| DB00910 | Paricalcitol | approved, investigational | unknown | substrate | Details |
| DB00831 | Trifluoperazine | approved, investigational | unknown | substrate | Details |
| DB00363 | Clozapine | approved | no | substrate | Details |
| DB00197 | Troglitazone | approved, investigational, withdrawn | unknown | substrate | Details |
| DB04953 | Ezogabine | approved, investigational | unknown | substrate | Details |
| DB06216 | Asenapine | approved | unknown | substrate | Details |
| DB00683 | Midazolam | approved, illicit | no | substrate | Details |
| DB00313 | Valproic acid | approved, investigational | unknown | substrate | Details |
| DB06401 | Bazedoxifene | approved, investigational | unknown | substrate | Details |
| DB09262 | Imidafenacin | investigational | no | substrate | Details |
| DB13874 | Enasidenib | approved, investigational | unknown | substrate | Details |
| DB11827 | Ertugliflozin | approved, investigational | no | inhibitor | Details |
| DB12020 | Tecovirimat | approved, investigational | unknown | substrate | Details |
| DB00334 | Olanzapine | approved, investigational | no | substrate | Details |
| DB12978 | Pexidartinib | approved, investigational | unknown | substrate | Details |
| DB00924 | Cyclobenzaprine | approved | unknown | substrate | Details |
| DB01217 | Anastrozole | approved, investigational | unknown | substrate | Details |
| DB00321 | Amitriptyline | approved | unknown | substrate | Details |
| DB06077 | Lumateperone | approved, investigational | no | substrate | Details |
| DB00252 | Phenytoin | approved, vet_approved | no | substrate | Details |
| DB00977 | Ethinylestradiol | approved | unknown | substrate | Details |
| DB09054 | Idelalisib | approved | unknown | substrateinhibitor | Details |
| DB11837 | Osilodrostat | approved, investigational | unknown | substrate | Details |
| DB09241 | Methylene blue | approved, investigational | unknown | inhibitor | Details |
| DB00920 | Ketotifen | approved | unknown | substrate | Details |
| DB00434 | Cyproheptadine | approved | unknown | substrate | Details |
| DB08804 | Nandrolone decanoate | approved, illicit | unknown | substrate | Details |
| DB00349 | Clobazam | approved, illicit | no | inhibitor | Details |