| DB00197 | Troglitazone | approved, investigational, withdrawn | unknown | substrate | Details |
| DB00295 | Morphine | approved, investigational | no | substrate | Details |
| DB00973 | Ezetimibe | approved | unknown | substrate | Details |
| DB06695 | Dabigatran etexilate | approved | unknown | substrate | Details |
| DB00316 | Acetaminophen | approved | unknown | substrate | Details |
| DB00842 | Oxazepam | approved | unknown | substrate | Details |
| DB00186 | Lorazepam | approved | unknown | substrate | Details |
| DB00313 | Valproic acid | approved, investigational | unknown | substrate | Details |
| DB11943 | Delafloxacin | approved, investigational | no | substrate | Details |
| DB13874 | Enasidenib | approved, investigational | unknown | substrate | Details |
| DB09288 | Propacetamol | experimental | no | substrate | Details |
| DB00455 | Loratadine | approved, investigational | unknown | | Details |
| DB06077 | Lumateperone | approved, investigational | no | substrate | Details |
| DB00983 | Formoterol | approved, investigational | unknown | substrate | Details |
| DB00783 | Estradiol | approved, investigational, vet_approved | unknown | inducer | Details |
| DB00514 | Dextromethorphan | approved | unknown | substrate | Details |
| DB09185 | Viloxazine | approved, investigational, withdrawn | no | substrate | Details |
| DB06045 | Trofinetide | approved, investigational | unknown | inhibitor | Details |
| DB06700 | Desvenlafaxine | approved, investigational | no | substrate | Details |