Did you mean ethyl estradiol norelgestromin?
Displaying drugs 1 - 25 of 95 in total
Estradiol
Estradiol is a naturally occurring hormone circulating endogenously in females. It is commercially available in several hormone therapy products for managing conditions associated with reduced estrogen, such as vulvovaginal atrophy and hot flashes. Some available forms of estradiol include oral tablets, injections, vaginal rings, transdermal patches, sprays, gels, and creams.[L11485,L11488,L11491,...
Approved
Investigational
Vet approved
Matched Synonyms: … Estradiol ... 17β-estradiol ... cis-Estradiol …
Matched Name: … Estradiol …
Matched Description: … Ethinyl estradiol is different from estradiol due to its higher biovailability and increased resistance ... Estradiol is a naturally occurring hormone circulating endogenously in females. ... Some available forms of estradiol include oral tablets, injections, vaginal rings, transdermal patches …
Matched Mixtures name: … Estradiol / Norethindrone Acetate ... Estradiol and Progesterone ... Estradiol and Norethindrone Acetate …
Matched Salts name: … Estradiol hemihydrate …
Matched Categories: … estradiol ... Estradiol Congeners ... Estradiol, agonists ... estradiol, combinations ... dienogest and estradiol …
Matched Products: … Estradiol ... Estradiol Vaginal ... PMS-estradiol …
Matched Name: … Estradiol …
Matched Description: … Ethinyl estradiol is different from estradiol due to its higher biovailability and increased resistance ... Estradiol is a naturally occurring hormone circulating endogenously in females. ... Some available forms of estradiol include oral tablets, injections, vaginal rings, transdermal patches …
Matched Mixtures name: … Estradiol / Norethindrone Acetate ... Estradiol and Progesterone ... Estradiol and Norethindrone Acetate …
Matched Salts name: … Estradiol hemihydrate …
Matched Categories: … estradiol ... Estradiol Congeners ... Estradiol, agonists ... estradiol, combinations ... dienogest and estradiol …
Matched Products: … Estradiol ... Estradiol Vaginal ... PMS-estradiol …
Ethinylestradiol
Ethinylestradiol was first synthesized in 1938 by Hans Herloff Inhoffen and Walter Hohlweg at Schering. It was developed in an effort to create an estrogen with greater oral bioavailability. These properties were achieved by the substitution of an ethinyl group at carbon 17 of estradiol. Ethinylestradiol soon replaced mestranol in...
Approved
Matched Synonyms: … Ethinyl estradiol ... 17-ethinyl-3,17-estradiol ... 17alpha-Ethinyl estradiol …
Matched Description: … [A191107] These properties were achieved by the substitution of an ethinyl group at carbon 17 of [estradiol …
Matched Mixtures name: … Norelgestromin and Ethinyl Estradiol ... Norelgestromin and Ethinyl Estradiol ... Norelgestromin and Ethinly Estradiol …
Matched Categories: … Estradiol Congeners ... norelgestromin and ethinylestradiol …
Matched Description: … [A191107] These properties were achieved by the substitution of an ethinyl group at carbon 17 of [estradiol …
Matched Mixtures name: … Norelgestromin and Ethinyl Estradiol ... Norelgestromin and Ethinyl Estradiol ... Norelgestromin and Ethinly Estradiol …
Matched Categories: … Estradiol Congeners ... norelgestromin and ethinylestradiol …
Estramustine
A nitrogen mustard linked to estradiol, usually as phosphate; used to treat prostatic neoplasms; also has radiation protective properties.
Approved
Investigational
Matched Synonyms: … 17β-Estradiol 3-(bis(2-chloroethyl)carbamate) ... Estradiol 3-(N,N-bis(2-chloroethyl)carbamate) …
Matched Description: … A nitrogen mustard linked to estradiol, usually as phosphate; used to treat prostatic neoplasms; also …
Matched Categories: … Estradiol Congeners …
Matched Description: … A nitrogen mustard linked to estradiol, usually as phosphate; used to treat prostatic neoplasms; also …
Matched Categories: … Estradiol Congeners …
Norgestrel
Norgestrel is synthetic steroidal progestin that is used in combination with ethinyl estradiol for oral contraception. Norgestrel is composed of a racemic mixture of two stereoisomers, dextronorgestrel and levonorgestrel. However, only the levorotary enantiomer (levonorgestrel) is biologically active.
Approved
Matched Description: … Norgestrel is synthetic steroidal progestin that is used in combination with ethinyl estradiol for oral …
Matched Mixtures name: … Norgestrel/Ethinyl Estradiol …
Matched Mixtures name: … Norgestrel/Ethinyl Estradiol …
Dienogest
Dienogest is an orally-active semisynthetic progestogen which also possesses the properties of 17α-hydroxyprogesterone. It is a derivative of 19-nortestosterone and has antiandrogenic properties. It is primarily used as a contraceptive in combination with ethinylestradiol, or in other combination form pills approved in United States and Europe however it is not...
Approved
Matched Mixtures name: … Estradiol Valerate and Estradiol Valerate/Dienogest ... Estradiol Valerate and Estradiol Valerate/Dienogest …
Matched Categories: … dienogest and estradiol …
Matched Categories: … dienogest and estradiol …
Estramustine phosphate
A nitrogen mustard linked to estradiol, usually as phosphate; used to treat prostatic neoplasms; also has radiation protective properties.
Approved
Investigational
Matched Description: … A nitrogen mustard linked to estradiol, usually as phosphate; used to treat prostatic neoplasms; also …
Nafarelin
Nafarelin is a potent synthetic agonist of gonadotropin-releasing hormone with 3-(2-naphthyl)-D-alanine substitution at residue 6. Nafarelin has been used in the treatments of central precocious puberty and endometriosis.
Approved
Buserelin
Buserelin is a synthetic peptide analog of the luteinizing hormone-releasing hormone (LHRH) agonist, which stimulates the pituitary gland's gonadotrophin-releasing hormone receptor (GnRHR). It is used in prostate cancer treatment.
Approved
Investigational
Nandrolone phenpropionate
C18 steroid with androgenic and anabolic properties. It is generally prepared from alkyl ethers of estradiol to resemble testosterone but less one carbon at the 19 position. It is a schedule III drug in the U.S.
Approved
Illicit
Investigational
Matched Description: … It is generally prepared from alkyl ethers of estradiol to resemble testosterone but less one carbon …
Linzagolix
Linzagolix is a non-peptide, selective antagonist of the gonadotropin-releasing hormone (GnRH) receptor. It has been studied for the treatment of estrogen-dependent conditions such as uterine fibroids and endometriosis.[A253642,A253647] It is similar to other GnRH receptor antagonists like cetrorelix, relugolix, and elagolix.
Uterine fibroids occur in >70% of women of reproductive...
Approved
Testosterone propionate
Testosterone propionate is a slower-releasing anabolic steroid with a short half-life. It is a synthetic androstane steroid derivative of testosterone in the form of 17β propionate ester of testosterone. Testosterone propionate was developed initially by Watson labs, and FDA approved on February 5, 1974. Currently, this drug has been discontinued...
Approved
Investigational
Vet approved
Withdrawn
Exemestane
Exemestane is an oral steroidal aromatase inhibitor used in the adjuvant treatment of hormonally-responsive (also called hormone-receptor-positive, estrogen-responsive) breast cancer in postmenopausal women. It irreversibly binds to the active site of the enzyme resulting in permanent inhibition.
Approved
Investigational
Estriol
A hydroxylated metabolite of estradiol or estrone that has a hydroxyl group at C3-beta, 16-alpha, and 17-beta position. Estriol is a major urinary estrogen. During pregnancy, large amount of estriol is produced by the placenta. Isomers with inversion of the hydroxyl group or groups are called epiestriol. Though estriol is...
Approved
Investigational
Vet approved
Matched Description: … A hydroxylated metabolite of estradiol or estrone that has a hydroxyl group at C3-beta, 16-alpha, and …
Matched Categories: … Estradiol Congeners …
Matched Categories: … Estradiol Congeners …
Triptorelin
Triptorelin is a synthetic decapeptide agonist analog of luteinizing hormone releasing hormone (LHRH). Possessing greater potency than endogenous LHRH, triptorelin reversibly represses gonadotropin secretion. After chronic, continuous administration, this agent effects sustained decreases in LH and FSH production and testicular and ovarian steroidogenesis. Serum testosterone concentrations may fall to levels...
Approved
Vet approved
Tamoxifen
Tamoxifen is a non-steroidal antiestrogen used to treat estrogen receptor positive breast cancers as well as prevent the incidence of breast cancer in high risk populations.[A1025,L7799,L7802] Tamoxifen is used alone or as an adjuvant in these treatments.[L7799,L7802] Tamoxifen may no longer be the preferred treatment for these types of cancers...
Approved
Testosterone cypionate
Testosterone cypionate is a synthetic derivative of testosterone in the form of an oil-soluble 17 (beta)-cyclopentylpropionate ester. Its benefit compared to other testosterone derivatives is the slow rate of release after injection and longer half-life. It was developed by the company Pharmacia and Upjohn and FDA approved on July 25,...
Approved
Elacestrant
Elacestrant is a non-steroidal small molecule and an estrogen receptor (ER) antagonist.[A256838,L44918] In January 2023, it was approved by the FDA for the treatment of ER-positive, HER2-negative, ESR1-mutated advanced or metastatic breast cancer.[L44918,L44948] It received a similar approval in the EU in September 2023. Elacestrant binds to estrogen receptor-alpha (ERα)...
Approved
Investigational
Enzacamene
Commonly known as 4-methylbenzylidene-camphor (4-MBC), enzacamene is a camphor derivative and an organic chemical UV-B filter. It is used in cosmetic products such as sunscreen to provide skin protection against UV rays. While its effects on the human reproductive system as an endocrine disruptor are being investigated, its use in...
Approved
Ganirelix
Ganirelix is a synthetic decapeptide and a competitive gonadotropin-releasing hormone (GnRH) antagonist. Derived from endogenous GnRH, ganirelix has amino acid substitutions. Ganirelix is indicated for controlled ovarian hyperstimulation in assisted reproduction techniques. The first case of pregnancy achieved after the use of ganirelix in an assisted reproduction program was reported...
Approved
Elagolix
Elagolix has been used in trials studying the basic science and treatment of Endometriosis, Folliculogenesis, Uterine Fibroids, Heavy Uterine Bleeding, and Heavy Menstrual Bleeding. As of 24 July 2018, however, the U.S. Food and Drug Administration (FDA) approved AbbVie's elagolix under the brand name Orilissa as the first and only...
Approved
Investigational
Matched Categories: … elagolix, estradiol and norethisterone …
Follitropin
Follitropin is a human follicle stimulating hormone (FSH) preparation of recombinant DNA origin, which consists of two non-covalently linked, non-identical glycoproteins designated as the alpha- and beta- subunits. The alpha- and beta- subunits have 92 and 111 amino acids. The alpha subunit is glycosylated at Asn 51 and Asn 78...
Approved
Matched Description: … pregnancy rate and the beta form tending towards a lower pregnancy rate, but with significantly higher estradiol …
Estradiol valerate
Estradiol Valerate (also known as E2V) is a pro-drug ester of DB00783, a naturally occurring hormone that circulates endogenously within the human body. Estradiol is the most potent form of all mammalian estrogenic steroids and acts as the major female sex hormone. As a pro-drug of estradiol, estradiol acetate therefore...
Approved
Investigational
Vet approved
Matched Synonyms: … Estradiol valerate …
Matched Name: … Estradiol valerate …
Matched Description: … As a pro-drug of estradiol, estradiol acetate therefore has the same downstream effects within the body ... Following absorption, the esters are cleaved, resulting in the release of endogenous estradiol, or 17β-estradiol ... with Estradiol Cypionate) through improved lipophilicity. …
Matched Mixtures name: … Estradiol Valerate and Estradiol Valerate/Dienogest ... Estradiol Valerate and Estradiol Valerate/Dienogest ... Estradiol Valerate and Estradiol Valerate/Dienogest …
Matched Categories: … Estradiol Congeners ... Estradiol, agonists …
Matched Products: … Estradiol Valerate ... Estradiol valerate ... ESTRADIOL FEM JENAPHARM …
Matched Name: … Estradiol valerate …
Matched Description: … As a pro-drug of estradiol, estradiol acetate therefore has the same downstream effects within the body ... Following absorption, the esters are cleaved, resulting in the release of endogenous estradiol, or 17β-estradiol ... with Estradiol Cypionate) through improved lipophilicity. …
Matched Mixtures name: … Estradiol Valerate and Estradiol Valerate/Dienogest ... Estradiol Valerate and Estradiol Valerate/Dienogest ... Estradiol Valerate and Estradiol Valerate/Dienogest …
Matched Categories: … Estradiol Congeners ... Estradiol, agonists …
Matched Products: … Estradiol Valerate ... Estradiol valerate ... ESTRADIOL FEM JENAPHARM …
Estradiol cypionate
Estradiol Cypionate is a pro-drug ester of DB00783, a naturally occurring hormone that circulates endogenously within the human body. Estradiol is the most potent form of all mammalian estrogenic steroids and acts as the major female sex hormone. As a pro-drug of estradiol, estradiol cypionate therefore has the same downstream...
Approved
Investigational
Vet approved
Matched Synonyms: … Estradiol cypionate …
Matched Name: … Estradiol cypionate …
Matched Description: … As a pro-drug of estradiol, estradiol cypionate therefore has the same downstream effects within the ... Estradiol cypionate is commercially available as Depo-Estradiol, an intramuscular depot injection used ... Following absorption, the esters are cleaved, resulting in the release of endogenous estradiol, or 17β-estradiol …
Matched Categories: … Estradiol Congeners …
Matched Products: … Depo-Estradiol …
Matched Name: … Estradiol cypionate …
Matched Description: … As a pro-drug of estradiol, estradiol cypionate therefore has the same downstream effects within the ... Estradiol cypionate is commercially available as Depo-Estradiol, an intramuscular depot injection used ... Following absorption, the esters are cleaved, resulting in the release of endogenous estradiol, or 17β-estradiol …
Matched Categories: … Estradiol Congeners …
Matched Products: … Depo-Estradiol …
Estradiol acetate
Estradiol acetate is a pro-drug ester of DB00783, a naturally occurring hormone that circulates endogenously within the human body. Estradiol is the most potent form of all mammalian estrogenic steroids and acts as the major female sex hormone. As a pro-drug of estradiol, estradiol acetate therefore has the same downstream...
Approved
Investigational
Vet approved
Matched Synonyms: … Estradiol acetate ... Estradiol 3-acetate ... Estradiol-3-acetate …
Matched Name: … Estradiol acetate …
Matched Description: … As a pro-drug of estradiol, estradiol acetate therefore has the same downstream effects within the body ... Following absorption, the esters are cleaved, resulting in the release of endogenous estradiol, or 17β-estradiol ... with Estradiol Cypionate) through improved lipophilicity. …
Matched Name: … Estradiol acetate …
Matched Description: … As a pro-drug of estradiol, estradiol acetate therefore has the same downstream effects within the body ... Following absorption, the esters are cleaved, resulting in the release of endogenous estradiol, or 17β-estradiol ... with Estradiol Cypionate) through improved lipophilicity. …
Estradiol benzoate
Estradiol Benzoate is a pro-drug ester of DB00783, a naturally occurring hormone that circulates endogenously within the human body. Estradiol is the most potent form of all mammalian estrogenic steroids and acts as the major female sex hormone. As a pro-drug of estradiol, estradiol benzoate therefore has the same downstream...
Approved
Investigational
Vet approved
Matched Synonyms: … Estradiol benzoate ... benzoato de estradiol …
Matched Name: … Estradiol benzoate …
Matched Description: … As a pro-drug of estradiol, estradiol benzoate therefore has the same downstream effects within the body ... Following absorption, the esters are cleaved, resulting in the release of endogenous estradiol, or 17β-estradiol ... with Estradiol Cypionate) through improved lipophilicity. …
Matched Categories: … Estradiol Congeners …
Matched Name: … Estradiol benzoate …
Matched Description: … As a pro-drug of estradiol, estradiol benzoate therefore has the same downstream effects within the body ... Following absorption, the esters are cleaved, resulting in the release of endogenous estradiol, or 17β-estradiol ... with Estradiol Cypionate) through improved lipophilicity. …
Matched Categories: … Estradiol Congeners …
Displaying drugs 1 - 25 of 95 in total