteoarthritis, ankylosing spondylitis, menstrual disorders, and headaches.
Dabigatran etexilateAn anticoagulant used for the prevention of venous thromboembolic events or stroke in patients with recent elective hip or knee replacement surgery and atrial fibrillation.
DexibuprofenA pharmacologically active enantiomer of racemic ibuprofen (NSAID) used to treat pain and inflammation.
GemfibrozilA lipid regulator that is used in the reduction of serum triglyceride levels in high-risk patients with hyperlipidemia.
AnastrozoleA competitive, selective, non-steroidal aromatase inhibitor used as adjuvant therapy for the treatment of hormone receptor-positive breast cancer in postmenopausal women.
LoxoprofenAn NSAID used to treat pain and inflammation in musculoskeletal conditions.
CenobamateA small molecule drug indicated to treat partial onset seizures in adults.
FormoterolAn inhaled long-acting beta2-adrenergic receptor agonist used as a bronchodilator in the management of asthma and COPD.
LetrozoleAn aromatase inhibitor used to treat breast cancer in postmenopausal women.
EthinylestradiolAn estradiol used as a contraceptive.
OsilodrostatAn oral inhibitor of cortisol synthesis used to treat Cushing's disease by normalizing hypercortisolism.
Bempedoic acidA drug used in conjunction with lifestyle modification and/or other agents for the treatment of refractory hypercholesterolemia.
EmpagliflozinAn SGLT2 inhibitor used to manage type 2 diabetes mellitus.
ArtesunateArtesunate is an artemesinin derivative indicated for the initial treatment of severe malaria.
DextromethorphanAn NMDA receptor antagonist used to treat cases of dry cough.
FebuxostatA xanthine oxidase inhibitor used for the management of chronic hyperuricemia in adults with gout who have an inadequate response or intolerance to allopurinol.
PonesimodA sphingosine 1-phosphate receptor modulator indicated to treat relapsing multiple sclerosis.
MirabegronA beta-3 adrenergic agonist used to treat overactive bladder and neurogenic detrusor overactivity.
EstetrolAn estrogen used in combination with drospirenone for oral contraception.
Nandrolone decanoateAn anabolic steroid indicated for the management of the anemia of renal insufficiency by increasing hemoglobin and red cell mass.
AsciminibAn inhibitor of ABL/BCR-ABL1 tyrosine kinase for the treatment of patients with Philadelphia chromosome-positive CML, including those with the T315I mutation.
SotagliflozinAn orally administered dual SGLT1/2 inhibitor used alongside insulin to improve glycemic control in patients with type 1 diabetes mellitus.
CannabidiolAn active cannabinoid used as an adjunctive treatment for the management of seizures associated with Lennox-Gastaut syndrome or Dravet syndrome and symptomatic relief of moderate to severe neuropathic pain or other painful conditions, like cancer.
CannabinolCannabinol (CBN) is a physiologically inactive constituent of Cannabis sativa.
Medical CannabisThe use of the plant species Cannabis sativa and Cannabis indica, popularly known as marijuana, has gained popularity in recent years for the management of a wide variety of medical...
CobimetinibAn antineoplastic agent and selective inhibitor of the mitogen-activated extracellular kinase (MEK) pathway used to treat unresectable or metastatic melanoma.
EdaravoneA free radical scavenger used to delay the progression of ALS.
MidazolamA short-acting benzodiazepine with rapid onset that is commonly used in seizures, anesthesia and anxiety disorders.
TretinoinA vitamin A derivative used to treat acne vulgaris and certain types of promyelocytic leukemia, as well as various skin conditions in over-the-counter medications.
VadadustatAn oral hypoxia-inducible factor prolyl-hydroxylase inhibitor used to treat symptomatic anemia associated with chronic kidney disease in adults on chronic maintenance dialysis.
VamoroloneA synthetic glucocorticoid used as an anti-inflammatory and immunosuppressant in the management of Duchenne muscular dystrophy (DMD).
CapivasertibA serine/threonine kinase inhibitor used to treat hormone receptor-positive, HER2-negative, locally advanced or metastatic breast cancer
Drugs & Drug Targets
DrugTargetType
HydromorphoneMu-type opioid receptortarget
HydromorphoneDelta-type opioid receptortarget
HydromorphoneKappa-type opioid receptortarget
HydromorphoneCytochrome P450 2C9enzyme
HydromorphoneUDP-glucuronosyltransferase 1-3enzyme
HydromorphoneUDP-glucuronosyltransferase 2B7enzyme
HydromorphoneSerum albumincarrier
LosartanType-1 angiotensin II receptortarget
LosartanCytochrome P450 3A4enzyme
LosartanCytochrome P450 2C9enzyme
LosartanP-glycoprotein 1transporter
LosartanSolute carrier family 22 member 6transporter
LosartanUDP-glucuronosyltransferase 1-1enzyme
LosartanUDP-glucuronosyltransferase 1-3enzyme
LosartanUDP-glucuronosyltransferase 1-10enzyme
LosartanUDP-glucuronosyltransferase 2B7enzyme
LosartanUDP-glucuronosyltransferase 2B17enzyme
LosartanCytochrome P450 2C19enzyme
LosartanSerum albumincarrier
LosartanSolute carrier family 22 member 12transporter
LosartanSolute carrier family 2, facilitated glucose transporter member 9transporter
LosartanBile salt export pumptransporter
LosartanCytochrome P450 2C8enzyme
DiclofenacProstaglandin G/H synthase 1target
DiclofenacProstaglandin G/H synthase 2target
DiclofenacTransthyretincarrier
DiclofenacCytochrome P450 2C9enzyme
DiclofenacCytochrome P450 2C19enzyme
DiclofenacCytochrome P450 1A2enzyme
DiclofenacCytochrome P450 2C8enzyme
DiclofenacSerum albumincarrier
DiclofenacMultidrug resistance-associated protein 4transporter
DiclofenacMultidrug resistance-associated protein 1transporter
DiclofenacSolute carrier family 22 member 6transporter
DiclofenacSolute carrier family 22 member 8transporter
DiclofenacSolute carrier organic anion transporter family member 1C1transporter
DiclofenacSolute carrier family 22 member 11transporter
DiclofenacUDP-glucuronosyltransferase 2B7enzyme
DiclofenacCytochrome P450 3A4enzyme
DiclofenacCytochrome P450 2B6enzyme
DiclofenacCytochrome P450 2C18enzyme
DiclofenacCytochrome P450 2E1enzyme
DiclofenacSolute carrier organic anion transporter family member 1B1transporter
DiclofenacBile salt export pumptransporter
DiclofenacUDP-glucuronosyltransferase 1-3enzyme
DiclofenacUDP-glucuronosyltransferase 1-9enzyme
DiclofenacUDP-glucuronosyltransferase 2B4enzyme
DiclofenacArachidonate 5-lipoxygenaseenzyme
DiclofenacSodium channel protein type 4 subunit alphatransporter
DiclofenacAcid-sensing ion channel 1transporter
DiclofenacPotassium voltage-gated channel subfamily KQT member 2transporter
DiclofenacPotassium voltage-gated channel subfamily KQT member 3transporter
DiclofenacPhospholipase A2, membrane associatedenzyme
DiclofenacP-glycoprotein 1transporter
EtodolacProstaglandin G/H synthase 1target
EtodolacProstaglandin G/H synthase 2target
EtodolacCytochrome P450 2C9enzyme
EtodolacUDP-glucuronosyltransferase 1-9enzyme
EtodolacRetinoic acid receptor RXR-alphatarget
EtodolacSerum albumincarrier
EtodolacSolute carrier family 22 member 6transporter
EtodolacUDP-glucuronosyltransferase 1-3enzyme
EtodolacUDP-glucuronosyltransferase 1-10enzyme
EtodolacUDP-glucuronosyltransferase 2B7enzyme
FlurbiprofenProstaglandin G/H synthase 2target
FlurbiprofenProstaglandin G/H synthase 1target
FlurbiprofenCytochrome P450 2C9enzyme
FlurbiprofenSerum albumincarrier
FlurbiprofenMultidrug resistance-associated protein 4transporter
FlurbiprofenSolute carrier family 22 member 6transporter
FlurbiprofenUDP-glucuronosyltransferase 2B7enzyme
FlurbiprofenUDP-glucuronosyltransferase 1-1enzyme
FlurbiprofenUDP-glucuronosyltransferase 1-3enzyme
FlurbiprofenUDP-glucuronosyltransferase 1-9enzyme
FlurbiprofenUDP-glucuronosyltransferase 2B4enzyme
IbuprofenProstaglandin G/H synthase 1target
IbuprofenProstaglandin G/H synthase 2target
IbuprofenCytochrome P450 2C9enzyme
IbuprofenSerum albumincarrier
IbuprofenMultidrug resistance-associated protein 4transporter
IbuprofenMultidrug resistance-associated protein 1transporter
IbuprofenSolute carrier organic anion transporter family member 1A2transporter
IbuprofenSolute carrier family 22 member 6transporter
IbuprofenSolute carrier family 22 member 8transporter
IbuprofenSolute carrier family 22 member 11transporter
IbuprofenSolute carrier organic anion transporter family member 2B1transporter
IbuprofenP-glycoprotein 1transporter
IbuprofenUDP-glucuronosyltransferase 1-3enzyme
IbuprofenUDP-glucuronosyltransferase 1-9enzyme
IbuprofenUDP-glucuronosyltransferase 2B4enzyme
IbuprofenUDP-glucuronosyltransferase 2B7enzyme
IbuprofenCytochrome P450 2C8enzyme
IbuprofenCytochrome P450 2C19enzyme
IbuprofenApoptosis regulator Bcl-2target
IbuprofenThrombomodulintarget
IbuprofenFatty acid-binding protein, intestinaltarget
IbuprofenPeroxisome proliferator-activated receptor gammatarget
IbuprofenCystic fibrosis transmembrane conductance regulatortarget
IbuprofenPeroxisome proliferator-activated receptor alphatarget
IbuprofenPlatelet glycoprotein Ib alpha chaintarget
IbuprofenProtein S100-A7target
IbuprofenAlpha-methylacyl-CoA racemaseenzyme
IbuprofenCytochrome P450 3A4enzyme
NaproxenProstaglandin G/H synthase 1target
NaproxenProstaglandin G/H synthase 2target
NaproxenSerum albumincarrier
NaproxenCytochrome P450 2C9enzyme
NaproxenCytochrome P450 1A2enzyme
NaproxenSolute carrier organic anion transporter family member 1A2transporter
NaproxenSolute carrier family 22 member 6transporter
NaproxenCytochrome P450 2C8enzyme
NaproxenUDP-glucuronosyltransferase 2B7enzyme
NaproxenPeptostreptococcal albumin-binding proteintarget
NaproxenBile salt export pumptransporter
NaproxenP-glycoprotein 1transporter
NaproxenUDP-glucuronosyltransferase 1-3enzyme
NaproxenUDP-glucuronosyltransferase 1-6enzyme
NaproxenUDP-glucuronosyltransferase 1-7enzyme
NaproxenUDP-glucuronosyltransferase 1-8enzyme
NaproxenUDP-glucuronosyltransferase 1-9enzyme
NaproxenUDP-glucuronosyltransferase 1-10enzyme
NaproxenSolute carrier family 22 member 8transporter
SuprofenProstaglandin G/H synthase 1target
SuprofenProstaglandin G/H synthase 2target
SuprofenCytochrome P450 2C9enzyme
SuprofenUDP-glucuronosyltransferase 1-1enzyme
SuprofenSolute carrier family 22 member 12transporter
SuprofenUDP-glucuronosyltransferase 2B7enzyme
SuprofenSerum albumincarrier
MitiglinideATP-binding cassette sub-family C member 8target
MitiglinidePeroxisome proliferator-activated receptor gammatarget
MitiglinideUDP-glucuronosyltransferase 1-3enzyme
MitiglinideUDP-glucuronosyltransferase 2B7enzyme
ZaltoprofenUDP-glucuronosyltransferase 2B7enzyme
ZaltoprofenCytochrome P450 2C9enzyme
ZaltoprofenProstaglandin G/H synthase 1enzyme
AmbrisentanEndothelin B receptortarget
AmbrisentanEndothelin-1 receptortarget
AmbrisentanCytochrome P450 2C19enzyme
AmbrisentanCytochrome P450 3A4enzyme
AmbrisentanUDP-glucuronosyltransferase 1-9enzyme
AmbrisentanUDP-glucuronosyltransferase 1-3enzyme
AmbrisentanUDP-glucuronosyltransferase 2B7enzyme
AmbrisentanP-glycoprotein 1transporter
AmbrisentanSolute carrier organic anion transporter family member 1B1transporter
AmbrisentanSolute carrier organic anion transporter family member 1B3transporter
AmbrisentanCytochrome P450 3A5enzyme
TroglitazonePeroxisome proliferator-activated receptor gammatarget
TroglitazoneLong-chain-fatty-acid--CoA ligase 4target
TroglitazonePlasminogen activator inhibitor 1target
TroglitazoneEquilibrative nucleoside transporter 1target
TroglitazoneCytochrome P450 3A4enzyme
TroglitazoneCytochrome P450 2C19enzyme
TroglitazoneUDP-glucuronosyltransferase 1-1enzyme
TroglitazoneCytochrome P450 2C8enzyme
TroglitazoneBile salt export pumptransporter
TroglitazoneSolute carrier organic anion transporter family member 1B1transporter
TroglitazoneEstrogen-related receptor gammatarget
TroglitazoneSteroid hormone receptor ERR1target
TroglitazoneCytochrome P450 19A1enzyme
TroglitazoneCytochrome P450 1A1enzyme
TroglitazoneCytochrome P450 2B6enzyme
TroglitazoneCytochrome P450 2C9enzyme
TroglitazoneCytochrome P450 3A5enzyme
TroglitazoneCytochrome P450 3A7enzyme
TroglitazoneUDP-glucuronosyltransferase 1-3enzyme
TroglitazoneUDP-glucuronosyltransferase 1-4enzyme
TroglitazoneUDP-glucuronosyltransferase 1-6enzyme
TroglitazoneUDP-glucuronosyltransferase 1-7enzyme
TroglitazoneUDP-glucuronosyltransferase 1-8enzyme
TroglitazoneUDP-glucuronosyltransferase 1-9enzyme
TroglitazoneUDP-glucuronosyltransferase 1-10enzyme
TroglitazoneUDP-glucuronosyltransferase 2B7enzyme
TroglitazoneUDP-glucuronosyltransferase 2B15enzyme
TroglitazonePeroxisome proliferator-activated receptor deltatarget
TroglitazonePeroxisome proliferator-activated receptor alphatarget
TroglitazoneGlutathione S-transferase Ptarget
MorphineMu-type opioid receptortarget
MorphineDelta-type opioid receptortarget
MorphineKappa-type opioid receptortarget
MorphineP-glycoprotein 1transporter
MorphineCytochrome P450 2C8enzyme
MorphineCytochrome P450 3A4enzyme
MorphineUDP-glucuronosyltransferase 2B7enzyme
MorphineUDP-glucuronosyltransferase 1-1enzyme
MorphineUDP-glucuronosyltransferase 1-8enzyme
MorphineUDP-glucuronosyltransferase 2B15enzyme
MorphineUDP-glucuronosyltransferase 2B4enzyme
MorphineUDP-glucuronosyltransferase 1-3enzyme
MorphineLymphocyte antigen 96target
MorphineSerum albumincarrier
IndomethacinProstaglandin G/H synthase 1target
IndomethacinProstaglandin G/H synthase 2target
IndomethacinCytochrome P450 2C19enzyme
IndomethacinUDP-glucuronosyltransferase 1-9enzyme
IndomethacinPhospholipase A2, membrane associatedtarget
IndomethacinProstaglandin reductase 2target
IndomethacinLactoylglutathione lyasetarget
IndomethacinProstaglandin D2 receptor 2target
IndomethacinPeroxisome proliferator-activated receptor gammatarget
IndomethacinSerum albumincarrier
IndomethacinCanalicular multispecific organic anion transporter 2transporter
IndomethacinMultidrug resistance-associated protein 4transporter
IndomethacinMultidrug resistance-associated protein 6transporter
IndomethacinP-glycoprotein 1transporter
IndomethacinMultidrug resistance-associated protein 1transporter
IndomethacinSolute carrier organic anion transporter family member 1A2transporter
IndomethacinSolute carrier family 22 member 6transporter
IndomethacinSolute carrier family 22 member 8transporter
IndomethacinCanalicular multispecific organic anion transporter 1transporter
IndomethacinATP-binding cassette sub-family C member 11transporter
IndomethacinSolute carrier family 22 member 11transporter
IndomethacinSodium/bile acid cotransportertransporter
IndomethacinSolute carrier family 22 member 7transporter
IndomethacinCytochrome P450 2C9enzyme
IndomethacinUDP-glucuronosyltransferase 1-1enzyme
IndomethacinLiver carboxylesterase 1enzyme
IndomethacinUDP-glucuronosyltransferase 2B7enzyme
IndomethacinPeroxisome proliferator-activated receptor alphatarget
IndomethacinAldo-keto reductase family 1 member C3target
IndomethacinSolute carrier organic anion transporter family member 1B1transporter
IndomethacinBile salt export pumptransporter
IndomethacinInterferon-induced, double-stranded RNA-activated protein kinasetarget
IndomethacinHuman Cyclooxygenasestarget
Mycophenolate mofetilInosine-5'-monophosphate dehydrogenase 2target
Mycophenolate mofetilInosine-5'-monophosphate dehydrogenase 1target
Mycophenolate mofetilUDP-glucuronosyltransferase 1-1enzyme
Mycophenolate mofetilUDP-glucuronosyltransferase 1-7enzyme
Mycophenolate mofetilUDP-glucuronosyltransferase 1-6enzyme
Mycophenolate mofetilUDP-glucuronosyltransferase 1-9enzyme
Mycophenolate mofetilUDP-glucuronosyltransferase 2B7enzyme
Mycophenolate mofetilUDP-glucuronosyltransferase 1-8enzyme
Mycophenolate mofetilUDP-glucuronosyltransferase 1-10enzyme
Mycophenolate mofetilLiver carboxylesterase 1enzyme
Mycophenolate mofetilCytochrome P450 3A4enzyme
Mycophenolate mofetilCytochrome P450 3A5enzyme
Mycophenolate mofetilCytochrome P450 2C8enzyme
Mycophenolate mofetilSolute carrier organic anion transporter family member 1B1transporter
Mycophenolate mofetilSolute carrier organic anion transporter family member 1B3transporter
Mycophenolate mofetilATP-binding cassette sub-family G member 2transporter
Mycophenolate mofetilP-glycoprotein 1transporter
Mycophenolate mofetil6-pyruvoyl tetrahydrobiopterin synthasetarget
Mycophenolate mofetilCarboxylic ester hydrolaseenzyme
Mycophenolate mofetilCanalicular multispecific organic anion transporter 1transporter
EzetimibeNiemann-Pick C1-like protein 1target
EzetimibeAminopeptidase Ntarget
EzetimibeSterol O-acyltransferase 1target
EzetimibeUDP-glucuronosyltransferase 1-1enzyme
EzetimibeUDP-glucuronosyltransferase 1-3enzyme
EzetimibeP-glycoprotein 1transporter
EzetimibeCanalicular multispecific organic anion transporter 1transporter
EzetimibeSolute carrier organic anion transporter family member 1B1transporter
EzetimibeUDP-glucuronosyltransferase 2B15enzyme
EzetimibeUDP-glucuronosyltransferase 2B7enzyme
EzetimibeCytochrome P450 3A4enzyme
EzetimibeCanalicular multispecific organic anion transporter 2transporter
EzetimibeATP-binding cassette sub-family G member 2transporter
EzetimibeCytochrome P450 2C8enzyme
EzetimibeBile salt export pumptransporter
Mycophenolic acidInosine-5'-monophosphate dehydrogenase 2target
Mycophenolic acidInosine-5'-monophosphate dehydrogenase 1target
Mycophenolic acidUDP-glucuronosyltransferase 1-1enzyme
Mycophenolic acidUDP-glucuronosyltransferase 1-9enzyme
Mycophenolic acidUDP-glucuronosyltransferase 2B7enzyme
Mycophenolic acidUDP-glucuronosyltransferase 1-7enzyme
Mycophenolic acidUDP-glucuronosyltransferase 1-6enzyme
Mycophenolic acidSerum albumincarrier
Mycophenolic acidUDP-glucuronosyltransferase 1-8enzyme
Mycophenolic acidUDP-glucuronosyltransferase 1-10enzyme
Mycophenolic acidCytochrome P450 3A4enzyme
Mycophenolic acidCytochrome P450 3A5enzyme
Mycophenolic acidCytochrome P450 2C8enzyme
VadimezanUDP-glucuronosyltransferase 1-9enzyme
VadimezanUDP-glucuronosyltransferase 2B7enzyme
VadimezanCytochrome P450 1A2enzyme
EpirubicinDNA topoisomerase 2-alphatarget
EpirubicinDNAtarget
EpirubicinMultidrug resistance-associated protein 1transporter
EpirubicinUDP-glucuronosyltransferase 2B7enzyme
EpirubicinCytosolic phospholipase A2enzyme
TapentadolMu-type opioid receptortarget
TapentadolKappa-type opioid receptortarget
TapentadolDelta-type opioid receptortarget
TapentadolSodium-dependent noradrenaline transportertarget
TapentadolUDP-glucuronosyltransferase 1-9enzyme
TapentadolUDP-glucuronosyltransferase 2B7enzyme
TapentadolCytochrome P450 2D6enzyme
TapentadolCytochrome P450 2C9enzyme
TapentadolCytochrome P450 2C19enzyme
TapentadolSodium-dependent serotonin transportertarget
PitavastatinSolute carrier organic anion transporter family member 1B1transporter
PitavastatinSolute carrier organic anion transporter family member 1B3transporter
PitavastatinUDP-glucuronosyltransferase 2B7enzyme
PitavastatinUDP-glucuronosyltransferase 1-3enzyme
PitavastatinCytochrome P450 2C9enzyme
PitavastatinCytochrome P450 2C8enzyme
Pitavastatin3-hydroxy-3-methylglutaryl-coenzyme A reductasetarget
PitavastatinSolute carrier organic anion transporter family member 2B1transporter
PitavastatinSodium/bile acid cotransportertransporter
PitavastatinATP-binding cassette sub-family G member 2transporter
PitavastatinP-glycoprotein 1transporter
PitavastatinCanalicular multispecific organic anion transporter 1transporter
PitavastatinSerum albumincarrier
PitavastatinAlpha-1-acid glycoprotein 1carrier
PitavastatinBile salt export pumptransporter
PitavastatinIntegrin alpha-Ltarget
SilodosinAlpha-1D adrenergic receptortarget
SilodosinCytochrome P450 3A4enzyme
SilodosinP-glycoprotein 1transporter
SilodosinMultidrug resistance protein 3transporter
SilodosinAlpha-1A adrenergic receptortarget
SilodosinAlpha-1B adrenergic receptortarget
SilodosinUDP-glucuronosyltransferase 2B7enzyme
SilodosinAldehyde dehydrogenase, mitochondrialenzyme
SilodosinAlcohol dehydrogenase [NADP(+)]enzyme
SilodosinHERG human cardiac K+ channeltarget
ZidovudineSerum albumincarrier
ZidovudineCytochrome P450 2A6enzyme
ZidovudineCytochrome P450 2C9enzyme
ZidovudineCytochrome P450 3A4enzyme
ZidovudineReverse transcriptase/RNaseHtarget
ZidovudineSolute carrier family 22 member 2transporter
ZidovudineSolute carrier family 22 member 6transporter
ZidovudineSolute carrier family 22 member 7transporter
ZidovudineSolute carrier family 22 member 8transporter
ZidovudineSolute carrier family 22 member 11transporter
ZidovudineSodium/nucleoside cotransporter 1transporter
ZidovudineEquilibrative nucleoside transporter 2transporter
ZidovudineP-glycoprotein 1transporter
ZidovudineMultidrug resistance-associated protein 4transporter
ZidovudineMultidrug resistance-associated protein 5transporter
ZidovudineATP-binding cassette sub-family G member 2transporter
ZidovudineTelomerase reverse transcriptasetarget
ZidovudineThymidine kinase, cytosolicenzyme
ZidovudineUDP-glucuronosyltransferase 2B7enzyme
ZidovudineUDP-glucuronosyltransferase 1-1enzyme
Lovastatin3-hydroxy-3-methylglutaryl-coenzyme A reductasetarget
LovastatinCytochrome P450 3A4enzyme
LovastatinCytochrome P450 2C8enzyme
LovastatinIntegrin alpha-Ltarget
LovastatinHistone deacetylase 2target
LovastatinSerum paraoxonase/lactonase 3enzyme
LovastatinP-glycoprotein 1transporter
LovastatinSolute carrier organic anion transporter family member 1A2transporter
LovastatinSolute carrier organic anion transporter family member 1B1transporter
LovastatinUDP-glucuronosyltransferase 1-1enzyme
LovastatinUDP-glucuronosyltransferase 1-3enzyme
LovastatinUDP-glucuronosyltransferase 2B7enzyme
LovastatinCanalicular multispecific organic anion transporter 1transporter
LovastatinBile salt export pumptransporter
LovastatinSerum albumincarrier
LovastatinCytochrome P450 2C19enzyme
LovastatinSolute carrier organic anion transporter family member 2B1transporter
LovastatinSolute carrier organic anion transporter family member 1B3transporter
Simvastatin3-hydroxy-3-methylglutaryl-coenzyme A reductasetarget
SimvastatinCytochrome P450 3A4enzyme
SimvastatinCytochrome P450 2C8enzyme
SimvastatinCytochrome P450 2C9enzyme
SimvastatinCytochrome P450 3A5enzyme
SimvastatinP-glycoprotein 1transporter
SimvastatinSolute carrier organic anion transporter family member 1A2transporter
SimvastatinSolute carrier organic anion transporter family member 1B1transporter
SimvastatinCytochrome P450 2B6enzyme
SimvastatinCytochrome P450 2D6enzyme
SimvastatinUDP-glucuronosyltransferase 1-1enzyme
SimvastatinUDP-glucuronosyltransferase 1-3enzyme
SimvastatinUDP-glucuronosyltransferase 2B7enzyme
SimvastatinCanalicular multispecific organic anion transporter 1transporter
SimvastatinIntegrin alpha-Ltarget
SimvastatinBile salt export pumptransporter
SimvastatinCytochrome P450 2C19enzyme
SimvastatinSolute carrier organic anion transporter family member 2B1transporter
SimvastatinSolute carrier organic anion transporter family member 1B3transporter
SimvastatinHistone deacetylase 2target
SimvastatinCocaine esteraseenzyme
SimvastatinLiver carboxylesterase 1enzyme
OxazepamUDP-glucuronosyltransferase 2B15enzyme
OxazepamUDP-glucuronosyltransferase 2B7enzyme
OxazepamUDP-glucuronosyltransferase 1-9enzyme
OxazepamGABA(A) Receptortarget
OxazepamGABA(A) Receptor Benzodiazepine Binding Sitetarget
OxazepamSerum albumincarrier
CarbamazepineVoltage-gated sodium channel alpha subunittarget
CarbamazepineCytochrome P450 2C8enzyme
CarbamazepineCytochrome P450 2B6enzyme
CarbamazepineCytochrome P450 3A4enzyme
CarbamazepineCytochrome P450 1A2enzyme
CarbamazepineCytochrome P450 2C19enzyme
CarbamazepineCytochrome P450 2C9enzyme
CarbamazepineP-glycoprotein 1transporter
CarbamazepineCytochrome P450 3A5enzyme
CarbamazepineUDP-glucuronosyltransferase 2B7enzyme
CarbamazepineRalA-binding protein 1transporter
CarbamazepineCanalicular multispecific organic anion transporter 1transporter
CarbamazepineNeuronal acetylcholine receptor subunit alpha-4target
CarbamazepineNuclear receptor subfamily 1 group I member 2target
CarbamazepineUDP-glucuronosyltransferase 1-1enzyme
CarbamazepineUDP-glucuronosyltransferase 1-6enzyme
CarbamazepineUDP-glucuronosyltransferase 1-7enzyme
CodeineMu-type opioid receptortarget
CodeineDelta-type opioid receptortarget
CodeineKappa-type opioid receptortarget
CodeineCytochrome P450 2D6enzyme
CodeineCytochrome P450 3A4enzyme
CodeineSolute carrier family 22 member 1transporter
CodeineUDP-glucuronosyltransferase 2B7enzyme
CodeineUDP-glucuronosyltransferase 2B4enzyme
Fluvastatin3-hydroxy-3-methylglutaryl-coenzyme A reductasetarget
FluvastatinCytochrome P450 2C9enzyme
FluvastatinCytochrome P450 3A4enzyme
FluvastatinCytochrome P450 2C8enzyme
FluvastatinCytochrome P450 2D6enzyme
FluvastatinCytochrome P450 2C19enzyme
FluvastatinCytochrome P450 1A1enzyme
FluvastatinSolute carrier organic anion transporter family member 1B1transporter
FluvastatinSolute carrier organic anion transporter family member 1B3transporter
FluvastatinSolute carrier organic anion transporter family member 2B1transporter
FluvastatinSolute carrier family 15 member 1transporter
FluvastatinCytochrome P450 3A5enzyme
FluvastatinUDP-glucuronosyltransferase 1-1enzyme
FluvastatinUDP-glucuronosyltransferase 1-3enzyme
FluvastatinUDP-glucuronosyltransferase 2B7enzyme
FluvastatinCanalicular multispecific organic anion transporter 1transporter
FluvastatinCytochrome P450 2B6enzyme
FluvastatinHistone deacetylase 2target
Valproic acidHistone deacetylase 9target
Valproic acidShort/branched chain specific acyl-CoA dehydrogenase, mitochondrialtarget
Valproic acidCytochrome P450 2A6enzyme
Valproic acidCytochrome P450 2B6enzyme
Valproic acidCytochrome P450 2C9enzyme
Valproic acidSolute carrier family 22 member 5transporter
Valproic acidSolute carrier family 22 member 6transporter
Valproic acidSolute carrier family 22 member 8transporter
Valproic acidMonocarboxylate transporter 1transporter
Valproic acidSolute carrier family 22 member 7transporter
Valproic acidCytochrome P450 3A5enzyme
Valproic acidUDP-glucuronosyltransferase 1-9enzyme
Valproic acidProstaglandin G/H synthase 1enzyme
Valproic acidCytochrome P450 1A2enzyme
Valproic acidCytochrome P450 2C19enzyme
Valproic acidCytochrome P450 3A4enzyme
Valproic acidUDP-glucuronosyltransferase 1-4enzyme
Valproic acidUDP-glucuronosyltransferase 1-8enzyme
Valproic acidUDP-glucuronosyltransferase 1-10enzyme
Valproic acidUDP-glucuronosyltransferase 1-6enzyme
Valproic acidUDP-glucuronosyltransferase 1-3enzyme
Valproic acidUDP-glucuronosyltransferase 2B7enzyme
Valproic acidUDP-glucuronosyltransferase 2B15enzyme
Valproic acid2-oxoglutarate dehydrogenase, mitochondrialtarget
Valproic acidSuccinate-semialdehyde dehydrogenase, mitochondrialtarget
Valproic acidSodium channel proteintarget
Valproic acidHistone deacetylase 2target
Valproic acidPeroxisome proliferator-activated receptor alphatarget
Valproic acidPeroxisome proliferator-activated receptor deltatarget
Valproic acidPeroxisome proliferator-activated receptor gammatarget
Valproic acidSerum albumincarrier
Valproic acidUDP-glucuronosyltransferase 1-1enzyme
Valproic acidSolute carrier organic anion transporter family member 2B1transporter
Valproic acidHistone deacetylasetarget
Valproic acidCyclin-dependent kinase inhibitor 1target
Valproic acidHepatocyte growth factortarget
Valproic acidOrnithine decarboxylasetarget
Valproic acidProgrammed cell death 1 ligand 1target
DapagliflozinSodium/glucose cotransporter 2target
DapagliflozinCytochrome P450 1A1enzyme
DapagliflozinCytochrome P450 1A2enzyme
DapagliflozinCytochrome P450 2A6enzyme
DapagliflozinCytochrome P450 2C9enzyme
DapagliflozinCytochrome P450 2D6enzyme
DapagliflozinCytochrome P450 3A4enzyme
DapagliflozinUDP-glucuronosyltransferase 1-9enzyme
DapagliflozinUDP-glucuronosyltransferase 2B4enzyme
DapagliflozinUDP-glucuronosyltransferase 2B7enzyme
DapagliflozinP-glycoprotein 1transporter
EnasidenibCytochrome P450 1A2enzyme
EnasidenibCytochrome P450 2B6enzyme
EnasidenibIsocitrate dehydrogenase [NADP], mitochondrialtarget
EnasidenibCytochrome P450 2C8enzyme
EnasidenibCytochrome P450 2C9enzyme
EnasidenibCytochrome P450 2C19enzyme
EnasidenibCytochrome P450 2D6enzyme
EnasidenibCytochrome P450 3A4enzyme
EnasidenibUDP-glucuronosyltransferase 1-1enzyme
EnasidenibUDP-glucuronosyltransferase 1-3enzyme
EnasidenibUDP-glucuronosyltransferase 1-4enzyme
EnasidenibUDP-glucuronosyltransferase 1-9enzyme
EnasidenibUDP-glucuronosyltransferase 2B7enzyme
EnasidenibUDP-glucuronosyltransferase 2B15enzyme
EnasidenibP-glycoprotein 1transporter
EnasidenibATP-binding cassette sub-family G member 2transporter
EnasidenibSolute carrier family 22 member 6transporter
EnasidenibSolute carrier organic anion transporter family member 1B1transporter
EnasidenibSolute carrier family 22 member 2transporter
EnasidenibSolute carrier organic anion transporter family member 1B3transporter
EnasidenibSolute carrier family 22 member 8transporter
EnasidenibSerum albumincarrier
NalmefeneMu-type opioid receptortarget
NalmefeneKappa-type opioid receptortarget
NalmefeneDelta-type opioid receptortarget
NalmefeneUDP-glucuronosyltransferase 2B7enzyme
NalmefeneUDP-glucuronosyltransferase 1-3enzyme
NalmefeneUDP-glucuronosyltransferase 1-8enzyme
NalmefeneCytochrome P450 3A4enzyme
NalmefeneCytochrome P450 3A5enzyme
AcemetacinProstaglandin G/H synthase 1target
AcemetacinProstaglandin G/H synthase 2target
AcemetacinUDP-glucuronosyltransferase 2B7enzyme
AcemetacinMultidrug resistance-associated protein 1transporter
ErtugliflozinUDP-glucuronosyltransferase 1-9enzyme
ErtugliflozinUDP-glucuronosyltransferase 2B7enzyme
ErtugliflozinSodium/glucose cotransporter 2target
ErtugliflozinP-glycoprotein 1transporter
ErtugliflozinATP-binding cassette sub-family G member 2transporter
ErtugliflozinSerum albumincarrier
ErtugliflozinUDP-glucuronosyltransferase 1-1enzyme
ErtugliflozinUDP-glucuronosyltransferase 1-4enzyme
ArtenimolActin, cytoplasmic 2target
ArtenimolAlpha-aminoadipic semialdehyde dehydrogenasetarget
ArtenimolAnnexin A2target
ArtenimolATP synthase subunit alpha, mitochondrialtarget
ArtenimolATP synthase subunit g, mitochondrialtarget
ArtenimolATP synthase subunit O, mitochondrialtarget
ArtenimolCalpastatintarget
ArtenimolT-complex protein 1 subunit gammatarget
ArtenimolCofilin-1target
ArtenimolChloride intracellular channel protein 1target
ArtenimolCysteine and glycine-rich protein 1target
ArtenimolDihydropyrimidinase-related protein 2target
ArtenimolDesmoplakintarget
ArtenimolElongation factor 1-alpha 1target
ArtenimolAlpha-enolasetarget
ArtenimolFilamin-Atarget
ArtenimolAlpha-ketoglutarate-dependent dioxygenase FTOtarget
ArtenimolGlucose-6-phosphate 1-dehydrogenasetarget
ArtenimolGlyceraldehyde-3-phosphate dehydrogenase, testis-specifictarget
ArtenimolGlucose-6-phosphate isomerasetarget
ArtenimolHeterogeneous nuclear ribonucleoproteins A2/B1target
ArtenimolHeterogeneous nuclear ribonucleoprotein D0target
ArtenimolHeterogeneous nuclear ribonucleoprotein Ktarget
ArtenimolHeterochromatin protein 1-binding protein 3target
ArtenimolHeat shock protein beta-1target
ArtenimolRas GTPase-activating-like protein IQGAP1target
ArtenimolFar upstream element-binding protein 2target
ArtenimolL-lactate dehydrogenase A chaintarget
ArtenimolL-lactate dehydrogenase B chaintarget
ArtenimolGalectin-1target
ArtenimolMicrotubule-associated protein 4target
ArtenimolMalate dehydrogenase, cytoplasmictarget
ArtenimolPuromycin-sensitive aminopeptidasetarget
ArtenimolProfilin-1target
ArtenimolPhosphoglycerate kinase 1target
ArtenimolPyruvate kinase PKMtarget
ArtenimolPeptidyl-prolyl cis-trans isomerase Atarget
ArtenimolPeroxiredoxin-1target
Artenimol60S ribosomal protein L10target
Artenimol60S ribosomal protein L14target
Artenimol60S ribosomal protein L18target
Artenimol60S ribosomal protein L23atarget
Artenimol60S ribosomal protein L35target
Artenimol60S ribosomal protein L4target
Artenimol40S ribosomal protein S13target
Artenimol40S ribosomal protein S17target
Artenimol40S ribosomal protein S18target
Artenimol40S ribosomal protein S19target
Artenimol40S ribosomal protein S28target
Artenimol40S ribosomal protein S5target
Artenimol40S ribosomal protein S6target
Artenimol40S ribosomal protein S8target
Artenimol40S ribosomal protein S9target
ArtenimolSplicing factor 1target
ArtenimolSplicing factor, proline- and glutamine-richtarget
ArtenimolSmall nuclear ribonucleoprotein Sm D2target
ArtenimolSignal recognition particle 14 kDa proteintarget
ArtenimolSerine/arginine-rich splicing factor 4target
ArtenimolTransgelintarget
ArtenimolTransgelin-2target
ArtenimolTriosephosphate isomerasetarget
ArtenimolTropomyosin alpha-1 chaintarget
ArtenimolTubulin alpha-1A chaintarget
ArtenimolVimentintarget
ArtenimolZyxintarget
ArtenimolHeat shock cognate 71 kDa proteintarget
ArtenimolTubulin beta-6 chaintarget
ArtenimolTubulin beta-4A chaintarget
ArtenimolTubulin beta chaintarget
ArtenimolFructose-bisphosphate aldolase Atarget
ArtenimolGlyceraldehyde-3-phosphate dehydrogenasetarget
ArtenimolCytochrome ctarget
ArtenimolPhosphoglycerate mutase 1target
ArtenimolMyosin-9target
ArtenimolProtein disulfide-isomerasetarget
ArtenimolProbable ATP-dependent RNA helicase DDX5target
ArtenimolSerine hydroxymethyltransferase, mitochondrialtarget
ArtenimolSpliceosome RNA helicase DDX39Btarget
ArtenimolNucleophosmintarget
ArtenimolTranslationally-controlled tumor protein homologtarget
ArtenimolP-type Ca2+-transporting ATPasetarget
ArtenimolOrnithine aminotransferasetarget
ArtenimolElongation factor 1-alphatarget
ArtenimolMultidrug resistance proteintarget
ArtenimolElongation factor 2target
ArtenimolActin-1target
ArtenimolGlyceraldehyde-3-phosphate dehydrogenasetarget
ArtenimolFructose-bisphosphate aldolasetarget
ArtenimolCell division cycle protein 48 homologue,putativetarget
ArtenimolHeat shock protein 90target
ArtenimolEukaryotic initiation factor 4Atarget
ArtenimolPyruvate kinasetarget
ArtenimolL-lactate dehydrogenasetarget
ArtenimolProtein disulfide-isomerasetarget
ArtenimolThioredoxin-related protein, putativetarget
ArtenimolSpermidine synthasetarget
ArtenimolProbable ATP-dependent 6-phosphofructokinasetarget
ArtenimolGlutamate dehydrogenasetarget
ArtenimolEndoplasmin homolog, putativetarget
ArtenimolHypoxanthine-guanine-xanthine phosphoribosyltransferasetarget
ArtenimolEnolasetarget
Artenimol40S ribosomal protein S3target
ArtenimolNon-SERCA-type Ca2+-transporting P-ATPasetarget
ArtenimolTubulin alpha chaintarget
ArtenimolKnob-associated histidine-rich proteintarget
ArtenimolS-adenosylmethionine synthasetarget
ArtenimolV-type H(+)-translocating pyrophosphatase, putativetarget
Artenimol60S ribosomal protein L4target
ArtenimolPhosphoethanolamine N-methyltransferasetarget
Artenimol40S ribosomal protein S3atarget
ArtenimolConserved Plasmodium membrane proteintarget
Artenimol60S ribosomal protein L3target
ArtenimolHigh molecular weight rhoptry protein 2target
ArtenimolSerine repeat antigen 5target
Artenimol40S ribosomal protein S19target
ArtenimolGlycophorin-binding proteintarget
ArtenimolCalcium-transporting ATPasetarget
ArtenimolV-type proton ATPase catalytic subunit Atarget
Artenimol60S ribosomal protein L2target
ArtenimolAcyl-CoA synthetasetarget
ArtenimolPlasmepsin IVtarget
ArtenimolPlasmepsin-1target
ArtenimolChloroquine resistance transportertarget
Artenimol14-3-3 proteintarget
ArtenimolIsoleucine--tRNA ligase, putativetarget
ArtenimolPlasmodium exported proteintarget
ArtenimolTubulin beta chaintarget
Artenimol60S ribosomal protein L27target
ArtenimolSec62, putativetarget
ArtenimolAutophagy-related protein 18, putativetarget
ArtenimolMature parasite-infected erythrocyte surface antigentarget
ArtenimolImportin-7, putativetarget
ArtenimolImportin subunit alphatarget
ArtenimolPeptidyl-prolyl cis-trans isomerasetarget
ArtenimolDnaJ protein, putativetarget
ArtenimolMerozoite surface protein 1target
ArtenimolGlutamate--tRNA ligasetarget
ArtenimolT-complex protein 1 subunit etatarget
ArtenimolPlasmepsin-2target
ArtenimolChaperone, putativetarget
ArtenimolRhoptry neck protein 3target
Artenimol40S ribosomal protein S5, putativetarget
ArtenimolSkeleton-binding protein 1target
ArtenimolPurine nucleotide phosphorylase, putativetarget
ArtenimolAdenosylhomocysteinasetarget
ArtenimolAdenosine deaminasetarget
ArtenimolMethionine--tRNA ligasetarget
ArtenimolCarbamoyl phosphate synthetasetarget
ArtenimolAspartate carbamoyltransferasetarget
ArtenimolSignal recognition particle receptor, beta subunittarget
ArtenimolParasite-infected erythrocyte surface proteintarget
ArtenimolCoatomer alpha subunit, putativetarget
ArtenimolHexokinasetarget
ArtenimolProteasome subunit alpha typetarget
ArtenimolHaloacid dehalogenase-like hydrolasetarget
ArtenimolInsulinase, putativetarget
Artenimol40S ribosomal protein S21target
ArtenimolUbiquitin-conjugating enzyme E2target
ArtenimolEukaryotic translation initiation factor 3 subunit Ctarget
Artenimol60S ribosomal protein L24, putativetarget
Artenimol60S ribosomal protein L23target
Artenimol60S ribosomal protein L17, putativetarget
ArtenimolHAP proteintarget
ArtenimolHeat shock protein 110, putativetarget
Artenimol60S ribosomal protein L10, putativetarget
ArtenimolLysophospholipase, putativetarget
ArtenimolPolyadenylate-binding proteintarget
ArtenimolUbiquitin-60S ribosomal protein L40target
ArtenimolPhosphoribosylpyrophosphate synthetasetarget
ArtenimolThioredoxin peroxidase 1target
ArtenimolProtein transport protein SEC31target
ArtenimolDipeptidyl aminopeptidase 1target
ArtenimolRing-infected erythrocyte surface antigentarget
ArtenimolATP-dependent RNA helicase UAP56target
ArtenimolCalcium-dependent protein kinase 4target
ArtenimolGTP-binding nuclear protein Rantarget
ArtenimolNucleoside transporter 2target
ArtenimolAnamorsin homologtarget
ArtenimolGlutamine synthetase, putativetarget
Artenimol60S ribosomal protein L30e, putativetarget
ArtenimolCasein kinase 2, alpha subunittarget
ArtenimolThreonine--tRNA ligasetarget
ArtenimolcAMP-dependent protein kinase regulatory subunittarget
ArtenimolElongation factor 1-gamma, putativetarget
ArtenimolThioredoxin-like proteintarget
Artenimol60S ribosomal protein L21target
Artenimol60S ribosomal protein L14, putativetarget
ArtenimolInner membrane complex sub-compartment protein 3target
ArtenimolHSP40, subfamily A, putativetarget
ArtenimolPyridoxal 5'-phosphate synthase subunit Pdx1target
ArtenimolUDP-glucuronosyltransferase 1-9enzyme
ArtenimolUDP-glucuronosyltransferase 2B7enzyme
ArtenimolSerum albumintarget
ArtenimolCytochrome P450 2D6enzyme
ArtenimolCytochrome P450 2C19enzyme
LabetalolAlpha-1 adrenergic receptorstarget
LabetalolBeta-1 adrenergic receptortarget
LabetalolBeta-2 adrenergic receptortarget
LabetalolCytochrome P450 2D6enzyme
LabetalolCytochrome P450 2C19enzyme
LabetalolSerum albumincarrier
Labetalolalpha1-acid glycoproteincarrier
LabetalolATP-binding cassette sub-family B member 5transporter
LabetalolUDP-glucuronosyltransferase 1-1enzyme
LabetalolUDP-glucuronosyltransferase 2B7enzyme
LabetalolUDP-glucuronosyltransferase 1-9enzyme
TamoxifenEstrogen receptor alphatarget
TamoxifenEstrogen receptor betatarget
TamoxifenCytochrome P450 2C9enzyme
TamoxifenCytochrome P450 3A4enzyme
TamoxifenCytochrome P450 2D6enzyme
TamoxifenCytochrome P450 2C8enzyme
TamoxifenCytochrome P450 2B6enzyme
TamoxifenLiver carboxylesterase 1enzyme
TamoxifenCytochrome P450 3A5enzyme
TamoxifenCytochrome P450 1A1enzyme
TamoxifenCytochrome P450 1B1enzyme
TamoxifenCytochrome P450 2C19enzyme
TamoxifenDimethylaniline monooxygenase [N-oxide-forming] 1enzyme
TamoxifenDimethylaniline monooxygenase [N-oxide-forming] 3enzyme
TamoxifenCytochrome P450 3A7enzyme
TamoxifenP-glycoprotein 1transporter
TamoxifenATP-binding cassette sub-family G member 2transporter
TamoxifenCytochrome P450 19A1enzyme
TamoxifenCytochrome P450 2A6enzyme
TamoxifenCytochrome P450 2E1enzyme
TamoxifenUDP-glucuronosyltransferase 1-10enzyme
TamoxifenSulfotransferase 1A1enzyme
TamoxifenCanalicular multispecific organic anion transporter 1transporter
Tamoxifen3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerasetarget
TamoxifenProtein kinase Ctarget
TamoxifenAndrogen receptortarget
TamoxifenPotassium voltage-gated channel subfamily H member 2target
TamoxifenNuclear receptor subfamily 1 group I member 2target
TamoxifenEstrogen-related receptor gammatarget
TamoxifenSex hormone-binding globulintarget
TamoxifenBile salt export pumptransporter
TamoxifenThyroxine-binding globulincarrier
TamoxifenBile salt sulfotransferaseenzyme
TamoxifenCytochrome P450 1A2enzyme
TamoxifenUDP-glucuronosyltransferase 2B7enzyme
TamoxifenUDP-glucuronosyltransferase 2B17enzyme
TamoxifenEstrogen sulfotransferaseenzyme
TamoxifenATP-binding cassette sub-family A member 1transporter
TamoxifenMitogen-activated protein kinase 8target
TamoxifenSerum albumincarrier
CarvedilolAlpha-1A adrenergic receptortarget
CarvedilolBeta-1 adrenergic receptortarget
CarvedilolNADH dehydrogenase [ubiquinone] 1 subunit C2target
CarvedilolBeta-2 adrenergic receptortarget
CarvedilolVascular endothelial growth factor Atarget
CarvedilolNatriuretic peptides Btarget
CarvedilolGap junction alpha-1 proteintarget
CarvedilolPotassium voltage-gated channel subfamily H member 2target
CarvedilolVascular cell adhesion protein 1target
CarvedilolCytochrome P450 2C9enzyme
CarvedilolCytochrome P450 2D6enzyme
CarvedilolXanthine dehydrogenase/oxidaseenzyme
CarvedilolP-glycoprotein 1transporter
CarvedilolCytochrome P450 1A2enzyme
CarvedilolCytochrome P450 3A4enzyme
CarvedilolCytochrome P450 1A1enzyme
CarvedilolCytochrome P450 2E1enzyme
CarvedilolAlpha-1D adrenergic receptortarget
CarvedilolAlpha-1B adrenergic receptortarget
CarvedilolAlpha-2C adrenergic receptortarget
CarvedilolAlpha-2B adrenergic receptortarget
CarvedilolAlpha-2A adrenergic receptortarget
CarvedilolE-selectintarget
CarvedilolHypoxia-inducible factor 1-alphatarget
CarvedilolInward rectifier potassium channel 4target
CarvedilolUDP-glucuronosyltransferase 1-1enzyme
CarvedilolSerum albumincarrier
CarvedilolUDP-glucuronosyltransferase 2B4enzyme
CarvedilolUDP-glucuronosyltransferase 2B7enzyme
CarvedilolInward rectifier potassium channel 2target
CarvedilolAlpha-1 adrenergic receptorstarget
KetorolacProstaglandin G/H synthase 1target
KetorolacProstaglandin G/H synthase 2target
KetorolacUDP-glucuronosyltransferase 2B7enzyme
KetorolacCytochrome P450 2C8enzyme
KetorolacCytochrome P450 2C9enzyme
Dabigatran etexilateProthrombintarget
Dabigatran etexilateP-glycoprotein 1transporter
Dabigatran etexilateLiver carboxylesterase 1enzyme
Dabigatran etexilateCocaine esteraseenzyme
Dabigatran etexilateUDP-glucuronosyltransferase 1-9enzyme
Dabigatran etexilateUDP-glucuronosyltransferase 2B7enzyme
Dabigatran etexilateUDP-glucuronosyltransferase 2B15enzyme
Dabigatran etexilateRibosyldihydronicotinamide dehydrogenase [quinone]enzyme
Dabigatran etexilateSerum albumincarrier
DexibuprofenProstaglandin G/H synthase 1target
DexibuprofenProstaglandin G/H synthase 2target
DexibuprofenApoptosis regulator Bcl-2target
DexibuprofenThrombomodulintarget
DexibuprofenTissue-type plasminogen activatortarget
DexibuprofenFatty acid-binding protein, intestinaltarget
DexibuprofenPeroxisome proliferator-activated receptor gammatarget
DexibuprofenCystic fibrosis transmembrane conductance regulatortarget
DexibuprofenCytochrome P450 2C9enzyme
DexibuprofenSerum albumincarrier
DexibuprofenMultidrug resistance-associated protein 4transporter
DexibuprofenMultidrug resistance-associated protein 1transporter
DexibuprofenSolute carrier organic anion transporter family member 1A2transporter
DexibuprofenSolute carrier family 22 member 6transporter
DexibuprofenSolute carrier family 22 member 8transporter
DexibuprofenSolute carrier family 22 member 11transporter
DexibuprofenSolute carrier organic anion transporter family member 2B1transporter
DexibuprofenP-glycoprotein 1transporter
DexibuprofenUDP-glucuronosyltransferase 1-1enzyme
DexibuprofenUDP-glucuronosyltransferase 1-3enzyme
DexibuprofenUDP-glucuronosyltransferase 1-9enzyme
DexibuprofenUDP-glucuronosyltransferase 2B4enzyme
DexibuprofenUDP-glucuronosyltransferase 2B7enzyme
DexibuprofenCytochrome P450 2C8enzyme
DexibuprofenCytochrome P450 2C19enzyme
DexibuprofenSolute carrier family 15 member 1target
DexibuprofenPeroxisome proliferator-activated receptor alphatarget
DexibuprofenPlatelet glycoprotein Ib alpha chaintarget
DexibuprofenProtein S100-A7target
DexibuprofenAlpha-methylacyl-CoA racemaseenzyme
GemfibrozilPeroxisome proliferator-activated receptor alphatarget
GemfibrozilCytochrome P450 2C9enzyme
GemfibrozilCytochrome P450 2C8enzyme
GemfibrozilCytochrome P450 1A2enzyme
GemfibrozilCytochrome P450 2C19enzyme
GemfibrozilUDP-glucuronosyltransferase 1-1enzyme
GemfibrozilCytochrome P450 3A4enzyme
GemfibrozilUDP-glucuronosyltransferase 1-3enzyme
GemfibrozilSolute carrier organic anion transporter family member 1B1target
GemfibrozilUDP-glucuronosyltransferase 2B7enzyme
GemfibrozilUDP-glucuronosyltransferase 1-9enzyme
GemfibrozilUDP-glucuronosyltransferase 2B4enzyme
GemfibrozilUDP-glucuronosyltransferase 2B17enzyme
GemfibrozilSerum albumincarrier
GemfibrozilSolute carrier family 22 member 8target
GemfibrozilSolute carrier organic anion transporter family member 2B1target
GemfibrozilSolute carrier organic anion transporter family member 1B3target
AnastrozoleCytochrome P450 19A1target
AnastrozoleP-glycoprotein 1transporter
AnastrozoleCytochrome P450 3A4enzyme
AnastrozoleCytochrome P450 3A5enzyme
AnastrozoleCytochrome P450 2C8enzyme
AnastrozoleUDP-glucuronosyltransferase 1-4enzyme
AnastrozoleUDP-glucuronosyltransferase 1-3enzyme
AnastrozoleUDP-glucuronosyltransferase 2B7enzyme
AnastrozoleCytochrome P450 1A2enzyme
AnastrozoleCytochrome P450 2C9enzyme
LoxoprofenProstaglandin G/H synthase 2target
LoxoprofenProstaglandin G/H synthase 1target
LoxoprofenCarbonyl reductase [NADPH] 1enzyme
LoxoprofenCytochrome P450 3A Subfamilyenzyme
LoxoprofenUDP-glucuronosyltransferase 2B7enzyme
CenobamateUDP-glucuronosyltransferase 2B7enzyme
CenobamateUDP-glucuronosyltransferase 2B4enzyme
CenobamateCytochrome P450 2E1enzyme
CenobamateCytochrome P450 2A6enzyme
CenobamateCytochrome P450 2B6enzyme
CenobamateCytochrome P450 2C19enzyme
CenobamateCytochrome P450 3A4enzyme
CenobamateCytochrome P450 3A5enzyme
CenobamateSerum albumincarrier
CenobamateCytochrome P450 2C8enzyme
FormoterolBeta-2 adrenergic receptortarget
FormoterolBeta-1 adrenergic receptortarget
FormoterolBeta-3 adrenergic receptortarget
FormoterolCytochrome P450 2D6enzyme
FormoterolCytochrome P450 2C19enzyme
FormoterolCytochrome P450 2C9enzyme
FormoterolCytochrome P450 2A6enzyme
FormoterolUDP-glucuronosyltransferase 1A1enzyme
FormoterolUDP-glucuronosyltransferase 1-8enzyme
FormoterolUDP-glucuronosyltransferase 1-9enzyme
FormoterolUDP-glucuronosyltransferase 2B7enzyme
FormoterolUDP-glucuronosyltransferase 2B15enzyme
FormoterolSolute carrier family 22 member 1transporter
FormoterolSolute carrier family 22 member 4transporter
FormoterolSolute carrier family 22 member 5transporter
FormoterolSolute carrier family 22 member 3transporter
FormoterolSerum albumincarrier
LetrozoleCytochrome P450 19A1target
LetrozoleCytochrome P450 3A4enzyme
LetrozoleCytochrome P450 2A6enzyme
LetrozoleCytochrome P450 19A1enzyme
LetrozoleCytochrome P450 2C19enzyme
LetrozoleUDP-glucuronosyltransferase 2B7enzyme
LetrozoleSerum albumincarrier
LetrozoleP-glycoprotein 1transporter
EthinylestradiolEstrogen receptor alphatarget
EthinylestradiolNuclear receptor subfamily 1 group I member 2target
EthinylestradiolCytochrome P450 3A4enzyme
EthinylestradiolCytochrome P450 2C8enzyme
EthinylestradiolBile salt export pumptransporter
EthinylestradiolSodium/bile acid cotransportertransporter
EthinylestradiolCanalicular multispecific organic anion transporter 1transporter
EthinylestradiolP-glycoprotein 1transporter
EthinylestradiolUDP-glucuronosyltransferase 1-1enzyme
EthinylestradiolCytochrome P450 2C19enzyme
EthinylestradiolUDP-glucuronosyltransferase 1-4enzyme
EthinylestradiolUDP-glucuronosyltransferase 1-9enzyme
EthinylestradiolCytochrome P450 2C9enzyme
EthinylestradiolCytochrome P450 1A2enzyme
EthinylestradiolEstrogen sulfotransferaseenzyme
EthinylestradiolSulfotransferase 1A3/1A4enzyme
EthinylestradiolCytochrome P450 3A5enzyme
EthinylestradiolUDP-glucuronosyltransferase 2B7enzyme
EthinylestradiolUDP-glucuronosyltransferase 1-3enzyme
EthinylestradiolCatechol O-methyltransferaseenzyme
EthinylestradiolSolute carrier organic anion transporter family member 1A2transporter
EthinylestradiolSerum albumincarrier
EthinylestradiolSex hormone-binding globulincarrier
OsilodrostatCytochrome P450 11B1, mitochondrialtarget
OsilodrostatCytochrome P450 11B2, mitochondrialtarget
OsilodrostatCytochrome P450 3A4enzyme
OsilodrostatCytochrome P450 2B6enzyme
OsilodrostatCytochrome P450 2D6enzyme
OsilodrostatUDP-glucuronosyltransferase 1-4enzyme
OsilodrostatUDP-glucuronosyltransferase 2B7enzyme
OsilodrostatUDP-glucuronosyltransferase 2B10enzyme
OsilodrostatCytochrome P450 3A5enzyme
OsilodrostatCytochrome P450 1A2enzyme
OsilodrostatCytochrome P450 2C19enzyme
OsilodrostatCytochrome P450 2E1enzyme
OsilodrostatUDP-glucuronosyltransferase 1A1enzyme
OsilodrostatSolute carrier organic anion transporter family member 1B1transporter
OsilodrostatSolute carrier family 22 member 1transporter
OsilodrostatSolute carrier family 22 member 2transporter
OsilodrostatSolute carrier family 22 member 6transporter
OsilodrostatSolute carrier family 22 member 8transporter
OsilodrostatMultidrug and toxin extrusion protein 1transporter
Bempedoic acidATP-citrate synthasetarget
Bempedoic acidVery long-chain acyl-CoA synthetaseenzyme
Bempedoic acidSolute carrier organic anion transporter family member 1B1transporter
Bempedoic acidCanalicular multispecific organic anion transporter 2transporter
Bempedoic acidSolute carrier organic anion transporter family member 1B3transporter
Bempedoic acidUDP-glucuronosyltransferase 2B7enzyme
Bempedoic acidNUAK family SNF1-like kinase 2enzyme
EmpagliflozinSodium/glucose cotransporter 2target
EmpagliflozinUDP-glucuronosyltransferase 2B7enzyme
EmpagliflozinUDP-glucuronosyltransferase 1-3enzyme
EmpagliflozinUDP-glucuronosyltransferase 1-8enzyme
EmpagliflozinUDP-glucuronosyltransferase 1-9enzyme
EmpagliflozinP-glycoprotein 1transporter
EmpagliflozinATP-binding cassette sub-family G member 2transporter
EmpagliflozinSolute carrier family 22 member 8transporter
EmpagliflozinSolute carrier organic anion transporter family member 1B1transporter
EmpagliflozinSolute carrier organic anion transporter family member 1B3transporter
ArtesunateMalaria protein EXP-1target
ArtesunateCytochrome P450 2A6enzyme
ArtesunateUDP-glucuronosyltransferase 2B7enzyme
ArtesunateUDP-glucuronosyltransferase 1-9enzyme
ArtesunateATP-binding cassette sub-family G member 2transporter
ArtesunateP-glycoprotein 1transporter
ArtesunateSolute carrier organic anion transporter family member 1B1transporter
ArtesunateSolute carrier family 22 member 8transporter
ArtesunateSerum albumincarrier
DextromethorphanSigma non-opioid intracellular receptor 1target
DextromethorphanNeuronal acetylcholine receptor subunit alpha-2target
DextromethorphanSodium-dependent serotonin transportertarget
DextromethorphanGlutamate receptor ionotropic, NMDA 3Atarget
DextromethorphanCytochrome P450 2D6enzyme
DextromethorphanCytochrome P450 3A4enzyme
DextromethorphanCytochrome P450 3A7enzyme
DextromethorphanCytochrome P450 2C9enzyme
DextromethorphanCytochrome P450 2B6enzyme
DextromethorphanCytochrome P450 2C19enzyme
DextromethorphanMembrane-associated progesterone receptor component 1target
DextromethorphanNeuronal acetylcholine receptor subunit alpha-3target
DextromethorphanNeuronal acetylcholine receptor subunit alpha-4target
DextromethorphanNeuronal acetylcholine receptor subunit beta-4target
DextromethorphanNeuronal acetylcholine receptor subunit beta-2target
DextromethorphanNeuronal acetylcholine receptor subunit alpha-7target
DextromethorphanMu-type opioid receptortarget
DextromethorphanDelta-type opioid receptortarget
DextromethorphanKappa-type opioid receptortarget
DextromethorphanNADPH oxidasetarget
DextromethorphanSodium-dependent noradrenaline transportertarget
DextromethorphanUDP-glucuronosyltransferase 2B4enzyme
DextromethorphanUDP-glucuronosyltransferase 2B7enzyme
DextromethorphanUDP-glucuronosyltransferase 2B15enzyme
DextromethorphanUDP-glucuronosyltransferase 2B17enzyme
FebuxostatSerum albumincarrier
FebuxostatXanthine dehydrogenase/oxidasetarget
FebuxostatUDP-glucuronosyltransferase 1-1enzyme
FebuxostatUDP-glucuronosyltransferase 1-3enzyme
FebuxostatUDP-glucuronosyltransferase 1-9enzyme
FebuxostatUDP-glucuronosyltransferase 2B7enzyme
FebuxostatCytochrome P450 1A2enzyme
FebuxostatCytochrome P450 2C8enzyme
FebuxostatCytochrome P450 2C9enzyme
FebuxostatATP-binding cassette sub-family G member 2transporter
PonesimodSphingosine 1-phosphate receptor 1target
PonesimodCytochrome P450 2J2enzyme
PonesimodCytochrome P450 3A4enzyme
PonesimodCytochrome P450 3A5enzyme
PonesimodCytochrome P450 4F3enzyme
PonesimodCytochrome P450 4F12enzyme
PonesimodUDP-glucuronosyltransferase 1-1enzyme
PonesimodUDP-glucuronosyltransferase 2B7enzyme
MirabegronCytochrome P450 3A4enzyme
MirabegronCytochrome P450 2D6enzyme
MirabegronP-glycoprotein 1transporter
MirabegronSolute carrier organic anion transporter family member 1A2transporter
MirabegronSerum albumincarrier
MirabegronAlpha-1-acid glycoprotein 1carrier
MirabegronCholinesteraseenzyme
MirabegronBeta-3 adrenergic receptortarget
MirabegronUDP-glucuronosyltransferase 2B7enzyme
MirabegronUDP-glucuronosyltransferase 1-3enzyme
MirabegronUDP-glucuronosyltransferase 1-8enzyme
MirabegronSolute carrier family 22 member 1transporter
MirabegronSolute carrier family 22 member 2transporter
MirabegronSolute carrier family 22 member 3transporter
MirabegronBeta-1 adrenergic receptortarget
EstetrolSerum albumincarrier
EstetrolCytochrome P450 3A4enzyme
EstetrolUDP-glucuronosyltransferase 2B7enzyme
EstetrolEstrogen receptor alphatarget
EstetrolEstrogen receptor betatarget
EstetrolAlpha-1-acid glycoprotein 1carrier
Nandrolone decanoateAndrogen receptortarget
Nandrolone decanoateCytochrome P450 19A1enzyme
Nandrolone decanoateAmine oxidase [flavin-containing] Benzyme
Nandrolone decanoateAmine oxidase [flavin-containing] Aenzyme
Nandrolone decanoateProto-oncogene c-Fostarget
Nandrolone decanoate5-hydroxytryptamine 2 receptortarget
Nandrolone decanoate5-hydroxytryptamine receptor 1Btarget
Nandrolone decanoateInsulin-like growth factor 1 receptortarget
Nandrolone decanoateDopamine receptortarget
Nandrolone decanoateUDP-glucuronosyltransferase 2B7enzyme
Nandrolone decanoateUDP-glucuronosyltransferase 1-4enzyme
Nandrolone decanoateUDP-glucuronosyltransferase 2B4enzyme
Nandrolone decanoateUDP-glucuronosyltransferase 1-3enzyme
Nandrolone decanoateUDP-glucuronosyltransferase 1-1enzyme
Nandrolone decanoateUDP-glucuronosyltransferase 1-10enzyme
Nandrolone decanoateSex hormone-binding globulincarrier
AsciminibCytochrome P450 3A4enzyme
AsciminibUDP-glucuronosyltransferase 2B7enzyme
AsciminibUDP-glucuronosyltransferase 2B17enzyme
AsciminibTyrosine-protein kinase ABL1target
AsciminibATP-binding cassette sub-family G member 2transporter
AsciminibUDP-glucuronosyltransferase 1-1enzyme
AsciminibCytochrome P450 2C19enzyme
AsciminibP-glycoprotein 1transporter
AsciminibSolute carrier organic anion transporter family member 1B1transporter
AsciminibSolute carrier organic anion transporter family member 1B3transporter
AsciminibSolute carrier family 22 member 1transporter
AsciminibCytochrome P450 2C9enzyme
SotagliflozinUDP-glucuronosyltransferase 1-9enzyme
SotagliflozinUDP-glucuronosyltransferase 1-1enzyme
SotagliflozinUDP-glucuronosyltransferase 2B7enzyme
SotagliflozinCytochrome P450 3A4enzyme
SotagliflozinSodium/glucose cotransporter 2target
SotagliflozinSodium/glucose cotransporter 1target
SotagliflozinCytochrome P450 2D6enzyme
SotagliflozinP-glycoprotein 1transporter
SotagliflozinATP-binding cassette sub-family G member 2transporter
SotagliflozinSolute carrier organic anion transporter family member 1B1transporter
SotagliflozinSolute carrier organic anion transporter family member 1B3transporter
SotagliflozinCanalicular multispecific organic anion transporter 1transporter
CannabidiolCytochrome P450 2C9enzyme
CannabidiolCytochrome P450 2C19enzyme
CannabidiolCytochrome P450 2D6enzyme
CannabidiolCytochrome P450 3A4enzyme
CannabidiolCannabinoid receptor 1target
CannabidiolCannabinoid receptor 2target
CannabidiolG-protein coupled receptor 12target
CannabidiolGlycine receptor subunit alpha-1target
CannabidiolGlycine receptor (alpha-1/beta)target
CannabidiolGlycine receptor subunit alpha-3target
CannabidiolN-arachidonyl glycine receptortarget
CannabidiolG-protein coupled receptor 55target
Cannabidiol5-hydroxytryptamine receptor 1Atarget
Cannabidiol5-hydroxytryptamine receptor 2Atarget
CannabidiolNeuronal acetylcholine receptor subunit alpha-7target
CannabidiolDelta-type opioid receptortarget
CannabidiolMu-type opioid receptortarget
CannabidiolPeroxisome proliferator-activated receptor gammatarget
CannabidiolCytochrome P450 3A5enzyme
CannabidiolSerotonin N-acetyltransferaseenzyme
CannabidiolCytochrome P450 1A1enzyme
CannabidiolFatty-acid amide hydrolase 1enzyme
CannabidiolArachidonate 5-lipoxygenaseenzyme
CannabidiolArachidonate 15-lipoxygenaseenzyme
CannabidiolQuinone oxidoreductaseenzyme
CannabidiolMultidrug resistance-associated protein 1transporter
CannabidiolATP-binding cassette sub-family G member 2transporter
CannabidiolEquilibrative nucleoside transporter 1transporter
CannabidiolTransient receptor potential cation channel subfamily V member 1target
CannabidiolVoltage-dependent T-type calcium channel subunit alpha-1Gtarget
CannabidiolVoltage-dependent T-type calcium channel subunit alpha-1Htarget
CannabidiolVoltage-dependent T-type calcium channel subunit alpha-1Itarget
CannabidiolTransient receptor potential cation channel subfamily A member 1target
CannabidiolTransient receptor potential cation channel subfamily M member 8target
CannabidiolTransient receptor potential cation channel subfamily V member 2target
CannabidiolTransient receptor potential cation channel subfamily V member 3target
CannabidiolTransient receptor potential cation channel subfamily V member 4target
CannabidiolVoltage-dependent anion-selective channel protein 1target
Cannabidiol5-hydroxytryptamine receptor 3Atarget
CannabidiolAdenosine receptor A1target
CannabidiolProstaglandin G/H synthase 1target
CannabidiolProstaglandin G/H synthase 2target
CannabidiolAcetyl-CoA acetyltransferase, mitochondrialtarget
CannabidiolSteroid 17-alpha-hydroxylase/17,20 lyasetarget
Cannabidiol3-hydroxy-3-methylglutaryl-coenzyme A reductasetarget
CannabidiolGlutathione reductase, mitochondrialtarget
CannabidiolGlutathione peroxidase 1target
CannabidiolIndoleamine 2,3-dioxygenase 1target
CannabidiolCytochrome P450 1B1target
CannabidiolNAD(P)H dehydrogenase [quinone] 1target
CannabidiolCatalasetarget
CannabidiolCytochrome P450 3A5target
CannabidiolCytochrome P450 2D6target
CannabidiolSuperoxide dismutase [Cu-Zn]target
CannabidiolCytochrome P450 1A2target
CannabidiolCytochrome P450 3A7target
CannabidiolSerotonin N-acetyltransferasetarget
CannabidiolN-acylethanolamine-hydrolyzing acid amidasetarget
CannabidiolCytochrome P450 1A2enzyme
CannabidiolCytochrome P450 1B1enzyme
CannabidiolCytochrome P450 2A6enzyme
CannabidiolCytochrome P450 2B6enzyme
CannabidiolCytochrome P450 2C8enzyme
CannabidiolCytochrome P450 2E1enzyme
CannabidiolCytochrome P450 3A7enzyme
CannabidiolUDP-glucuronosyltransferase 1-7enzyme
CannabidiolUDP-glucuronosyltransferase 1-9enzyme
CannabidiolUDP-glucuronosyltransferase 2B7enzyme
CannabidiolUDP-glucuronosyltransferase 2B17enzyme
CannabidiolP-glycoprotein 1transporter
CannabidiolCytochrome P450 2J2enzyme
CannabidiolLiver carboxylesterase 1enzyme
CannabinolCytochrome P450 3A4enzyme
CannabinolCytochrome P450 2C19enzyme
CannabinolCytochrome P450 1A1enzyme
CannabinolCytochrome P450 1A2enzyme
CannabinolCytochrome P450 1B1enzyme
CannabinolCytochrome P450 2A6enzyme
CannabinolCytochrome P450 2B6enzyme
CannabinolCytochrome P450 2C9enzyme
CannabinolCytochrome P450 2D6enzyme
CannabinolCytochrome P450 3A5enzyme
CannabinolCytochrome P450 3A7enzyme
CannabinolUDP-glucuronosyltransferase 1-7enzyme
CannabinolUDP-glucuronosyltransferase 1-8enzyme
CannabinolUDP-glucuronosyltransferase 1-9enzyme
CannabinolUDP-glucuronosyltransferase 1-10enzyme
CannabinolUDP-glucuronosyltransferase 2B7enzyme
CannabinolP-glycoprotein 1transporter
CannabinolATP-binding cassette sub-family G member 2transporter
CannabinolMultidrug resistance-associated protein 1transporter
CannabinolCytochrome P450 2E1enzyme
CannabinolCytochrome P450 2J2enzyme
CannabinolLiver carboxylesterase 1enzyme
Medical CannabisCannabinoid receptor 1target
Medical CannabisCannabinoid receptor 2target
Medical CannabisCytochrome P450 2C9enzyme
Medical CannabisCytochrome P450 2C19enzyme
Medical CannabisCytochrome P450 2D6enzyme
Medical CannabisCytochrome P450 3A4enzyme
Medical CannabisG-protein coupled receptor 12target
Medical CannabisGlycine receptor subunit alpha-1target
Medical CannabisGlycine receptor (alpha-1/beta)target
Medical CannabisGlycine receptor subunit alpha-3target
Medical CannabisN-arachidonyl glycine receptortarget
Medical CannabisG-protein coupled receptor 55target
Medical Cannabis5-hydroxytryptamine receptor 1Atarget
Medical Cannabis5-hydroxytryptamine receptor 2Atarget
Medical CannabisNeuronal acetylcholine receptor subunit alpha-7target
Medical CannabisDelta-type opioid receptortarget
Medical CannabisMu-type opioid receptortarget
Medical CannabisPeroxisome proliferator-activated receptor gammatarget
Medical CannabisCytochrome P450 3A5enzyme
Medical CannabisCytochrome P450 3A7enzyme
Medical CannabisCytochrome P450 1A1enzyme
Medical CannabisCytochrome P450 1A2enzyme
Medical CannabisCytochrome P450 1B1enzyme
Medical CannabisArachidonate 5-lipoxygenaseenzyme
Medical CannabisArachidonate 15-lipoxygenaseenzyme
Medical CannabisSuperoxide dismutase [Cu-Zn]enzyme
Medical CannabisMultidrug resistance-associated protein 1transporter
Medical CannabisATP-binding cassette sub-family G member 2transporter
Medical CannabisEquilibrative nucleoside transporter 1transporter
Medical CannabisTransient receptor potential cation channel subfamily V member 1target
Medical CannabisVoltage-dependent T-type calcium channel subunit alpha-1Gtarget
Medical CannabisVoltage-dependent T-type calcium channel subunit alpha-1Htarget
Medical CannabisVoltage-dependent T-type calcium channel subunit alpha-1Itarget
Medical CannabisTransient receptor potential cation channel subfamily A member 1target
Medical CannabisTransient receptor potential cation channel subfamily M member 8target
Medical CannabisTransient receptor potential cation channel subfamily V member 2target
Medical CannabisTransient receptor potential cation channel subfamily V member 3target
Medical CannabisTransient receptor potential cation channel subfamily V member 4target
Medical CannabisVoltage-dependent anion-selective channel protein 1target
Medical CannabisN-acyl-phosphatidylethanolamine-hydrolyzing phospholipase Dtarget
Medical CannabisN-acylethanolamine-hydrolyzing acid amidasetarget
Medical CannabisSerotonin N-acetyltransferasetarget
Medical CannabisPhospholipase A2target
Medical CannabisSuperoxide dismutase [Cu-Zn]target
Medical CannabisFatty-acid amide hydrolase 1target
Medical CannabisCatalasetarget
Medical CannabisQuinone oxidoreductasetarget
Medical CannabisSphingomyelin phosphodiesterasetarget
Medical CannabisGlutathione peroxidase 1target
Medical CannabisGlutathione reductase, mitochondrialtarget
Medical Cannabis3-hydroxy-3-methylglutaryl-coenzyme A reductasetarget
Medical CannabisIndoleamine 2,3-dioxygenase 1target
Medical CannabisProstaglandin G/H synthase 1target
Medical CannabisProstaglandin G/H synthase 2target
Medical CannabisSteroid 17-alpha-hydroxylase/17,20 lyasetarget
Medical CannabisAcetyl-CoA acetyltransferase, mitochondrialtarget
Medical CannabisCytochrome P450 2A6enzyme
Medical CannabisCytochrome P450 2B6enzyme
Medical CannabisCytochrome P450 2C8enzyme
Medical CannabisCytochrome P450 2E1enzyme
Medical CannabisCytochrome P450 2J2enzyme
Medical CannabisUDP-glucuronosyltransferase 1-7enzyme
Medical CannabisUDP-glucuronosyltransferase 1-8enzyme
Medical CannabisUDP-glucuronosyltransferase 1-9enzyme
Medical CannabisUDP-glucuronosyltransferase 1-10enzyme
Medical CannabisUDP-glucuronosyltransferase 2B17enzyme
Medical CannabisLiver carboxylesterase 1enzyme
Medical CannabisP-glycoprotein 1transporter
Medical CannabisUDP-glucuronosyltransferase 2B7enzyme
CobimetinibDual specificity mitogen-activated protein kinase kinase 1target
CobimetinibCytochrome P450 3A4enzyme
CobimetinibSolute carrier organic anion transporter family member 1B1transporter
CobimetinibSolute carrier organic anion transporter family member 1B3transporter
CobimetinibATP-binding cassette sub-family G member 2transporter
CobimetinibP-glycoprotein 1transporter
CobimetinibUDP-glucuronosyltransferase 2B7enzyme
CobimetinibCytochrome P450 2D6enzyme
CobimetinibCytochrome P450 3A5enzyme
CobimetinibAlpha-1-acid glycoprotein 1carrier
EdaravoneSolute carrier family 22 member 6transporter
EdaravoneSolute carrier family 22 member 8transporter
EdaravoneUDP-glucuronosyltransferase 1-1enzyme
EdaravoneUDP-glucuronosyltransferase 1-6enzyme
EdaravoneUDP-glucuronosyltransferase 1-7enzyme
EdaravoneUDP-glucuronosyltransferase 1-8enzyme
EdaravoneUDP-glucuronosyltransferase 1-9enzyme
EdaravoneUDP-glucuronosyltransferase 1-10enzyme
EdaravoneUDP-glucuronosyltransferase 2B7enzyme
EdaravoneUDP-glucuronosyltransferase 2B17enzyme
EdaravoneSulfotransferaseenzyme
EdaravoneSerum albumincarrier
MidazolamCytochrome P450 3A4enzyme
MidazolamCytochrome P450 3A5enzyme
MidazolamUDP-glucuronosyltransferase 1-4enzyme
MidazolamCytochrome P450 3A7enzyme
MidazolamGABA(A) Receptortarget
MidazolamGABA(A) Receptor Benzodiazepine Binding Sitetarget
MidazolamP-glycoprotein 1transporter
MidazolamSerum albumincarrier
MidazolamAlpha-1-acid glycoprotein 1carrier
MidazolamAdenosine receptor A2atarget
MidazolamExcitatory amino acid transporter 2transporter
MidazolamUDP-glucuronosyltransferase 2B7enzyme
MidazolamUDP-glucuronosyltransferase 2B4enzyme
TretinoinRetinoic acid receptor gammatarget
TretinoinRetinoic acid receptor RXR-betatarget
TretinoinRetinal dehydrogenase 1target
TretinoinRetinoic acid-induced protein 3target
TretinoinRetinoic acid receptor RXR-gammatarget
TretinoinRetinal dehydrogenase 2target
TretinoinRetinoic acid receptor responder protein 1target
TretinoinCytochrome P450 2C8enzyme
TretinoinCellular retinoic acid-binding protein 1transporter
TretinoinCellular retinoic acid-binding protein 2transporter
TretinoinCytochrome P450 2B6enzyme
TretinoinCytochrome P450 3A4enzyme
TretinoinCytochrome P450 3A5enzyme
TretinoinCytochrome P450 2A6enzyme
TretinoinCytochrome P450 3A7enzyme
TretinoinCytochrome P450 2C18enzyme
TretinoinCytochrome P450 2C9enzyme
TretinoinCytochrome P450 4A11enzyme
TretinoinCytochrome P450 1A1enzyme
TretinoinRetinoic acid receptor alphatarget
TretinoinRetinoic acid receptor betatarget
TretinoinLipocalin-1target
TretinoinOdorant-binding protein 2atarget
TretinoinRetinol-binding protein 4target
TretinoinSerum albumincarrier
Tretinoin[Pyruvate dehydrogenase [lipoamide]] kinase isozyme 4, mitochondrialtarget
TretinoinRetinoic acid receptor RXR-alphatarget
TretinoinCarcinoembryonic antigentarget
TretinoinUDP-glucuronosyltransferase 2B7enzyme
TretinoinCytochrome P450 2E1enzyme
TretinoinCytochrome P450 26A1enzyme
TretinoinCellular retinoic acid-binding protein 1target
VadadustatEgl nine homolog 2target
VadadustatEgl nine homolog 3target
VadadustatEgl nine homolog 1target
VadadustatHypoxia-inducible factor 1-alphatarget
VadadustatEndothelial PAS domain-containing protein 1target
VadadustatUDP-glucuronosyltransferase 1-1enzyme
VadadustatUDP-glucuronosyltransferase 1-7enzyme
VadadustatUDP-glucuronosyltransferase 1-8enzyme
VadadustatUDP-glucuronosyltransferase 1-9enzyme
VadadustatUDP-glucuronosyltransferase 2B7enzyme
VadadustatCytochrome P450 2B6enzyme
VadadustatCytochrome P450 2C8enzyme
VadadustatCytochrome P450 3A4enzyme
VadadustatATP-binding cassette sub-family G member 2transporter
VadadustatSolute carrier family 22 member 8transporter
VadadustatSolute carrier family 22 member 6transporter
VadadustatSerum albumincarrier
VadadustatCytochrome P450 2C9enzyme
VamoroloneGlucocorticoid receptortarget
VamoroloneCytochrome P450 3A4enzyme
VamoroloneCytochrome P450 3A5enzyme
VamoroloneCytochrome P450 2C8enzyme
VamoroloneUDP-glucuronosyltransferase 1-3enzyme
VamoroloneUDP-glucuronosyltransferase 2B7enzyme
VamoroloneUDP-glucuronosyltransferase 2B17enzyme
VamoroloneMineralocorticoid receptortarget
CapivasertibCytochrome P450 3A4enzyme
CapivasertibUDP-glucuronosyltransferase 2B7enzyme
CapivasertibRAC-alpha serine/threonine-protein kinasetarget
CapivasertibRAC-beta serine/threonine-protein kinasetarget
CapivasertibRAC-gamma serine/threonine-protein kinasetarget
CapivasertibATP-binding cassette sub-family G member 2transporter
CapivasertibSolute carrier organic anion transporter family member 1B1transporter
CapivasertibSolute carrier organic anion transporter family member 1B3transporter
CapivasertibSolute carrier family 22 member 8transporter
CapivasertibMultidrug and toxin extrusion protein 1transporter
CapivasertibMultidrug and toxin extrusion protein 2transporter
CapivasertibSolute carrier family 22 member 2transporter