| DB00588 | Fluticasone propionate | approved | unknown | inhibitor | Details |
| DB01103 | Quinacrine | investigational | yes | inhibitor | Details |
| DB06311 | Darapladib | investigational | unknown | | Details |
| DB04552 | Niflumic acid | experimental | unknown | | Details |
| DB00411 | Carbamoylcholine | approved | unknown | inducer | Details |
| DB04827 | Urethane | approved, withdrawn | unknown | substrate | Details |
| DB00578 | Carbenicillin | approved, investigational | unknown | inhibitor | Details |
| DB05029 | Lancovutide | investigational | unknown | inhibitor | Details |
| DB00445 | Epirubicin | approved | unknown | inhibitor | Details |
| DB01083 | Orlistat | approved, investigational | unknown | inhibitor | Details |
| DB00086 | Streptokinase | approved, investigational | unknown | inducer | Details |
| DB04786 | Suramin | investigational | unknown | inhibitor | Details |
| DB00041 | Aldesleukin | approved | unknown | inducer | Details |
| DB00721 | Procaine | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB13867 | Fluticasone | approved, experimental | unknown | inhibitor | Details |