| DB01181 | Ifosfamide | approved | unknown | substrate | Details |
| DB01424 | Aminophenazone | approved, withdrawn | unknown | substrate | Details |
| DB00682 | Warfarin | approved | unknown | substrate | Details |
| DB07670 | N,4-Dimethyl-N-(1-phenyl-1H-pyrazol-5-yl)benzenesulfonamide | experimental | unknown | | Details |
| DB00921 | Buprenorphine | approved, illicit, investigational, vet_approved | unknown | substrate | Details |
| DB00349 | Clobazam | approved, illicit | unknown | substrate | Details |
| DB01559 | Clotiazepam | approved, illicit | unknown | substrate | Details |
| DB00531 | Cyclophosphamide | approved, investigational | unknown | substrate | Details |
| DB00250 | Dapsone | approved, investigational | unknown | substrate | Details |
| DB00829 | Diazepam | approved, illicit, investigational, vet_approved | unknown | substrate | Details |
| DB00586 | Diclofenac | approved, vet_approved | unknown | substrate | Details |
| DB00458 | Imipramine | approved | unknown | substrate | Details |
| DB00448 | Lansoprazole | approved, investigational | unknown | substrate | Details |
| DB00333 | Methadone | approved | unknown | substrate | Details |
| DB00338 | Omeprazole | approved, investigational, vet_approved | unknown | substrate | Details |
| DB00850 | Perphenazine | approved | unknown | substrate | Details |
| DB01435 | Antipyrine | approved, investigational | unknown | substrate | Details |
| DB00818 | Propofol | approved, investigational, vet_approved | unknown | substrate | Details |
| DB01124 | Tolbutamide | approved, investigational | unknown | substrate | Details |
| DB00755 | Tretinoin | approved, investigational, nutraceutical | unknown | substrate | Details |
| DB01174 | Phenobarbital | approved, investigational | unknown | substrate | Details |
| DB09166 | Etizolam | experimental | unknown | substrate | Details |
| DB08496 | (R)-warfarin | experimental | unknown | substrate | Details |
| DB14055 | (S)-Warfarin | experimental, investigational | unknown | substrate | Details |
| DB11757 | Istradefylline | approved, investigational | unknown | substrate | Details |
| DB00661 | Verapamil | approved | unknown | substrate | Details |
| DB00252 | Phenytoin | approved, vet_approved | yes | substrate | Details |
| DB00986 | Glycopyrronium | approved, investigational, vet_approved | unknown | substrate | Details |
| DB01183 | Naloxone | approved, vet_approved | unknown | substrate | Details |