| Serotonin (5-HT) 1F Receptor Agonists | Agents acting as agonists at serotonin (5-HT) receptor 1F. | 1 | 7 | Details |
| Serotonin (5HT1) receptor agonists, sumatriptan and derivatives | Not Available | 0 | 0 | Details |
| Serotonin 1b Receptor Agonists | Not Available | 7 | 60 | Details |
| Serotonin 1d Receptor Agonists | Not Available | 7 | 60 | Details |
| Serotonin 2c Receptor Agonists | Not Available | 1 | 9 | Details |
| Serotonin 3 Receptor Antagonists | Not Available | 5 | 35 | Details |
| Serotonin 4 Receptor Agonists | Not Available | 2 | 15 | Details |
| Serotonin 4 Receptor Antagonists | Not Available | 0 | 0 | Details |
| Serotonin 5-HT1 Receptor Agonists | Endogenous compounds and drugs that specifically stimulate SEROTONIN 5-HT1 RECEPTORS. I... more | 27 | 367 | Details |
| Serotonin 5-HT1 Receptor Antagonists | Drugs that bind to but do not activate SEROTONIN 5-HT1 RECEPTORS, thereby blocking the ... more | 45 | 633 | Details |
| Serotonin 5-HT1A Receptor Antagonists | Entities that are capable of exerting an antagonistic effect on 5-HT1A receptors. | 35 | 483 | Details |
| Serotonin 5-HT1D Receptor Antagonists | Entities that are capable of exerting an antagonistic effect on 5-HT1D receptors. | 9 | 187 | Details |
| Serotonin 5-HT2 Receptor Agonists | Endogenous compounds and drugs that specifically stimulate SEROTONIN 5-HT2 RECEPTORS. I... more | 17 | 248 | Details |
| Serotonin 5-HT2 Receptor Antagonists | Drugs that bind to but do not activate SEROTONIN 5-HT2 RECEPTORS, thereby blocking the ... more | 103 | 1305 | Details |
| Serotonin 5-HT2A Receptor Agonists | Not Available | 0 | 0 | Details |
| Serotonin 5-HT2A Receptor Antagonists | Entities that are capable of exerting an antagonistic effect on 5-HT2A receptors. | 85 | 1159 | Details |
| Serotonin 5-HT2B Receptor Agonists | Not Available | 0 | 0 | Details |
| Serotonin 5-HT2C Receptor Agonists | Not Available | 2 | 12 | Details |
| Serotonin 5-HT2C Receptor Antagonists | Entities that are capable of exerting an antagonistic effect on 5-HT2C receptors. | 56 | 954 | Details |
| Serotonin 5-HT3 Receptor Antagonists | Drugs that bind to but do not activate SEROTONIN 5-HT3 RECEPTORS, thereby blocking the ... more | 9 | 76 | Details |
| Serotonin 5-HT4 Receptor Agonists | Endogenous compounds and drugs that specifically stimulate SEROTONIN 5-HT4 RECEPTORS. | 5 | 9 | Details |
| Serotonin Agents | Drugs used for their effects on serotonergic systems. Among these are drugs that affect... more | 244 | 2302 | Details |
| Serotonin and Noradrenaline Reuptake Inhibitors | Drugs that selectively block or suppress the plasma membrane transport of SEROTONIN and... more | 7 | 66 | Details |
| Serotonin antagonist and reuptake inhibitors (SARIs) | A class of drugs that are mainly used as antidepressants, but are also anxiolytics and ... more | 3 | 36 | Details |
| Serotonin Modulators | Not Available | 79 | 968 | Details |