Cytochrome P-450 Enzyme Inhibitors

Name
Cytochrome P-450 Enzyme Inhibitors
Accession Number
DBCAT000394
Description

Drugs and compounds which inhibit or antagonize the biosynthesis or actions of CYTOCHROME P-450 ENZYMES.

Drugs
DrugDrug Description
(5-(PYRIDIN-3-YL)FURAN-2-YL)METHANAMINENot Available
1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine (PEPAP) is a synthetic analogue of meperidine. It is sold as a "synthetic heroin."
6-Deoxyerythronolide BNot Available
AbametapirA pediculicide metalloproteinase used topically in the treatment of head lice infection.
AbemaciclibA medication used to treat HR+ HER2- advanced or metastatic breast cancer.
AbirateroneAn antiandrogen used in the treatment of metastatic castration-resistant prostate cancer and metastatic high-risk castration-sensitive prostate cancer.
AcalabrutinibA Bruton tyrosine kinase inhibitor used to treat mantle cell lymphoma, chronic lymphocytic leukemia, and small lymphocytic lymphoma.
AcebutololA selective β1-receptor antagonist used for the management of hypertension and ventricular premature beats in adults.
AcetaminophenAn analgesic drug used alone or in combination with opioids for pain management, and as an antipyretic agent.
AcetazolamideA carbonic anhydrase inhibitor used to treat edema from heart failure or medications, certain types of epilepsy, and glaucoma.
Acetyl sulfisoxazoleAcute, recurrent or chronic urinary tract infections (primarily pyelonephritis, pyelitis and cystitis) due to susceptible organisms (usually Escherichia coli, Klebsiella-Enterobacter, staphylococcus, Proteus mirabilis and, less frequently, Proteus vulgaris) in the...
AcoramidisA small molecule transthyretin stabilizer for use in patients with cardiomyopathy caused by transthyretin amyloidosis.
AdagrasibA KRAS inhibitor indicated for the treatment of locally advanced or metastatic KRAS G12C-mutated non-small cell lung cancer in patients who have received at least one prior systemic therapy.
AdemetionineS-Adenosylmethionine (SAMe) is used as a drug in Europe for the treatment of depression, liver disorders, fibromyalgia, and osteoarthritis. It has also been introduced into the United States market as...
AgomelatineAgomelatine is indicated to treat major depressive episodes in adults.
Albinterferon Alfa-2BInvestigated for use/treatment in hepatitis (viral, C).
AlbuterolA beta-2 adrenergic receptor agonist used to treat asthma, bronchitis, COPD, as well as prevent exercise induced bronchospasms.
AldesleukinA recombinant analog of interleukin-2 used to induce an adaptive immune response in the treatment of renal cell carcinoma.
AllicinAllicin has been used in trials studying the treatment of Follicular Lymphoma.
AllopurinolA xanthine oxidase inhibitor used to reduce urinary and serum uric acid concentrations in patients with gout, recurrent calcium oxalate calculi, and various malignancies.
AlmonertinibA third-generation, irreversible epidermal growth factor receptor (EGFR) tyrosine kinase inhibitor (TKI) indicated for the treatment of patients with metastatic EGFR T790M mutation-positive non-small cell lung cancer (NSCLC).
AlosetronA 5-HT3 antagonist used to treat diarrhea-predominant IBS.
AlpelisibAlpelisib is indicated in combination with fulvestrant to treat postmenopausal women, and men, with advanced or metastatic breast cancer. This cancer must be hormone receptor (HR)-positive, human epidermal growth factor...
AlpibectirAlpibectir is a small molecule drug. Alpibectir is under investigation in clinical trial NCT06748937 (A Study of the Early Effects, Safety, and Acceptability of Oral Alpibectir in Combination With Ethionamide)....
AminophenazoneAn analgesic drug used to treat acute migraine attacks in combination with ergotamine and caffeine.
AmiodaroneA class III antiarrhythmic indicated for the treatment of recurrent hemodynamically unstable ventricular tachycardia and recurrent ventricular fibrillation.
AmitriptylineA tricyclic antidepressant indicated in the treatment of depressive illness, either endogenous or psychotic, and to relieve depression associated anxiety.
AmlodipineA calcium channel blocker used to treat hypertension and angina.
AmodiaquineAn antimalarial drug.
AmoxapineA tricyclic antidepressant used in the treatment of neurotic or reactive depressive disorders and endogenous or psychotic depression.
AmoxicillinA penicillin derivative used for the treatment of infections caused by gram-positive bacteria, in particular streptococcal bacteria causing upper respiratory tract infections.
AmphetamineA CNS stimulant and sympathomimetic agent indicated for the treatment of Attention Deficit Hyperactivity Disorder (ADHD).
AmprenavirA protease inhibitor used to treat HIV infection.
AnacaulaseA mix of proteolytic enzymes indicated for eschar removal in adults with deep partial thickness and/or full-thickness thermal burns.
AnagrelideA platelet-reducing agent used to treat thrombocythemia, and its related complications, secondary to myeloproliferative neoplasms.
AnastrozoleA competitive, selective, non-steroidal aromatase inhibitor used as adjuvant therapy for the treatment of hormone receptor-positive breast cancer in postmenopausal women.
Angelica sinensis rootAngelica sinensis root is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.
AntipyrineAn antipyretic agent used for the symptomatic treatment of acute otitis media, most commonly in combination with benzocaine.
AprepitantA substance P/neurokinin 1 receptor antagonist used to treat nausea and vomiting caused by chemotherapy and surgery.
AprocitentanAn endothelin receptor antagonist used for the treatment of uncontrolled hypertension in patients inadequately controlled on other treatments.
ArmodafinilA stimulant used to improve wakefulness in adult patients with excessive sleepiness associated with obstructive sleep apnea, narcolepsy, or shift work disorder.
Arsenic trioxideA chemotherapeutic agent used in the treatment of refractory or relapsed acute promyelocytic leukemia in patients with prior retinoid and anthracycline chemotherapy.
ArtefenomelArtefenomel has been investigated for the treatment of Malaria.
ArtenimolFor the treatment of uncomplicated Plasmodium falciparum infection in adults, children, and infants aged 6 months and up weighing over 5 kg [FDA Label]. Used in combination with DB13941.
AsciminibAn inhibitor of ABL/BCR-ABL1 tyrosine kinase for the treatment of patients with Philadelphia chromosome-positive CML, including those with the T315I mutation.
AsenapineAn atypical antipsychotic used to treat patients with bipolar I disorder and patients with schizophrenia.
AstemizoleA second generation antihistamine used to treat allergy symptoms.
AsunaprevirAn NS3 protease inhibitor used to treat hepatitis C genotype 1b.
AtazanavirAn antiviral protease inhibitor used in combination with other antiretrovirals for the treatment of HIV.
AtomoxetineA selective norepinephrine reuptake inhibitor (SNRI) used in the management of Attention Deficit Hyperactivity Disorder (ADHD).
AtorvastatinAn HMG-CoA reductase inhibitor used to lower lipid levels and reduce the risk of cardiovascular disease including myocardial infarction and stroke.
AtovaquoneAn antimicrobial indicated for the prevention and treatment of Pneumocystis jirovecii pneumonia (PCP) and for the prevention and treatment of Plasmodium falciparum malaria.
AtrasentanAn endothelin A receptor antagonist used to reduce proteinuria in patients with primary IgA nephropathy.
AvacopanAn orally bioavailable complement 5a receptor (C5aR) antagonist for the treatment of severe anti-neutrophil cytoplasmic (auto)antibody (ANCA)-associated vasculitis.
AvapritinibA selective tyrosine kinase inhibitor being investigated for the treatment of multidrug resistant gastrointestinal tumors.
AvasimibeInvestigated for use/treatment in peripheral vascular disease.
AVE9633Investigated for use/treatment in leukemia (myeloid).
AzamulinAzamulin is a small molecule drug. Azamulin has a monoisotopic molecular weight of 478.26 Da.
AzelastineA histamine H1-receptor antagonist used intranasally to treat allergic and vasomotor rhinitis and in an ophthalmic solution to treat allergic conjunctivitis.
AzithromycinA macrolide antibiotic used to treat a variety of bacterial infections.
BalaglitazoneBalaglitazone has been used in trials studying the treatment of Diabetes Mellitus, Type 2.
Baloxavir marboxilA polymerase acidic endonuclease inhibitor used to treat uncomplicated influenza.
BarnidipineA calcium channel blocker used to treat various forms of hypertension.
BelinostatA histone deacetylase (HDAC) inhibitor used for the treatment of patients with relapsed or refractory peripheral T-cell lymphoma (PTCL).
BelumosudilAn oral inhibitor of rho-associated coiled-coil-containing protein kinases (ROCK) used in the treatment of chronic graft-versus-host disease (GVHD).
BenidipineA synthetic dihydropyridine calcium channel blocker used to treat hypertension and angina pectoris.
BenzbromaroneA uricosuric agent which is taken daily for the prevention of gout flares.
BenznidazoleA trypanocidal agent used to treat Chagas disease.
BepridilFor the treatment of hypertension, and chronic stable angina (classic effort-associated angina).
BergaptenBergapten is under investigation in clinical trial NCT00533195 (Comparison of UVA1 Phototherapy Versus Photochemotherapy for Patients With Severe Generalized Atopic Dermatitis).
BerotralstatAn inhibitor of plasma kallikrein used for prophylaxis of angioedema attacks in patients with hereditary angioedema.
BesifloxacinA fluoroquinolone antibiotic agent used for the treatment of bacterial conjunctivitis.
BesigomsinBesigomsin is a small molecule drug. Besigomsin has a monoisotopic molecular weight of 416.18 Da.
BexaroteneA retinoid drug used for cutaneous manifestations of T-cell lymphoma in patients who have not responded well to previous systemic therapy.
BezafibrateA lipid-lowering fibrate used in the management of primary and secondary hyperlipidaemia, when there is a lack of clinical improvement following lifestyle modifications or correction of the underlying disorder.
BicalutamideAn androgen receptor inhibitor used to treat Stage D2 metastatic carcinoma of the prostate.
BifonazoleAn azole antifungal drug used to treat fungal skin infections, such as dermatomycosis.
BiperidenA muscarinic receptor antagonist used to treat parkinsonism and control extrapyramidal side effects of neuroleptic drugs.
Birch bark extractA herbal medicinal product used to treat partial thickness wounds.
Black cohoshA herbal product indicated in the symptomatic treatment of menopause.
BoceprevirA hepatitis C virus NS3/4A protease inhibitor used in combination with other medications to treat chronic hepatitis C genotype 1 infection. Boceprevir is not indicated as monotherapy.
BortezomibA proteasome inhibitor used to treat multiple myeloma in patients who have not been successfully treated with at least two previous therapies.
BosutinibAn antineoplastic agent used for the treatment of chronic, accelerated, or blast phase Philadelphia chromosome-positive (Ph+) chronic myelogenous leukemia (CML) in adults with inadequate clinical response to other treatments.
Brefeldin AA metabolite from Penicillium brefeldianum that exhibits a wide range of antibiotic activity.
Brentuximab vedotinA CD30-directed antibody-drug conjugate used to treat various types of lymphoma.
BrincidofovirAn oral lipid prodrug of cidofovir used in the treatment of human smallpox disease.
BromazepamA short-acting benzodiazepine with intermediate onset commonly used to treat panic disorders and severe anxiety.
BromocriptineA dopamine D2 receptor agonist used for the treatment of galactorrhea due to hyperprolactinemia and other prolactin-related conditions, as well as in early Parkinsonian Syndrome.
Bryostatin 1Bryostatin 1 has been investigated for the treatment of HIV Infection and Alzheimer's Disease.
BuprenorphineA partial opioid agonist used for management of severe pain that is not responsive to alternative treatments. Also used for maintenance treatment of opioid addiction.
BupropionA norepinephrine and dopamine reuptake inhibitor used in the treatment of major depressive disorder (MDD), seasonal affective disorder (SAD), and as an aid to smoking cessation.
BW-A 58CBW-A 58C, also known as 2-(4-tert-butylcyclohexyl)-3-hydroxy-1,4-naphthoquinone, is an experimental naphthoquinone antimalarial drug which undergoes extensive alkyl hydroxylation to a single t-butylhydroxy metabolite in man in vivo and also in human...
CabergolineA dopamine receptor agonist used for the treatment of hyperprolactinemic conditions due to various causes.
CabozantinibA tyrosine kinase inhibitor used to treat advanced renal cell carcinoma, hepatocellular carcinoma, and medullary thyroid cancer.
CaffeineA stimulant present in tea, coffee, cola beverages, analgesic drugs, and agents used to increase alertness. It is also used in to prevent and treat pulmonary complications of premature birth.
CandesartanAn angiotensin-receptor blocker indicated in the treatment of hypertension.
Candesartan cilexetilAn angiotensin receptor blocker used to treat hypertension, systolic hypertension, left ventricular hypertrophy, and delay progression of diabetic nephropathy.
CandicidinUsed in the topical treatment of vulvovaginal candidiasis.
CannabidiolAn active cannabinoid used as an adjunctive treatment for the management of seizures associated with Lennox-Gastaut syndrome or Dravet syndrome and symptomatic relief of moderate to severe neuropathic pain or other painful conditions, like cancer.
CannabinolCannabinol (CBN) is a physiologically inactive constituent of Cannabis sativa.
CapecitabineA nucleoside metabolic inhibitor indicated to treat different gastrointestinal, including pancreatic cancer, and breast cancer.
CapmatinibA kinase inhibitor targeting c-Met receptor tyrosine kinase in the treatment of non-small cell lung cancer with MET exon 14 skipping.
CapsaicinA topical analgesic agent used for the symptomatic relief of neuropathic pain associated with post-herpetic neuralgia, as well as other muscle and joint pain.
CarbamazepineAn anticonvulsant used to treat various types of seizures and pain resulting from trigeminal neuralgia.
CarbazochromeIndicated for capillary and parenchymal hemorrhage (trauma, tonsillectomy, during surgery), intestinal bleeding, and thrombocytopenic purpura.
CarbomycinCarbomycin, also called magnamycin, is crystalline macrolide antibiotic. This antibacterial is obtained from Streptomyces halstedii and it presents a large inhibitory effect against Gram-positive bacteria and some Mycoplasma strains. The...
CariprazineAn atypical antipsychotic used to treat schizophrenia and acute manic or mixed episodes due to bipolar I disorder.
CasimersenAn antisense phosphorodiamidate morpholino oligonucleotide used to treat Duchenne muscular dystrophy patients with mutations amenable to exon 45 skipping.
CaspofunginAn echinocandin used to treat a variety of fungal infections.
CathineUsed to decrease appetite.
CelecoxibAn NSAID used to treat osteoarthritis, rheumatoid arthritis, acute pain, menstrual symptoms, and to reduce polyps is familial adenomatous polyposis.
CenobamateA small molecule drug indicated to treat partial onset seizures in adults.
Cepeginterferon alfa-2BCepeginterferon alfa-2B is under investigation in clinical trial NCT01889433 (An Open-label Comparative Efficacy and Safety Study of Algeron (Cepeginterferon Alfa-2b) in Treatment-naive Patients With Chronic Hepatitis C).
CeritinibAn antineoplastic kinase inhibitor used to treat anaplastic lymphoma kinase (ALK)-positive metastatic non-small cell lung cancer (NSCLC) in patients with inadequate clinical response or intolerance to crizotinib.
CerivastatinA statin (or HMG CoA reductase inhibitor) used with dietary changes to decrease lipid levels and reduce the risk of cardiovascular events.
CethromycinA ketolide antibiotic with broad-spectrum activity against Gram-positive, Gram-negative, and atypical bacteria that may be useful for treating several conditions including community-acquired pneumonia, inhalation anthrax, plague, and tularemia.
ChamazuleneNot Annotated
ChloramphenicolA broad spectrum antibiotic that is effective against a variety of susceptible and serious bacterial infections but is not frequently used because of its high risk of bone marrow toxicity.
ChloroquineAn antimalarial drug used to treat susceptible infections with P. vivax, P. malariae, P. ovale, and P. falciparum. It is also used for second line treatment for rheumatoid arthritis.
ChlorpheniramineA histamine-H1 receptor antagonist indicated for the management of symptoms associated with upper respiratory allergies.
ChlorpromazineA phenothiazine antipsychotic used to treat nausea, vomiting, preoperative anxiety, schizophrenia, bipolar disorder, and severe behavioral problems in children.
ChlorzoxazoneA drug with muscle relaxant properties that is used as an adjunct to physical therapy and analgesics to treat stiffness and pain caused by a variety of musculoskeletal conditions.
CholecalciferolA form of Vitamin D used in the treatment of specific medical conditions such as refractory rickets, hypoparathyroidism, and familial hypophosphatemia, as well as osteoporosis and chronic kidney disease.
CiglitazoneDeveloped by Takeda Pharmaceuticals in the early 1980s, it is considered the prototypical compound for the thiazolidinedione class. Ciglitazone was never used as a medication, but it sparked interest in...
CimetidineA histamine H2 receptor antagonist used to manage GERD, peptic ulcer disease, and indigestion.
CinacalcetA calcium sensing receptor agonist used to treat secondary hyperparathyroidism in chronic kidney disease and hypercalcemia in parathyroid carcinoma.
CinchonidineNot Annotated
Cinnamon oilNot Annotated
CinoxacinFor the treatment of initial and recurrent urinary tract infections in adults caused by the following susceptible microorganisms: Escherichia coli, Proteus mirabilis, Proteus vulgaris, Klebsiella species (including K. pneumoniae), and...
CiprofloxacinA second generation fluoroquinolone used to treat various susceptible bacterial infections.
CisaprideA medication used to treat heartburn associated with GERD.
CisplatinA platinum based chemotherapy agent used to treat various sarcomas, carcinomas, lymphomas, and germ cell tumors.
CitalopramA selective serotonin reuptake inhibitor (SSRI) used in the treatment of depression.
ClarithromycinA macrolide antibiotic used for the treatment of a wide variety of bacterial infections such as acute otitis, pharyngitis, tonsillitis, respiratory tract infections, uncomplicated skin infections, and helicobacter pylori infection.
ClascoteroneAn androgen receptor antagonist used for the topical treatment of acne vulgaris in patients 12 years of age and older.
ClemastineAn antihistamine with sedative and anticholinergic effects used to treat the symptoms of allergic rhinitis.
ClevidipineA dihydropyridine L-type calcium channel blocker used to lower blood pressure when oral antihypertensive therapy is not feasible or not desirable.
ClinafloxacinClinafloxacin is a fluoroquinolone antibacterial currently under research. It has been proven to present good antibiotic properties. However, its approval and release have been halted due to the presence of...
ClindamycinA lincosamide antibiotic used to treat serious infections caused by susceptible anaerobic, streptococcal, staphylococcal, and pneumococcal bacteria.
ClobazamA benzodiazepine used as adjunct treatment in seizures associated with Lennox-Gastaut syndrome.
ClofazimineA riminophenazine antimycobacterial used to treat leprosy.
ClofibrateA fibric acid derivative used to treat hypertriglyceridemia and high cholesterol.
ClomipramineA tricyclic antidepressant used in the treatment of obsessive-compulsive disorder and disorders with an obsessive-compulsive component, such as depression, schizophrenia, and Tourette’s disorder.
ClonazepamA long-acting benzodiazepine with intermediate onset commonly used to treat panic disorders, severe anxiety, and seizures.
CloperidoneCloperidone is a small molecule drug. Cloperidone has a monoisotopic molecular weight of 398.15 Da.
ClopidogrelAn antiplatelet agent used to prevent blood clots in peripheral vascular disease, coronary artery disease, and cerebrovascular disease.
ClotrimazoleA topical broad-spectrum antifungal agent used for the treatment of a wide variety of dermatophyte infections and candidiasis.
ClozapineAn atypical or second-generation antipsychotic drug used in treatment-resistant schizophrenia and to decrease suicide risk in schizophrenic patients.
Cobalt chlorideNot Annotated
CobicistatA CYP3A inhibitor used to increase the systemic exposure of atazanavir or darunavir in combination with other antiretroviral agents in the treatment of HIV-1 infection.
CobimetinibAn antineoplastic agent and selective inhibitor of the mitogen-activated extracellular kinase (MEK) pathway used to treat unresectable or metastatic melanoma.
CocaineAn ester local anesthetic used during diagnostic procedures and surgeries in or through the nasal cavities.
ColchicineAn alkaloid used to treat gout and Familial Mediterranean Fever as well as prevent major cardiovascular events.
Coltuximab ravtansineInvestigated for use/treatment in lymphoma (non-hodgkin's).
ConivaptanAn antidiuretic hormone inhibitor used to raise serum sodium levels.
Conjugated estrogensA mixture of estrogens used in estrogen replacement therapy for menopause and hypoestrogenism, used in the treatment of various malignancies, and used in the treatment of postmenopausal osteoporosis.
CrisaboroleA non-steroidal topical medication used for the treatment of mild-moderate atopic dermatitis.
CrizotinibA receptor tyrosine kinase inhibitor used to treat metastatic non-small cell lung cancer (NSCLC) where the tumors have been confirmed to be anaplastic lymphoma kinase (ALK), or ROS1-positive.
CryptotanshinoneNot Annotated
CurcuminNo approved therapeutic indications.
Curcumin sulfateNo approved therapeutic indications.
CyclizineAn antihistamine and antiemetic drug used for the prevention and treatment of nausea, vomiting, and dizziness associated with motion sickness, and vertigo.
CyclosporineA steroid-sparing immunosuppressant used in organ and bone marrow transplants as well as inflammatory conditions such as ulcerative colitis, rheumatoid arthritis, and atopic dermatitis.
Cyproterone acetateA steroid used in combination with ethinyl estradiol to treat women with severe acne and symptoms of androgenization. Also used alone at much higher doses for palliative treatment of patients with prostate cancer
DabrafenibA kinase inhibitor used to treat patients with specific types of melanoma, non-small cell lung cancer, and thyroid cancer.
DacomitinibA medication used to treat non small cell lung cancer with EGFR exon 19 deletion of exon 21 L858R substitution.
DalfopristinAn antibiotic used with quinupristin to treat severe or life-threatening infections of vancomycin-resistant Enterococcus faecium (VREF), and skin infections caused by methicillin susceptible staphylococcus aureus or streptococcus pyogenes.
DanazolA synthetic steroid and pituitary gonadotropin inhibitor used in the treatment of endometriosis and symptomatic treatment of severe pain and tenderness associated with benign fibrocystic breasts.
DanoprevirDanoprevir has been used in trials studying the treatment of Hepatitis C, Chronic.
DapoxetineA selective serotonin reuptake inhibitor used in the treatment of premature ejaculation.
DaprodustatA small-molecule hypoxia-inducible factor prolyl hydroxylase inhibitor used for the treatment of anemia in patients with chronic kidney disease.
DarifenacinAn M3 muscarinic receptor blocker used to treat urinary incontinence.
DarunavirA HIV protease inhibitor used in the treatment of human immunodeficiency virus (HIV) infection in patients with history of prior antiretroviral therapies.
DasatinibA tyrosine kinase inhibitor used for the treatment of Philadelphia chromosome-positive acute lymphoblastic leukemia or chronic myeloid leukemia.
DaunorubicinAn anthracycline aminoglycoside used to induce remission of nonlymphocytic leukemia and acute lymphocytic leukemia.
DefactinibAn inhibitor of FAK used alongside a MEK1/RAF inhibitor for the treatment of recurrent low-grade serous ovarian cancer.
DeferasiroxAn iron chelator used to treat chronic iron overload caused by blood transfusions. Also used in patients with non-transfusion-dependent thalassemia syndromes, and in patients with elevated liver iron concentration and serum ferritin.
DelavirdineA non-nucleoside reverse transcriptase inhibitor used to treat HIV infection.
DeltamethrinNot Annotated
DeramciclaneInvestigated for use/treatment in anxiety disorders.
DesipramineA tricyclic antidepressant used in the treatment of depression.
DesmethylprodineDesmethylprodine, a derivative of meperidine, is an opioid analgesic with the potency of morphine. It has been listed as a Schedule I controlled drug in the United States, and thus...
DesogestrelA synthetic progestin used in contraception, often in combination with ethinyl estradiol.
DesvenlafaxineAn antidepressant agent and SNRI used for the treatment of major depressive disorders in adults.
DeutivacaftorA CFTR potentiator used to treat cystic fibrosis in patients with responsive mutations (e.g. F508del).
DexamethasoneA glucocorticoid available in various modes of administration that is used for the treatment of various inflammatory conditions, including bronchial asthma, as well as endocrine and rheumatic disorders.
Dexamethasone acetateCommonly known as decadron, dexamethasone acetate is a glucocorticosteroid previously marketed in the USA for the treatment of inflammatory respiratory, allergic, autoimmune, and other conditions. Developed in 1957, dexamethasone is...
Dexamethasone isonicotinateDexamethasone isonicotinate is an anti-inflammatory, anti-allergic glucocorticoid that can be administered orally, by inhalation, topically, and parenterally. Its unintended mineralocorticoid action may cause salt and water retention.
DexchlorpheniramineA chlorpheniramine enantiomer antihistamine indicated in the treatment of sunburns, insect bites, and allergic reactions of the skin.
Dexchlorpheniramine maleateA first generation antihistamine used to treat allergic and vasomotor rhinitis, allergic conjunctivitis, and mild urticaria and angioedema.
DexfenfluramineFor the management of obesity including weight loss and maintenance of weight loss in patients on a reduced calorie diet
DexlansoprazoleA proton pump inhibitor used to treat erosive esophagitis, heartburn, and gastroesophageal reflux disease (GERD).
DexloxiglumideFor the treatment of Irritable Bowel Syndrome (IBS) and Gastroesophageal Reflux Disease (GERD).
DexmedetomidineAn alpha-2 agonist used for sedation during various procedures.
DextropropoxypheneAn opioid analgesic used to treat mild to moderate pain.
DiacereinAn slow-onset anthraquinone IL-1 inhibitor used in the treatment of degenerative joint diseases like osteoarthritis.
DiazepamA long-acting benzodiazepine with rapid onset commonly used to treat panic disorders, severe anxiety, alcohol withdrawal, and seizures.
DiazoxideA non diuretic benzothiadiazine indicated for the management of hypoglycemia in patients who produce an excess of insulin caused by a variety of conditions.
DiclofenacAn NSAID used to treat the signs and symptoms of osteoarthritis and rheumatoid arthritis.
DiethylstilbestrolUsed in the treatment of prostate cancer. Previously used in the prevention of miscarriage or premature delivery in pregnant women prone to miscarriage or premature delivery.
DifloxacinDifloxacin is a synthetic fluoroquinolone used in veterinary. As an antibacterial, it presents a broad bactericidal spectrum and its effects are dependent on its concentration. However, it presents a reduced...
DihydralazineDihydralazine is under investigation in clinical trial NCT00311974 (The Effect of Dihydralazine on Kidney Function and Hormones in Healthy Individuals).
DihydroergotamineAn ergot alkaloid used in the acute treatment of migraine headache and cluster headache.
DiltiazemA calcium channel blocker used to treat hypertension and to manage chronic stable angina.
Dimethyl sulfoxideA reversible mitogen-activated extracellular signal-regulated kinase-1 (MEK1) and MEK2 inhibitor used to treat certain types of melanoma, metastatic non-small cell lung cancer, and locally advanced or metastatic anaplastic thyroid cancer.
DiosminA citrus flavonoid medication used to support vascular health.
DiphenhydramineA H1 receptor antihistamine used in the treatment of seasonal allergies, and various allergic reactions including sneezing, runny nose, itchy/watery eyes, itching of nose or throat, pruritus, urticaria, insect bites/stings, and allergic rashes.
DirithromycinAn antibiotic used to treat a variety of respiratory, skin, and other infections.
DisulfiramA carbamate derivative used to treat alcohol addiction.
DitiocarbA chelating agent that has been used to mobilize toxic metals from the tissues of man and experimental animals. It is the main metabolite of DISULFIRAM.
Ditiocarb zincDitiocarb Zinc is approved for use within allergenic epicutaneous patch tests which are indicated for use as an aid in the diagnosis of allergic contact dermatitis (ACD) in persons 6...
DocetaxelA taxoid antineoplastic agent used in the treatment of various cancers, such as locally advanced or metastatic breast cancer, metastatic prostate cancer, gastric adenocarcinoma, and head and neck cancer.
DoconexentAn omega 3 fatty acid used in a variety of nutritional supplements to support central nervous system and cardiovascular health.
DoramectinDoramectin is a veterinary drug approved by the Food and Drug Administration for the treatment of parasites such as gastrointestinal roundworms, lungworms, eyeworms, grubs, sucking lice and mange mites in...
DordaviproneA protease inhibitor used to treat diffuse midline glioma with a H3 K27M mutation.
DosulepinA tricyclic antidepressant commonly used only in patients for whom alternative therapies are ineffective due to its toxicity potential.
DovitinibInvestigated for use/treatment in multiple myeloma and solid tumors.
DoxepinA psychotropic agent used for the treatment of depression, anxiety, manic-depressive disorder, and insomnia.
DoxorubicinA medication used to treat various cancers, including AIDS-associated Kaposi's Sarcoma and metastatic cancers.
DoxycyclineA tetracycline antibiotic used to treat a wide variety of bacterial infections.
DronabinolA synthetic delta-9-THC used in the treatment of anorexia and weight loss in HIV patients as well as nausea and vomiting in cancer chemotherapy.
DronedaroneAn antiarrhythmic agent used in the reduce the risk of hospitalization in patients with paroxysmal or persistent atrial fibrillation.
DuloxetineA serotonin norepinephrine reuptake inhibitor used to treat generalized anxiety disorder, neuropathic pain, osteoarthritis, and stress incontinence.
EconazoleA topical antifungal used to treat tinea pedis, tinea cruris, tinea corporis, cutaneous candidiasis and tinea versicolor.
Edetate calcium disodium anhydrousA chelating agent used to treat lead poisoning.
Edetate disodium anhydrousA polyvalent ion chelator indicated for emergency treatment of hypercalcemia and digitalis toxicity associated ventricular arrhythmias.
EfavirenzA non-nucleoside reverse transcriptase inhibitor used to treat HIV infection or prevent the spread of HIV.
EfonidipineFor the treatment of hypertension.
ElagolixA gonadotropin releasing hormone receptor antagonist used to treat moderate to severe pain in endometriosis.
ElbasvirAn antiviral and NS5A inhibitor used to treat hepatitis C infections.
ElexacaftorA small molecule CFTR corrector used in combination with tezacaftor and ivacaftor for the treatment of cystic fibrosis patients with one F508del-CFTR mutation.
EliglustatA glucosylceramide synthase used to treat type 1 Gaucher disease in patients who are CYP2D6 extensive, intermediate, or poor metabolizers.
ElinzanetantA selective, dual neurokinin 1 (NK-1) and 3 (NK-3) receptor antagonist used to treat vasomotor symptoms associated with menopause.
Ellagic acidEllagic acid is being investigated for use in follicular lymphoma, brain injury in intrauterine growth restricted babies, obese adolescents, and solar lentigines.
EltrombopagA thrombopoietin receptor agonist used to treat thrombocytopenia or aplastic anemia associated with various etiologies.
ElvitegravirAn antiretroviral agent used in combination with other antiretrovirals for the treatment of HIV-1 infection in antiretroviral treatment-experienced adults.
EnasidenibAn isocitrate dehydrogenase-2 inhibitor used to treat relapsed or refractory acute myeloid leukemia with an isocitrate dehydrogenase-2 mutation.
EncorafenibA kinase inhibitor used to treat unresectable or metastatic melanoma with BRAF mutations.
EnmetazobactamA beta-lactamase inhibitor used to treat complicated urinary tract infections in combination with cefepime.
EnoxacinFor the treatment of adults (≥18 years of age) with the following infections caused by susceptible strains of the designated microorganisms: (1) uncomplicated urethral or cervical gonorrhea due to Neisseria...
EnrofloxacinEnrofloxacin is an antibiotic agent from the fluoroquinolone family produced by the Bayer Corporation. Enrofloxacin is approved by the FDA for its veterinary use. Due to the identification of fluoroquinolone-resistant...
EnsitrelvirEnsitrelvir is indicated for post-exposure prophylaxis of coronavirus disease 2019 (COVID-19) in adults and adolescents 12 years of age and older following contact with an individual who has COVID-19.
EntacaponeA selective reversible catechol-O-methyltransferase inhibitor for the treatment of Parkinson's disease.
EnzalutamideA second-generation androgen receptor inhibitor used to treat castration-resistant prostate cancer and metastatic castration-sensitive prostate cancer.
EpinastineAn H1 receptor antagonist used to prevent itching in allergic conjunctivitis.
EpinephrineA hormone and neurotransmitter used to treat allergic reactions, to restore cardiac rhythm, and to control mucosal congestion, glaucoma, and asthma.
EpofolateEpofolate has been used in trials studying the treatment of Advanced Solid Tumors. Epofolate (BMS-753493) is a folate conjugate of the epothilone analog BMS-748285 that was designed to selectively target...
Epothilone DInvestigated for use/treatment in colorectal cancer, lung cancer, breast cancer, solid tumors, and prostate cancer.
EprinomectinNot Annotated
ErdafitinibA fibroblast growth factor receptor tyrosine kinase inhibitor used to treat locally advanced or metastatic urothelial carcinoma.
ErgometrineAn ergot alkaloid used for the treatment of postpartum haemorrhage and post abortion hemorrhage in patients with uterine atony.
ErgotamineAn alpha-1 selective adrenergic agonist vasoconstrictor used to treat migraines with or without aura and cluster headaches.
ErlotinibAn EGFR tyrosine kinase inhibitor used to treat certain small cell lung cancers or advanced metastatic pancreatic cancers.
ErythromycinA macrolide antibiotic used to treat and prevent a variety of bacterial infections.
EscitalopramA selective serotonin re-uptake inhibitor used in the treatment of major depressive disorder (MDD), generalized anxiety disorder (GAD), and other select psychiatric disorders such as obsessive-compulsive disorder (OCD).
EslicarbazepineAn antiepileptic indicated as a monotherapy or adjunct therapy in the treatment of epilepsy.
Eslicarbazepine acetateAn anticonvulsant agent used as an adjunct to treat partial-onset seizures in patients with inadequate clinical response to conventional antiepileptic therapy.
EsomeprazoleA proton pump inhibitor used to treat GERD, reduce the risk of NSAID associated gastric ulcers, eradicate H. pylori, and to treat conditions causing gastric acid hypersecretion.
EstradiolAn estrogenic steroid used to treat vasomotor symptoms of vulvar and vaginal atrophy in menopause, hypoestrogenism, prevention of postmenopausal osteoporosis, treatment of breast cancer, and advanced androgen-dependent carcinoma of the prostate.
Estradiol acetateAn estrogen used to treat vasomotor symptoms and moderate to severe vulvar and vaginal atrophy from menopause.
Estradiol benzoateAn estrogen indicated in combination with progesterone for the treatment of irregular menstruation.
Estradiol cypionateAn estradiol prodrug used to treat vasomotor symptoms and hypoestrogenisms from hypogonadism.
Estradiol dienanthateAn estrogen used in some combined hormonal oral contraceptives.
Estradiol valerateAn estradiol prodrug used to treat some effects of menopause, hypoestrogenism, androgen dependant carcinoma of the prostate, and in combination products for endometriosis and contraception.
Estrone sulfateAn estrogen used as monotherapy or in several combination hormone replacement products for managing menopause symptoms and hormone disorders.
EthambutolAn antituberculosis agent used in the prophylaxis and treatment of tuberculosis (TB).
EthanolFor therapeutic neurolysis of nerves or ganglia for the relief of intractable chronic pain in such conditions as inoperable cancer and trigeminal neuralgia (tic douloureux), in patients for whom neurosurgical...
EthinylestradiolAn estradiol used as a contraceptive.
EtoposideA podophyllotoxin derivative used to treat testicular and small cell lung tumors.
EtoricoxibA selective COX-2 inhibitor used to relieve moderate post-surgical dental pain as a short-term treatment and inflammatory and painful symptoms of various forms of arthritis.
EtravirineA non-nucleoside reverse transcriptase inhibitor (NNRTI) used in the treatment of HIV-1 infections in combination with other antiretroviral agents.
EtripamilAn L-type calcium channel blocker used to convert acute symptomatic episodes of paroxysmal supraventricular tachycardia to sinus rhythm in adults.
Evening primrose oilEvening primrose oil is used as part of over-the-counter dietary supplements. It is also used for the treatment of systemic inflammatory diseases and for women's health conditions such as cyclical...
EverolimusA mammalian target of rapamycin (mTOR) kinase inhibitor used to treat various types of malignancies.
EzetimibeA cholesterol absorption inhibitor used to lower total cholesterol, LDL-C, Apo-B, and non-HDL-C in primary hyperlipidemia and familial cholesterolemia.
FamotidineA histamine H2 receptor antagonist used to treat duodenal ulcers, benign gastric ulcers, GERD, and Zollinger-Ellison syndrome.
FavipiravirAn antiviral used to manage influenza, and that has the potential to target other viral infections.
FedratinibFedratinib is indicated for the treatment of adult patients with intermediate-2 or high-risk primary or secondary (post-polycythemia vera or post-essential thrombocythemia) myelofibrosis.
FelbamateAn anticonvulsant used to treat severe epilepsy.
FelodipineA calcium channel blocker used to treat hypertension.
FenfluramineFenfluramine is a phenethylamine that is structurally similar to serotonin. Due to its ability to increase extracellular serotonin levels, modulate serotonergic and other neurologic receptors, and control neurotransmission, it is effective in treating pharmacoresistant seizures.
FennelNot Annotated
FenofibrateA peroxisome proliferator receptor alpha activator used to lower LDL-C, total-C, triglycerides, and Apo B, while increasing HDL-C in hypercholesterolemia, dyslipidemia, and hypertriglyceridemia.
FenvalerateNot Annotated
FerrohemeNot Annotated
FexinidazoleAn orally bioavailable 2-substituted 5-nitroimidazole used to treat early- and late-stage human African trypanosomiasis caused by Trypanosoma brucei gambiense.
FidaxomicinA macrolide antibiotic used to treat diarrhea associated with Clostridium difficile infection.
FlecainideA class Ic antiarrhythmic agent used to manage atrial fibrillation and paroxysmal supraventricular tachycardias (PSVT).
FloxuridineAn antimetabolite used as palliative management for liver metastases of gastrointestinal malignancy.
FluconazoleA triazole antifungal used to treat various fungal infections including candidiasis.
FlumequineFlumequine is a synthetic chemotherapeutic antibiotic of the fluoroquinolone drug class used to treat bacterial infections.
FlunitrazepamA benzodiazepine used to manage anxiety disorders and insomnia.
FluorouracilA pyrimidine analog used to treat basal cell carcinomas, and as an injection in palliative cancer treatment.
FluoxetineA selective serotonin reuptake inhibitor used to treat major depressive disorder, bulimia, OCD, premenstrual dysphoric disorder, panic disorder, and bipolar I.
FluphenazineA phenothiazine used to treat patients requiring long-term neuroleptic therapy.
FlurazepamA long-acting benzodiazepine with a rapid onset of action that is commonly used to treat insomnia.
FlurithromycinNot Annotated
FluticasoneA corticosteroid indicated in the treatment of corticosteroid responsive dermatoses, asthma, and COPD.
Fluticasone furoateAn inhaled corticosteroid that can be used as maintenance treatment of asthma and/or chronic obstructive pulmonary disease (COPD) depending on the product. Also available as a nasal spray to manage symptoms of allergic rhinitis.
Fluticasone propionateA glucocorticoid used to treat asthma, inflammatory pruritic dermatoses, and nonallergic rhinitis.
FluvastatinAn HMG-CoA reductase inhibitor used to lower lipid levels and reduce the risk of cardiovascular disease including myocardial infarction and stroke.
FluvoxamineA selective serotonin-reuptake inhibitor used to treat obsessive-compulsive disorder.
FomepizoleAn inhibitor of alcohol dehydrogenase used as an antidote in confirmed or suspected methanol or ethylene glycol poisoning.
FosamprenavirAn antiretroviral agent used for the treatment and postexposure prophylaxis of human immunodeficiency virus (HIV-1) infection.
FosaprepitantAn antiemetic drug used in combination with other antiemetic agents for the prevention of acute and delayed nausea and vomiting caused by chemotherapy.
FosfluconazoleFosfluconazole is a small molecule drug. Fosfluconazole has a monoisotopic molecular weight of 386.07 Da.
FosnetupitantA medication used in combination with others to prevent chemotherapy associated nausea and vomiting.
FostamatinibA spleen tyrosine kinase inhibitor used to treat chronic immune thrombocytopenia after attempting one other treatment.
FurafyllineFurafylline is a derivative of methylxanthine derivative. It was developed on the context of asthma as a long-acting alternative for theophylline.
Fusidic acidA topical antibacterial agent used to prevent and treat mild to moderate skin infections caused by susceptible bacteria.
GarenoxacinInvestigated for use/treatment in bacterial infection.
Garlic oilNot Annotated
GatifloxacinA fourth generation fluoroquinolone used to treat a wide variety of infections in the body.
GefitinibA tyrosine kinase inhibitor used as first-line therapy to treat non-small cell lung carcinoma (NSCLC) that meets certain genetic mutation criteria.
GemfibrozilA lipid regulator that is used in the reduction of serum triglyceride levels in high-risk patients with hyperlipidemia.
GemifloxacinA quinolone antibacterial agent used for the treatment of acute bacterial exacerbation of chronic bronchitis and mild to moderate community-acquired pneumonia caused by susceptible bacteria.
GenisteinCurrently Genistein is being studied in clinical trials as a treatment for prostate cancer.
GestodeneGestodene is a progestogen hormonal contraceptive. Products containing gestoden include Meliane, which contains 20 mcg of ethinylestradiol and 75 mcg of gestodene; and Gynera, which contains 30 mcg of ethinylestradiol...
Ginkgo bilobaA herbal supplement found in over-the-counter or unapproved homeopathic products for various health conditions, such as cognitive, neurodegenerative, cardiovascular, and reproductive health disorders.
Ginsenoside CNot Available
GivinostatA histone deacetylase inhibitor indicated for the treatment of Duchenne Muscular Dystrophy (DMD).
GlecaprevirA Hepatitis C NS3/4A protease inhibitor used to treat Hepatitis C.
GlyburideA sulfonylurea used in the treatment of non insulin dependent diabetes mellitus.
Glycerol phenylbutyrateA nitrogen-binding agent used to manage patients with urea cycle disorders who cannot be sufficiently managed amino acid supplementation and/or dietary restrictions.
GoldensealNot Annotated
GPI-1485Investigated for use/treatment in erectile dysfunction and parkinson's disease.
GrapefruitAn extract from Grapefruit used in allergy testing.
GrazoprevirAn antiviral and NS3/4A protease inhibitor used to treat hepatitis C infections.
GrepafloxacinA fluoroquinolone antibiotic used to treat various gram positive and gram negative bacterial infections.
GuaiazulenNot Annotated
HalofantrineAn antimalarial used for the treatment of severe malaria.
HaloperidolAn antipsychotic agent used to treat schizophrenia and other psychoses, as well as symptoms of agitation, irritability, and delirium.
Hippuric acidNot Annotated
HistamineAn ingredient of topical drugs for the relief of joint pain or muscle aches and pains.
HomochlorcyclizineNot Annotated
Human placenta hydrolysateNot Annotated
HydralazineAn antihypertensive agent used for the management of essential hypertension or severe hypertension associated with conditions requiring immediate action, heart failure, and pre-eclampsia or eclampsia .
HydrastineNot Annotated
HydrastinineNot Annotated
HydroxychloroquineAn antimalarial medication used to treat uncomplicated cases of malaria and for chemoprophylaxis in specific regions. Also a disease modifying anti-rheumatic drug (DMARD) indicated for treatment of rheumatoid arthritis and lupus erythematosus.
HydroxyureaAn antimetabolite used to treat sickle cell anemia crisis, resistant chronic myeloid leukemia, and Locally advanced squamous cell carcinomas of the head and neck (excluding the lip).
HydroxyzineAn antihistamine used to treat anxiety and tension associated with psychoneuroses, as well as allergic conditions such as pruritus and chronic urticaria.
IbrexafungerpA triterpene antifungal indicated in the treatment of vulvovaginal candidiasis and prevention of recurrent vulvovaginal candidiasis in post-menarchal patients.
IbuprofenAn NSAID and non-selective COX inhibitor used to treat mild-moderate pain, fever, and inflammation.
IdelalisibAn antineoplastic kinase inhibitor used to treat chronic lymphocytic leukemia (CLL), relapsed follicular B-cell non-Hodgkin lymphoma (FL), and relapsed small lymphocytic lymphoma (SLL).
IfosfamideAn alkylating and immunosuppressive agent used in chemotherapy for the treatment of cancers, including testicular cancer, ovarian cancer, cervical cancer, osteocarcinoma, bladder cancer, small cell lung cancer, and non-Hodgkin's lymphoma.
ImatinibA tyrosine kinase inhibitor used to treat a number of leukemias, myelodysplastic/myeloproliferative disease, systemic mastocytosis, hypereosinophilic syndrome, dermatofibrosarcoma protuberans, and gastrointestinal stromal tumors.
ImipramineA tricyclic antidepressant indicated for the treatment of depression and to reduce childhood enuresis.
ImlunestrantAn estrogen receptor antagonist used to treat estrogen receptor (ER)-positive, human epidermal growth factor receptor 2 (HER2)-negative, estrogen receptor-1 (ESR1)-mutated advanced or metastatic breast cancer in adults with previous endocrine therapy.
IndalpineIndalpine was one of the first selective serotonin reuptake inhibitors to reach the American market. It was initially marketed by Pharmuka. However, after the emergence of widespread concern regarding adverse...
IndinavirA protease inhibitor used to treat HIV infection.
IndisulamInvestigated for use/treatment in lung cancer.
IndomethacinA nonsteroidal anti-inflammatory (NSAID) used for symptomatic management of chronic musculoskeletal pain conditions and to induce closure of a hemodynamically significant patent ductus arteriosus in premature infants.
Interferon alfaAn immunomodulator used to treat hepatitis B and C as well as certain types of cancer including cutaneous T-cell lymphoma and renal cell carcinoma.
Interferon alfa-2aA form of recombinant human interferon used to stimulate the innate antiviral response in the treatment of hepatitis B and C viruses.
Interferon alfa-2bA form of recombinant human interferon used to treat hepatitis B and C infection, genital warts, hairy cell leukemia, follicular lymphoma, malignant melanoma, and AIDs-related Kaposi's sarcoma.
Interferon alfa-2cInterferon alfa-2c is under investigation in clinical trial NCT00485563 (A Phase II Study of EC17 (Folate-hapten Conjugate) in Patients With Progressive Metastatic Renal Cell Carcinoma).
Interferon alfa-n1A purified form of human interferon used to stimulate the innate antiviral response in the treatment of genital warts due to human papilloma virus.
Interferon alfa-n3A purified form of human interferon used to stimulate the innate antiviral response in the treatment of genital warts due to human papilloma virus.
Interferon alfacon-1A recombinant interferon similar the interferon alfa subtype which is used to treat hepatitis C infections.
Interferon beta-1aA form of recombinant human interferon used to slow disease progression and reduce the frequency of clinical symptoms in patients who have relapsing multiple sclerosis.
Interferon beta-1bA form of recombinant human interferon used to slow the progression of relapsing multiple sclerosis and to reduce the frequency of clinical symptoms.
Interferon gamma-1bA form of recombinant human interferon used to treat infections associated with chronic granulomatous disease and to slow the progression of severe malignant osteopetrosis.
IpriflavoneNot Annotated
IproniazidFor the treatment of depression (originally intended to treat tuberculosis).
IrbesartanAn angiotensin receptor blocker used to treat hypertension, delay progression of diabetic nephropathy, and treat congestive heart failure.
IrinotecanA topoisomerase inhibitor used to treat metastatic carcinoma of the colon or rectum and pancreatic adenocarcinoma.
IsavuconazoleIndicated for patients 18 years of age and older for the treatment of invasive aspergillosis [FDA Label]. Indicated for patients 18 years of age and older for the treatment of...
IsavuconazoniumA triazole antifungal used for the treatment of invasive aspergillosis and mucormycosis.
IsoliquiritigeninIsoliquiritigenin is a precursor to several flavonones in many plants.
IsoniazidAn antibiotic used to treat mycobacterial infections; most commonly use in combination with other antimycobacterial agents for the treatment of active or latent tuberculosis.
Isosorbide dinitrateA vasodilator used to treat angina in coronary artery disease.
IsradipineA dihydropyridine calcium channel blocker used for the treatment of hypertension.
ItraconazoleA triazole antifungal agent used to treat various fungal infections, such as blastomycosis and onychomycosis.
IvacaftorA cystic fibrosis transmembrane conductance regulator (CFTR) potentiator used alone or in combination products to treat cystic fibrosis in patients who have specific genetic mutations that are responsive to the medication.
JPC-3210JPC-3210 is a potent antimalarial agent. It is an erythrocytic schizonticide with potent in vitro antimalarial activity against multidrug-resistant Plasmodium falciparum lines, low cytotoxicity, potent in vivo efficacy against murine...
KavaNot Available
KetazolamA long-acting benzodiazepine used to manage anxiety and insomnia.
KetoconazoleA broad spectrum antifungal used to treat seborrheic dermatitis and fungal skin infections.
KetoprofenAn NSAID used to treat rheumatoid arthritis, osteoarthritis, ankylosing spondylitis, dysmenorrhea, mild to moderate muscle pain, postoperative pain, and postpartum pain.
KitasamycinKitasamycin is a macrolide antibiotic derived from Streptomyces kitasatoensis.
KOS-1584Investigated for use/treatment in solid tumors.
LabetalolAn alpha and beta adrenergic antagonist used to treat hypertension, angina, and sympathetic overactivity syndrome.
LandiololA rapid-acting selective beta-blocker used to reduce ventricular rate in supraventricular tachycardia in adults.
LanreotideA somatostatin analog used for the treatment of unresectable, well- or moderately-differentiated, locally advanced or metastatic gastroenteropancreatic neuroendocrine tumors and acromegaly.
LansoprazoleA proton pump inhibitor used to help gastrointestinal ulcers heal, to treat symptoms of gastroesophageal reflux disease (GERD), to eradicate Helicobacter pylori, and to treat hypersecretory conditions such as Zollinger-Ellison Syndrome.
LapatinibAn antineoplastic agent and tyrosine kinase inhibitor used for the treatment of advanced or metastatic HER-positive breast cancer in patients who received prior chemotherapeutic treatments.
LaromustineInvestigated for use/treatment in brain cancer, cancer/tumors (unspecified), colorectal cancer, leukemia (lymphoid), leukemia (myeloid), lung cancer, myelodysplastic syndrome, pediatric indications, and solid tumors.
LasmiditanAn oral 5HT1F agonist used for the acute treatment of migraine headache with or without aura.
LazertinibA tyrosine kinase inhibitor used in combiantion with amivantamab to treat non-small cell lung cancer with EGFR mutations.
LeflunomideA pyrimidine synthesis inhibitor indicated to treat rheumatoid arthritis.
LemborexantA dual orexin antagonist indicated for the treatment of sleep-onset and/or sleep maintenance insomnia.
LenacapavirA first-in-class capsid inhibitor being investigated for use in HIV-1 treatment.
LeniolisibA phosphoinositide 3-kinase-delta inhibitor that is used to treat activated phosphoinositide 3-kinase delta syndrome.
LenvatinibA receptor tyrosine kinase inhibitor used for the treatment of metastatic thyroid cancer, advanced renal cell carcinoma in combination with everolimus, and unresectable hepatocellular carcinoma.
LercanidipineA calcium channel blocker for the management of hypertension.
LestaurtinibInvestigated for use/treatment in pancreatic cancer, prostate cancer, and leukemia (myeloid).
LetermovirAn antiviral medication used for prophylaxis in adult transplant recipients at risk of cytomegalovirus (CMV) infection and disease.
LetrozoleAn aromatase inhibitor used to treat breast cancer in postmenopausal women.
LevofloxacinA fluoroquinolone antibiotic used to treat infections caused by susceptible bacteria of the upper respiratory tract, skin and skin structures, urinary tract, and prostate, as well as for post-exposure treatment of inhaled anthrax and the plague.
LevoketoconazoleOne of two enantiomeric forms of racemic ketoconazole that strongly inhibits multiple steroidogenic enzymes and is used for the symptomatic treatment of endogenous Cushing's syndrome.
LevosalbutamolA beta-2 adrenergic receptor agonist used to treat COPD and asthma.
LevothyroxineA synthetic T4 hormone used to treat hypothyroidism that can be used along with surgery and radioiodine therapy to manage thyrotropin-dependent well-differentiated thyroid cancer.
LicofeloneFor the management of osteoarthritis.
LidocaineA local anesthetic used in a wide variety of superficial and invasive procedures.
LifitegrastA medication used to treat dry eye disease.
LimnetrelvirLimnetrelvir is a small molecule drug. The usage of the INN stem '-trelvir' in the name indicates that Limnetrelvir is a antiviral 3CL protease inhibitor. Limnetrelvir has a monoisotopic molecular...
LinagliptinA dipeptidyl peptidase-4 (DPP-4) inhibitor used to manage hyperglycemia in patients with type 2 diabetes mellitus.
LinerixibatAn ileal bile acid transporter (IBAT) inhibitor indicated for the treatment of cholestatic pruritus in adult patients with primary biliary cholangitis.
LinzagolixA selective gonadotropin-releasing hormone (GnRH) receptor antagonist used for the symptomatic treatment of uterine fibroids.
LiotrixMay be used to treat primary, secondary or tertiary hypothyroidism. May also be used to suppress thyroid stimulating hormone (TSH) secretion in patients with simple (nontoxic) goiter, subacute or chronic...
LobeglitazoneLobeglitazone was approved by the Ministry of Food and Drug Safety (South Korea) in 2013, and is being monitored by postmarketing surveillance until 2019. Lobeglitazone is not approved for use...
LomefloxacinA fluoroquinolone used to prevent and treat a wide variety of infections in the body.
LomitapideA microsomal triglyceride transfer protein inhibitor used to lower cholesterol associated with homozygous familial hypercholesterolemia (HoFH), reducing risk of cardiovascular events such as myocardial infarction and stroke.
LomustineAn alkylating agent used as a part of chemotherapeutic regimens for the treatment of primary and metastatic brain tumors as well as refractory or relapsed Hodgkin's disease in addition to surgical and/or radiotherapeutic treatments.
LonafarnibA potent farnesyl transferase inhibitor used to reduce mortality associated with Hutchinson-Gilford progeria syndrome (HGPS) and other progeroid laminopathies.
LonapegsomatropinA human growth hormone indicated in the treatment of growth failure due to inadequate endogenous growth hormone secretion.
LoperamideA long acting antidiarrheal used to control nonspecific diarrhea and chronic diarrhea caused by inflammatory bowel disease, or gastroenteritis.
LopinavirAn HIV-1 protease inhibitor used in combination with ritonavir to treat human immunodeficiency virus (HIV) infection.
LoratadineA second generation antihistamine used to manage the symptoms of allergic rhinitis.
LorcaserinA serotonin 2C receptor agonist used in conjunction with physical activity and calorie restriction for weight loss in obese patients with a body mass index (BMI) of 30 and above, and in overweight patients with weight-related comorbidities.
LorlatinibAn anaplastic lymphoma kinase inhibitor used to treat anaplastic lymphoma kinase positive metastatic non small cell lung cancer.
Lorvotuzumab mertansineLorvotuzumab mertansine has been used in trials studying the treatment of SCLC, Leukemia, Ovarian Cancer, Multiple Myeloma, and Merkel Cell Carcinoma, among others.
LosartanAn angiotensin receptor blocker used to treat hypertension and diabetic nephropathy, and is used to reduce the risk of stroke.
LuliconazoleA topical antifungal agent used to treat fungal infections.
LumacaftorA protein chaperone used in combination with ivacaftor for the treatment of cystic fibrosis in patients who are homozygous for the F508del mutation in the CFTR gene.
LumasiranLumasiran is an interfering RNA that silences hydroxyacid oxidase 1 for the treatment of primary hypoxaluria type 1.
LumefantrineAn antimalarial agent used in combination with artemether for the treatment of acute uncomplicated malaria caused by Plasmodium falciparum.
LynestrenolA progestin used for contraception and in the treatment of menstrual disorders.
Madecassic acidNot Annotated
MafosfamideMafosfamide has been used in trials studying the treatment of Lymphoma, Leukemia, Meningeal Neoplasm, and Brain and Central Nervous System Tumors.
ManidipineA dihydropyridine calcium channel blocker used to treat hypertension.
MaralixibatAn ileal bile acid transporter inhibitor indicated to treat cholestatic pruritus in patients with Alagille syndrome.
MavorixaforA CXC chemokine receptor 4 antagonist used to treat WHIM syndrome.
Medical CannabisThe use of the plant species Cannabis sativa and Cannabis indica, popularly known as marijuana, has gained popularity in recent years for the management of a wide variety of medical...
Medroxyprogesterone acetateA progestin used as a contraceptive and in the treatment of secondary amenorrhea, abnormal uterine bleeding, pain from endometriosis, endometrial and renal carcinomas, paraphilia in males, and GnRH-dependent precocious puberty.
Mefenamic acidAn NSAID used to treat mild to moderate pain for no more than a week, and primary dysmenorrhea.
MefloquineAn antimalarial agent used in the prophylaxis and treatment of malaria caused by Plasmodium falciparum and Plasmodium vivax.
MelperoneAn atypical butyrophenone antipsychotic used to treat sleep disorders, confusion, and psychomotor dysfunction associated with geriatric, psychiatric, and alcohol-dependent patients.
MemantineAn NMDA receptor antagonist used to treat moderate to severe dementia in Alzheimer's.
MenadioneThe primary known function of vitamin K is to assist in the normal clotting of blood, but it may also play a role in normal bone calcification.
MephenytoinA phenylhydantoin used to treat refractory partial epilepsy.
MepyramineAn antihistamine agent used for the symptomatic treatment of allergy, hypersensitivity reactions, and pruritic skin disorders.
MequitazineFor the treatment of Hay fever, urticaria (hives) and allergic rhinitis
MetacetamolMetacetamol is a small molecule drug. Metacetamol has a monoisotopic molecular weight of 151.06 Da.
MethadoneAn opioid analgesic indicated for management of severe pain that is not responsive to alternative treatments. Also used to aid in detoxification and maintenance treatment of opioid addiction.
MethimazoleA thionamide antithyroid agent that inhibits the actions of thyroid peroxidase, leading to a reduction in thyroid hormone synthesis and amelioration of hyperthyroidism.
MethotrimeprazineA phenothiazine used in the management of psychosis, particular those of schizophrenia, and manic phases of bipolar disorder.
MethoxsalenA furocoumarin used to treat psoriasis and vitiligo.
MethsuximideA succinimide anticonvulsant that increases the seizure threshold. Primarily used for childhood absence seizures. Functions by suppressing paroxysmal spike-and-wave patterns associated with lapses of consciousness in absence seizures.
Methylene blueAn oxidation-reduction agent used for the treatment of pediatric and adult patients with acquired methemoglobinemia.
MethylergometrineAn ergot alkaloid used to prevent and control uterine atony and hemorrhage before and after delivery.
MethyloneMethylone is under investigation in clinical trial NCT05741710 (A Study to Assess the use of Methylone in the Treatment of PTSD).
MetoclopramideAn antiemetic agent and dopamine D2 antagonist used in the treatment of gastroesophageal reflux disease, prevention of nausea and vomiting, and to stimulate gastric emptying.
MetoprololA beta-blocker used in the treatment of hypertension and angina, and used to reduce mortality due to myocardial infarction.
MetronidazoleA nitroimidazole used to treat trichomoniasis, amebiasis, inflammatory lesions of rosacea, and bacterial infections, as well as prevent postoperative infections.
MetyraponeA steroid 11-beta-monooxygenase inhibitor used to test hypothalamic-pituitary ACTH function.
MexiletineA class 1B antiarrhythmic agent used in the treatment of documented ventricular arrhythmias that warrant treatment.
MibefradilFor the treatment of angina and high blood pressure.
MiconazoleAn azole antifungal with broad-spectrum activity used to treat fungal infections affecting the vagina, mouth and skin, including candidiasis.
MidazolamA short-acting benzodiazepine with rapid onset that is commonly used in seizures, anesthesia and anxiety disorders.
MidecamycinA macrolide antibiotic used to treat a variety of infections caused by susceptible bacteria.
MidostaurinAn antineoplastic agent used to treat high-risk acute myeloid leukemia (AML) with specific mutations, aggressive systemic mastocytosis (ASM), systemic mastocytosis with associated hematologic neoplasm (SM-AHN), or mast cell leukemia (MCL).
MifentidineMifentidine is a small molecule drug. The usage of the INN stem '-tidine' in the name indicates that Mifentidine is a histamine- H2​-receptor antagonist, cimetidine derivative. Mifentidine has a monoisotopic...
MifepristoneA cortisol receptor blocker used to treat Cushing's syndrome, and to terminate pregnancies up to 70 days gestation.
MilnacipranA selective serotonin and norepinephrine reuptake inhibitor (SNRI) used for the treatment of fibromyalgia and a short-term treatment of major depressive disorder.
MiocamycinMiocamycin is a macrolide type antimicrobial . This drug may be marketed in Japan for clinical use as it is listed in the Japanese pharmacopeia . It has shown to...
MirabegronA beta-3 adrenergic agonist used to treat overactive bladder and neurogenic detrusor overactivity.
MiricorilantMiricorilant is under investigation in clinical trial NCT03818256 (Study Evaluating the Safety, Efficacy, and Pharmacokinetics of Miricorilant (CORT118335) in Obese Adult Patients With Schizophrenia and Recent Weight Gain While Taking...
MirtazapineA tetracyclic antidepressant used in the treatment of major depression and is used off-label as a drug for insomnia and to increase appetite.
MitemcinalInvestigated for use/treatment in gastroparesis and irritable bowel syndrome (IBS).
MitoxantroneA chemotherapeutic agent used for the treatment of secondary progressive, progressive relapsing, or worsening relapsing-remitting multiple sclerosis.
MizolastineA second-generation non-sedating antihistamine used to treat symptoms of allergic rhinoconjunctivitis and urticaria.
MoclobemideA monoamine oxidase inhibitor used in the treatment of major depressive disorder and bipolar disorder.
ModafinilA stimulant used to improve wakefulness in patients with sleep apnea, narcolepsy, or shift work disorder.
MomelotinibA Janus Kinase inhibitor used to treat intermediate or high-risk myelofibrosis.
MometasoneA corticosteroid with no indications.
Mometasone furoateA corticosteroid used to treat asthma, allergic rhinitis, nasal congestion, nasal polyps, dermatitis, and pruritus.
MontelukastA leukotriene receptor antagonist used as part of an asthma therapy regimen, to prevent exercise induced bronchoconstriction, and to treat seasonal allergic rhinitis.
MoxifloxacinA fluoroquinolone antibiotic used to treat various bacterial infections.
NabiloneA synthetic delta-9-THC used in the treatment of anorexia and weight loss in HIV patients as well as nausea and vomiting in cancer chemotherapy.
NabiximolsIn Canada, Sativex has received a Notice of Compliance (NOC) for use as an as adjunctive treatment for symptomatic relief of spasticity in patients with multiple sclerosis (MS) who have...
NafimidoneNafimidone is a small molecule drug. Nafimidone has a monoisotopic molecular weight of 236.09 Da.
NafithromycinNafithromycin is under investigation in clinical trial NCT02903836 (Phase II Study of Oral Nafithromycin in CABP).
Nalidixic acidA quinolone antibiotic used to treat urinary tract infections.
NaloxegolA peripherally-selective opioid antagonist used to treat opioid-induced constipation (OIC) in adult patients with chronic non-cancer pain.
NaloxoneAn opioid receptor antagonist used to rapidly reverse an opioid overdose. Also included in some drug formulations as an abuse deterrent to prevent injection.
NaringinNot Annotated
NefazodoneAn antidepressant used in the treatment of depression.
NelfinavirA viral protease inhibitor used in the treatment of HIV infection.
NemonoxacinInvestigated for use/treatment in bacterial infection and pneumonia.
NetoglitazoneNetoglitazone (MCC-555) is a hypoglycemic agent.
NetupitantAn antiemetic agent used in combination with palonosetron to prevent acute and delayed vomiting and nausea caused by chemotherapy.
NevirapineA non-nucleoside reverse transcriptase inhibitor used as part of a management regimen for HIV-1 virus infection.
NiacinA B vitamin used to treat hypertriglyceridemia and pellagra.
NicardipineA calcium channel blocker used for the short-term treatment of hypertension and chronic stable angina.
NiclosamideAn anthelmintic indicated in the treatment of beef, pork, fish, and dwarf tapeworm infections in adults and children.
NicotinamideAn ingredient found in a variety of cosmetic products.
NicotineA stimulatory alkaloid found in tobacco products that is often used for the relief of nicotine withdrawal symptoms and as an aid to smoking cessation.
NifedipineA dihydropyridine calcium channel blocker indicated for the management of several subtypes of angina pectoris, and hypertension.
NilotinibA kinase inhibitor used for the chronic phase treatment of Chronic Myeloid Leukemia (CML) that is Philadelphia chromosome positive and for the treatment of CML that is resistant to therapy containing imatinib.
NilutamideAn antineoplastic hormone used to treat prostate cancer.
NilvadipineA calcium channel blocker used to manage arterial hypertension.
NirmatrelvirAn oral protease inhibitor with emergency use authorization for the treatment of mild-to-moderate COVID-19.
NitisinoneA hydroxyphenylpyruvate dioxygenase inhibitor used as an adjunct to dietary restrictions for the treatment of hereditary tyrosinemia type 1 (HT-1) and Alkaptonuria, which cause intolerance to tyrosine containing foods.
NitrazepamA long-acting benzodiazepine with intermediate onset commonly used to treat panic disorders, severe anxiety, insomnia, and seizures.
Nitric OxideA vasodilating agent used in the treatment of hypoxic respiratory failure in premature neonates.
NivasorexantNivasorexant is a small molecule drug. The usage of the INN stem '-orexant' in the name indicates that Nivasorexant is a orexin receptor antagonist. Nivasorexant has a monoisotopic molecular weight...
Nix-0699Not Annotated
NorfloxacinA broad-spectrum fluoroquinolone antibiotic with variable activity against gram-positive and gram-negative bacteria. Typically reserved for the treatment of UTIs due to accumulation in the urine.
NortriptylineA tricyclic antidepressant used in the treatment of depression.
NoscapineA non-sedating isoquinoline alkaloid used primarily for its antitussive properties.
Obeticholic acidA bile acid analog and farnesoid X receptor agonist used to treat primary biliary cholangitis in adult patients with inadequate clinical response or intolerance to UDCA.
OctreotideA peptide drug used to treat acromegaly as well as diarrhea associated with metastatic carcinoid tumors and vasoactive intestinal peptide secreting tumors.
OfloxacinAn antibacterial agent used for the treatment of bacterial infections in many parts of the body, including the respiratory tract, kidney, skin, soft tissue, and urinary tract.
OlanzapineAn antipsychotic drug used in the management of schizophrenia, bipolar 1 disorder, and agitation associated with these disorders.
OlaparibA poly (ADP-ribose) polymerase (PARP) inhibitor used to treat ovarian cancer, breast cancer, pancreatic cancer, and prostate cancer.
OleandomycinOleandomycin is a macrolide antibiotic, though it is less effective than erythromycin. It is synthesized from strains of Streptomyces antibioticus.
OlorofimOlorofim is under investigation in clinical trial NCT03340597 (Assessment of Varying Oral Dosing Regimens for F901318 in Healthy Subjects).
OmeprazoleA proton pump inhibitor used to treat GERD associated conditions such as heartburn and gastric acid hypersecretion, and to promote healing of tissue damage and ulcers caused by gastric acid and H. pylori infection.
OndansetronA serotonin 5-HT3 receptor antagonist used to prevent nausea and vomiting in cancer chemotherapy and postoperatively.
OpelconazoleNot Annotated
OpicaponeA catechol-O-methyltransferase inhibitor used as an adjunct treatment for Parkinson's Disease in adults currently receiving levodopa and a dopa decarboxylase inhibitor.
OrbifloxacinOrbifloxacin is a fluoroquinolone antibiotic. It is marketed by Schering-Plough Animal Health and approved for certain infections in dogs.
OritavancinAn antibacterial agent used to treat acute bacterial skin and skin structure infections caused by susceptible Gram-positive bacteria.
OrphenadrineA muscarinic antagonist used as an adjunct for the symptomatic relief of musculoskeletal pain and discomfort.
OsilodrostatAn oral inhibitor of cortisol synthesis used to treat Cushing's disease by normalizing hypercortisolism.
OsimertinibA tyrosine kinase inhibitor used in the treatment of certain types of non-small cell lung carcinoma.
OspemifeneA non-hormonal estrogen receptor modulator (SERM) used to treat moderate to severe dyspareunia, a symptom of vulvar and vaginal atrophy, due to menopause.
OSU-6162OSU-6162 is under investigation in clinical trial NCT05641623 (OSU6162 as Add-on in Ssri/snri-resistant Depression).
OxamniquineFor treatment of Schistosomiasis caused by Schistosoma mansoni
OxandroloneAn androgenic hormone used to treat muscle loss from prolonged corticosteroid treatment and to treat bone pain associated with osteoporosis.
OxcarbazepineAn anti-epileptic used in the treatment of partial-onset seizures.
OxethazaineAn antacid used to treat gastritis, peptic ulcer disease, heartburn, esophagitis, hiatus hernia, and anorexia.
OxprenololA non-selective beta-adrenergic antagonist used to treat hypertension, angina pectoris, arrhythmias, and anxiety.
OxybutyninAn antimuscarinic agent that reduces detrusor muscle activity, relaxing the bladder and preventing the urge to void.
OxymetholoneAn anabolic steroid used for the treatment of types of anemia, such as acquired aplastic anemia, congenital aplastic anemia, myelofibrosis, and the hypoplastic anemias.
P-57AS3Investigated for use/treatment in obesity.
PacritinibA kinase inhibitor used for the treatment of primary and secondary myelofibrosis in adult patients with significantly reduced platelet counts.
PalbociclibAn endocrine-based chemotherapeutic agent used in combination with other antineoplastic agents to treat HER2-negative and HR-positive advanced or metastatic breast cancer.
PaltusotineA somatostatin receptor agonist used to treat acromegaly in adults whose surgery is not an option or has not been effective.
PanobinostatA non-selective histone deacetylase inhibitor used to treat multiple myeloma in combination with other antineoplastic agents.
PantoprazoleA proton pump inhibitor used to treat erosive esophagitis, gastric acid hypersecretion, and to promote healing of tissue damage caused by gastric acid.
ParamethasoneFor the treatment of all conditions in which corticosteroid therapy is indicated except adrenal-deficiency states for which its lack of sodium-retaining properties makes it less suitable than hydrocortisone with supplementary...
ParoxetineA selective serotonin reuptake inhibitor used to treat major depressive disorder, panic disorder, OCD, social phobia, generalized anxiety disorder, the vasomotor symptoms of menopause, and premenstrual dysphoric disorder.
PasireotideA somatostatin analog used in the treatment of Cushing’s disease, specifically for those patients whom pituitary surgery is not appropriate.
PatupiloneInvestigated for use/treatment in ovarian cancer, lung cancer, brain cancer, breast cancer, and gastric cancer.
PazopanibAn antineoplastic agent used in the treatment of advanced renal cell cancer and advanced soft tissue sarcoma in patients with prior chemotherapy.
PazufloxacinPazufloxacin is under investigation in clinical trial NCT02592096 (Pazufloxacin Mesilate Ear Drops Clinical Trial Protocol).
PefloxacinAn antibiotic used to treat a variety of bacterial infections.
Peginterferon alfa-2aA modified form of recombinant human interferon used to stimulate the innate antiviral response in the treatment of hepatitis B and C viruses.
Peginterferon alfa-2bA purified form of human interferon used to stimulate the innate antiviral response in the treatment of hepatitis B and C, genital warts, and some cancers.
Peppermint oilAn ingredient used in a variety of natural health products and is not an approved medication.
PerampanelA non-competitive AMPA glutamate receptor antagonist used to treat partial-onset seizures with or without secondarily generalized seizures, and as adjunctive treatment of primary generalized tonic-clonic seizures in patients with epilepsy.
PergolideA long-acting dopamine agonist that is uncommonly used for the management of Parkinson's disease, due to the risk for cardiac valvulopathy.
PerhexilineFor the management of severe angina pectoris.
PerphenazineA phenothiazine used to treat schizophrenia as well as nausea and vomiting.
PexidartinibAn antitumor agent that is used for the treatment of rare disease tenosynovial giant cell tumors (TGCT) by inhibiting colony-stimulating factor 1 and its receptor.
PhencyclidineA hallucinogen formerly used as a veterinary anesthetic, and briefly as a general anesthetic for humans. Phencyclidine is similar to ketamine in structure and in many of its effects. Like...
PhenelzineA monoamine oxidase inhibitor used to treat atypical, nonendogenous, or neurotic depression.
PhenylbutazoneAn NSAID used to treat backache and ankylosing spondylitis.
Phenylbutyric acidAn agent indicated for the adjunctive therapy for the management of chronic urea cycle disorders due to deficiencies in specific enzymes, including the neonatal-onset deficiency and late-onset disease with a history of hyperammonemic encephalopathy.
PhenytoinAn anticonvulsant drug used in the prophylaxis and control of various types of seizures.
Phloxine BFor use in dental disclosing products, allowing for highlighting of bacterial placques.
PibrentasvirA Hepatitis C NS5A inhibitor used to treat Hepatitis C.
PilocarpineA muscarinic agonist used to treat dry mouth and various ophthalmic conditions, such as presbyopia, increased intraocular pressure, and angle-closure glaucoma.
PimozideAn antipsychotic used to manage debilitating motor and phonic tics in patients with Tourette's Disorder.
PindololA beta adrenoceptor antagonist used to treat hypertension, edema, ventricular tachycardias, and atrial fibrillation.
PioglitazoneA thiazolidinedione used adjunctively with diet and exercise to normalize glycemic levels in adults with type 2 diabetes mellitus.
Pipemidic acidA quinolone antibiotic indicated in the treatment of susceptible urinary tract infections.
PiperaquineFor the treatment of uncomplicated Plasmodium falciparum infection in adults, children, and infants aged 6 months and up weighing over 5 kg [FDA Label]. Used in combination with DB11638.
PiperineBioperine has been used in trials studying the treatment of Multiple Myeloma and Deglutition Disorders.
Piperonyl butoxideA pesticide used as a potentiator ingredient in the treatment of pediculosis (head lice, body lice or crabs) to boost efficacy of treatment.
PipotiazineAn antipsychotic indicated for the management of chronic, non-agitated schizophrenic patients.
PirfenidoneAn agent used for the treatment of idiopathic pulmonary fibrosis (IPF).
PiroxicamAn NSAID used to treat the symptoms of osteoarthritis and rheumatoid arthritis.
PirtobrutinibA kinase inhibitor used to treat relapsed or refractory mantle cell lymphoma (MCL) after at least two lines of systemic therapy. It is also used in adults with relapsed or refractory CLL/SLL who have previously received a covalent BTK inhibitor.
PitolisantAn antagonist and inverse agonist at the histamine H3 receptor that is used to treat narcolepsy in adults.
Poloxamer 188A medication used to clean wounds.
Polysorbate 80It is used as a solubilizer, antimicrobial preservative and disinfectant .
PosaconazoleA triazole antifungal drug that is used to treat invasive infections by Candida species and Aspergillus species in severely immunocompromised patients.
PralsetinibA RET receptor tyrosine kinase inhibitor for the treatment of metastatic RET-driven non-small cell lung cancer.
PranlukastA leukotriene receptor antagonist for the treatment of allergic rhinitis and asthma symptoms.
PrasteroneA steroid formulated as a vaginal insert indicated for the treatment of moderate to severe dyspareunia associated with menopausal vulvar and vaginal atrophy.
PrimaquineAn antimalarial indicated to prevent relapse of vivax malaria.
ProbenecidA medication used to treat gouty arthritis, tophaceous gout, and hyperuricemia.
ProgesteroneA hormone used for a variety of functions, including contraception, control of abnormal uterine bleeding, maintenance of pregnancy, and prevention of endometrial hyperplasia.
ProguanilA medication indicated for prophylaxis and treatment of Plasmodium falciparum malaria.
PromazineA phenothiazine used to manage schizophrenia.
PromethazineA first-generation antihistamine used for the treatment of allergic conditions, nausea and vomiting, and motion sickness.
PropacetamolPropacetamol is a paracetamol prodrug of intravenous administration used to control fever and pain of perioperative period in multimodal analgesia therapy.
PropafenoneA Class 1C antiarrhythmic agent used in the management of paroxysmal atrial fibrillation/flutter and ventricular arrhythmias.
PropofolA medication used in general anesthesia and for sedation.
PropranololA non-selective beta adrenergic antagonist used to treat hypertension, angina, atrial fibrillation, myocardial infarction, migraine, essential tremor, hypertrophic subaortic stenosis, and pheochromocytoma.
PrulifloxacinA broad-spectrum fluoroquinolone antibiotic used to treat a variety of susceptible bacterial infections.
PyrimethamineAn antiparasitic drug used in the prevention and treatment of toxoplasmosis and malaria.
QuazepamA long-acting benzodiazepine used to manage insomnia.
QuercetinA natural flavonoid found in foods and natural supplement products.
QuinidineA medication used to restore normal sinus rhythm, treat atrial fibrillation and flutter, and treat ventricular arrhythmias.
QuinineAn alkaloid used to treat uncomplicated Plasmodium falciparum malaria.
QuinupristinAn antibiotic agent used in the treatment of serious vancomycin-resistant Enterococcus faecium bacteremia as well as complicated skin and skin structure infections.
RabeprazoleA proton pump inhibitor used to help gastrointestinal ulcers heal, to treat symptoms of gastroesophageal reflux disease (GERD), to eradicate Helicobacter pylori, and to treat hypersecretory conditions such as Zollinger-Ellison Syndrome.
RaloxifeneA selective estrogen receptor modulator that is used to prevent and treat osteoporosis and reduce the risk of invasive breast cancer in high-risk postmenopausal women.
RanitidineA histamine H2 antagonist used to treat duodenal ulcers, Zollinger-Ellison syndrome, gastric ulcers, GERD, and erosive esophagitis.
RanolazineAn anti-anginal drug used for the treatment of chronic angina.
ReboxetineA drug used for the acute treatment of major depression and for maintenance therapy of depression.
RegorafenibA kinase inhibitor used to treat patients with metastatic colorectal cancer, unresectable, locally advanced, or metastatic gastrointestinal stromal tumors, and hepatocellular carcinoma.
RelacorilantA selective glucocorticoid receptor antagonist that reverses glucocorticoid-mediated anti-apoptotic signaling to restore chemosensitivity in platinum-resistant ovarian, fallopian tube, and primary peritoneal cancers.
RemacemideInvestigated for use/treatment in epilepsy, huntington's disease, and parkinson's disease.
RemdesivirA nucleoside analog used to treat RNA virus infections including COVID-19.
RemibrutinibA Bruton's tyrosine kinase inhibitor used to treat chronic spontaneous urticaria in adults.
RemoxiprideAn discontinued atypical antipsychotic selective for dopamine D2 receptors.
RepotrectinibA tyrosine kinase inhibitor used to treat locally active or metastatic non-small cell lung cancer
ResmetiromA thyroid hormone receptor-beta agonist used to treat noncirrhotic nonalcoholic steatohepatitis (NASH) with moderate to advanced liver fibrosis in adults.
ResveratrolBeing investigated for the treatment of Herpes labialis infections (cold sores).
RevumenibA small molecule menin inhibitor for the treatment of relapsed/refractory leukemia with KMT2A translocation.
RheinNo approved indication.
RibociclibA cyclin-dependent kinase inhibitor used to treat HR+, HER2- breast cancer.
RidaforolimusInvestigated for use/treatment in solid tumors, sarcoma, cancer/tumors (unspecified), endometrial cancer, prostate cancer, and bone metastases.
RifampinAn antibiotic used alone or in combination with other antimicrobial drugs to treat tuberculosis and asymptomatic carriers of Neisseria meningitidis.
RifamycinAn antibacterial used to treat traveler's diarrhea.
RilpivirineA non-nucleoside reverse transcriptase inhibitor (NNRTI) used in combination with other antiretrovirals to specifically treat human immunodeficiency virus type 1 (HIV-1).
RilzabrutinibA kinase inhibitor used to treat persistent or chronic immune thrombocytopenia (ITP) who have had an insufficient response to a previous treatment.
RimegepantAn oral CGRP receptor antagonist used for the acute treatment of migraines with or without aura in adults.
RipretinibA kinase inhibitor used to treat advanced gastrointestinal stromal tumor (GIST).
RisperidoneA second-generation antipsychotic medication used to treat a number of mental health disorders including schizophrenia, bipolar mania, psychosis, or as an adjunct in severe depression.
RitanserinRitanserin has been used in trials studying the treatment of Cocaine-Related Disorders.
RitlecitinibA kinase inhibitor used to treat severe alopecia areata in adults and adolescents 12 years and older.
RitonavirAn HIV protease inhibitor used in combination with other antivirals in the treatment of HIV infection.
RivoglitazoneRivoglitazone (INN) is a thiazolidinedione undergoing research for use in the treatment of type 2 diabetes. It is being developed by Daiichi Sankyo Co.
RizatriptanA triptan used to treat migraines with or without aura.
RofecoxibA COX-2 inhibitor NSAID used to treat osteoarthritis, rheumatoid arthritis, acute pain, primary dysmenorrhea, and migraine attacks.
RokitamycinNot Annotated
RolapitantA neurokinin-1 (NK-1) receptor antagonist used in combination with other antiemetics for the prevention of delayed nausea and vomiting associated with emetogenic chemotherapy.
Ropeginterferon alfa-2bA mono-pegylated type I interferon used to treat polycythemia vera.
RosiglitazoneA thiazolidinedione indicated as an adjunct to diet and exercise to maintain glycemic control in type 2 diabetes.
RosoxacinFor the treatment of bacterial infection of respiratory tract, urinary tract, GI, CNS and immuno compromised patients.
RosuvastatinAn HMG-CoA reductase inhibitor used to lower lipid levels and reduce the risk of cardiovascular disease including myocardial infarction and stroke.
RotigotineA non-selective dopamine agonist used for the treatment of Parkinson's Disease and Restless Leg Syndrome.
RoxithromycinAn antibiotic used to treat a variety of susceptible bacterial infections.
RucaparibA poly (ADP-ribose) polymerase (PARP) inhibitor used to treat recurrent ovarian and prostate cancers in previously treated adults.
RufinamideAn antiepileptic drug used as adjunctive therapy to treat seizures associated with Lennox-Gastaut Syndrome (LGS).
RufloxacinA fluoroquinolone antibiotic indicated in the treatment of susceptible respiratory infections and uncomplicated cystitis.
RutinA flavonoid found in over-the-counter vitamin supplements.
SafinamideA MAO-B inhibitor used as an add-on treatment to levodopa/carbidopa for Parkinson's disease during "off" episodes.
SagopiloneSagopilone has been used in trials studying the treatment of Melanoma, Neoplasms, CNS Disease, Breast Cancer, and Breast Neoplasms, among others. It is a so-called fully synthetic epothilone and is...
SalmeterolA long-acting beta-2 adrenergic receptor agonist used to treat asthma and COPD.
SaquinavirAn HIV protease inhibitor used in combination with other antiretroviral agents for the treatment of HIV-1 with advanced immunodeficiency.
SaracatinibSaracatinib has been investigated for the treatment of Cancer, Osteosarcoma, Ovarian Cancer, Fallopian Tube Cancer, and Primary Peritoneal Cancer.
SarafloxacinSarafloxacin is a quinolone antibiotic drug, which was discontinued by its manufacturer, Abbott Laboratories, before receiving approval for use in the US or Canada.
SarilumabA monoclonal antibody used to treat moderate to severe rheumatoid arthritis who have responded poorly or are intolerant of other DMARDs.
Saw palmettoSaw palmetto is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.
SebetralstatA plasma kallikrein inhibitor indicated for the oral on-demand treatment of acute hereditary angioedema attacks in adults and pediatric patients aged 12 years and older, shown in phase 3 trials to provide faster symptom relief, reduced attack severity, and quicker resolution compared to placebo.
SecnidazoleA nitroimidazole antibiotic used to treat bacterial vaginosis.
SelamectinSelamectin is a topical parasiticide and antihelminthic used on dogs and cats to treat and prevent infections of heartworms, fleas, ear mites, sarcoptic mange, and certain types of ticks in...
SelegilineA monoamine oxidase inhibitor used to treat major depressive disorder and Parkinson's.
SelpercatinibA RET receptor tyrosine kinase inhibitor for the treatment of RET-driven non-small cell lung cancer, medullary thyroid cancer, and thyroid cancer in appropriate patient populations.
SeproxetineSeproxetine is also known as (S)-norfluoxetine. It is a selective serotonin reuptake inhibitor (SSRI). It is an active metabolite of fluoxetine. Seproxetine was being investigated by Eli Lilly as an...
SeratrodastSeratrodast (INN) is a thromboxane receptor antagonist used primarily in the treatment of asthma.
SertralineA selective serotonin reuptake inhibitor (SSRI) indicated to treat major depressive disorder, social anxiety disorder and many other psychiatric conditions.
SevabertinibA HER2 kinase inhibitor used to treat non-squamous non-small cell lung cancer with HER2 (ERBB2) tyrosine kinase domain (TKD) activating mutations.
SeviteronelSeviteronel has been used in trials studying the treatment of CRPC, Prostate Cancer, and Castration-resistant Prostate Cancer.
SildenafilA phosphodiesterase inhibitor used for the treatment of erectile dysfunction.
SiltuximabAn interleukin antagonist used to treat multicentric Castleman's disease (MCD) in patients who are HIV and HHV-8 negative.
SimeprevirA direct-acting antiviral agent that inhibits HCV NS3/4A protease to treat chronic hepatitis C virus (HCV) infection in adults with HCV genotype 1 or 4.
SimvastatinAn HMG-CoA reductase inhibitor used to lower lipid levels and reduce the risk of cardiovascular events including myocardial infarction and stroke.
SitafloxacinA fluoroquinolone antibiotic indicated in the treatment of susceptible bacterial infections.
SitaxentanInvestigated for use/treatment in pulmonary hypertension, connective tissue diseases, hypertension, and congestive heart failure.
SN-38Investigated for use/treatment in colorectal cancer.
SofpironiumA topical anticholinergic used to treat primary axillary hyperhidrosis.
SolithromycinInvestigated for the treatment of community-acquired pneumonia (CAP).
SomapacitanA human growth hormone analog subcutaneous injection indicated for adults with growth hormone deficiency.
SomatostatinA natural peptide hormone used to treat acute bleeding from esophageal varices, gastrointestinal ulcers, and gastritis; prevent pancreatic complications after surgery; and restrict secretions of the upper intestine, pancreas, and biliary tract.
SomatotropinA recombinant human growth hormone used as replacement therapy in various conditions of growth failure, growth hormone deficiency, and weakness in children and adults.
SonrotoclaxA selective oral BCL-2 inhibitor indicated for relapsed or refractory mantle cell lymphoma who have already tried a BTK inhibitor.
Sophora flavescens rootNot Annotated
SorafenibA kinase inhibitor used to treat unresectable liver carcinoma, advanced renal carcinoma, and differentiated thyroid carcinoma.
SotagliflozinAn orally administered dual SGLT1/2 inhibitor used alongside insulin to improve glycemic control in patients with type 1 diabetes mellitus.
SparfloxacinA fluoroquinolone antibiotic used to treat bacterial respiratory infections and sinusitis.
SparsentanAn endothelin and angiotensin II receptor antagonist indicated to reduce proteinuria in adults with primary immunoglobulin A nephropathy at risk of rapid disease progression.
SparteineSparteine is a plant alkaloid derived from Cytisus scoparius and Lupinus mutabilis which may chelate calcium and magnesium. It is a sodium channel blocker, so it falls in the category...
SpiramycinA macrolide antimicrobial agent used in the treatment of various bacterial infections.
SpironolactoneAn aldosterone receptor antagonist used to treat edema, hypertension, heart failure, and aldosteronism.
St. John's WortAn herbal ingredient used in non-prescription therapeutic products for the short-term treatment of minor skin irritations, insomnia, depression, and anxiety.
StiripentolAn antiepileptic agent used in combination with other anticonvulsants to treat seizures associated with Dravet syndrome.
SulconazoleA topical antifungal agent used for the treatment of tinea cruris, tinea corporis, and tinea versicolor caused by susceptible fungal strains.
SulfadiazineA sulfonamide antibiotic used in a variety of infections, such as urinary tract infections, trachoma, and chancroid.
SulfadimethoxineFor use in the treatment of infections.
SulfamethizoleA sulfonamide antibiotic used to treat a wide variety of susceptible bacterial infections.
SulfamethoxazoleAn oral sulfonamide antibiotic, given in combination with trimethoprim, used to treat a variety of infections of the urinary tract, respiratory system, and gastrointestinal tract.
SulfamoxoleFor the treatment of bacterial infection.
SulfanilamideA sulfonamide anti-infective used to treat vulvovaginal candidiasis caused by Candida albicans.
SulfaphenazoleFor the treatment bacterial infections.
SulfapyridineA sulfonamide antibiotic used to treat dermatitis herpetiformis, benign mucous membrane pemphigoid and pyoderma gangrenosum.
SulfinpyrazoneA platelet inhibitory and uricosuric agent used to inhibit thrombotic and embolic processes and to manage the chronic phases of gout .
SulfisoxazoleA sulfonamide antibiotic used with other antibiotics to prevent and treat a variety of bacterial infections.
SulforaphaneSulforaphane is under investigation for the treatment of Autism Spectrum Disorder. It is a naturally occurring isothiocyanate found in high concentration in a variety of broccoli.
SunitinibA receptor tyrosine kinase inhibitor and chemotherapeutic agent used for the treatment of renal cell carcinoma (RCC) and imatinib-resistant gastrointestinal stromal tumor (GIST).
SuprofenAn NSAID used to prevent pupil constriction in ocular surgery.
SuvorexantA orexin receptor antagonist used to treat insomnia that is characterized by difficulties with sleep onset and/or sleep maintenance.
SuzetrigineA sodium channel blocker used to treat moderate to severe acute pain in adults.
TabimorelinTabimorelin is a small molecule drug. The usage of the INN stem '-relin' in the name indicates that Tabimorelin is a pituitary hormone-release stimulating peptide. Tabimorelin has a monoisotopic molecular...
TacrolimusA calcineurin inhibitor used to prevent organ transplant rejection and to treat moderate to severe atopic dermatitis.
TalarozoleTalarozole has been investigated for the treatment of Psoriasis and Cutaneous Inflammation.
TaletrectinibA small molecule ROS1 inhibitor for use in patients with advanced forms of ROS1-positive non-small cell lung cancer.
TamoxifenA selective estrogen receptor modulator used to treat estrogen receptor positive breast cancer, reduce the risk of invasive breast cancer following surgery, or reduce the risk of breast cancer in high risk women.
Tanshinone INot Annotated
TasisulamTasisulam has been used in trials studying the treatment and basic science of Melanoma, Lymphoma, Solid Tumors, Breast Cancer, and Ovarian Cancer, among others.
Technetium Tc-99m ciprofloxacinInvestigated for use/treatment in infectious and parasitic disease (unspecified).
TecovirimatAn antiviral medication used to treat smallpox, monkeypox, and cowpox.
TegaserodA serotonin-4 (5-HT4) receptor agonist indicated for the treatment of constipation predominant irritable bowel syndrome (IBS-C) specifically in women under the age of 65. There is currently no safety or efficacy data for use of tegaserol in men.
TelaprevirAn NS3/4A viral protease inhibitor used in combination with other antivirals for the curative treatment of chronic Hepatitis C Virus infections.
Telisotuzumab vedotinAn chemotherapeutic antibody-drug conjugate comprising a c-Met-directed antibody with a microtubule-disrupting small molecule payload.
TelithromycinAn ketolide used to treat community acquired pneumonia of mild to moderate severity.
TelmisartanAn ARB used to treat hypertension, diabetic nephropathy, and congestive heart failure.
Telotristat ethylA tryptophan hydroxylase inhibitor that is used to treat carcinoid syndrome diarrhea.
TemafloxacinFor the treatment of lower respiratory tract infections, genital and urinary infections like prostatitis, and skin infections.
TemsirolimusA antineoplastic agent used in the treatment of renal cell carcinoma (RCC) that works by inhibiting mTOR.
TeniposideA cytotoxic drug used as an adjunct for chemotherapy induction in the treatment of refractory childhood acute lymphoblastic leukemia.
TepotinibAn oral tyrosine kinase inhibitor targeted against MET for the treatment of metastatic non-small cell lung cancer in patients exhibiting MET exon 14 skipping mutations.
TerbinafineAn allylamine antifungal used to treat dermatophyte infections of toenails and fingernails as well as other fungal skin infections.
TerfenadineAn antihistamine for the treatment of allergy symptoms.
TeriflunomideA pyrimidine synthesis inhibitor with anti-inflammatory and immunomodulatory properties used to treat patients with the relapsing-remitting form of multiple sclerosis.
TesmilifeneIntended for the treatment of various forms of cancer.
Testosterone cypionateAn androgen used to treat low or absent testosterone.
Testosterone enanthateAn androgen used to treat low or absent testosterone.
Testosterone undecanoateAn androgen indicated for testosterone replacement therapy in adult males with primary hypogonadism and hypogonadotropic hypogonadism.
TetracyclineAn antibiotic used to treat a wide variety of susceptible infections.
TezacaftorA CFTR corrector used to treat cystic fibrosis in patients with susceptible mutations (e.g. F508del).
ThalidomideA medication used to treat cancers, particularly newly diagnosed multiple myeloma, and erythema nodosum leprosum.
ThiabendazoleA benzimidazole used in the treatment of strongyloides, cutaneous larva migrans, visceral larva migrans, and trichinosis infections.
ThiopentalA barbiturate used to induce general anesthesia, treat convulsions, and reduce intracranial pressure.
ThioridazineA phenothiazine antipsychotic used to treat schizophrenia and generalized anxiety disorder.
ThiotepaAn alkylating agent used to prevent graft rejection in stem cell transplantation and to treat a variety of malignancies including certain types of adenocarcinoma and superficial bladder carcinomas.
ThiothixeneAn antipsychotic indicated for the management of schizophrenia.
TiamulinTiamulin is a pleuromutilin antibiotic drug that is used in veterinary medicine particularly for pigs and poultry.
TicagrelorA P2Y12 platelet inhibitor used in patients with a history of myocardial infarction or with acute coronary syndrome (ACS) to prevent future myocardial infarction, stroke and cardiovascular death.
TiclopidineA platelet aggregation inhibitor used in the prevention of conditions associated with thrombi, such as stroke and transient ischemic attacks (TIA).
Tienilic acidFor the treatment of hypertension.
TildipirosinTildipirosin is a veterinary antibiotic.
TilidineA synthetic opioid indicated in the treatment of severe pain.
TioconazoleAn imidazole antifungal used to treat vulvovaginal candidiasis.
TipranavirA protease inhibitor used to treat HIV-1 resistant to more than 1 protease inhibitor.
TirbanibulinA tyrosine kinase and tubulin inhibitor used to treat actinic keratosis on the face or scalp.
TocainideAn orally active class 1b antiarrhythmic agent that interferes with cardiac sodium channels and typically used to treat ventricular arrhythmias.
TofisopamFor the treatment of anxiety and alcohol withdrawal.
TolbutamideA sulfonylurea used to treat hyperglycemia in patients with type 2 diabetes mellitus.
TolcaponeA catechol-O-methyltransferase (COMT) inhibitor used as adjunct therapy in the symptomatic management of idiopathic Parkinson's disease.
TopiramateAn anticonvulsant drug used in the control of epilepsy and in the prophylaxis and treatment of migraines.
TopiroxostatIndicated for the treatment of gout and hyperurcemia in Japan.
TopotecanAn antineoplastic agent used to treat ovarian cancer, small cell lung cancer, or cervical cancer.
TorasemideA diuretic used to treat hypertension and edema associated with heart failure, renal failure, or liver disease.
ToremifeneA first generation nonsteroidal selective estrogen receptor modulator used to treat certain breast cancers.
TovorafenibA type II RAF inhibitor used to treat pediatric low-grade glioma with BRAF gene mutations.
TradipitantA substance P receptor antagonist used to prevent motion-induced vomiting in adults.
TrametinibA kinase inhibitor used alone or in combination with dabrafenib to treat patients with cancers with specific BRAF mutations, such as melanoma and non-small cell lung cancer.
TranylcypromineA monoamine oxidase inhibitor used to treat major depressive disorder.
TrazodoneA serotonin uptake inhibitor used to treat major depressive disorder.
TreosulfanA DNA alkylating agent used in the context of myeloablative conditioning prior to allogeneic hemoatopoietic stem cell transplantation.
TriazolamA benzodiazepine used for short term treatment of insomnia.
TrichloroethyleneTrichloroethylene is a halocarbon commonly used as an industrial solvent, not to be confused with the similar 1,1,1-trichloroethane, also known as chlorothene. It has been sold under a variety of...
TriclabendazoleAn anthelmintic drug used to treat fascioliasis.
TrilaciclibA CDK4 and CDK6 inhibitor to reduce the risk of chemotherapy induced myelosuppression.
TrimethoprimAn antifolate antibiotic often used in combination with sulfamethoxazole to treat a number of infections, including those of the urinary tract, respiratory tract, and gastrointestinal tract.
TripelennamineA histamine H1 antagonist used to treat hypersensitivity reactions, coughs, and the common cold.
TrofinetideA drug used to treat Rett syndrome in children and adults.
TroglitazoneFor the treatment of Type II diabetes mellitus. It is used alone or in combination with a sulfonylurea, metformin, or insulin as an adjunct to diet and exercise.
TroleandomycinFor the treatment of bacterial infection.
TrospiumAn antimuscarinic agent used to treat the symptoms of overactive bladder (OAB).
TrovafloxacinAn antibiotic used to treat gonorrhea and chlamydia.
TucatinibA kinase inhibitor used to treat certain types of unresectable/metastatic HER-2 positive breast cancer.
UbrogepantAn oral CGRP antagonist used in the acute treatment of migraine with or without aura.
VadadustatAn oral hypoxia-inducible factor prolyl-hydroxylase inhibitor used to treat symptomatic anemia associated with chronic kidney disease in adults on chronic maintenance dialysis.
ValdecoxibA COX-2 inhibitor used to treat osteoarthritis and dysmenorrhoea.
Valproic acidAn anticonvulsant used to control complex partial seizures and both simple and complex absence seizures.
ValsartanAn angiotensin-receptor blocker used to manage hypertension alone or in combination with other antihypertensive agents and to manage heart failure in patients who are intolerant to ACE inhibitors.
VapreotideFor the treatment of esophageal variceal bleeding in patients with cirrhotic liver disease and has also shown efficacy in the treatment of patients with AIDS-related diarrhea.
VardenafilA phosphodiesterase 5 inhibitor used to treat erectile dysfunction.
VayarinADHD in children, hypertriglyceridemia .
VemurafenibA kinase inhibitor used to treat patients with Erdheim-Chester Disease who have the BRAF V600 mutation, and melanoma in patients who have the BRAF V600E mutation.
VenetoclaxA BCL-2 inhibitor used to treat chronic lymphocytic leukemia, small lymphocytic lymphoma, or acute myeloid leukemia.
VenlafaxineA selective serotonin and norepinephrine reuptake inhibitor (SNRI) used for the treatment of major depression, generalized or social anxiety disorder, and panic disorder.
VepdegestrantAn oral proteolysis-targeting chimera (PROTAC) estrogen receptor degrader used to treat adults with estrogen receptor (ER)-positive, human epidermal growth factor receptor 2 (HER2)-negative, ESR1-mutated advanced or metastatic breast cancer.
VerapamilA non-dihydropyridine calcium channel blocker used in the treatment of angina, arrhythmia, and hypertension.
VernakalantAn antiarrhythmic medication used to treat patients with atrial fibrillation.
VilazodoneAn antidepressant agent used for the treatment of major depressive disorder that targets the 5-HT transporter and 5-HT1A receptors.
ViloxazineA selective norepinephrine reuptake inhibitor indicated for the treatment of Attention Deficit Hyperactivity Disorder (ADHD) in adults in children.
VinblastineA vinca alkaloid used to treat breast cancer, testicular cancer, neuroblastoma, Hodgkin's and non-Hodgkins lymphoma, mycosis fungoides, histiocytosis, and Kaposi's sarcoma.
VinorelbineA vinca alkaloid used in the treatment of metastatic non-small cell lung carcinoma (NSLC) and in conjunction with other drugs in locally advanced NSCLC.
VismodegibA hedgehog pathway inhibitor used to treat patients with locally advanced or metastatic basal cell carcinoma.
Vitis vinifera seedNot Annotated
VoclosporinA calcineurin inhibitor for the treatment of lupus nephritis (LN) in patients diagnosed with systemic lupus erythematosus (SLE).
VonoprazanA potassium-competitive acid blocker used in the treatment of acid-related disorders and as an adjunct to Helicobacter pylori eradication.
VoriconazoleA triazole compound used to treat fungal infections.
WarfarinA vitamin K antagonist used to treat venous thromboembolism, pulmonary embolism, thromboembolism with atrial fibrillation, thromboembolism with cardiac valve replacement, and thromboembolic events post myocardial infarction.
WIN 55212-2WIN 55,212-2 is a chemical described as an aminoalkylindole derivative, which produces effects similar to those of cannabinoids such as tetrahydrocannabinol (THC) but has an entirely different chemical structure. It...
XanomelineA muscarinic agonist used in conjunction with trospium, a muscarinic antagonist, to treat schizophrenia.
ZafirlukastA leukotriene receptor antagonist used for prophylaxis and chronic treatment of asthma.
ZileutonA leukotriene synthesis inhibitor used in the prophylaxis and treatment of chronic asthma.
ZimelidineFor the treatment of depression.
ZiprasidoneAn atypical antipsychotic used to manage schizophrenia, bipolar mania, and agitation in patients with schizophrenia.
ZonisamideA sulfonamide anticonvulsant used to treat partial seizures.
ZucapsaicinA topical analgesic used as an adjunct to relieve severe pain of osteoarthritis of the knee in selected adult patients.
Drugs & Drug Targets
DrugTargetType
(5-(PYRIDIN-3-YL)FURAN-2-YL)METHANAMINECytochrome P450 2D6target
(5-(PYRIDIN-3-YL)FURAN-2-YL)METHANAMINECytochrome P450 2A6target
1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidineCytochrome P450 2D6enzyme
6-Deoxyerythronolide B6-deoxyerythronolide B hydroxylasetarget
6-Deoxyerythronolide BCytochrome P450 3A4enzyme
AbametapirCytochrome P450 2B6enzyme
AbametapirCytochrome P450 3A4enzyme
AbametapirCytochrome P450 1A2enzyme
AbemaciclibCytochrome P450 2D6enzyme
AbemaciclibCytochrome P450 2C9enzyme
AbemaciclibCytochrome P450 2C8enzyme
AbemaciclibCytochrome P450 2B6enzyme
AbemaciclibCytochrome P450 1A2enzyme
AbemaciclibSolute carrier family 22 member 2transporter
AbemaciclibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
AbemaciclibATP-dependent translocase ABCB1transporter
AbemaciclibCytochrome P450 3A4enzyme
Abemaciclibalpha1-acid glycoproteincarrier
AbemaciclibAlbumincarrier
AbemaciclibCyclin-dependent kinase 6target
AbemaciclibCyclin-dependent kinase 4target
AbemaciclibMultidrug and toxin extrusion protein 2transporter
AbemaciclibMultidrug and toxin extrusion protein 1transporter
AbirateroneCytochrome P450 2C8enzyme
AbirateroneCytochrome P450 2D6enzyme
AbirateroneMultidrug resistance-associated protein 1transporter
Abiraterone3-oxo-5-alpha-steroid 4-dehydrogenasetarget
AbirateroneAndrogen receptortarget
AbirateroneSolute carrier organic anion transporter family member 1B1transporter
AbirateroneCytochrome P450 3A5enzyme
AbirateroneCytochrome P450 2C9enzyme
AbirateroneCytochrome P450 2C19enzyme
AbirateroneCytochrome P450 1A2enzyme
AbirateroneSteroid 17-alpha-hydroxylase/17,20 lyasetarget
AbirateroneAlbumincarrier
AbirateroneAlpha-1-acid glycoprotein 1carrier
AbirateroneCytochrome P450 3A4enzyme
AbirateroneSulfotransferase 2A1enzyme
AcalabrutinibCytochrome P450 3A Subfamilyenzyme
AcalabrutinibTyrosine-protein kinase BTKtarget
AcalabrutinibCytochrome P450 3A4enzyme
Acalabrutinibalpha1-acid glycoproteincarrier
AcalabrutinibAlbumincarrier
AcalabrutinibCytochrome P450 3A5enzyme
AcebutololATP-dependent translocase ABCB1transporter
AcebutololBeta-2 adrenergic receptortarget
AcebutololCytochrome P450 2D6enzyme
AcebutololBeta-1 adrenergic receptortarget
AcetaminophenUDP-glucuronosyltransferase 1A6enzyme
AcetaminophenUDP-glucuronosyltransferase 1A9enzyme
AcetaminophenUDP-glucuronosyltransferase 2B15enzyme
AcetaminophenSulfotransferase 1A1enzyme
AcetaminophenSulfotransferase 1A3enzyme
AcetaminophenArylamine N-acetyltransferase 2enzyme
AcetaminophenProstaglandin E synthase 3target
AcetaminophenTransient receptor potential cation channel subfamily V member 1target
AcetaminophenAlbumincarrier
AcetaminophenFatty-acid amide hydrolase 1enzyme
AcetaminophenGlutathione S-transferase Penzyme
AcetaminophenGlutathione S-transferase Mu 1enzyme
AcetaminophenSodium-dependent noradrenaline transportertarget
AcetaminophenSodium-dependent serotonin transportertarget
AcetaminophenHuman Cyclooxygenasestarget
AcetaminophenFatty-acid amide hydrolase 1target
AcetaminophenUDP-glucuronosyltransferase 1A1enzyme
AcetaminophenCytochrome P450 3A4enzyme
AcetaminophenCytochrome P450 2A6enzyme
AcetaminophenCytochrome P450 2D6enzyme
AcetaminophenATP-dependent translocase ABCB1transporter
AcetaminophenCytochrome P450 2E1enzyme
AcetaminophenCytochrome P450 1A2enzyme
AcetaminophenProstaglandin G/H synthase 2target
AcetaminophenProstaglandin G/H synthase 1target
AcetazolamideCarbonic anhydrase 1target
AcetazolamideAquaporin-1target
AcetazolamideCarbonic anhydrase 14target
AcetazolamideSolute carrier family 22 member 6transporter
AcetazolamideCarbonic anhydrase 2target
AcetazolamideCarbonic anhydrase 3target
AcetazolamideCarbonic anhydrase 4target
AcetazolamideCytochrome P450 3A4enzyme
AcetazolamideCarbonic anhydrase 7target
AcetazolamideCarbonic anhydrase 12target
Acetyl sulfisoxazoleCytochrome P450 2C9enzyme
Acetyl sulfisoxazoleDihydropteroate synthasetarget
AcoramidisOrganic anion transporter 3transporter
AcoramidisBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
AcoramidisSolute carrier family 22 member 6transporter
AcoramidisUDP-glucuronosyltransferase 2B7enzyme
AcoramidisUDP-glucuronosyltransferase 1A1enzyme
AcoramidisUDP-glucuronosyltransferase 1A9enzyme
AcoramidisCytochrome P450 2C9enzyme
AcoramidisTransthyretintarget
AdagrasibATP-dependent translocase ABCB1transporter
AdagrasibCytochrome P450 2D6enzyme
AdagrasibCytochrome P450 2C9enzyme
AdagrasibCytochrome P450 2B6enzyme
AdagrasibCytochrome P450 1A2enzyme
AdagrasibCytochrome P450 2C8enzyme
AdagrasibCytochrome P450 3A4enzyme
AdagrasibGTPase KRastarget
AdemetionineS-adenosylmethionine decarboxylase proenzymetarget
AdemetionineGlycine N-methyltransferasetarget
AdemetionineS-adenosylmethionine synthase isoform type-2target
AdemetionineCystathionine beta-synthasetarget
AdemetionineS-adenosylmethionine synthase isoform type-1target
AdemetionineCytochrome P450 2E1enzyme
AdemetionineCatechol O-methyltransferasetarget
AdemetionineSpermidine synthaseenzyme
AdemetionineCap-specific mRNA (nucleoside-2'-O-)-methyltransferase 1target
AdemetionineArsenite methyltransferasetarget
AgomelatineCytochrome P450 1A2enzyme
AgomelatineCytochrome P450 2C9enzyme
AgomelatineMelatonin receptor type 1Atarget
AgomelatineMelatonin receptor type 1Btarget
Agomelatine5-hydroxytryptamine receptor 2Ctarget
Albinterferon Alfa-2BCytochrome P450 1A2enzyme
AlbuterolBeta-2 adrenergic receptortarget
AlbuterolBeta-3 adrenergic receptortarget
AlbuterolCytochrome P450 3A4enzyme
AlbuterolBeta-1 adrenergic receptortarget
AldesleukinInterleukin-2target
AldesleukinCytochrome P450 2E1enzyme
AldesleukinXanthine dehydrogenase/oxidaseenzyme
AldesleukinCytochrome P450 3A4enzyme
AldesleukinCytosolic phospholipase A2enzyme
AldesleukinProstaglandin G/H synthase 2enzyme
AldesleukinCytokine receptor common subunit gammatarget
AldesleukinInterleukin-2 receptor subunit alphatarget
AldesleukinInterleukin-2 receptor subunit betatarget
AllicinTransient receptor potential cation channel subfamily A member 1target
AllicinTransient receptor potential cation channel subfamily V member 1target
AllicinATP-dependent translocase ABCB1transporter
AllicinCytochrome P450 3A4enzyme
AllicinAcetylcholinesterasetarget
AllicinCholinesterasetarget
AllopurinolAldehyde oxidaseenzyme
AllopurinolCytochrome P450 1A2enzyme
AllopurinolSolute carrier family 22 member 2transporter
AllopurinolBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
AllopurinolXanthine dehydrogenase/oxidaseenzyme
AllopurinolXanthine dehydrogenase/oxidasetarget
AllopurinolOrganic anion transporter 3transporter
AllopurinolSolute carrier family 22 member 7transporter
AlmonertinibCytochrome P450 1A2enzyme
AlmonertinibCytochrome P450 2A6enzyme
AlmonertinibAlbumincarrier
AlmonertinibAlpha-1-acid glycoprotein 1carrier
AlmonertinibSolute carrier organic anion transporter family member 1B1transporter
AlmonertinibSolute carrier family 22 member 6transporter
AlmonertinibSolute carrier family 22 member 2transporter
AlmonertinibATP-dependent translocase ABCB1transporter
AlmonertinibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
AlmonertinibUDP-glucuronosyltransferase 1A1enzyme
AlmonertinibUDP-glucuronosyltransferase 2B7enzyme
AlmonertinibMultidrug and toxin extrusion protein 1transporter
AlmonertinibSolute carrier family 22 member 1transporter
AlmonertinibCytochrome P450 3A5enzyme
AlmonertinibCytochrome P450 3A4enzyme
AlmonertinibEpidermal growth factor receptortarget
AlmonertinibReceptor protein-tyrosine kinasetarget
Alosetron5-hydroxytryptamine receptor 3Atarget
AlosetronCytochrome P450 1A2enzyme
AlosetronCytochrome P450 2C9enzyme
AlosetronCytochrome P450 3A4enzyme
AlosetronCytochrome P450 2E1enzyme
Alosetron5-hydroxytryptamine receptor 3Btarget
AlpelisibEstrogen receptortarget
AlpelisibPhosphatidylinositol 3-kinasetarget
AlpelisibATP-dependent translocase ABCB1transporter
AlpelisibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
AlpelisibCytochrome P450 2C19enzyme
AlpelisibCytochrome P450 2C8enzyme
AlpelisibCytochrome P450 2C9enzyme
AlpelisibCytochrome P450 3A4enzyme
AlpelisibPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoformtarget
AlpibectirBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
AlpibectirATP-dependent translocase ABCB1transporter
AlpibectirCytochrome P450 3A4enzyme
AminophenazoneMyeloperoxidaseenzyme
AminophenazoneCytochrome P450 2C19enzyme
AminophenazoneCytochrome P450 1A2enzyme
AminophenazoneCytochrome P450 2C8enzyme
AminophenazoneSolute carrier family 22 member 6transporter
AminophenazoneCytochrome P450 2C9enzyme
AminophenazoneCytochrome P450 2D6enzyme
AminophenazoneCytochrome P450 3A4enzyme
AminophenazoneProstaglandin G/H synthase 1target
AminophenazoneSteroid 17-alpha-hydroxylase/17,20 lyaseenzyme
AminophenazoneCytochrome P450 2C18enzyme
AmiodaroneAlbumincarrier
AmiodaroneVoltage-gated inwardly rectifying potassium channel KCNH2target
AmiodaronePeroxisome proliferator-activated receptor gamma coactivator 1-betatarget
AmiodaronePeroxisome proliferator-activated receptor alphatarget
AmiodaroneCytochrome P450 2J2enzyme
AmiodaroneSolute carrier family 22 member 2transporter
AmiodaroneBile salt export pumptransporter
AmiodaronePeroxisome proliferator-activated receptor gammatarget
AmiodaroneThyroid hormone receptortarget
AmiodaroneCytochrome P450 2A6enzyme
AmiodaroneCytochrome P450 2C19enzyme
AmiodaroneATP-dependent translocase ABCB1transporter
AmiodaroneCytochrome P450 1A1enzyme
AmiodaroneCytochrome P450 1A2enzyme
AmiodaroneCytochrome P450 3A4enzyme
AmiodaroneVoltage gated L-type calcium channeltarget
AmiodaroneVoltage-dependent T-type calcium channel subunit alpha-1Itarget
AmiodaroneCytochrome P450 2D6enzyme
AmiodaroneBeta adrenergic receptortarget
AmiodaroneHERG human cardiac K+ channeltarget
AmiodaroneCytochrome P450 2C8enzyme
AmiodaroneCytochrome P450 2C9enzyme
Amitriptyline5-hydroxytryptamine receptor 1Dtarget
Amitriptyline5-hydroxytryptamine receptor 7target
AmitriptylineAlpha-1B adrenergic receptortarget
Amitriptyline5-hydroxytryptamine receptor 2Ctarget
AmitriptylineSigma non-opioid intracellular receptor 1target
AmitriptylineHistamine H4 receptortarget
AmitriptylineHistamine H2 receptortarget
AmitriptylineCytochrome P450 2C8enzyme
AmitriptylineCytochrome P450 2B6enzyme
AmitriptylineCytochrome P450 2C9enzyme
AmitriptylineBDNF/NT-3 growth factors receptortarget
AmitriptylineHigh affinity nerve growth factor receptortarget
AmitriptylineKappa-type opioid receptortarget
AmitriptylineDelta-type opioid receptortarget
AmitriptylineAlpha-1D adrenergic receptortarget
AmitriptylinePotassium voltage-gated channel subfamily A member 1target
AmitriptylineCytochrome P450 3A5enzyme
AmitriptylineCytochrome P450 3A4enzyme
AmitriptylineAlpha-1A adrenergic receptortarget
Amitriptyline5-hydroxytryptamine receptor 1Atarget
Amitriptyline5-hydroxytryptamine receptor 2Atarget
AmitriptylineMu-type opioid receptortarget
Amitriptyline5-hydroxytryptamine receptor 1Btarget
Amitriptyline5-hydroxytryptamine receptor 6target
AmitriptylinePotassium voltage-gated channel subfamily KQT member 3target
AmitriptylineHistamine H1 receptortarget
AmitriptylineAlpha-1-acid glycoprotein 1carrier
AmitriptylineAlbumincarrier
AmitriptylineCytochrome P450 2D6enzyme
AmitriptylineCytochrome P450 2C19enzyme
AmitriptylineCytochrome P450 1A2enzyme
AmitriptylineAlpha-2A adrenergic receptortarget
AmitriptylinePotassium voltage-gated channel subfamily KQT member 2target
AmitriptylineSodium-dependent noradrenaline transportertarget
AmitriptylineSodium-dependent serotonin transportertarget
AmitriptylineUDP-glucuronosyltransferase 2B10enzyme
Amitriptyline5-hydroxytryptamine receptor 2Ctarget
AmitriptylineMuscarinic acetylcholine receptortarget
AmitriptylineHERG human cardiac K+ channeltarget
AmitriptylineATP-dependent translocase ABCB1transporter
AmitriptylineUDP-glucuronosyltransferase 1A4enzyme
AmitriptylineGlutathione S-transferases (Cytosolic)enzyme
AmlodipineVoltage gated L-type calcium channeltarget
AmlodipineVoltage-dependent calcium channel subunit alpha-2/delta-1target
AmlodipineCytochrome P450 2C9enzyme
AmlodipineCytochrome P450 2C19enzyme
AmlodipineVoltage-dependent N-type calcium channeltarget
AmlodipineVoltage-dependent T-type calcium channel subunit alpha-1Itarget
AmlodipineSphingomyelin phosphodiesterasetarget
AmlodipineCytochrome P450 2D6enzyme
AmlodipineCytochrome P450 2C8enzyme
AmlodipineATP-dependent translocase ABCB1transporter
AmlodipineCytochrome P450 3A5enzyme
AmlodipineVoltage-dependent calcium channel subunit alpha-2/delta-3target
AmlodipineVoltage-dependent L-type calcium channel subunit beta-1target
AmlodipineVoltage-dependent N-type calcium channel subunit alpha-1Btarget
AmlodipineCytochrome P450 2B6enzyme
AmlodipineCytochrome P450 1A1enzyme
AmlodipineVoltage-dependent L-type calcium channel subunit alpha-1Ctarget
AmlodipineCytochrome P450 3A4enzyme
AmlodipineCarbonic anhydrase 1target
AmodiaquineATP-dependent translocase ABCB1transporter
AmodiaquineCytochrome P450 2C9enzyme
AmodiaquineCytochrome P450 1B1enzyme
AmodiaquineCytochrome P450 1A1enzyme
AmodiaquineFe(II)-protoporphyrin IXtarget
AmodiaquineCytochrome P450 2D6enzyme
AmodiaquineCytochrome P450 2C8enzyme
AmodiaquineHistamine N-methyltransferasetarget
AmoxapineGamma-aminobutyric acid receptor subunit alpha-1target
Amoxapine5-hydroxytryptamine receptor 7target
AmoxapineSodium-dependent dopamine transportertarget
AmoxapineGABA(A) Receptortarget
AmoxapineHistamine H4 receptortarget
AmoxapineAlpha-2 adrenergic receptorstarget
Amoxapine5-hydroxytryptamine receptor 1Btarget
Amoxapine5-hydroxytryptamine receptor 1Atarget
Amoxapine5-hydroxytryptamine receptor 3Atarget
Amoxapine5-hydroxytryptamine receptor 2Btarget
AmoxapineMuscarinic acetylcholine receptortarget
AmoxapineAlpha-1 adrenergic receptorstarget
AmoxapineHistamine H1 receptortarget
AmoxapineD(4) dopamine receptortarget
AmoxapineD(3) dopamine receptortarget
Amoxapine5-hydroxytryptamine receptor 6target
Amoxapine5-hydroxytryptamine receptor 2Ctarget
Amoxapine5-hydroxytryptamine receptor 2Atarget
AmoxapineCytochrome P450 2D6enzyme
AmoxapineAlpha-1-acid glycoprotein 1carrier
AmoxapineMuscarinic acetylcholine receptor M1target
AmoxapineD(1A) dopamine receptortarget
AmoxapineAlpha-1A adrenergic receptortarget
AmoxapineD(2) dopamine receptortarget
AmoxapineAlpha-2A adrenergic receptortarget
AmoxapineSodium-dependent noradrenaline transportertarget
AmoxapineSodium-dependent serotonin transportertarget
AmoxapineDopamine receptortarget
AmoxicillinSolute carrier family 15 member 2transporter
AmoxicillinPenicillin-binding proteintarget
AmoxicillinPenicillin binding proteintarget
AmoxicillinMetallo-beta-lactamase type 2enzyme
AmoxicillinAlbumincarrier
AmoxicillinCytochrome P450 2C8enzyme
AmoxicillinSolute carrier family 22 member 6transporter
AmoxicillinSolute carrier family 15 member 1transporter
AmphetamineD(2) dopamine receptortarget
AmphetamineBeta adrenergic receptortarget
AmphetamineAlpha adrenergic receptortarget
AmphetamineSodium-dependent noradrenaline transportertarget
AmphetamineCytochrome P450 2A6enzyme
AmphetamineSynaptic vesicular amine transportertarget
AmphetamineOrganic cation/carnitine transporter 2transporter
AmphetamineSolute carrier family 22 member 3transporter
AmphetamineCytochrome P450 2D6enzyme
AmphetamineTrace amine-associated receptor 1target
AmphetamineCocaine- and amphetamine-regulated transcript proteintarget
AmphetamineSodium-dependent dopamine transportertarget
AmphetamineAmine oxidase [flavin-containing] Btarget
AmphetamineSodium-dependent serotonin transportertarget
AmphetamineMonoamine oxidasetarget
AmprenavirCytochrome P450 2C19enzyme
AmprenavirPol polyproteintarget
AmprenavirCytochrome P450 3A4enzyme
AmprenavirATP-dependent translocase ABCB1transporter
AmprenavirMultidrug resistance-associated protein 1transporter
AmprenavirCytochrome P450 2B6enzyme
AmprenavirCytochrome P450 2C9enzyme
AmprenavirCytochrome P450 2D6enzyme
AmprenavirCytochrome P450 3A5enzyme
AmprenavirSolute carrier organic anion transporter family member 1B1transporter
AmprenavirGag-Pol polyproteintarget
AnacaulaseAlpha-1-antichymotrypsintarget
AnacaulaseAlpha-2-macroglobulintarget
AnacaulaseCytochrome P450 2C9enzyme
AnacaulaseCytochrome P450 2C8enzyme
AnagrelidecGMP-inhibited 3',5'-cyclic phosphodiesterase 3Atarget
AnagrelideCytochrome P450 1A2enzyme
AnagrelidePhosphodiesterase 3target
AnastrozoleCytochrome P450 2C9enzyme
AnastrozoleCytochrome P450 1A2enzyme
AnastrozoleUDP-glucuronosyltransferase 2B7enzyme
AnastrozoleUDP-glucuronosyltransferase 1A3enzyme
AnastrozoleUDP-glucuronosyltransferase 1A4enzyme
AnastrozoleCytochrome P450 2C8enzyme
AnastrozoleCytochrome P450 3A5enzyme
AnastrozoleCytochrome P450 3A4enzyme
AnastrozoleATP-dependent translocase ABCB1transporter
AnastrozoleAromatasetarget
Angelica sinensis rootCytochrome P450 2C19enzyme
Angelica sinensis rootCytochrome P450 2C11enzyme
AntipyrineCytochrome P450 2C8enzyme
AntipyrineCytochrome P450 2C9enzyme
AntipyrineCytochrome P450 1A2enzyme
AntipyrineCytochrome P450 2C19enzyme
AntipyrineCytochrome P450 3A4enzyme
AntipyrineSolute carrier family 22 member 6transporter
AntipyrineCytochrome P450 2A6enzyme
AntipyrineCytochrome P450 2B6enzyme
AntipyrineCytochrome P450 2C18enzyme
AntipyrineCytochrome P450 2D6enzyme
AntipyrineCytochrome P450 2E1enzyme
AntipyrineProstaglandin G/H synthase 2target
AntipyrineProstaglandin G/H synthase 1target
AprepitantCytochrome P450 2C19enzyme
AprepitantCytochrome P450 2C9enzyme
AprepitantCytochrome P450 3A4enzyme
AprepitantSubstance-P receptortarget
AprocitentanBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
AprocitentanATP-dependent translocase ABCB1transporter
AprocitentanCytochrome P450 2C19enzyme
AprocitentanCytochrome P450 2C18enzyme
AprocitentanCytochrome P450 2C9enzyme
AprocitentanCytochrome P450 2C8enzyme
AprocitentanCytochrome P450 3A4enzyme
AprocitentanAlbumincarrier
AprocitentanUDP-glucuronosyltransferase 2B7enzyme
AprocitentanUDP-glucuronosyltransferase 1A1enzyme
AprocitentanEndothelin receptor type Btarget
AprocitentanEndothelin-1 receptortarget
AprocitentanBile salt export pumptransporter
AprocitentanHepatic sodium/bile acid cotransportertransporter
ArmodafinilAlpha-1D adrenergic receptortarget
ArmodafinilSodium-dependent dopamine transportertarget
ArmodafinilCytochrome P450 2C9enzyme
ArmodafinilCytochrome P450 3A5enzyme
ArmodafinilCytochrome P450 2B6enzyme
ArmodafinilCytochrome P450 1A2enzyme
ArmodafinilCytochrome P450 3A4enzyme
ArmodafinilCytochrome P450 2C19enzyme
Arsenic trioxideProtein PMLtarget
Arsenic trioxideInhibitor of nuclear factor kappa-B kinase subunit betatarget
Arsenic trioxideTranscription factor Juntarget
Arsenic trioxideG1/S-specific cyclin-D1target
Arsenic trioxideMitogen-activated protein kinase 3target
Arsenic trioxideMitogen-activated protein kinase 1target
Arsenic trioxideRAC-alpha serine/threonine-protein kinasetarget
Arsenic trioxideATP-binding cassette sub-family C member 2transporter
Arsenic trioxideThioredoxin reductase 1, cytoplasmictarget
Arsenic trioxideATP-dependent translocase ABCB1transporter
Arsenic trioxideCytochrome P450 3A4enzyme
Arsenic trioxideCyclin-dependent kinase inhibitor 1target
Arsenic trioxideAlbumincarrier
ArtefenomelCytochrome P450 3A4enzyme
ArtefenomelCytochrome P450 3A Subfamilyenzyme
ArtenimolSmall ribosomal subunit protein eS19target
ArtenimolSmall ribosomal subunit protein uS13target
ArtenimolSmall ribosomal subunit protein eS17target
ArtenimolSmall ribosomal subunit protein uS15target
ArtenimolLarge ribosomal subunit protein uL4target
ArtenimolLarge ribosomal subunit protein uL29target
ArtenimolLarge ribosomal subunit protein uL23target
ArtenimolLarge ribosomal subunit protein eL18target
ArtenimolLarge ribosomal subunit protein eL14target
ArtenimolLarge ribosomal subunit protein uL16target
ArtenimolPeroxiredoxin-1target
ArtenimolPeptidyl-prolyl cis-trans isomerase Atarget
ArtenimolPyruvate kinase PKMtarget
ArtenimolPhosphoglycerate kinase 1target
ArtenimolProfilin-1target
ArtenimolPuromycin-sensitive aminopeptidasetarget
ArtenimolMalate dehydrogenase, cytoplasmictarget
ArtenimolMicrotubule-associated protein 4target
ArtenimolGalectin-1target
ArtenimolL-lactate dehydrogenase B chaintarget
ArtenimolL-lactate dehydrogenase A chaintarget
ArtenimolFar upstream element-binding protein 2target
ArtenimolRas GTPase-activating-like protein IQGAP1target
ArtenimolHeat shock protein beta-1target
ArtenimolHeterochromatin protein 1-binding protein 3target
ArtenimolHeterogeneous nuclear ribonucleoprotein Ktarget
ArtenimolHeterogeneous nuclear ribonucleoprotein D0target
ArtenimolHeterogeneous nuclear ribonucleoproteins A2/B1target
ArtenimolGlucose-6-phosphate isomerasetarget
ArtenimolGlyceraldehyde-3-phosphate dehydrogenase, testis-specifictarget
ArtenimolGlucose-6-phosphate 1-dehydrogenasetarget
ArtenimolAlpha-ketoglutarate-dependent dioxygenase FTOtarget
ArtenimolFilamin-Atarget
ArtenimolAlpha-enolasetarget
ArtenimolElongation factor 1-alpha 1target
ArtenimolDesmoplakintarget
ArtenimolDihydropyrimidinase-related protein 2target
ArtenimolCysteine and glycine-rich protein 1target
ArtenimolChloride intracellular channel protein 1target
ArtenimolCofilin-1target
ArtenimolT-complex protein 1 subunit gammatarget
ArtenimolCalpastatintarget
ArtenimolATP synthase peripheral stalk subunit OSCP, mitochondrialtarget
ArtenimolATP synthase F(0) complex subunit g, mitochondrialtarget
ArtenimolATP synthase F(1) complex subunit alpha, mitochondrialtarget
ArtenimolAnnexin A2target
ArtenimolAlpha-aminoadipic semialdehyde dehydrogenasetarget
ArtenimolActin, cytoplasmic 2target
ArtenimolSmall ribosomal subunit protein eS28target
ArtenimolSmall ribosomal subunit protein uS7target
ArtenimolSmall ribosomal subunit protein eS6target
ArtenimolSmall ribosomal subunit protein eS8target
ArtenimolSmall ribosomal subunit protein uS4target
ArtenimolSplicing factor 1target
ArtenimolSplicing factor, proline- and glutamine-richtarget
ArtenimolSmall nuclear ribonucleoprotein Sm D2target
ArtenimolSignal recognition particle 14 kDa proteintarget
ArtenimolSerine/arginine-rich splicing factor 4target
ArtenimolTransgelintarget
ArtenimolTransgelin-2target
ArtenimolTriosephosphate isomerasetarget
ArtenimolTropomyosin alpha-1 chaintarget
ArtenimolTubulin alpha-1A chaintarget
ArtenimolVimentintarget
ArtenimolZyxintarget
ArtenimolHeat shock cognate 71 kDa proteintarget
ArtenimolTubulin beta-6 chaintarget
ArtenimolTubulin beta-4A chaintarget
ArtenimolTubulin beta chaintarget
ArtenimolFructose-bisphosphate aldolase Atarget
ArtenimolGlyceraldehyde-3-phosphate dehydrogenasetarget
ArtenimolCytochrome ctarget
ArtenimolPhosphoglycerate mutase 1target
ArtenimolMyosin-9target
ArtenimolProtein disulfide-isomerasetarget
ArtenimolProbable ATP-dependent RNA helicase DDX5target
ArtenimolSerine hydroxymethyltransferase, mitochondrialtarget
ArtenimolSpliceosome RNA helicase DDX39Btarget
ArtenimolNucleophosmintarget
ArtenimolTranslationally-controlled tumor protein homologtarget
ArtenimolP-type Ca(2+) transportertarget
ArtenimolOrnithine aminotransferasetarget
ArtenimolElongation factor 1-alphatarget
ArtenimolMultidrug resistance protein 1target
ArtenimolElongation factor 2target
ArtenimolActin-1target
ArtenimolGlyceraldehyde-3-phosphate dehydrogenasetarget
ArtenimolFructose-bisphosphate aldolasetarget
ArtenimolCell division cycle protein 48 homologue, putativetarget
ArtenimolHeat shock protein 90target
ArtenimolRNA helicasetarget
ArtenimolPyruvate kinasetarget
ArtenimolL-lactate dehydrogenasetarget
ArtenimolProtein disulfide-isomerasetarget
ArtenimolThioredoxin-related protein, putativetarget
ArtenimolSpermidine synthasetarget
ArtenimolProbable ATP-dependent 6-phosphofructokinasetarget
ArtenimolGlutamate dehydrogenasetarget
ArtenimolEndoplasmin, putativetarget
ArtenimolHypoxanthine-guanine-xanthine phosphoribosyltransferasetarget
ArtenimolEnolasetarget
Artenimol40S ribosomal protein S3target
ArtenimolP-type sodium-transporting ATPase4target
ArtenimolTubulin alpha chaintarget
ArtenimolKnob-associated histidine-rich proteintarget
ArtenimolS-adenosylmethionine synthasetarget
ArtenimolH(+)-exporting diphosphatasetarget
ArtenimolLarge ribosomal subunit protein uL4target
ArtenimolPhosphoethanolamine N-methyltransferasetarget
ArtenimolSmall ribosomal subunit protein eS1target
ArtenimolProtein ARVtarget
Artenimol60S ribosomal protein L3target
ArtenimolHigh molecular weight rhoptry protein 2target
ArtenimolSerine repeat antigen 5target
Artenimol40S ribosomal protein S19target
ArtenimolGlycophorin-binding protein 130target
ArtenimolCalcium-transporting ATPasetarget
ArtenimolV-type proton ATPase catalytic subunit Atarget
Artenimol60S ribosomal protein L2target
ArtenimolAcyl-CoA synthetasetarget
ArtenimolPlasmepsin IVtarget
ArtenimolPlasmepsin Itarget
ArtenimolChloroquine resistance transportertarget
Artenimol14-3-3 protein Itarget
ArtenimolIsoleucine--tRNA ligase, putativetarget
ArtenimolPlasmodium RESA N-terminal domain-containing proteintarget
ArtenimolTubulin beta chaintarget
Artenimol60S ribosomal protein L27target
ArtenimolTranslocation protein SEC62target
ArtenimolAutophagy-related protein 18target
ArtenimolMature parasite-infected erythrocyte surface antigentarget
ArtenimolImportin-7, putativetarget
ArtenimolImportin subunit alphatarget
ArtenimolPeptidyl-prolyl cis-trans isomerasetarget
ArtenimolDnaJ protein, putativetarget
ArtenimolMerozoite surface protein 1target
ArtenimolGlutamate--tRNA ligasetarget
ArtenimolT-complex protein 1 subunit etatarget
ArtenimolPlasmepsin IItarget
ArtenimolChaperone, putativetarget
ArtenimolRhoptry neck protein 3target
Artenimol40S ribosomal protein S5, putativetarget
ArtenimolSkeleton-binding protein 1target
ArtenimolPurine nucleoside phosphorylasetarget
ArtenimolAdenosylhomocysteinasetarget
ArtenimolAdenosine deaminasetarget
ArtenimolMethionine--tRNA ligasetarget
Artenimolcarbamoyl-phosphate synthase (ammonia)target
ArtenimolSignal recognition particle receptor subunit betatarget
ArtenimolN-acetylgalactosaminide beta-1,3-galactosyltransferasetarget
ArtenimolCoatomer alpha subunit, putativetarget
ArtenimolHexokinasetarget
ArtenimolProteasome subunit alpha typetarget
ArtenimolHaloacid dehalogenase-like hydrolasetarget
ArtenimolInsulinase, putativetarget
Artenimol40S ribosomal protein S21target
ArtenimolUbiquitin-conjugating enzyme E2target
ArtenimolEukaryotic translation initiation factor 3 subunit Ctarget
Artenimol60S ribosomal protein L24, putativetarget
Artenimol60S ribosomal protein L23target
ArtenimolLarge ribosomal subunit protein uL22target
ArtenimolPlasmepsin IIItarget
ArtenimolEndoplasmic reticulum chaperone GRP170target
Artenimol60S ribosomal protein L10, putativetarget
ArtenimolEsterase, putativetarget
ArtenimolPolyadenylate-binding proteintarget
ArtenimolUbiquitin-60S ribosomal protein L40target
Artenimolribose-phosphate diphosphokinasetarget
Artenimol2-Cys peroxiredoxintarget
ArtenimolProtein transport protein SEC31target
ArtenimolDipeptidyl aminopeptidase 1target
ArtenimolRing-infected erythrocyte surface antigentarget
ArtenimolRNA helicasetarget
ArtenimolCalcium-dependent protein kinase 4target
ArtenimolGTP-binding nuclear protein Rantarget
ArtenimolNucleoside transporter 2target
ArtenimolAnamorsin homologtarget
ArtenimolGlutamine synthetase, putativetarget
Artenimol60S ribosomal protein L30e, putativetarget
Artenimolnon-specific serine/threonine protein kinasetarget
ArtenimolThreonine--tRNA ligasetarget
ArtenimolcAMP-dependent protein kinase regulatory subunittarget
ArtenimolThioredoxin-like protein 1target
Artenimol60S ribosomal protein L21target
Artenimol60S ribosomal protein L14, putativetarget
ArtenimolInner membrane complex sub-compartment protein 3target
ArtenimolHSP40, subfamily Atarget
ArtenimolPyridoxal 5'-phosphate synthase subunit Pdx1target
ArtenimolUDP-glucuronosyltransferase 1A9enzyme
ArtenimolUDP-glucuronosyltransferase 2B7enzyme
ArtenimolAlbumintarget
ArtenimolCytochrome P450 2D6enzyme
ArtenimolCytochrome P450 2C19enzyme
AsciminibCytochrome P450 3A4enzyme
AsciminibCytochrome P450 2C9enzyme
AsciminibSolute carrier family 22 member 1transporter
AsciminibSolute carrier organic anion transporter family member 1B3transporter
AsciminibSolute carrier organic anion transporter family member 1B1transporter
AsciminibATP-dependent translocase ABCB1transporter
AsciminibCytochrome P450 2C19enzyme
AsciminibUDP-glucuronosyltransferase 1A1enzyme
AsciminibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
AsciminibUDP-glucuronosyltransferase 2B7enzyme
AsciminibUDP-glucuronosyltransferase 2B17enzyme
AsciminibTyrosine-protein kinase ABL1target
AsenapineHistamine H1 receptortarget
AsenapineD(4) dopamine receptortarget
AsenapineD(3) dopamine receptortarget
AsenapineD(2) dopamine receptortarget
AsenapineD(1A) dopamine receptortarget
AsenapineAlpha-1A adrenergic receptortarget
AsenapineAlpha-2C adrenergic receptortarget
AsenapineAlpha-2B adrenergic receptortarget
AsenapineAlpha-2A adrenergic receptortarget
Asenapine5-hydroxytryptamine receptor 7target
Asenapine5-hydroxytryptamine receptor 6target
Asenapine5-hydroxytryptamine receptor 2Ctarget
Asenapine5-hydroxytryptamine receptor 2Btarget
Asenapine5-hydroxytryptamine receptor 2Atarget
Asenapine5-hydroxytryptamine receptor 1Btarget
Asenapine5-hydroxytryptamine receptor 1Atarget
AsenapineHistamine H2 receptortarget
AsenapineCytochrome P450 1A2enzyme
AsenapineCytochrome P450 2D6enzyme
Asenapine5-hydroxytryptamine receptor 5Atarget
AsenapineUDP-glucuronosyltransferase 1A4enzyme
AsenapineCytochrome P450 3A4enzyme
AsenapineBeta-1 adrenergic receptortarget
AsenapineBeta-2 adrenergic receptortarget
AsenapineAlbumincarrier
Asenapinealpha1-acid glycoproteincarrier
AstemizoleBile salt export pumptransporter
AstemizoleMicrotubule-associated protein tautarget
AstemizoleVoltage-gated delayed rectifier potassium channel KCNH1target
AstemizoleCytochrome P450 2J2enzyme
AstemizoleCytochrome P450 2D6enzyme
AstemizoleATP-dependent translocase ABCB1transporter
AstemizoleCytochrome P450 3A7enzyme
AstemizoleCytochrome P450 3A5enzyme
AstemizoleCytochrome P450 3A4enzyme
AstemizoleVoltage-gated inwardly rectifying potassium channel KCNH2target
AstemizoleHistamine H1 receptortarget
AsunaprevirGenome polyproteintarget
AsunaprevirGag-Pol polyproteintarget
AsunaprevirATP-dependent translocase ABCB1transporter
AsunaprevirSolute carrier organic anion transporter family member 2B1transporter
AsunaprevirSolute carrier organic anion transporter family member 1B3transporter
AsunaprevirSolute carrier organic anion transporter family member 1B1transporter
AsunaprevirCytochrome P450 2D6enzyme
AsunaprevirCytochrome P450 2C19enzyme
AsunaprevirCytochrome P450 2C9enzyme
AsunaprevirCytochrome P450 2B6enzyme
AsunaprevirCytochrome P450 2A6enzyme
AsunaprevirCytochrome P450 3A5enzyme
AsunaprevirCytochrome P450 3A4enzyme
AtazanavirPol polyproteintarget
AtazanavirCytochrome P450 3A4enzyme
AtazanavirCytochrome P450 2C9enzyme
AtazanavirATP-dependent translocase ABCB1transporter
AtazanavirGag-Pol polyproteintarget
AtazanavirCytochrome P450 3A7enzyme
AtazanavirCytochrome P450 3A5enzyme
AtazanavirSolute carrier organic anion transporter family member 2B1transporter
AtazanavirCytochrome P450 1A2enzyme
AtazanavirMultidrug resistance-associated protein 1transporter
AtazanavirAlbumincarrier
AtazanavirUDP-glucuronosyltransferase 1A1enzyme
AtazanavirSolute carrier organic anion transporter family member 1B1transporter
AtazanavirSolute carrier organic anion transporter family member 1B3transporter
AtazanavirCytochrome P450 2C8enzyme
AtazanavirBile salt export pumptransporter
Atazanaviralpha1-acid glycoproteincarrier
AtomoxetineCytochrome P450 2C19enzyme
AtomoxetineSodium-dependent serotonin transportertarget
AtomoxetineCytochrome P450 2D6enzyme
AtomoxetineSodium-dependent noradrenaline transportertarget
AtomoxetineNMDA receptortarget
AtomoxetineAlbumincarrier
Atomoxetinealpha1-acid glycoproteincarrier
AtomoxetineHigh affinity immunoglobulin gamma Fc receptor Icarrier
AtomoxetineG protein-activated inward rectifier potassium channel 1target
AtomoxetineKappa-type opioid receptortarget
Atorvastatin3-hydroxy-3-methylglutaryl-coenzyme A reductasetarget
AtorvastatinCytochrome P450 3A4enzyme
AtorvastatinDipeptidyl peptidase 4target
AtorvastatinCytochrome P450 2D6enzyme
AtorvastatinCytochrome P450 2C9enzyme
AtorvastatinCytochrome P450 2C19enzyme
AtorvastatinCytochrome P450 3A5enzyme
AtorvastatinCytochrome P450 3A7enzyme
AtorvastatinATP-dependent translocase ABCB1transporter
AtorvastatinSolute carrier organic anion transporter family member 1A2transporter
AtorvastatinSolute carrier organic anion transporter family member 1B1transporter
AtorvastatinATP-binding cassette sub-family C member 4transporter
AtorvastatinATP-binding cassette sub-family C member 5transporter
AtorvastatinMultidrug resistance-associated protein 1transporter
AtorvastatinCytochrome P450 2B6enzyme
AtorvastatinCytochrome P450 2C8enzyme
AtorvastatinAryl hydrocarbon receptortarget
AtorvastatinSolute carrier organic anion transporter family member 2B1transporter
AtorvastatinSolute carrier organic anion transporter family member 1B3transporter
AtorvastatinUDP-glucuronosyltransferase 1A1enzyme
AtorvastatinUDP-glucuronosyltransferase 1A3enzyme
AtorvastatinATP-binding cassette sub-family C member 2transporter
AtorvastatinBile salt export pumptransporter
AtorvastatinAlbumincarrier
AtorvastatinHistone deacetylase 2target
AtorvastatinNuclear receptor subfamily 1 group I member 3target
AtovaquoneATP-dependent translocase ABCB1transporter
AtovaquoneCytochrome P450 3A4enzyme
AtovaquoneCytochrome P450 2C9enzyme
AtovaquoneCytochrome btarget
AtovaquoneDihydroorotate dehydrogenase (quinone), mitochondrialtarget
AtovaquoneDihydroorotate dehydrogenase (quinone), mitochondrialtarget
AtrasentanSolute carrier organic anion transporter family member 1B3transporter
AtrasentanAlbumincarrier
AtrasentanCytochrome P450 3A Subfamilyenzyme
AtrasentanEndothelin receptor type Btarget
AtrasentanEndothelin-1 receptortarget
AtrasentanCytochrome P450 2B6enzyme
AtrasentanSolute carrier organic anion transporter family member 1B1transporter
AtrasentanATP-dependent translocase ABCB1transporter
AtrasentanUDP-glucuronosyltransferases (UGTs)enzyme
AtrasentanCytochrome P450 2C9enzyme
AtrasentanCytochrome P450 2C8enzyme
AvacopanC5a anaphylatoxin chemotactic receptor 1target
AvacopanCytochrome P450 3A4enzyme
AvacopanCytochrome P450 2C9enzyme
AvacopanCytochrome P450 2B6enzyme
AvacopanCytochrome P450 1A2enzyme
AvacopanATP-dependent translocase ABCB1transporter
AvapritinibATP-dependent translocase ABCB1transporter
AvapritinibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
AvapritinibCytochrome P450 3A4enzyme
AvapritinibCytochrome P450 2C9enzyme
AvapritinibBile salt export pumptransporter
AvapritinibMultidrug and toxin extrusion protein 1transporter
AvapritinibMultidrug and toxin extrusion protein 2transporter
AvapritinibPlatelet-derived growth factor receptor alphatarget
AvapritinibMast/stem cell growth factor receptor Kittarget
AvasimibeLiver carboxylesterase 1target
AvasimibeCytochrome P450 3A4enzyme
AvasimibeCytochrome P450 2C9enzyme
AvasimibeCytochrome P450 2C19enzyme
AvasimibeCytochrome P450 1A2enzyme
AVE9633Myeloid cell surface antigen CD33target
AVE9633Cytochrome P450 3A4enzyme
AzamulinCytochrome P450 3A4target
AzamulinCytochrome P450 3A5target
AzamulinCytochrome P450 3A Subfamilytarget
AzelastineCytochrome P450 2B6enzyme
AzelastineLeukotriene C4 synthasetarget
AzelastinePhospholipase A2target
AzelastineHistamine H2 receptortarget
AzelastineCytochrome P450 2E1enzyme
AzelastineCytochrome P450 2A6enzyme
AzelastineATP-dependent translocase ABCB1transporter
AzelastineCytochrome P450 2C8enzyme
AzelastineCytochrome P450 2C9enzyme
AzelastineCytochrome P450 3A5enzyme
AzelastineCytochrome P450 1A1enzyme
AzelastineCytochrome P450 2C19enzyme
AzelastineCytochrome P450 3A4enzyme
AzelastineHistamine H1 receptortarget
AzelastineCytochrome P450 1A2enzyme
AzelastineCytochrome P450 2D6enzyme
AzithromycinATP-binding cassette sub-family C member 2transporter
AzithromycinProtein-arginine deiminase type-4target
AzithromycinCytochrome P450 3A4enzyme
Azithromycin23S ribosomal RNAtarget
AzithromycinATP-dependent translocase ABCB1transporter
BalaglitazonePeroxisome proliferator-activated receptor gammatarget
BalaglitazoneCytochrome P450 2C8enzyme
BalaglitazoneCytochrome P450 3A4enzyme
Baloxavir marboxilBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
Baloxavir marboxilUDP-glucuronosyltransferase 1A3enzyme
Baloxavir marboxilCytochrome P450 3A4enzyme
Baloxavir marboxilPolymerase acidic proteintarget
Baloxavir marboxilATP-dependent translocase ABCB1transporter
Baloxavir marboxilCytochrome P450 2B6enzyme
Baloxavir marboxilCytochrome P450 2C8enzyme
BarnidipineVoltage-dependent L-type calcium channel subunit alpha-1Ctarget
BarnidipineCytochrome P450 3A4enzyme
BarnidipineVoltage-dependent T-type calcium channel subunit alpha-1Gtarget
BarnidipineVoltage-dependent T-type calcium channel subunit alpha-1Htarget
BarnidipineVoltage gated L-type calcium channeltarget
BelinostatHistone deacetylasetarget
BelinostatCytochrome P450 1A2enzyme
BelinostatUDP-glucuronosyltransferase 1A1enzyme
BelinostatCytochrome P450 2C8enzyme
BelinostatCytochrome P450 2C9enzyme
BelinostatATP-dependent translocase ABCB1transporter
BelinostatCytochrome P450 3A4enzyme
BelumosudilCytochrome P450 3A4enzyme
BelumosudilCytochrome P450 2C8enzyme
BelumosudilCytochrome P450 2D6enzyme
BelumosudilRho-associated protein kinase 1target
BelumosudilCytochrome P450 1A2enzyme
BelumosudilCytochrome P450 2C19enzyme
BelumosudilUDP-glucuronosyltransferase 1A1enzyme
BelumosudilATP-dependent translocase ABCB1transporter
BelumosudilBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
BelumosudilSolute carrier organic anion transporter family member 1B1transporter
BelumosudilAlpha-1-acid glycoprotein 1carrier
BelumosudilAlbumincarrier
BelumosudilRho-associated protein kinase 2target
BelumosudilUDP-glucuronosyltransferase 1A9enzyme
BenidipineVoltage-dependent L-type calcium channeltarget
BenidipineVoltage-dependent N-type calcium channel subunit alpha-1Btarget
BenidipineVoltage-dependent T-type calcium channeltarget
BenidipineCytochrome P450 3A4enzyme
BenidipineCytochrome P450 3A5enzyme
BenidipineVoltage gated L-type calcium channeltarget
BenzbromaroneCytochrome P450 2C9target
BenzbromaroneCytochrome P450 2C19target
BenzbromaroneSolute carrier organic anion transporter family member 1B1transporter
BenzbromaroneSolute carrier organic anion transporter family member 2B1transporter
BenzbromaroneBile salt export pumptransporter
BenzbromaroneCytochrome P450 2C19enzyme
BenzbromaroneMultidrug resistance-associated protein 1target
BenzbromaroneAnoctamin-1target
BenzbromaroneSolute carrier family 22 member 12target
BenznidazoleNuclear receptor subfamily 1 group I member 2target
BenznidazoleInhibitor of nuclear factor kappa-B kinase subunit betatarget
BenznidazoleNuclear factor erythroid 2-related factor 2target
BenznidazoleATP-dependent translocase ABCB1transporter
BenznidazoleCytochrome P450 3A4target
BepridilCalmodulintarget
BepridilCytochrome P450 3A4enzyme
BepridilVoltage-gated inwardly rectifying potassium channel KCNH2target
BepridilCytochrome P450 2D6enzyme
BepridilATP-dependent translocase ABCB1transporter
BepridilDual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1Atarget
BepridilDual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1Btarget
BepridilVoltage-dependent calcium channel subunit alpha-2/delta-2target
BepridilVoltage-dependent T-type calcium channel subunit alpha-1Htarget
BepridilTroponin C, slow skeletal and cardiac musclestarget
BepridilPotassium voltage-gated channel subfamily KQT member 1target
BepridilSodium/potassium-transporting ATPase subunit alpha-1target
BepridilVoltage-dependent P/Q-type calcium channel subunit alpha-1Atarget
BergaptenCytochrome P450 3A4enzyme
BerotralstatPlasma kallikreintarget
BerotralstatBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
BerotralstatATP-dependent translocase ABCB1transporter
BerotralstatCytochrome P450 3A4enzyme
BerotralstatCytochrome P450 2D6enzyme
BesifloxacinDNA gyrase subunit Btarget
BesifloxacinDNA gyrase subunit Atarget
BesifloxacinCytochrome P450 1A2enzyme
BesifloxacinDNA gyrase subunit Atarget
BesifloxacinDNA gyrase subunit Atarget
BesifloxacinDNA topoisomerase 4 subunit Atarget
BesifloxacinDNA topoisomerase 4 subunit Atarget
BesigomsinCytochrome P450 2C8enzyme
BesigomsinAcetylcholinesterasetarget
BesigomsinATP-dependent translocase ABCB1transporter
BesigomsinBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
BesigomsinCytochrome P450 3A4enzyme
BesigomsinTransient receptor potential cation channel subfamily V member 1target
BesigomsinCytochrome P450 2C19enzyme
BesigomsinCytochrome P450 2C9enzyme
BexaroteneRetinoic acid receptor RXR-betatarget
BexaroteneCytochrome P450 3A4enzyme
BexaroteneRetinoic acid receptor RXR-alphatarget
BexaroteneRetinoic acid receptor RXR-gammatarget
BexaroteneCytochrome P450 2C8enzyme
BexaroteneHuman Retinoid X Receptors (RXRs)target
BezafibratePeroxisome proliferator-activated receptor alphatarget
BezafibrateSolute carrier organic anion transporter family member 1B1transporter
BezafibratePeroxisome proliferator-activated receptor deltatarget
BezafibratePeroxisome proliferator-activated receptor gammatarget
BezafibrateCytochrome P450 1A1enzyme
BezafibrateCytochrome P450 2C8enzyme
BezafibrateCytochrome P450 3A4enzyme
BezafibrateNuclear receptor subfamily 1 group I member 2target
BezafibrateRetinoic acid receptor RXR-alphatarget
BezafibrateRetinoic acid receptor RXR-betatarget
BezafibrateRetinoic acid receptor RXR-gammatarget
BezafibratePeroxisome proliferator-activated receptorstarget
BicalutamideAndrogen receptortarget
BicalutamideATP-dependent translocase ABCB1transporter
BicalutamideCytochrome P450 2D6enzyme
BicalutamideCytochrome P450 2C9enzyme
BicalutamideCytochrome P450 2C19enzyme
BicalutamideCytochrome P450 3A4enzyme
BifonazoleCytochrome P450 2E1enzyme
BifonazoleCytochrome P450 2B6target
BifonazoleLanosterol 14-alpha demethylasetarget
BifonazoleAromataseenzyme
BifonazoleCytochrome P450 3A4enzyme
BiperidenCytochrome P450 2D6enzyme
BiperidenMuscarinic acetylcholine receptor M1target
Birch bark extractCytochrome P450 2C8enzyme
Birch bark extractCytochrome P450 3A Subfamilyenzyme
Black cohoshCytochrome P450 3A4enzyme
Black cohoshCytochrome P450 3A2enzyme
Black cohoshCytochrome P450 1A2enzyme
Black cohoshCytochrome P450 2C9enzyme
Black cohoshCytochrome P450 2D6enzyme
BoceprevirGenome polyproteintarget
BoceprevirGenome polyproteintarget
BoceprevirATP-dependent translocase ABCB1transporter
BoceprevirCytochrome P450 3A5enzyme
BoceprevirCytochrome P450 3A4enzyme
BortezomibCytochrome P450 3A4enzyme
BortezomibCytochrome P450 2C19enzyme
BortezomibCytochrome P450 1A2enzyme
BortezomibCytochrome P450 2D6enzyme
BortezomibCytochrome P450 2C9enzyme
BortezomibProteasome subunit beta type-5target
BortezomibProteasome subunit beta type-1target
BortezomibATP-dependent translocase ABCB1transporter
BortezomibSolute carrier organic anion transporter family member 1B3transporter
BortezomibSerine protease 1target
BosutinibSTE20-like serine/threonine-protein kinasetarget
BosutinibTyrosine-protein kinase Tectarget
BosutinibTyrosine-protein kinase HCKtarget
BosutinibTyrosine-protein kinase Fgrtarget
BosutinibCytochrome P450 2C8enzyme
BosutinibCalcium/calmodulin-dependent protein kinase type II subunit gammatarget
BosutinibMitogen-activated protein kinase kinase kinase 2target
BosutinibDual specificity mitogen-activated protein kinase kinase 2target
BosutinibDual specificity mitogen-activated protein kinase kinase 1target
BosutinibCytochrome P450 3A4enzyme
BosutinibATP-dependent translocase ABCB1transporter
BosutinibProto-oncogene tyrosine-protein kinase Srctarget
BosutinibTyrosine-protein kinase Lyntarget
BosutinibTyrosine-protein kinase ABL1target
Brefeldin ACytohesin-2target
Brefeldin AADP-ribosylation factor 1target
Brefeldin ACytochrome P450 3A4enzyme
Brentuximab vedotinATP-binding cassette sub-family B member 5transporter
Brentuximab vedotinCytochrome P450 3A4enzyme
Brentuximab vedotinTumor necrosis factor receptor superfamily member 8target
BrincidofovirBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
BrincidofovirATP-binding cassette sub-family C member 2transporter
BrincidofovirBile salt export pumptransporter
BrincidofovirSolute carrier organic anion transporter family member 1B1transporter
BrincidofovirSolute carrier family 22 member 6transporter
BrincidofovirOrganic anion transporter 3transporter
BrincidofovirSolute carrier organic anion transporter family member 1B3transporter
BrincidofovirVariola virus DNAtarget
BrincidofovirSphingomyelin phosphodiesteraseenzyme
BrincidofovirDNA polymerase betatarget
BrincidofovirDNA polymerase subunit gamma-2target
BrincidofovirDNA polymerase subunit gamma-1target
BrincidofovirDNA polymerase epsilon subunit 2target
BrincidofovirDNA polymerase nutarget
BrincidofovirDNA polymerase delta subunit 4target
BrincidofovirDNA polymerase delta catalytic subunittarget
BrincidofovirCytochrome P450 2D6enzyme
BrincidofovirCytochrome P450 2C19enzyme
BrincidofovirCytochrome P450 2C9enzyme
BrincidofovirCytochrome P450 2C8enzyme
BrincidofovirCytochrome P450 2B6enzyme
BrincidofovirCytochrome P450 1A2enzyme
BrincidofovirDNA polymerasetarget
BrincidofovirCytochrome P450 4F2enzyme
BrincidofovirDNA polymerase thetatarget
BromazepamGABA(A) Receptor Benzodiazepine Binding Sitetarget
BromazepamCytochrome P450 1A2enzyme
BromazepamCytochrome P450 2C19enzyme
BromazepamCytochrome P450 2E1enzyme
BromazepamGABA(A) Receptortarget
BromazepamGamma-aminobutyric acid receptor subunit alpha-2target
Bromocriptine5-hydroxytryptamine receptor 2Ctarget
BromocriptineAlpha-2B adrenergic receptortarget
BromocriptineAlpha-2C adrenergic receptortarget
Bromocriptine5-hydroxytryptamine receptor 1Atarget
BromocriptineD(3) dopamine receptortarget
BromocriptineATP-dependent translocase ABCB1transporter
Bromocriptine5-hydroxytryptamine receptor 7target
BromocriptineAlpha-1D adrenergic receptortarget
BromocriptineAlpha-1B adrenergic receptortarget
BromocriptineAlpha-1A adrenergic receptortarget
BromocriptineD(1A) dopamine receptortarget
BromocriptineD(1B) dopamine receptortarget
BromocriptineAlpha-2A adrenergic receptortarget
Bromocriptine5-hydroxytryptamine receptor 1Btarget
Bromocriptine5-hydroxytryptamine receptor 2Atarget
BromocriptineD(4) dopamine receptortarget
Bromocriptine5-hydroxytryptamine receptor 1Dtarget
BromocriptineCytochrome P450 3A4enzyme
BromocriptineD(2) dopamine receptortarget
Bromocriptine5-hydroxytryptamine receptor 2Btarget
Bryostatin 1Cytochrome P450 3A4enzyme
Bryostatin 1Protein kinase C alpha typetarget
Bryostatin 1Protein kinase C epsilon typetarget
Bryostatin 1Caspase-8target
Bryostatin 1Protein unc-13 homolog Btarget
Bryostatin 1Serine/threonine-protein kinase D1target
Bryostatin 1T-lymphocyte activation antigen CD86target
Bryostatin 1Prostaglandin G/H synthase 2target
Bryostatin 1G1/S-specific cyclin-D1target
Bryostatin 1Tumor necrosis factortarget
BuprenorphineKappa-type opioid receptortarget
BuprenorphineMu-type opioid receptortarget
BuprenorphineCytochrome P450 3A4enzyme
BuprenorphineCytochrome P450 2D6enzyme
BuprenorphineATP-dependent translocase ABCB1transporter
BuprenorphineBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
BuprenorphineCytochrome P450 2C9enzyme
BuprenorphineCytochrome P450 3A5enzyme
BuprenorphineCytochrome P450 2C8enzyme
BuprenorphineCytochrome P450 3A7enzyme
BuprenorphineDelta-type opioid receptortarget
BuprenorphineCytochrome P450 2C18enzyme
BuprenorphineCytochrome P450 2C19enzyme
BuprenorphineNociceptin receptortarget
BupropionSolute carrier family 22 member 2transporter
BupropionSodium-dependent serotonin transportertarget
Bupropion5-hydroxytryptamine receptor 3Atarget
BupropionCytochrome P450 2E1enzyme
BupropionCytochrome P450 2C9enzyme
BupropionNeuronal acetylcholine receptor subunit alpha-3target
BupropionAlpha-1-acid glycoprotein 1carrier
BupropionCytochrome P450 2D6enzyme
BupropionCytochrome P450 2B6enzyme
BupropionSodium-dependent noradrenaline transportertarget
BupropionSodium-dependent dopamine transportertarget
BW-A 58CCytochrome P450 2C9enzyme
CabergolineAlpha-2B adrenergic receptortarget
CabergolineATP-dependent translocase ABCB1transporter
CabergolineD(1) dopamine receptortarget
CabergolineBeta-2 adrenergic receptortarget
CabergolineBeta-1 adrenergic receptortarget
CabergolineAlpha-1D adrenergic receptortarget
CabergolineAlpha-1B adrenergic receptortarget
CabergolineAlpha-1A adrenergic receptortarget
Cabergoline5-hydroxytryptamine receptor 7target
CabergolineCytochrome P450 3A4enzyme
Cabergoline5-hydroxytryptamine receptor 2Ctarget
Cabergoline5-hydroxytryptamine receptor 1Btarget
CabergolineD(1A) dopamine receptortarget
CabergolineD(1B) dopamine receptortarget
CabergolineAlpha-2C adrenergic receptortarget
Cabergoline5-hydroxytryptamine receptor 1Atarget
Cabergoline5-hydroxytryptamine receptor 2Btarget
CabergolineD(3) dopamine receptortarget
Cabergoline5-hydroxytryptamine receptor 2Atarget
CabergolineD(2) dopamine receptortarget
Cabergoline5-hydroxytryptamine receptor 1Dtarget
CabergolineD(4) dopamine receptortarget
CabergolineAlpha-2A adrenergic receptortarget
CabozantinibTyrosine-protein kinase Mertarget
CabozantinibTyrosine-protein kinase receptor TYRO3target
CabozantinibProto-oncogene tyrosine-protein kinase ROStarget
CabozantinibTyrosine-protein kinase receptor UFOtarget
CabozantinibReceptor-type tyrosine-protein kinase FLT3target
CabozantinibBDNF/NT-3 growth factors receptortarget
CabozantinibMast/stem cell growth factor receptor Kittarget
CabozantinibVascular endothelial growth factor receptor 3target
CabozantinibVascular endothelial growth factor receptor 1target
CabozantinibCytochrome P450 2C8enzyme
CabozantinibProto-oncogene tyrosine-protein kinase receptor Rettarget
CabozantinibVascular endothelial growth factor receptor 2target
CabozantinibHepatocyte growth factor receptortarget
CabozantinibCytochrome P450 2C9enzyme
CabozantinibCytochrome P450 3A4enzyme
CabozantinibAngiopoietin-1 receptortarget
CaffeineCytochrome P450 2C9enzyme
CaffeineAdenosine receptortarget
Caffeine5'-nucleotidasetarget
CaffeinePhosphodiesterase enzymestarget
CaffeineAdenosine receptor A3target
CaffeineAdenosine receptor A2btarget
CaffeineBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
CaffeineSerine-protein kinase ATMtarget
CaffeineInositol 1,4,5-trisphosphate receptortarget
CaffeinePhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoformtarget
CaffeinePhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoformtarget
CaffeineAdenosine receptor A1target
Caffeine3',5'-cyclic-AMP phosphodiesterase 4Btarget
CaffeineAdenosine receptor A2atarget
CaffeineCytochrome P450 1A2enzyme
CaffeineRyanodine receptor 1target
CaffeineCytochrome P450 3A4enzyme
CaffeineCytochrome P450 2E1enzyme
CaffeineCytochrome P450 2C8enzyme
CaffeinePhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoformtarget
CaffeineCytochrome P450 1A1enzyme
CaffeineCytochrome P450 1B1enzyme
CaffeineCytochrome P450 2D6enzyme
CaffeineCyclic nucleotide phosphodiesterasetarget
CaffeineDNA-dependent protein kinase catalytic subunittarget
CandesartanType-1 angiotensin II receptortarget
CandesartanCytochrome P450 2C8enzyme
CandesartanCytochrome P450 2C9enzyme
CandesartanATP-dependent translocase ABCB1transporter
CandesartanUDP-glucuronosyltransferase 1A3enzyme
CandesartanProstaglandin G/H synthase 1enzyme
CandesartanSolute carrier organic anion transporter family member 1B1transporter
Candesartan cilexetilProstaglandin G/H synthase 1enzyme
Candesartan cilexetilUDP-glucuronosyltransferase 1A3enzyme
Candesartan cilexetilATP-dependent translocase ABCB1transporter
Candesartan cilexetilCytochrome P450 2C9enzyme
Candesartan cilexetilCytochrome P450 2C8enzyme
Candesartan cilexetilType-1 angiotensin II receptortarget
CandicidinErgosteroltarget
CandicidinCytochrome P450 3A4enzyme
Cannabidiol5-hydroxytryptamine receptor 1Atarget
CannabidiolG protein-coupled receptor 55target
CannabidiolN-arachidonyl glycine receptortarget
CannabidiolGlycine receptor subunit alpha-3target
CannabidiolGlycine receptor (alpha-1/beta)target
CannabidiolGlycine receptor subunit alpha-1target
CannabidiolG protein-coupled receptor 12target
CannabidiolCannabinoid receptor 2target
CannabidiolCannabinoid receptor 1target
CannabidiolCytochrome P450 3A4enzyme
CannabidiolCytochrome P450 2D6enzyme
CannabidiolCytochrome P450 2C19enzyme
CannabidiolCytochrome P450 2C9enzyme
Cannabidiol5-hydroxytryptamine receptor 2Atarget
CannabidiolNeuronal acetylcholine receptor subunit alpha-7target
CannabidiolDelta-type opioid receptortarget
CannabidiolMu-type opioid receptortarget
CannabidiolPeroxisome proliferator-activated receptor gammatarget
CannabidiolCytochrome P450 3A5enzyme
CannabidiolSerotonin N-acetyltransferaseenzyme
CannabidiolCytochrome P450 1A1enzyme
CannabidiolFatty-acid amide hydrolase 1enzyme
CannabidiolPolyunsaturated fatty acid 5-lipoxygenaseenzyme
CannabidiolPolyunsaturated fatty acid lipoxygenase ALOX15enzyme
CannabidiolZeta-crystallinenzyme
CannabidiolMultidrug resistance-associated protein 1transporter
CannabidiolBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
CannabidiolEquilibrative nucleoside transporter 1transporter
CannabidiolTransient receptor potential cation channel subfamily V member 1target
CannabidiolVoltage-dependent T-type calcium channel subunit alpha-1Gtarget
CannabidiolVoltage-dependent T-type calcium channel subunit alpha-1Htarget
CannabidiolVoltage-dependent T-type calcium channel subunit alpha-1Itarget
CannabidiolTransient receptor potential cation channel subfamily A member 1target
CannabidiolTransient receptor potential cation channel subfamily M member 8target
CannabidiolTransient receptor potential cation channel subfamily V member 2target
CannabidiolTransient receptor potential cation channel subfamily V member 3target
CannabidiolTransient receptor potential cation channel subfamily V member 4target
CannabidiolNon-selective voltage-gated ion channel VDAC1target
Cannabidiol5-hydroxytryptamine receptor 3Atarget
CannabidiolAdenosine receptor A1target
CannabidiolProstaglandin G/H synthase 1target
CannabidiolProstaglandin G/H synthase 2target
CannabidiolAcetyl-CoA acetyltransferase, mitochondrialtarget
CannabidiolSteroid 17-alpha-hydroxylase/17,20 lyasetarget
Cannabidiol3-hydroxy-3-methylglutaryl-coenzyme A reductasetarget
CannabidiolGlutathione reductase, mitochondrialtarget
CannabidiolGlutathione peroxidase 1target
CannabidiolIndoleamine 2,3-dioxygenase 1target
CannabidiolNAD(P)H dehydrogenase [quinone] 1target
CannabidiolCatalasetarget
CannabidiolSuperoxide dismutase [Cu-Zn]target
CannabidiolSerotonin N-acetyltransferasetarget
CannabidiolN-acylethanolamine-hydrolyzing acid amidasetarget
CannabidiolCytochrome P450 1A2enzyme
CannabidiolCytochrome P450 1B1enzyme
CannabidiolCytochrome P450 2A6enzyme
CannabidiolCytochrome P450 2B6enzyme
CannabidiolCytochrome P450 2C8enzyme
CannabidiolCytochrome P450 2E1enzyme
CannabidiolCytochrome P450 3A7enzyme
CannabidiolUDP-glucuronosyltransferase 1A7enzyme
CannabidiolUDP-glucuronosyltransferase 1A9enzyme
CannabidiolUDP-glucuronosyltransferase 2B7enzyme
CannabidiolUDP-glucuronosyltransferase 2B17enzyme
CannabidiolATP-dependent translocase ABCB1transporter
CannabidiolCytochrome P450 2J2enzyme
CannabidiolLiver carboxylesterase 1enzyme
CannabinolCytochrome P450 3A4enzyme
CannabinolCytochrome P450 2C19enzyme
CannabinolCytochrome P450 1A1enzyme
CannabinolCytochrome P450 1A2enzyme
CannabinolCytochrome P450 1B1enzyme
CannabinolCytochrome P450 2A6enzyme
CannabinolCytochrome P450 2B6enzyme
CannabinolCytochrome P450 2C9enzyme
CannabinolCytochrome P450 2D6enzyme
CannabinolCytochrome P450 3A5enzyme
CannabinolCytochrome P450 3A7enzyme
CannabinolUDP-glucuronosyltransferase 1A7enzyme
CannabinolUDP-glucuronosyltransferase 1A8enzyme
CannabinolUDP-glucuronosyltransferase 1A9enzyme
CannabinolUDP-glucuronosyltransferase 1A10enzyme
CannabinolUDP-glucuronosyltransferase 2B7enzyme
CannabinolATP-dependent translocase ABCB1transporter
CannabinolBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
CannabinolMultidrug resistance-associated protein 1transporter
CannabinolCytochrome P450 2E1enzyme
CannabinolCytochrome P450 2J2enzyme
CannabinolLiver carboxylesterase 1enzyme
CannabinolCannabinoid receptor 1target
CapecitabineThymidylate synthasetarget
CapecitabineThymidylate synthasetarget
CapecitabineUridine phosphorylase 2enzyme
CapecitabineUridine phosphorylase 1enzyme
CapecitabineAlbumincarrier
CapecitabineRNAtarget
CapecitabineDNAtarget
CapecitabineCytochrome P450 2C9enzyme
CapecitabineLiver carboxylesterase 1enzyme
CapecitabineCytidine deaminaseenzyme
CapecitabineThymidine phosphorylaseenzyme
CapmatinibCytochrome P450 3A4enzyme
CapmatinibAldehyde oxidaseenzyme
CapmatinibHepatocyte growth factor receptortarget
CapmatinibATP-dependent translocase ABCB1transporter
CapmatinibMultidrug and toxin extrusion protein 1transporter
CapmatinibMultidrug and toxin extrusion protein 2transporter
CapmatinibCytochrome P450 1A2enzyme
CapmatinibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
CapsaicinCytochrome P450 3A4enzyme
CapsaicinProstaglandin G/H synthase 2enzyme
CapsaicinMyeloperoxidaseenzyme
CapsaicinCytochrome P450 1A2enzyme
CapsaicinCytochrome P450 2E1enzyme
CapsaicinAmine oxidase [flavin-containing] Aenzyme
CapsaicinDopamine beta-hydroxylaseenzyme
CapsaicinGlutamine synthetaseenzyme
CapsaicinCholinesteraseenzyme
CapsaicinTransient receptor potential cation channel subfamily V member 1target
CapsaicinProhibitin-2target
CarbamazepineNeuronal acetylcholine receptor subunit alpha-4target
CarbamazepineCytochrome P450 2C8enzyme
CarbamazepineCytochrome P450 2B6enzyme
CarbamazepineCytochrome P450 3A4enzyme
CarbamazepineCytochrome P450 1A2enzyme
CarbamazepineCytochrome P450 2C19enzyme
CarbamazepineCytochrome P450 2C9enzyme
CarbamazepineATP-dependent translocase ABCB1transporter
CarbamazepineCytochrome P450 3A5enzyme
CarbamazepineUDP-glucuronosyltransferase 2B7enzyme
CarbamazepineRalA-binding protein 1transporter
CarbamazepineATP-binding cassette sub-family C member 2transporter
CarbamazepineVoltage-gated sodium channel alpha subunittarget
CarbamazepineNuclear receptor subfamily 1 group I member 2target
CarbamazepineUDP-glucuronosyltransferase 1A1enzyme
CarbamazepineUDP-glucuronosyltransferase 1A6enzyme
CarbamazepineUDP-glucuronosyltransferase 1A7enzyme
CarbazochromeGlutathione S-transferase Mu 1enzyme
CarbazochromeGlutathione S-transferase Mu 2enzyme
CarbazochromeNADPH--cytochrome P450 reductaseenzyme
CarbazochromeCytochrome P450 3A4enzyme
CarbazochromeRibosyldihydronicotinamide dehydrogenase [quinone]enzyme
CarbomycinCytochrome P450 3A4enzyme
Carbomycin23S ribosomal RNAtarget
CariprazineCytochrome P450 2C9enzyme
CariprazineCytochrome P450 2E1enzyme
CariprazineCytochrome P450 2C19enzyme
CariprazineCytochrome P450 3A4enzyme
CariprazineCytochrome P450 2D6enzyme
CariprazineATP-dependent translocase ABCB1transporter
CariprazineCytochrome P450 3A5enzyme
CariprazineD(3) dopamine receptortarget
CariprazineD(2) dopamine receptortarget
Cariprazine5-hydroxytryptamine receptor 1Atarget
Cariprazine5-hydroxytryptamine receptor 2Btarget
Cariprazine5-hydroxytryptamine receptor 2Atarget
CariprazineHistamine H1 receptortarget
Cariprazine5-hydroxytryptamine receptor 2Ctarget
CariprazineAlpha-1A adrenergic receptortarget
CariprazineCytochrome P450 1A2enzyme
CasimersenDMD gene (exon 45 casimersen target site)target
CasimersenCytochrome P450 2C19enzyme
CasimersenCytochrome P450 2C9enzyme
CasimersenCytochrome P450 3A5enzyme
CasimersenCytochrome P450 3A4enzyme
CaspofunginATP-dependent translocase ABCB1transporter
Caspofungin1,3-beta-glucan synthase component GSC2target
Caspofungin1,3-beta-glucan synthase component FKS1target
CaspofunginCytochrome P450 3A4enzyme
CaspofunginSolute carrier organic anion transporter family member 1B3transporter
CaspofunginSolute carrier organic anion transporter family member 1B1transporter
CaspofunginSolute carrier family 22 member 6transporter
CaspofunginSolute carrier family 22 member 1transporter
CathineSolute carrier family 22 member 2transporter
CathineSodium-dependent noradrenaline transportertarget
CathineSodium-dependent dopamine transportertarget
CathineCytochrome P450 2A6enzyme
CathineCytochrome P450 3A4enzyme
CelecoxibATP-dependent translocase ABCB1transporter
CelecoxibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
CelecoxibProstaglandin G/H synthase 2enzyme
CelecoxibSialidase-1target
CelecoxibSignal transducer and activator of transcription 3target
CelecoxibCadherin-11target
CelecoxibProstaglandin G/H synthase 2target
Celecoxib3-phosphoinositide-dependent protein kinase 1target
CelecoxibCytochrome P450 2C9enzyme
CelecoxibCytochrome P450 2D6enzyme
CelecoxibATP-binding cassette sub-family C member 4transporter
CelecoxibCytochrome P450 3A4enzyme
CelecoxibCytochrome P450 2C8enzyme
CelecoxibCarbonic anhydrase 2target
CelecoxibCarbonic anhydrase 3target
CelecoxibBile salt export pumptransporter
CenobamateCytochrome P450 2C8enzyme
CenobamateAlbumincarrier
CenobamateCytochrome P450 3A5enzyme
CenobamateCytochrome P450 3A4enzyme
CenobamateCytochrome P450 2C19enzyme
CenobamateCytochrome P450 2B6enzyme
CenobamateCytochrome P450 2A6enzyme
CenobamateCytochrome P450 2E1enzyme
CenobamateUDP-glucuronosyltransferase 2B4enzyme
CenobamateUDP-glucuronosyltransferase 2B7enzyme
CenobamateVoltage-gated sodium channel alpha subunittarget
CenobamateGamma-aminobutyric acid receptor subunit alpha-1target
Cepeginterferon alfa-2BCytochrome P450 1A2enzyme
Cepeginterferon alfa-2BInterferon alpha/beta receptor (IFNAR)target
CeritinibCytochrome P450 3A4enzyme
CeritinibALK tyrosine kinase receptortarget
CeritinibATP-dependent translocase ABCB1transporter
CeritinibCytochrome P450 2C9enzyme
CerivastatinSolute carrier organic anion transporter family member 1B1transporter
CerivastatinCytochrome P450 2B6enzyme
CerivastatinUDP-glucuronosyltransferase 1A1enzyme
CerivastatinBile salt export pumptransporter
CerivastatinCytochrome P450 2C8enzyme
CerivastatinCytochrome P450 3A4enzyme
CerivastatinCytochrome P450 2D6enzyme
CerivastatinCytochrome P450 2C9enzyme
CerivastatinCytochrome P450 3A5enzyme
CerivastatinCytochrome P450 3A7enzyme
CerivastatinATP-dependent translocase ABCB1transporter
Cerivastatin3-hydroxy-3-methylglutaryl-coenzyme A reductasetarget
CerivastatinATP-binding cassette sub-family C member 2transporter
CerivastatinBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
CethromycinCytochrome P450 3A5enzyme
CethromycinCytochrome P450 3A4enzyme
CethromycinATP-dependent translocase ABCB1transporter
Cethromycin23S ribosomal RNAtarget
ChamazuleneCytochrome P450 2D6enzyme
ChamazuleneCytochrome P450 1A2enzyme
ChamazuleneCytochrome P450 3A4enzyme
ChloramphenicolComplement decay-accelerating factortarget
ChloramphenicolDr hemagglutinin structural subunittarget
ChloramphenicolCytochrome P450 2C19enzyme
ChloramphenicolCytochrome P450 3A4enzyme
ChloramphenicolCytochrome P450 3A5enzyme
ChloramphenicolCytochrome P450 3A7enzyme
ChloramphenicolSolute carrier family 22 member 6transporter
ChloramphenicolLarge ribosomal subunit protein uL16target
ChloramphenicolChloramphenicol acetyltransferase 3enzyme
ChloramphenicolChloramphenicol 3-O phosphotransferaseenzyme
ChloramphenicolChloramphenicol acetyltransferaseenzyme
ChloroquineTumor necrosis factortarget
ChloroquineToll-like receptor 9target
ChloroquineGlutathione S-transferase A2target
ChloroquineCytochrome P450 2D6enzyme
ChloroquineCytochrome P450 3A4enzyme
ChloroquineCytochrome P450 1A1enzyme
ChloroquineCytochrome P450 2C8enzyme
ChloroquineCytochrome P450 3A5enzyme
ChloroquineGlutathione S-transferasetarget
ChloroquineATP-dependent translocase ABCB1transporter
ChloroquineAlbumincarrier
Chloroquinealpha1-acid glycoproteincarrier
ChloroquineHigh mobility group protein B1target
ChloroquineGlutathione S-transferase Mu 1target
ChloroquineAngiotensin-converting enzyme 2target
ChloroquineAtypical chemokine receptor 1target
ChlorpheniramineHistamine H1 receptortarget
ChlorpheniramineCytochrome P450 3A4enzyme
ChlorpheniramineCytochrome P450 2D6enzyme
ChlorpheniramineSodium-dependent serotonin transportertarget
ChlorpheniramineSodium-dependent noradrenaline transportertarget
ChlorpheniramineSodium-dependent dopamine transportertarget
ChlorpheniramineCytochrome P450 3A5enzyme
ChlorpheniramineCytochrome P450 3A7enzyme
ChlorpheniramineSolute carrier family 22 member 2transporter
ChlorpheniramineSolute carrier family 22 member 1transporter
ChlorpromazineAlpha-1 adrenergic receptorstarget
ChlorpromazineCalmodulintarget
ChlorpromazineBile salt export pumptransporter
ChlorpromazineD(2) dopamine receptortarget
Chlorpromazine5-hydroxytryptamine receptor 2Atarget
ChlorpromazineCytochrome P450 2D6enzyme
ChlorpromazineCholinesteraseenzyme
ChlorpromazineCytochrome P450 1A2enzyme
ChlorpromazineAlbumincarrier
ChlorpromazineATP-dependent translocase ABCB1transporter
ChlorpromazineD(1A) dopamine receptortarget
Chlorpromazine5-hydroxytryptamine receptor 1Atarget
ChlorpromazineAlpha-1A adrenergic receptortarget
ChlorpromazineAlpha-1B adrenergic receptortarget
ChlorpromazineCytochrome P450 2E1enzyme
ChlorpromazineCytochrome P450 3A4enzyme
ChlorpromazineHistamine H1 receptortarget
ChlorpromazineVoltage-gated inwardly rectifying potassium channel KCNH2target
ChlorpromazineD(1) dopamine receptortarget
ChlorpromazineD(3) dopamine receptortarget
ChlorpromazineD(4) dopamine receptortarget
ChlorpromazineD(1B) dopamine receptortarget
Chlorpromazine5-hydroxytryptamine receptor 2Ctarget
Chlorpromazine5-hydroxytryptamine 2 receptortarget
ChlorpromazineHistamine H4 receptortarget
ChlorpromazineAlpha-2 adrenergic receptorstarget
ChlorpromazineMuscarinic acetylcholine receptor M1target
ChlorpromazineMuscarinic acetylcholine receptor M3target
ChlorpromazineSphingomyelin phosphodiesterasetarget
Chlorpromazinealpha1-acid glycoproteintarget
Chlorpromazine5-hydroxytryptamine receptor 6target
Chlorpromazine5-hydroxytryptamine receptor 7target
ChlorzoxazoneCalcium-activated potassium channel subunit alpha-1target
ChlorzoxazoneCytochrome P450 2E1enzyme
ChlorzoxazoneCytochrome P450 1A2enzyme
ChlorzoxazoneCytochrome P450 2A6enzyme
ChlorzoxazoneCytochrome P450 1A1enzyme
ChlorzoxazoneCytochrome P450 2D6enzyme
ChlorzoxazoneCytochrome P450 3A4enzyme
ChlorzoxazoneIntermediate conductance calcium-activated potassium channel protein 4target
CholecalciferolCytochrome P450 2C8enzyme
CholecalciferolCytochrome P450 1A1enzyme
CholecalciferolVitamin D3 receptortarget
CholecalciferolCytochrome P450 3A4enzyme
CholecalciferolCytochrome P450 2J2enzyme
CholecalciferolSterol 26-hydroxylase, mitochondrialenzyme
CholecalciferolVitamin D 25-hydroxylaseenzyme
CholecalciferolCholesterol side-chain cleavage enzyme, mitochondrialenzyme
CholecalciferolVitamin D-binding proteincarrier
CiglitazonePeroxisome proliferator-activated receptor gammatarget
CiglitazoneCytochrome P450 3A4enzyme
CiglitazoneCytochrome P450 2C8enzyme
CimetidineCytochrome P450 3A5enzyme
CimetidineAlbumincarrier
CimetidineMultidrug and toxin extrusion protein 2transporter
CimetidineBile salt export pumptransporter
CimetidineFlavin-containing monooxygenase 1enzyme
CimetidineFlavin-containing monooxygenase 3enzyme
CimetidineCytochrome P450 2E1enzyme
CimetidineCytochrome P450 2C9enzyme
CimetidineCytochrome P450 2C8enzyme
CimetidineCytochrome P450 11B1, mitochondrialenzyme
CimetidineSolute carrier family 22 member 7transporter
CimetidineSolute carrier family 22 member 11transporter
CimetidineHistamine H2 receptortarget
CimetidineCytochrome P450 1A2enzyme
CimetidineCytochrome P450 2D6enzyme
CimetidineCytochrome P450 2C19enzyme
CimetidineCytochrome P450 3A4enzyme
CimetidineATP-dependent translocase ABCB1transporter
CimetidineSolute carrier family 22 member 4transporter
CimetidineMultidrug and toxin extrusion protein 1transporter
CimetidineOrganic anion transporter 3transporter
CimetidineSolute carrier family 22 member 6transporter
CimetidineOrganic cation/carnitine transporter 2transporter
CimetidineSolute carrier family 22 member 3transporter
CimetidineSolute carrier family 22 member 1transporter
CimetidineSolute carrier family 22 member 2transporter
CinacalcetExtracellular calcium-sensing receptortarget
CinacalcetCytochrome P450 3A4enzyme
CinacalcetCytochrome P450 2D6enzyme
CinacalcetCytochrome P450 1A2enzyme
CinchonidineCytochrome P450 2D6target
Cinnamon oilAryl hydrocarbon receptortarget
Cinnamon oilNuclear receptor subfamily 1 group I member 2target
Cinnamon oilXanthine dehydrogenase/oxidasetarget
Cinnamon oilCytochrome P450 1A2enzyme
Cinnamon oilCytochrome P450 2C9enzyme
CinoxacinDNA topoisomerase 2-betatarget
CinoxacinDNAtarget
CinoxacinDNA gyrase subunit Atarget
CinoxacinSolute carrier family 22 member 6transporter
CinoxacinCytochrome P450 1A2enzyme
CinoxacinDNA topoisomerase 2-alphatarget
CiprofloxacinMultidrug and toxin extrusion protein 2transporter
CiprofloxacinDNA gyrase subunit Atarget
CiprofloxacinDNA topoisomerase 4 subunit Atarget
CiprofloxacinDNA topoisomerase 2-alphatarget
CiprofloxacinCytochrome P450 1A2enzyme
CiprofloxacinCytochrome P450 3A4enzyme
CiprofloxacinCytochrome P450 3A5enzyme
CiprofloxacinCytochrome P450 3A7enzyme
CiprofloxacinATP-dependent translocase ABCB1transporter
CiprofloxacinVoltage-gated inwardly rectifying potassium channel KCNH2target
CiprofloxacinDNA gyrase subunit Atarget
CiprofloxacinDNA topoisomerase 4 subunit Atarget
CiprofloxacinDNA topoisomerase 4 subunit Btarget
CiprofloxacinDNA gyrase subunit Atarget
CiprofloxacinMultidrug resistance protein MdtKtarget
CiprofloxacinGyrase Atarget
CiprofloxacinDNA gyrase subunit Atarget
CiprofloxacinMultidrug and toxin extrusion protein 1transporter
CiprofloxacinDNA gyrase subunit Btarget
CiprofloxacinAlbumincarrier
CiprofloxacinThymidylate synthasetarget
CisaprideCytochrome P450 2C19enzyme
CisaprideCytochrome P450 2B6enzyme
CisaprideCytochrome P450 2C8enzyme
CisaprideCytochrome P450 2C9enzyme
CisaprideCytochrome P450 2D6enzyme
CisaprideCytochrome P450 2A6enzyme
CisaprideCytochrome P450 3A7enzyme
CisaprideCytochrome P450 3A5enzyme
CisaprideCytochrome P450 3A4enzyme
Cisapride5-hydroxytryptamine receptor 2Atarget
CisaprideVoltage-gated inwardly rectifying potassium channel KCNH2target
Cisapride5-hydroxytryptamine receptor 3Atarget
Cisapride5-hydroxytryptamine receptor 4target
CisplatinGlutathione S-transferase theta-1enzyme
CisplatinMetallothionein-1Aenzyme
CisplatinMetallothionein-2enzyme
CisplatinSuperoxide dismutase [Cu-Zn]enzyme
CisplatinGlutathione S-transferase Penzyme
CisplatinNAD(P)H dehydrogenase [quinone] 1enzyme
CisplatinGlutathione S-transferase Mu 1enzyme
CisplatinDNA-3-methyladenine glycosylasetarget
CisplatinAlpha-2-macroglobulintarget
CisplatinAlbumincarrier
CisplatinSerotransferrintarget
CisplatinCopper transport protein ATOX1target
CisplatinBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
CisplatinCytochrome P450 4A11enzyme
CisplatinCholinesteraseenzyme
CisplatinCytochrome P450 2B6enzyme
CisplatinCytochrome P450 2C9enzyme
CisplatinArylamine N-acetyltransferaseenzyme
CisplatinXanthine dehydrogenase/oxidaseenzyme
CisplatinMyeloperoxidaseenzyme
CisplatinProstaglandin G/H synthase 2enzyme
CisplatinCopper-transporting ATPase 1transporter
CisplatinCopper-transporting ATPase 2transporter
CisplatinATP-binding cassette sub-family C member 6transporter
CisplatinProtein SLC31A2transporter
CisplatinHigh affinity copper uptake protein 1transporter
CisplatinSolute carrier family 22 member 2transporter
CisplatinATP-binding cassette sub-family C member 2transporter
CisplatinATP-binding cassette sub-family C member 5transporter
CisplatinATP-binding cassette sub-family C member 3transporter
CisplatinDNAtarget
CitalopramAldehyde oxidaseenzyme
CitalopramAmine oxidase [flavin-containing] Benzyme
CitalopramAmine oxidase [flavin-containing] Aenzyme
CitalopramHistamine H1 receptortarget
CitalopramCytochrome P450 1A2enzyme
CitalopramATP-dependent translocase ABCB1transporter
CitalopramCytochrome P450 3A4enzyme
CitalopramCytochrome P450 2D6enzyme
CitalopramCytochrome P450 2C19enzyme
CitalopramSodium-dependent serotonin transportertarget
ClarithromycinLarge ribosomal subunit protein uL10target
ClarithromycinCytochrome P450 3A4enzyme
ClarithromycinCytochrome P450 3A5enzyme
ClarithromycinATP-dependent translocase ABCB1transporter
ClarithromycinSolute carrier family 22 member 7transporter
ClarithromycinVoltage-gated inwardly rectifying potassium channel KCNH2target
ClarithromycinSolute carrier organic anion transporter family member 1B1target
ClarithromycinSolute carrier organic anion transporter family member 1B3target
ClarithromycinBile salt export pumptransporter
ClarithromycinSolute carrier organic anion transporter family member 1B1transporter
ClarithromycinSolute carrier organic anion transporter family member 1B3transporter
ClascoteroneCytochrome P450 2C8enzyme
ClascoteroneCytochrome P450 3A4enzyme
ClascoteroneCytochrome P450 2E1enzyme
ClascoteroneCytochrome P450 2D6enzyme
ClascoteroneCytochrome P450 2C19enzyme
ClascoteroneCytochrome P450 2C9enzyme
ClascoteroneCytochrome P450 2B6enzyme
ClascoteroneCytochrome P450 1A2enzyme
ClascoteroneAndrogen receptortarget
ClemastineHistamine H1 receptortarget
ClemastineCytochrome P450 2D6enzyme
ClevidipineVoltage-dependent L-type calcium channel subunit alpha-1Ftarget
ClevidipineVoltage-dependent L-type calcium channel subunit alpha-1Starget
ClevidipineVoltage-dependent L-type calcium channel subunit alpha-1Dtarget
ClevidipineVoltage-dependent L-type calcium channel subunit alpha-1Ctarget
ClevidipineCytochrome P450 2C9enzyme
ClevidipineCytochrome P450 2D6enzyme
ClevidipineCytochrome P450 2E1enzyme
ClevidipineVoltage gated L-type calcium channeltarget
ClevidipineCholinesteraseenzyme
ClevidipineCytochrome P450 3A4enzyme
ClevidipineCytochrome P450 2C19enzyme
ClinafloxacinDNA gyrase subunit Btarget
ClinafloxacinDNA gyrase subunit Atarget
ClinafloxacinCytochrome P450 2C9enzyme
ClinafloxacinCytochrome P450 2D6enzyme
ClinafloxacinCytochrome P450 2C19enzyme
ClinafloxacinCytochrome P450 1A2enzyme
ClindamycinCytochrome P450 3A4enzyme
ClindamycinCytochrome P450 3A5enzyme
ClindamycinAlpha-1-acid glycoprotein 1carrier
ClindamycinATP-dependent translocase ABCB1transporter
ClindamycinLarge ribosomal subunit protein uL1target
ClobazamCytochrome P450 2C19enzyme
ClobazamCytochrome P450 3A4enzyme
ClobazamCytochrome P450 2B6enzyme
ClobazamCytochrome P450 2C18enzyme
ClobazamATP-dependent translocase ABCB1transporter
ClobazamGABA(A) Receptortarget
ClobazamCytochrome P450 2D6enzyme
ClobazamGABA(A) Receptor Benzodiazepine Binding Sitetarget
ClobazamAlbumincarrier
ClobazamAlpha-1-acid glycoprotein 1carrier
ClobazamCytochrome P450 2C9enzyme
ClobazamUDP-glucuronosyltransferase 1A4enzyme
ClobazamUDP-glucuronosyltransferase 1A6enzyme
ClobazamUDP-glucuronosyltransferase 2B4enzyme
ClobazamUDP-glucuronosyltransferase 1A1enzyme
ClobazamCytochrome P450 1A2enzyme
ClobazamCytochrome P450 2C8enzyme
ClobazamGamma-aminobutyric acid receptor subunit gamma-3target
ClobazamGamma-aminobutyric acid receptor subunit alpha-1target
ClobazamCytochrome P450 3A7enzyme
ClobazamCytochrome P450 3A5enzyme
ClofazimineCytochrome P450 3A4enzyme
ClofaziminePeroxisome proliferator-activated receptor gammatarget
ClofazimineCytochrome P450 2C8enzyme
ClofazimineCytochrome P450 2D6enzyme
ClofazimineMultidrug resistance-associated protein 1transporter
ClofazimineBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
ClofazimineATP-dependent translocase ABCB1transporter
ClofazimineAlbumincarrier
ClofaziminePotassium voltage-gated channel subfamily A member 3target
ClofazimineCytochrome P450 3A5enzyme
ClofibrateLipoprotein lipasetarget
ClofibrateThyroxine-binding globulincarrier
ClofibrateCytochrome P450 4A11enzyme
ClofibrateCytochrome P450 1A1enzyme
ClofibratePeroxisome proliferator-activated receptor alphatarget
ClofibrateCytochrome P450 3A4enzyme
ClofibrateGlutathione S-transferase A2enzyme
ClofibrateCytochrome P450 2E1enzyme
ClomipramineSodium-dependent serotonin transportertarget
ClomipramineSodium-dependent noradrenaline transportertarget
ClomipramineGlutathione S-transferase Ptarget
Clomipramine5-hydroxytryptamine receptor 2Atarget
ClomipramineCytochrome P450 1A2enzyme
ClomipramineCytochrome P450 2D6enzyme
ClomipramineCytochrome P450 2C19enzyme
ClomipramineATP-dependent translocase ABCB1transporter
ClomipramineCytochrome P450 3A4enzyme
Clomipramine5-hydroxytryptamine receptor 2Btarget
Clomipramine5-hydroxytryptamine receptor 2Ctarget
ClomipramineAlbumincarrier
ClonazepamCytochrome P450 3A4enzyme
ClonazepamAlbumincarrier
ClonazepamCytochrome P450 2E1enzyme
ClonazepamArylamine N-acetyltransferase 2enzyme
ClonazepamNuclear receptor subfamily 1 group I member 2target
ClonazepamGABA(A) Receptor Benzodiazepine Binding Sitetarget
CloperidoneCytochrome P450 2C9enzyme
ClopidogrelCytochrome P450 2C19enzyme
ClopidogrelSolute carrier family 22 member 1transporter
ClopidogrelATP-dependent translocase ABCB1transporter
ClopidogrelLiver carboxylesterase 1enzyme
ClopidogrelCytochrome P450 2C8enzyme
ClopidogrelCytochrome P450 1A2enzyme
ClopidogrelCytochrome P450 2C9enzyme
ClopidogrelSolute carrier family 22 member 2transporter
ClopidogrelCytochrome P450 3A5enzyme
ClopidogrelCytochrome P450 2B6enzyme
ClopidogrelCytochrome P450 3A4enzyme
ClopidogrelP2Y purinoceptor 12target
ClopidogrelAlbumincarrier
ClotrimazoleCytochrome P450 2E1enzyme
ClotrimazoleIntermediate conductance calcium-activated potassium channel protein 4target
ClotrimazoleCytochrome P450 2D6enzyme
ClotrimazoleCytochrome P450 2C8enzyme
ClotrimazoleCytochrome P450 3A4enzyme
ClotrimazoleCytochrome P450 2B6enzyme
ClotrimazoleATP-dependent translocase ABCB1transporter
ClotrimazoleCytochrome P450 2A6enzyme
ClotrimazoleCytochrome P450 2C9enzyme
ClotrimazoleCytochrome P450 3A7enzyme
ClotrimazoleLanosterol 14-alpha demethylasetarget
ClotrimazoleNuclear receptor subfamily 1 group I member 2target
ClotrimazoleHydroxycarboxylic acid receptor 2target
ClotrimazoleBile salt export pumptransporter
ClotrimazoleSolute carrier organic anion transporter family member 1B1transporter
ClotrimazoleSolute carrier organic anion transporter family member 1B3transporter
ClotrimazoleErgosteroltarget
ClotrimazoleC-X-C chemokine receptor type 2target
ClozapineGamma-aminobutyric acid type B receptor subunit 2target
ClozapineGamma-aminobutyric acid receptor subunit alpha-1target
ClozapineGamma-aminobutyric acid receptor subunit gamma-1target
ClozapineGamma-aminobutyric acid receptor subunit beta-1target
ClozapineSolute carrier family 22 member 3transporter
ClozapineSolute carrier family 22 member 2transporter
ClozapineSolute carrier family 22 member 1transporter
ClozapineGamma-aminobutyric acid type B receptor subunit 1target
ClozapineD(1B) dopamine receptortarget
ClozapineAlbumincarrier
ClozapineAlpha-1-acid glycoprotein 1carrier
ClozapineGlutathione S-transferase Ptarget
ClozapineCytochrome P450 2C8enzyme
ClozapineCytochrome P450 2A6enzyme
ClozapineCytochrome P450 1A1enzyme
ClozapineUDP-glucuronosyltransferase 1A4enzyme
ClozapineFlavin-containing monooxygenase 3enzyme
ClozapineD(4) dopamine receptortarget
ClozapineHistamine H1 receptortarget
ClozapineD(2) dopamine receptortarget
ClozapineNeuron-specific vesicular protein calcyontarget
ClozapineHistamine H4 receptortarget
Clozapine5-hydroxytryptamine receptor 2Atarget
Clozapine5-hydroxytryptamine receptor 1Atarget
Clozapine5-hydroxytryptamine receptor 2Ctarget
ClozapineD(1A) dopamine receptortarget
ClozapineCytochrome P450 1A2enzyme
ClozapineCytochrome P450 2D6enzyme
ClozapineD(3) dopamine receptortarget
ClozapineMuscarinic acetylcholine receptor M1target
ClozapineMuscarinic acetylcholine receptor M2target
ClozapineMuscarinic acetylcholine receptor M3target
ClozapineMuscarinic acetylcholine receptor M4target
ClozapineMuscarinic acetylcholine receptor M5target
Clozapine5-hydroxytryptamine receptor 1Btarget
Clozapine5-hydroxytryptamine receptor 1Dtarget
Clozapine5-hydroxytryptamine receptor 1Etarget
Clozapine5-hydroxytryptamine receptor 3Atarget
Clozapine5-hydroxytryptamine receptor 6target
Clozapine5-hydroxytryptamine receptor 7target
ClozapineAlpha-1A adrenergic receptortarget
ClozapineAlpha-1B adrenergic receptortarget
ClozapineAlpha-2A adrenergic receptortarget
ClozapineAlpha-2B adrenergic receptortarget
ClozapineAlpha-2C adrenergic receptortarget
ClozapineCytochrome P450 2C9enzyme
ClozapineATP-dependent translocase ABCB1transporter
ClozapineCytochrome P450 3A4enzyme
ClozapineCytochrome P450 2C19enzyme
Cobalt chlorideCytochrome P450 1A2enzyme
Cobalt chlorideProlyl hydroxylase EGLN3target
Cobalt chlorideProlyl hydroxylase EGLN2target
Cobalt chlorideEgl nine homolog 1target
CobicistatSolute carrier organic anion transporter family member 1B1transporter
CobicistatSolute carrier organic anion transporter family member 1B3transporter
CobicistatCytochrome P450 3A4target
CobicistatCytochrome P450 3A4enzyme
CobicistatCytochrome P450 3A5target
CobicistatCytochrome P450 3A7target
CobicistatCytochrome P450 3A Subfamilytarget
CobicistatCytochrome P450 3A7enzyme
CobicistatCytochrome P450 3A5enzyme
CobicistatBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
CobicistatATP-dependent translocase ABCB1transporter
CobicistatCytochrome P450 2D6enzyme
CobimetinibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
CobimetinibATP-dependent translocase ABCB1transporter
CobimetinibUDP-glucuronosyltransferase 2B7enzyme
CobimetinibCytochrome P450 2D6enzyme
CobimetinibCytochrome P450 3A5enzyme
CobimetinibAlpha-1-acid glycoprotein 1carrier
CobimetinibDual specificity mitogen-activated protein kinase kinase 2target
CobimetinibSolute carrier organic anion transporter family member 1B3transporter
CobimetinibSolute carrier organic anion transporter family member 1B1transporter
CobimetinibCytochrome P450 3A4enzyme
CobimetinibDual specificity mitogen-activated protein kinase kinase 1target
CocaineCytochrome P450 3A4enzyme
CocaineSodium-dependent dopamine transportertarget
CocaineSodium-dependent serotonin transportertarget
CocaineSodium channel proteintarget
CocaineSodium-dependent noradrenaline transportertarget
CocaineMuscarinic acetylcholine receptor M1target
CocaineMuscarinic acetylcholine receptor M2target
CocaineCytochrome P450 2D6enzyme
CocaineCytochrome P450 2C8enzyme
CocaineSigma non-opioid intracellular receptor 1target
CocaineLiver carboxylesterase 1target
CocaineCholinesteraseenzyme
CocaineSodium-dependent dopamine transportertransporter
Cocainealpha1-acid glycoproteincarrier
CocaineLiver carboxylesterase 1enzyme
CocaineVoltage-gated sodium channel alpha subunittarget
CocaineSolute carrier family 22 member 2transporter
ColchicineAlbumincarrier
ColchicineCytochrome P450 2E1enzyme
ColchicineCytochrome P450 2C8enzyme
ColchicineCytochrome P450 2B6enzyme
ColchicineATP-dependent translocase ABCB1transporter
ColchicineCytochrome P450 3A4enzyme
ColchicineTubulin beta chaintarget
Coltuximab ravtansineB-lymphocyte antigen CD19target
Coltuximab ravtansineCytochrome P450 3A4enzyme
ConivaptanVasopressin V1a receptortarget
ConivaptanVasopressin V2 receptortarget
ConivaptanCytochrome P450 3A4enzyme
ConivaptanATP-dependent translocase ABCB1transporter
Conjugated estrogensMultidrug resistance-associated protein 1transporter
Conjugated estrogensEstrogen receptortarget
Conjugated estrogensCytochrome P450 3A4enzyme
Conjugated estrogensCytochrome P450 1A2enzyme
Conjugated estrogensCatechol O-methyltransferaseenzyme
Conjugated estrogensATP-binding cassette sub-family C member 3transporter
Conjugated estrogensATP-binding cassette sub-family C member 4transporter
Conjugated estrogensBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
Conjugated estrogensThyroxine-binding globulincarrier
Conjugated estrogensSex hormone-binding globulincarrier
Conjugated estrogensAlbumincarrier
Conjugated estrogensEstrogen receptor betatarget
Conjugated estrogensSolute carrier organic anion transporter family member 3A1transporter
Conjugated estrogensSolute carrier family 22 member 11transporter
Conjugated estrogensSolute carrier organic anion transporter family member 1B3transporter
Conjugated estrogensATP-binding cassette sub-family C member 11transporter
Conjugated estrogensSolute carrier organic anion transporter family member 4A1transporter
Conjugated estrogensATP-binding cassette sub-family C member 2transporter
Conjugated estrogensOrganic solute transporter subunit betatransporter
Conjugated estrogensOrganic solute transporter subunit alphatransporter
Conjugated estrogensHepatic sodium/bile acid cotransportertransporter
Conjugated estrogensSolute carrier family 22 member 10transporter
Conjugated estrogensOrganic anion transporter 3transporter
Conjugated estrogensSolute carrier organic anion transporter family member 1C1transporter
Conjugated estrogensSolute carrier organic anion transporter family member 1B1transporter
Conjugated estrogensSolute carrier organic anion transporter family member 1A2transporter
Conjugated estrogensSolute carrier organic anion transporter family member 2B1transporter
Conjugated estrogensATP-dependent translocase ABCB1transporter
Conjugated estrogensSolute carrier family 22 member 6transporter
CrisaboroleCytochrome P450 2B6enzyme
CrisaboroleCytochrome P450 2C8enzyme
CrisaboroleCytochrome P450 2C9enzyme
CrisaborolePhosphodiesterase 4target
Crisaborole3',5'-cyclic-AMP phosphodiesterase 4Dtarget
Crisaborole3',5'-cyclic-AMP phosphodiesterase 4Atarget
Crisaborole3',5'-cyclic-AMP phosphodiesterase 4Btarget
Crisaborole3',5'-cyclic-AMP phosphodiesterase 4Ctarget
CrizotinibALK tyrosine kinase receptortarget
CrizotinibCytochrome P450 3A4enzyme
CrizotinibCytochrome P450 3A5enzyme
CrizotinibATP-dependent translocase ABCB1transporter
CrizotinibHepatocyte growth factor receptortarget
CrizotinibCytochrome P450 2B6enzyme
CrizotinibCytochrome P450 3A Subfamilyenzyme
CrizotinibAlbumincarrier
Crizotinibalpha1-acid glycoproteincarrier
CrizotinibProto-oncogene tyrosine-protein kinase ROStarget
CrizotinibMacrophage-stimulating protein receptortarget
CryptotanshinoneAcetylcholinesterasetarget
CryptotanshinoneCholinesterasetarget
CryptotanshinoneCytochrome P450 2C9enzyme
CryptotanshinoneCytochrome P450 1A2enzyme
CryptotanshinoneProstaglandin G/H synthase 2target
Cryptotanshinone5'-AMP-activated protein kinasetarget
CryptotanshinoneEstrogen receptortarget
CryptotanshinoneCytochrome P450 2D6enzyme
CurcuminXanthine dehydrogenase/oxidasetarget
CurcuminCarbonic anhydrase 1target
CurcuminGlutathione S-transferase Penzyme
CurcuminGlutathione S-transferase Mu 1enzyme
CurcuminGlutathione S-transferase A1enzyme
CurcuminCytochrome P450 2D6enzyme
CurcuminCytochrome P450 1A2enzyme
CurcuminCytochrome P450 2B6enzyme
CurcuminCytochrome P450 3A4enzyme
CurcuminCytochrome P450 2C9enzyme
CurcuminGlutathione S-transferase Ptarget
CurcuminCarbonyl reductase [NADPH] 1target
CurcuminATP-binding cassette sub-family C member 5target
CurcuminVitamin D3 receptortarget
CurcuminPeroxisome proliferator-activated receptor gammatarget
CurcuminCarbonic anhydrase 2target
CurcuminAmyloid-beta precursor proteintarget
CurcuminCarbonic anhydrase 4target
CurcuminProstaglandin G/H synthase 2target
CurcuminMatrix metalloproteinase-9target
CurcuminProstaglandin G/H synthase 1target
CurcuminDNA (cytosine-5)-methyltransferase 3Btarget
CurcuminCollagenase 3target
CurcuminATP-dependent translocase ABCB1transporter
CurcuminCarbonic anhydrase 14target
CurcuminNitric oxide synthase, inducibletarget
CurcuminCytochrome P450 3A4target
CurcuminCarbonic anhydrase 9target
CurcuminCarbonic anhydrase 6target
CurcuminCarbonic anhydrase 12target
Curcumin sulfateUDP-glucuronosyltransferases (UGTs)enzyme
Curcumin sulfateCytochrome P450 3A5enzyme
Curcumin sulfateCytochrome P450 3A4enzyme
Curcumin sulfateATP-dependent translocase ABCB1transporter
Curcumin sulfateCytochrome P450 2D6enzyme
Curcumin sulfateCytochrome P450 1A2enzyme
Curcumin sulfateCytochrome P450 2B6enzyme
Curcumin sulfateCytochrome P450 2C9enzyme
Curcumin sulfateGlutathione S-transferase Ptarget
Curcumin sulfateCarbonyl reductase [NADPH] 1target
Curcumin sulfateATP-binding cassette sub-family C member 5target
Curcumin sulfateVitamin D3 receptortarget
Curcumin sulfatePeroxisome proliferator-activated receptor gammatarget
Curcumin sulfateCytochrome P450 2C19enzyme
Curcumin sulfateSulfotransferase 1A3enzyme
Curcumin sulfateSulfotransferase 1B1enzyme
Curcumin sulfateSulfotransferase 1E1enzyme
Curcumin sulfateSulfotransferase 1C4enzyme
CyclizineAlbumincarrier
CyclizineCytochrome P450 2C9enzyme
CyclizineSulfotransferase 1E1target
CyclizineHistamine H1 receptortarget
CyclosporineHepatic sodium/bile acid cotransportertransporter
CyclosporineIleal sodium/bile acid cotransportertransporter
CyclosporineBile salt export pumptransporter
CyclosporineATP-dependent translocase ABCB1transporter
CyclosporineCytochrome P450 3A4enzyme
CyclosporineCytochrome P450 3A5enzyme
CyclosporineCalcineurin subunit B type 2target
CyclosporinePeptidyl-prolyl cis-trans isomerase Atarget
CyclosporineGuided entry of tail-anchored proteins factor CAMLGtarget
CyclosporineATP-binding cassette sub-family C member 2transporter
CyclosporineBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
CyclosporineSolute carrier organic anion transporter family member 1B1transporter
CyclosporineCytochrome P450 2C19enzyme
CyclosporineCytochrome P450 2D6enzyme
CyclosporinePeptidyl-prolyl cis-trans isomerase F, mitochondrialtarget
CyclosporineSolute carrier organic anion transporter family member 1B3transporter
CyclosporineProtein phosphatase 3 catalytic subunit alphatarget
CyclosporineATP-binding cassette sub-family C member 10transporter
CyclosporineSolute carrier family 22 member 6transporter
Cyproterone acetateAndrogen receptortarget
Cyproterone acetateProstate-specific antigentarget
Cyproterone acetateCytochrome P450 3A4enzyme
Cyproterone acetateAromataseenzyme
Cyproterone acetateGlucocorticoid receptortarget
Cyproterone acetateProgesterone receptortarget
DabrafenibLIM domain kinase 1target
DabrafenibSerine/threonine-protein kinase SIK1target
DabrafenibSolute carrier organic anion transporter family member 1B1transporter
DabrafenibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
DabrafenibATP-dependent translocase ABCB1transporter
DabrafenibCytochrome P450 2C8enzyme
DabrafenibCytochrome P450 3A4enzyme
DabrafenibCytochrome P450 2C9enzyme
DabrafenibCytochrome P450 2C19enzyme
DabrafenibCytochrome P450 1A2enzyme
DabrafenibAlbumincarrier
DabrafenibSolute carrier organic anion transporter family member 1A2transporter
DabrafenibSolute carrier family 22 member 2transporter
DabrafenibCytochrome P450 2B6enzyme
DabrafenibOrganic anion transporter 3transporter
DabrafenibSerine/threonine-protein kinase B-raftarget
DabrafenibRAF proto-oncogene serine/threonine-protein kinasetarget
DabrafenibSolute carrier family 22 member 6transporter
DabrafenibUDP-glucuronosyltransferase 1A1enzyme
DabrafenibSolute carrier organic anion transporter family member 1B3transporter
DabrafenibSerine/threonine-protein kinase Nek11target
DacomitinibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
DacomitinibReceptor tyrosine-protein kinase erbB-2target
DacomitinibReceptor tyrosine-protein kinase erbB-4target
DacomitinibEpidermal growth factor receptortarget
DacomitinibCytochrome P450 2D6enzyme
DacomitinibAlbumincarrier
DacomitinibCytochrome P450 3A4enzyme
DacomitinibCytochrome P450 2C9enzyme
DacomitinibUDP-glucuronosyltransferase 1A1enzyme
DacomitinibATP-dependent translocase ABCB1transporter
DacomitinibSolute carrier family 22 member 1transporter
DalfopristinBacterial 50S ribosomal proteintarget
DalfopristinCytochrome P450 3A4enzyme
DalfopristinStreptogramin A acetyltransferasetarget
DanazolCytochrome P450 3A4enzyme
DanazolEstrogen receptortarget
DanazolGonadotropin-releasing hormone receptortarget
DanazolPutative gonadotropin-releasing hormone II receptortarget
DanazolSex hormone-binding globulincarrier
DanazolC-C motif chemokine 2target
DanazolAromataseenzyme
DanazolAndrogen receptortarget
DanazolProgesterone receptortarget
DanoprevirGenome polyproteintarget
DanoprevirCytochrome P450 3A4enzyme
DanoprevirGag-Pol polyproteintarget
DapoxetineCytochrome P450 2D6enzyme
DapoxetineSodium-dependent serotonin transportertarget
Dapoxetine5-hydroxytryptamine receptor 2Ctarget
Dapoxetine5-hydroxytryptamine receptor 1Btarget
Dapoxetine5-hydroxytryptamine receptor 1Atarget
DapoxetineCytochrome P450 3A4enzyme
DaprodustatCytochrome P450 2C8enzyme
DaprodustatCytochrome P450 3A4enzyme
DaprodustatSolute carrier organic anion transporter family member 1B1transporter
DaprodustatSolute carrier organic anion transporter family member 1B3transporter
DaprodustatSolute carrier family 22 member 6transporter
DaprodustatOrganic anion transporter 3transporter
DaprodustatProlyl hydroxylase EGLN3target
DaprodustatBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
DaprodustatProlyl hydroxylase EGLN2target
DaprodustatEgl nine homolog 1target
DarifenacinCytochrome P450 2D6enzyme
DarifenacinMuscarinic acetylcholine receptor M3target
DarifenacinCytochrome P450 3A4enzyme
DarifenacinMuscarinic acetylcholine receptor M1target
DarifenacinMuscarinic acetylcholine receptor M2target
DarifenacinMuscarinic acetylcholine receptor M4target
DarifenacinMuscarinic acetylcholine receptor M5target
DarunavirGag-Pol polyproteintarget
DarunavirCytochrome P450 2D6enzyme
DarunavirAlpha-1-acid glycoprotein 1carrier
DarunavirAlbumincarrier
DarunavirSolute carrier organic anion transporter family member 1B1transporter
DarunavirCytochrome P450 3A4enzyme
DarunavirPol polyproteintarget
DarunavirATP-dependent translocase ABCB1transporter
DasatinibTyrosine-protein kinase Fgrtarget
DasatinibTyrosine-protein kinase FRKtarget
DasatinibHeat shock cognate 71 kDa proteintarget
DasatinibTyrosine-protein kinase Lyntarget
DasatinibMitogen-activated protein kinase kinase kinase 20target
DasatinibMitogen-activated protein kinase 14target
DasatinibAmidophosphoribosyltransferasetarget
DasatinibEphrin type-B receptor 4target
DasatinibTyrosine-protein kinase ABL1target
DasatinibEphrin type-A receptor 5target
DasatinibTyrosine-protein kinase CSKtarget
DasatinibBreakpoint cluster region proteintarget
DasatinibNuclear receptor subfamily 4 group A member 3target
DasatinibTyrosine-protein kinase BTKtarget
DasatinibFlavin-containing monooxygenase 3enzyme
DasatinibCytochrome P450 3A5enzyme
DasatinibCytochrome P450 1B1enzyme
DasatinibCytochrome P450 1A2enzyme
DasatinibCytochrome P450 1A1enzyme
DasatinibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
DasatinibATP-dependent translocase ABCB1transporter
DasatinibCytochrome P450 3A4enzyme
DasatinibSignal transducer and activator of transcription 5Btarget
DasatinibEphrin type-A receptor 2target
DasatinibPlatelet-derived growth factor receptor betatarget
DasatinibMast/stem cell growth factor receptor Kittarget
DasatinibTyrosine-protein kinase Yestarget
DasatinibTyrosine-protein kinase Lcktarget
DasatinibTyrosine-protein kinase Fyntarget
DasatinibProto-oncogene tyrosine-protein kinase Srctarget
DasatinibTyrosine-protein kinase ABL2target
DaunorubicinATP-binding cassette sub-family C member 10transporter
DaunorubicinCarbonyl reductase [NADPH] 3enzyme
DaunorubicinCarbonyl reductase [NADPH] 1enzyme
DaunorubicinAldo-keto reductase family 1 member B1enzyme
DaunorubicinCytochrome P450 3A4enzyme
DaunorubicinCytochrome P450 1B1enzyme
DaunorubicinDNA topoisomerase 2-betatarget
DaunorubicinDNA topoisomerase 2-alphatarget
DaunorubicinBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
DaunorubicinATP-binding cassette sub-family C member 6transporter
DaunorubicinMultidrug resistance-associated protein 1transporter
DaunorubicinATP-dependent translocase ABCB1transporter
DaunorubicinNADPH--cytochrome P450 reductaseenzyme
DaunorubicinCytochrome P450 3A5enzyme
DaunorubicinDNAtarget
DefactinibMultidrug and toxin extrusion protein 2transporter
DefactinibFocal adhesion kinase 1target
DefactinibProtein-tyrosine kinase 2-betatarget
DefactinibCytochrome P450 3A4enzyme
DefactinibCytochrome P450 2C9enzyme
DefactinibCytochrome P450 2B6enzyme
DefactinibCytochrome P450 1A2enzyme
DefactinibUDP-glucuronosyltransferase 1A1enzyme
DefactinibATP-binding cassette sub-family B member 5transporter
DefactinibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
DefactinibSolute carrier organic anion transporter family member 1B1transporter
DefactinibSolute carrier organic anion transporter family member 1B3transporter
DeferasiroxUDP-glucuronosyltransferase 1A1enzyme
DeferasiroxCytochrome P450 1A2enzyme
DeferasiroxCytochrome P450 2C8enzyme
DeferasiroxUDP-glucuronosyltransferase 1A9enzyme
DeferasiroxUDP-glucuronosyltransferase 1A3enzyme
DeferasiroxCytochrome P450 3A4enzyme
DeferasiroxIrontarget
DelavirdineGag-Pol polyproteintarget
DelavirdineCytochrome P450 3A4enzyme
DelavirdineCytochrome P450 2C9enzyme
DelavirdineCytochrome P450 2D6enzyme
DelavirdineCytochrome P450 3A5enzyme
DelavirdineCytochrome P450 3A7enzyme
DelavirdineCytochrome P450 2C19enzyme
DelavirdineReverse transcriptase/RNaseHtarget
DeltamethrinProtein phosphatase 3 catalytic subunit alphatarget
DeltamethrinSerine/threonine-protein phosphatase 2B catalytic subunit beta isoformtarget
DeltamethrinHuman Carboxylesterasesenzyme
DeltamethrinCytochrome P450 2D6enzyme
DeltamethrinAcetylcholinesterasetarget
DeramciclaneCytochrome P450 2D6enzyme
Deramciclane5-hydroxytryptamine receptor 2Ctarget
Deramciclane5-hydroxytryptamine receptor 2Atarget
DesipramineMuscarinic acetylcholine receptor M2target
DesipramineMuscarinic acetylcholine receptor M1target
DesipramineSodium-dependent noradrenaline transportertarget
DesipramineBeta-2 adrenergic receptortarget
DesipramineSodium-dependent serotonin transportertarget
DesipramineSolute carrier family 22 member 3transporter
DesipramineHistamine H1 receptortarget
DesipramineBeta-1 adrenergic receptortarget
DesipramineCytochrome P450 2D6enzyme
DesipramineMuscarinic acetylcholine receptor M3target
DesipramineMuscarinic acetylcholine receptor M4target
DesipramineMuscarinic acetylcholine receptor M5target
DesipramineAlpha-1 adrenergic receptorstarget
DesipramineAlpha-2 adrenergic receptorstarget
DesipramineD(2) dopamine receptortarget
Desipramine5-hydroxytryptamine receptor 2Ctarget
Desipramine5-hydroxytryptamine receptor 1Atarget
DesipramineSphingomyelin phosphodiesterasetarget
DesipramineCytochrome P450 2E1enzyme
DesipramineCytochrome P450 1A2enzyme
DesipramineSolute carrier family 22 member 4transporter
Desipramine5-hydroxytryptamine receptor 2Atarget
DesipramineAlpha-1-acid glycoprotein 1carrier
DesipramineCytochrome P450 2B6enzyme
DesipramineCytochrome P450 3A4enzyme
DesipramineSolute carrier family 22 member 2transporter
DesipramineSolute carrier family 22 member 1transporter
DesipramineATP-dependent translocase ABCB1transporter
DesipramineOrganic cation/carnitine transporter 2transporter
DesmethylprodineCytochrome P450 2D6enzyme
DesogestrelProgesterone receptortarget
DesogestrelEstrogen receptortarget
DesogestrelCytochrome P450 3A4enzyme
DesogestrelAlbumincarrier
DesogestrelSex hormone-binding globulincarrier
DesogestrelCytochrome P450 2C9enzyme
DesogestrelUDP-glucuronosyltransferase 1A1enzyme
DesvenlafaxineUDP-glucuronosyltransferase 1A1enzyme
DesvenlafaxineCytochrome P450 3A4enzyme
DesvenlafaxineUDP-glucuronosyltransferase 1A3enzyme
DesvenlafaxineUDP-glucuronosyltransferase 2B4enzyme
DesvenlafaxineUDP-glucuronosyltransferase 2B15enzyme
DesvenlafaxineUDP-glucuronosyltransferase 2B17enzyme
DesvenlafaxineCytochrome P450 2C19enzyme
DesvenlafaxineSodium-dependent dopamine transportertarget
DesvenlafaxineCytochrome P450 2D6enzyme
DesvenlafaxineSodium-dependent noradrenaline transportertarget
DesvenlafaxineSodium-dependent serotonin transportertarget
DeutivacaftorCystic fibrosis transmembrane conductance regulatortarget
DeutivacaftorCytochrome P450 3A Subfamilyenzyme
DeutivacaftorAlpha-1-acid glycoprotein 1carrier
DeutivacaftorAlbumincarrier
DeutivacaftorBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
DeutivacaftorATP-binding cassette sub-family B member 5transporter
DeutivacaftorCytochrome P450 2C8enzyme
DeutivacaftorCytochrome P450 2C9enzyme
DeutivacaftorCytochrome P450 3A4enzyme
DexamethasoneAnnexin A1target
DexamethasoneOrganic anion transporter 3transporter
Dexamethasone11-beta-hydroxysteroid dehydrogenase 1enzyme
Dexamethasone11-beta-hydroxysteroid dehydrogenase type 2enzyme
DexamethasoneAlbumincarrier
DexamethasoneCytochrome P450 11B1, mitochondrialenzyme
DexamethasoneNuclear receptor subfamily 1 group I member 2target
DexamethasoneCytochrome P450 4A11enzyme
DexamethasoneCytochrome P450 3A43enzyme
DexamethasoneCytochrome P450 2E1enzyme
DexamethasoneCytochrome P450 2C8enzyme
DexamethasoneCytochrome P450 2C19enzyme
DexamethasoneCytochrome P450 2B6enzyme
DexamethasoneCytochrome P450 2A6enzyme
DexamethasoneCytochrome P450 1A1enzyme
DexamethasoneSteroid 17-alpha-hydroxylase/17,20 lyaseenzyme
DexamethasoneBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
DexamethasoneSolute carrier organic anion transporter family member 1A2transporter
DexamethasoneATP-binding cassette sub-family C member 2transporter
DexamethasoneATP-dependent translocase ABCB1transporter
DexamethasoneBile salt export pumptransporter
DexamethasoneCytochrome P450 3A7enzyme
DexamethasoneCytochrome P450 3A5enzyme
DexamethasoneCytochrome P450 3A4enzyme
DexamethasoneNuclear receptor subfamily 0 group B member 1target
DexamethasoneNitric oxide synthase, inducibletarget
DexamethasoneGlucocorticoid receptortarget
Dexamethasone acetateOrganic anion transporter 3transporter
Dexamethasone acetate11-beta-hydroxysteroid dehydrogenase 1enzyme
Dexamethasone acetate11-beta-hydroxysteroid dehydrogenase type 2enzyme
Dexamethasone acetateAlbumincarrier
Dexamethasone acetateCytochrome P450 11B1, mitochondrialenzyme
Dexamethasone acetateNuclear receptor subfamily 1 group I member 2target
Dexamethasone acetateCytochrome P450 4A11enzyme
Dexamethasone acetateCytochrome P450 3A43enzyme
Dexamethasone acetateCytochrome P450 2E1enzyme
Dexamethasone acetateCytochrome P450 2C8enzyme
Dexamethasone acetateGlucocorticoid receptortarget
Dexamethasone acetateAnnexin A1target
Dexamethasone acetateNitric oxide synthase, inducibletarget
Dexamethasone acetateNuclear receptor subfamily 0 group B member 1target
Dexamethasone acetateCytochrome P450 3A4enzyme
Dexamethasone acetateCytochrome P450 3A5enzyme
Dexamethasone acetateCytochrome P450 3A7enzyme
Dexamethasone acetateBile salt export pumptransporter
Dexamethasone acetateATP-dependent translocase ABCB1transporter
Dexamethasone acetateATP-binding cassette sub-family C member 2transporter
Dexamethasone acetateSolute carrier organic anion transporter family member 1A2transporter
Dexamethasone acetateBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
Dexamethasone acetateSteroid 17-alpha-hydroxylase/17,20 lyaseenzyme
Dexamethasone acetateCytochrome P450 1A1enzyme
Dexamethasone acetateCytochrome P450 2A6enzyme
Dexamethasone acetateCytochrome P450 2B6enzyme
Dexamethasone acetateCytochrome P450 2C19enzyme
Dexamethasone isonicotinateCytochrome P450 3A4enzyme
Dexamethasone isonicotinateCytochrome P450 3A5enzyme
DexchlorpheniramineHistamine H1 receptortarget
DexchlorpheniramineCytochrome P450 2D6enzyme
Dexchlorpheniramine maleateCytochrome P450 3A4enzyme
Dexchlorpheniramine maleateSolute carrier family 22 member 2carrier
Dexchlorpheniramine maleateSolute carrier family 22 member 1carrier
Dexchlorpheniramine maleateHistamine H1 receptortarget
Dexchlorpheniramine maleateCytochrome P450 2D6enzyme
DexfenfluramineSodium-dependent serotonin transportertarget
Dexfenfluramine5-hydroxytryptamine receptor 2Ctarget
DexfenfluramineCytochrome P450 2D6enzyme
DexfenfluramineCytochrome P450 1A2enzyme
DexfenfluramineCytochrome P450 2E1enzyme
DexlansoprazolePotassium-transporting ATPase alpha chain 1target
DexlansoprazoleCytochrome P450 2C19enzyme
DexlansoprazoleCytochrome P450 3A4enzyme
DexlansoprazolePotassium-transporting ATPase subunit betatarget
DexlansoprazoleN(G),N(G)-dimethylarginine dimethylaminohydrolase 1target
DexloxiglumideCholecystokinin receptor type Atarget
DexloxiglumideCytochrome P450 3A4enzyme
DexloxiglumideCytochrome P450 2C9enzyme
DexloxiglumideCytochrome P450 3A5enzyme
DexloxiglumideCytochrome P450 2B6enzyme
DexloxiglumideCytochrome P450 2E1enzyme
DexloxiglumideGastrin/cholecystokinin type B receptortarget
DexmedetomidineAlpha-2A adrenergic receptortarget
DexmedetomidineCytochrome P450 2E1enzyme
DexmedetomidineCytochrome P450 1A2enzyme
DexmedetomidineCytochrome P450 1A1enzyme
DexmedetomidineCytochrome P450 2D6enzyme
DexmedetomidineAlpha-2 adrenergic receptorstarget
DextropropoxypheneDelta-type opioid receptortarget
DextropropoxypheneMu-type opioid receptortarget
DextropropoxypheneKappa-type opioid receptortarget
DextropropoxypheneLiver carboxylesterase 1enzyme
DextropropoxypheneNMDA receptortarget
DextropropoxypheneUDP-glucuronosyltransferase 2B4enzyme
DextropropoxypheneCytochrome P450 3A Subfamilyenzyme
DextropropoxypheneCytochrome P450 3A4enzyme
DextropropoxypheneCytochrome P450 2D6enzyme
DiacereinInterleukin-1 betatarget
DiacereinCytochrome P450 2D6target
DiacereinCytochrome P450 2C9target
DiacereinCytochrome P450 2E1target
DiacereinCytochrome P450 3A Subfamilytarget
DiacereinCytochrome P450 1A2target
DiacereinPolyunsaturated fatty acid 5-lipoxygenasetarget
DiacereinArylamine N-acetyltransferasetarget
DiacereinOxysterols receptor LXR-betatarget
DiacereinOxysterols receptor LXR-alphatarget
DiazepamCytochrome P450 2C18enzyme
DiazepamCytochrome P450 2C8enzyme
DiazepamGABA(A) Receptortarget
DiazepamGABA(A) Receptor Benzodiazepine Binding Sitetarget
DiazepamTranslocator proteintarget
DiazepamProstaglandin G/H synthase 1enzyme
DiazepamCytochrome P450 2B6enzyme
DiazepamATP-dependent translocase ABCB1transporter
DiazepamCytochrome P450 3A5enzyme
DiazepamCytochrome P450 2C19enzyme
DiazepamCytochrome P450 2C9enzyme
DiazepamAlbumincarrier
DiazepamCytochrome P450 3A4enzyme
DiazepamCytochrome P450 3A7enzyme
DiazoxideATP-sensitive inward rectifier potassium channel 8target
DiazoxideBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
DiazoxideCytochrome P450 3A4enzyme
DiazoxideCytochrome P450 1A2enzyme
DiazoxideMitochondrial ATP synthase F1 domaintarget
DiazoxideAlbumincarrier
DiazoxideATP-sensitive inward rectifier potassium channel 11target
DiazoxideOrganic anion transporter 3transporter
DiazoxideSolute carrier family 22 member 6transporter
DiclofenacCytochrome P450 3A4enzyme
DiclofenacHuman Cyclooxygenasestarget
DiclofenacATP-dependent translocase ABCB1transporter
DiclofenacPhospholipase A2, membrane associatedenzyme
DiclofenacPotassium voltage-gated channel subfamily KQT member 3transporter
DiclofenacPotassium voltage-gated channel subfamily KQT member 2transporter
DiclofenacProstaglandin G/H synthase 1target
DiclofenacProstaglandin G/H synthase 2target
DiclofenacTransthyretincarrier
DiclofenacCytochrome P450 2C9enzyme
DiclofenacCytochrome P450 2C19enzyme
DiclofenacCytochrome P450 1A2enzyme
DiclofenacCytochrome P450 2C8enzyme
DiclofenacAlbumincarrier
DiclofenacATP-binding cassette sub-family C member 4transporter
DiclofenacMultidrug resistance-associated protein 1transporter
DiclofenacSolute carrier family 22 member 6transporter
DiclofenacOrganic anion transporter 3transporter
DiclofenacSolute carrier organic anion transporter family member 1C1transporter
DiclofenacSolute carrier family 22 member 11transporter
DiclofenacUDP-glucuronosyltransferase 2B7enzyme
DiclofenacAcid-sensing ion channel 1transporter
DiclofenacCytochrome P450 2B6enzyme
DiclofenacCytochrome P450 2C18enzyme
DiclofenacCytochrome P450 2E1enzyme
DiclofenacSolute carrier organic anion transporter family member 1B1transporter
DiclofenacBile salt export pumptransporter
DiclofenacUDP-glucuronosyltransferase 1A3enzyme
DiclofenacUDP-glucuronosyltransferase 1A9enzyme
DiclofenacUDP-glucuronosyltransferase 2B4enzyme
DiclofenacPolyunsaturated fatty acid 5-lipoxygenaseenzyme
DiclofenacSodium channel protein type 4 subunit alphatransporter
DiethylstilbestrolBile salt export pumptransporter
DiethylstilbestrolSolute carrier organic anion transporter family member 2B1transporter
DiethylstilbestrolSolute carrier organic anion transporter family member 1B1transporter
DiethylstilbestrolSex hormone-binding globulintarget
DiethylstilbestrolEstrogen receptortarget
DiethylstilbestrolNuclear receptor subfamily 1 group I member 2target
DiethylstilbestrolNuclear receptor coactivator 2target
DiethylstilbestrolSteroid hormone receptor ERR2target
DiethylstilbestrolSteroid hormone receptor ERR1target
DiethylstilbestrolCytochrome P450 2E1enzyme
DiethylstilbestrolCytochrome P450 2C9enzyme
DiethylstilbestrolCytochrome P450 2C8enzyme
DiethylstilbestrolCytochrome P450 3A4enzyme
DiethylstilbestrolEstrogen receptor betatarget
DiethylstilbestrolATP-dependent translocase ABCB1transporter
DiethylstilbestrolBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
DiethylstilbestrolAromataseenzyme
DiethylstilbestrolCatechol O-methyltransferaseenzyme
DiethylstilbestrolTransthyretincarrier
DiethylstilbestrolEstrogen-related receptor gammatarget
DiethylstilbestrolEstrogen receptortarget
DiethylstilbestrolAndrogen receptortarget
DifloxacinCytochrome P450 1A1enzyme
DifloxacinMultidrug resistance-associated protein 1transporter
DifloxacinNeuronal Acetylcholine (nACh) Receptor Subunitstarget
DifloxacinCytochrome P450 1A2enzyme
DihydralazineDiamine oxidase [copper-containing]target
DihydralazineCytochrome P450 1A2enzyme
DihydralazineMyeloperoxidasetarget
DihydralazineCytochrome P450 3A4enzyme
DihydroergotamineBeta-3 adrenergic receptortarget
DihydroergotamineCytochrome P450 3A4enzyme
Dihydroergotamine5-hydroxytryptamine receptor 1Ftarget
DihydroergotamineD(4) dopamine receptortarget
DihydroergotamineD(3) dopamine receptortarget
DihydroergotamineD(2) dopamine receptortarget
DihydroergotamineAlpha-2 adrenergic receptorstarget
DihydroergotamineAlpha-1 adrenergic receptorstarget
Dihydroergotamine5-hydroxytryptamine receptor 2Ctarget
Dihydroergotamine5-hydroxytryptamine receptor 2Atarget
Dihydroergotamine5-hydroxytryptamine receptor 1Etarget
Dihydroergotamine5-hydroxytryptamine receptor 1Atarget
DihydroergotamineATP-dependent translocase ABCB1transporter
Dihydroergotamine5-hydroxytryptamine receptor 2Btarget
DihydroergotamineAlpha-2A adrenergic receptortarget
Dihydroergotamine5-hydroxytryptamine receptor 4target
Dihydroergotamine5-hydroxytryptamine receptor 1Dtarget
Dihydroergotamine5-hydroxytryptamine receptor 1Btarget
DiltiazemAlpha-1-acid glycoprotein 1carrier
DiltiazemAlbumincarrier
DiltiazemVoltage-dependent L-type calcium channel subunit alpha-1Ctarget
DiltiazemATP-dependent translocase ABCB1transporter
DiltiazemCytochrome P450 3A7enzyme
DiltiazemCytochrome P450 3A5enzyme
DiltiazemCytochrome P450 2D6enzyme
DiltiazemCytochrome P450 2C19enzyme
DiltiazemCytochrome P450 3A4enzyme
DiltiazemVoltage-dependent calcium channel gamma-1 subunittarget
DiltiazemVoltage-dependent calcium channel subunit alpha-2/delta-1target
DiltiazemVoltage gated L-type calcium channeltarget
DiltiazemCytochrome P450 2C8enzyme
Dimethyl sulfoxideTransthyretincarrier
Dimethyl sulfoxideCytochrome P450 2C19enzyme
Dimethyl sulfoxideCytochrome P450 2D6enzyme
Dimethyl sulfoxideCytochrome P450 3A4enzyme
Dimethyl sulfoxideInterleukin-5 receptor subunit alphatarget
Dimethyl sulfoxideMucin-16target
Dimethyl sulfoxideMyc proto-oncogene proteintarget
DiosminAryl hydrocarbon receptortarget
DiosminATP-dependent translocase ABCB1transporter
DiosminSolute carrier organic anion transporter family member 1B1transporter
DiosminSolute carrier organic anion transporter family member 1B3transporter
DiosminSolute carrier organic anion transporter family member 2B1transporter
DiosminCytochrome P450 1A1enzyme
DiosminCytochrome P450 2C9enzyme
DiosminCytochrome P450 2E1enzyme
DiosminCytochrome P450 3A4enzyme
DiosminAlbumincarrier
DiphenhydramineHistamine H1 receptortarget
DiphenhydramineHistamine N-methyltransferasetarget
DiphenhydramineMuscarinic acetylcholine receptor M2target
DiphenhydramineProstaglandin G/H synthase 1enzyme
DiphenhydramineOrganic cation/carnitine transporter 2transporter
DiphenhydramineSolute carrier family 22 member 2transporter
DiphenhydramineCytochrome P450 2C19enzyme
DiphenhydramineCytochrome P450 2C9enzyme
DiphenhydramineCytochrome P450 2D6enzyme
Dirithromycin23S ribosomal RNAtarget
DirithromycinCytochrome P450 3A4enzyme
DisulfiramAldehyde dehydrogenase family 3 member A2target
DisulfiramBile salt export pumptransporter
DisulfiramCytochrome P450 3A5enzyme
DisulfiramCytochrome P450 3A4enzyme
DisulfiramDopamine beta-hydroxylasetarget
DisulfiramCytochrome P450 2E1enzyme
DisulfiramAldehyde dehydrogenase, mitochondrialtarget
DitiocarbCytochrome P450 2E1enzyme
DitiocarbCytochrome P450 3A4enzyme
DitiocarbCytochrome P450 3A5enzyme
DitiocarbDopamine beta-hydroxylasetarget
DitiocarbSuperoxide dismutase [Cu-Zn]target
DitiocarbTyrosinasetarget
DitiocarbCytochrome P450 2A6enzyme
DitiocarbCatalasetarget
Ditiocarb zincMetal regulatory transcription factor 1target
Ditiocarb zincCytochrome P450 2E1target
Ditiocarb zincCytochrome P450 2A6target
Ditiocarb zincSuperoxide dismutase [Cu-Zn]target
Ditiocarb zincDopamine beta-hydroxylasetarget
DocetaxelApoptosis regulator Bcl-2target
DocetaxelTubulin beta-1 chaintarget
DocetaxelCytochrome P450 3A4enzyme
DocetaxelCytochrome P450 3A5enzyme
DocetaxelCytochrome P450 3A7enzyme
DocetaxelATP-dependent translocase ABCB1transporter
DocetaxelATP-binding cassette sub-family C member 10transporter
DocetaxelCytochrome P450 1B1enzyme
DocetaxelSolute carrier organic anion transporter family member 1B3transporter
DocetaxelSolute carrier family 22 member 7transporter
DocetaxelBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
DocetaxelMultidrug resistance-associated protein 1transporter
DocetaxelATP-binding cassette sub-family C member 2transporter
DocetaxelNuclear receptor subfamily 1 group I member 2target
DoconexentRetinoic acid receptor RXR-gammatarget
DoconexentProstaglandin G/H synthase 1target
DoconexentProstaglandin G/H synthase 2target
DoconexentMyc proto-oncogene proteintarget
DoconexentRetinoic acid receptor RXR-betatarget
DoconexentRetinoic acid receptor RXR-alphatarget
DoconexentCytochrome P450 2C9enzyme
DoconexentPeroxisome proliferator-activated receptor alphatarget
DoconexentPeroxisome proliferator-activated receptor gammatarget
DoconexentSterol regulatory element-binding protein 1target
DoramectinCytochrome P450 3A4enzyme
DoramectinSolute carrier organic anion transporter family member 1B1transporter
DoramectinAnoctamin-1target
DoramectinATP-dependent translocase ABCB1transporter
DordaviproneSolute carrier organic anion transporter family member 1B3transporter
DordaviproneSolute carrier family 22 member 1transporter
DordaviproneSolute carrier organic anion transporter family member 1B1transporter
DordaviproneOrganic anion transporter 3transporter
DordaviproneSolute carrier family 22 member 6transporter
DordaviproneMultidrug and toxin extrusion protein 2transporter
DordaviproneMultidrug and toxin extrusion protein 1transporter
DordaviproneCytochrome P450 2C19enzyme
DordaviproneCytochrome P450 1A2enzyme
DordaviproneATP-dependent Clp protease proteolytic subunit, mitochondrialtarget
DordaviproneCytochrome P450 3A5enzyme
DordaviproneCytochrome P450 2D6enzyme
DordaviproneCytochrome P450 2C9enzyme
DordaviproneCytochrome P450 2C8enzyme
DordaviproneCytochrome P450 2B6enzyme
DordaviproneCytochrome P450 3A4enzyme
DordaviproneD(2) dopamine receptortarget
DordaviproneD(3) dopamine receptortarget
DosulepinMuscarinic acetylcholine receptor M2target
DosulepinCytochrome P450 2C19enzyme
DosulepinCytochrome P450 2C9enzyme
DosulepinCytochrome P450 3A4enzyme
DosulepinCytochrome P450 1A2enzyme
DosulepinAlpha-2 adrenergic receptorstarget
DosulepinAlpha-1 adrenergic receptorstarget
DosulepinSodium-dependent serotonin transportertarget
DosulepinSodium-dependent noradrenaline transportertarget
DosulepinMuscarinic acetylcholine receptor M5target
DosulepinMuscarinic acetylcholine receptor M4target
DosulepinMuscarinic acetylcholine receptor M3target
DosulepinMuscarinic acetylcholine receptor M1target
DosulepinHistamine H1 receptortarget
DosulepinCytochrome P450 2D6enzyme
Dosulepin5-hydroxytryptamine receptor 2Atarget
Dosulepin5-hydroxytryptamine receptor 1Atarget
DovitinibCytochrome P450 2C19enzyme
DovitinibCytochrome P450 1A1enzyme
DovitinibCytochrome P450 1A2enzyme
DovitinibATP-binding cassette sub-family C member 3transporter
DovitinibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
DovitinibUDP-glucuronosyltransferase 1A3enzyme
DovitinibUDP-glucuronosyltransferase 2B7enzyme
DovitinibNuclear receptor subfamily 1 group I member 2target
DovitinibSolute carrier organic anion transporter family member 1B1transporter
DovitinibSolute carrier organic anion transporter family member 2B1transporter
DovitinibVascular endothelial growth factor receptortarget
DovitinibMast/stem cell growth factor receptor Kittarget
DovitinibReceptor-type tyrosine-protein kinase FLT3target
DovitinibFibroblast growth factor receptor 3target
DovitinibATP-dependent translocase ABCB1transporter
DovitinibSolute carrier organic anion transporter family member 1B3transporter
DovitinibCytochrome P450 3A4enzyme
DoxepinCytochrome P450 1A2enzyme
DoxepinCytochrome P450 2C9enzyme
DoxepinCytochrome P450 2C19enzyme
Doxepin5-hydroxytryptamine receptor 2Atarget
Doxepin5-hydroxytryptamine receptor 1Atarget
DoxepinAlpha-1A adrenergic receptortarget
DoxepinMuscarinic acetylcholine receptor M5target
DoxepinATP-dependent translocase ABCB1transporter
DoxepinMuscarinic acetylcholine receptor M3target
DoxepinMuscarinic acetylcholine receptor M2target
DoxepinMuscarinic acetylcholine receptor M1target
DoxepinCytochrome P450 2D6enzyme
DoxepinHistamine H2 receptortarget
DoxepinHistamine H1 receptortarget
DoxepinSodium-dependent noradrenaline transportertarget
DoxepinSodium-dependent serotonin transportertarget
Doxepin5-hydroxytryptamine receptor 2Btarget
Doxepin5-hydroxytryptamine receptor 2Ctarget
DoxepinAlpha-1B adrenergic receptortarget
DoxepinAlpha-1D adrenergic receptortarget
DoxepinCytochrome P450 3A4enzyme
Doxepin5-hydroxytryptamine receptor 6target
DoxepinHistamine H4 receptortarget
DoxepinVoltage-gated inwardly rectifying potassium channel KCNH2target
DoxepinAlbumincarrier
DoxepinAlpha-1-acid glycoprotein 1carrier
DoxepinMuscarinic acetylcholine receptor M4target
DoxorubicinATP-binding cassette sub-family C member 6transporter
DoxorubicinATP-binding cassette sub-family C member 3transporter
DoxorubicinATP-dependent translocase ABCB1transporter
DoxorubicinCytochrome P450 2B6enzyme
DoxorubicinCytochrome P450 2D6enzyme
DoxorubicinCytochrome P450 3A4enzyme
DoxorubicinDNAtarget
DoxorubicinDNA topoisomerase 2-alphatarget
DoxorubicinNADH dehydrogenase [ubiquinone] iron-sulfur protein 2, mitochondrialenzyme
DoxorubicinNADH dehydrogenase [ubiquinone] iron-sulfur protein 3, mitochondrialenzyme
DoxorubicinNADH dehydrogenase [ubiquinone] iron-sulfur protein 7, mitochondrialenzyme
DoxorubicinNADPH--cytochrome P450 reductaseenzyme
DoxorubicinRalA-binding protein 1transporter
DoxorubicinATP-binding cassette sub-family C member 2transporter
DoxorubicinAlbumincarrier
DoxorubicinMultidrug resistance-associated protein 1transporter
DoxorubicinDNA topoisomerase 1target
DoxorubicinDNA topoisomerase 2-betatarget
DoxorubicinAldo-keto reductase family 1 member B1enzyme
DoxorubicinAldo-keto reductase family 1 member B10enzyme
DoxorubicinAldo-keto reductase family 1 member C4enzyme
DoxorubicinTelomerase reverse transcriptasetarget
DoxorubicinNitric oxide synthase 1enzyme
DoxorubicinNitric oxide synthase, inducibleenzyme
DoxorubicinNitric oxide synthase 3enzyme
DoxorubicinXanthine dehydrogenase/oxidaseenzyme
DoxorubicinNAD(P)H dehydrogenase [quinone] 1enzyme
DoxorubicinAldo-keto reductase family 1 member C3enzyme
DoxorubicinAldo-keto reductase family 1 member A1enzyme
DoxorubicinCarbonyl reductase [NADPH] 3enzyme
DoxorubicinCarbonyl reductase [NADPH] 1enzyme
DoxorubicinCytochrome P450 1B1enzyme
DoxorubicinMitochondrial potassium channel ATP-binding subunittransporter
DoxorubicinSolute carrier family 22 member 16transporter
DoxorubicinBile salt export pumptransporter
DoxorubicinBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
DoxorubicinATP-binding cassette sub-family C member 10transporter
DoxorubicinNucleolar and coiled-body phosphoprotein 1target
DoxycyclineNeutrophil collagenasetarget
DoxycyclineAlbumincarrier
DoxycyclineATP-binding cassette sub-family B member 5transporter
DoxycyclineCytochrome P450 3A4enzyme
DoxycyclineSolute carrier family 22 member 6transporter
DoxycyclineInterstitial collagenasetarget
DoxycyclineCollagenase 3target
DoxycyclineMatrilysintarget
Doxycycline30S ribosomal proteintarget
DronabinolCytochrome P450 2D6enzyme
DronabinolCytochrome P450 2B6enzyme
DronabinolCytochrome P450 2A6enzyme
DronabinolCytochrome P450 1B1enzyme
DronabinolCytochrome P450 1A2enzyme
DronabinolCytochrome P450 1A1enzyme
DronabinolCytochrome P450 2C19enzyme
DronabinolProstaglandin G/H synthase 1enzyme
DronabinolBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
DronabinolATP-dependent translocase ABCB1transporter
DronabinolCannabinoid receptor 2target
DronabinolCytochrome P450 2C9enzyme
DronabinolCytochrome P450 3A4enzyme
DronabinolCannabinoid receptor 1target
DronabinolUDP-glucuronosyltransferase 1A10enzyme
DronabinolUDP-glucuronosyltransferase 1A9enzyme
DronabinolUDP-glucuronosyltransferase 1A3enzyme
DronabinolUDP-glucuronosyltransferase 1A1enzyme
DronabinolLiver carboxylesterase 1enzyme
DronabinolMultidrug resistance-associated protein 1transporter
DronabinolCytochrome P450 3A7enzyme
DronabinolCytochrome P450 3A5enzyme
DronabinolCytochrome P450 2J2enzyme
DronedaroneVoltage-dependent L-type calcium channel subunit alpha-1Ctarget
DronedaroneVoltage-gated inwardly rectifying potassium channel KCNH2target
DronedaroneAlpha-2C adrenergic receptortarget
DronedaroneAlpha-2B adrenergic receptortarget
DronedaroneAlpha-2A adrenergic receptortarget
DronedaroneAlpha-1D adrenergic receptortarget
DronedaroneAlpha-1B adrenergic receptortarget
DronedaroneBeta-1 adrenergic receptortarget
DronedaroneAlpha-1A adrenergic receptortarget
DronedaronePotassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 4target
DronedaroneCytochrome P450 2J2enzyme
DronedaroneVoltage-dependent L-type calcium channel subunit alpha-1Ftarget
DronedaroneVoltage-dependent L-type calcium channel subunit alpha-1Starget
DronedaroneVoltage-dependent L-type calcium channel subunit beta-1target
DronedaroneVoltage-dependent L-type calcium channel subunit beta-2target
DronedaroneVoltage-dependent L-type calcium channel subunit beta-3target
DronedaroneVoltage-dependent L-type calcium channel subunit beta-4target
DronedaroneCytochrome P450 2D6enzyme
DronedaroneCytochrome P450 3A4enzyme
DronedaroneATP-dependent translocase ABCB1transporter
DronedaronePotassium channel subfamily K member 2target
DronedaroneAlbumincarrier
DronedaroneSolute carrier family 22 member 2transporter
DronedaroneSolute carrier family 22 member 1transporter
DronedaroneSolute carrier organic anion transporter family member 1B1transporter
DronedaroneSolute carrier organic anion transporter family member 1B3transporter
DronedaroneOrganic anion transporter 3transporter
DronedaroneCytochrome P450 3A5enzyme
DronedaroneVoltage-dependent L-type calcium channel subunit alpha-1Dtarget
DronedaroneThyroid hormone receptor alphatarget
DronedaroneSodium channel protein type 5 subunit alphatarget
DronedaroneG protein-activated inward rectifier potassium channel 1target
DronedaronePotassium voltage-gated channel subfamily KQT member 1target
DronedaroneInward rectifier potassium channeltarget
DronedaroneSodium/calcium exchanger 1target
DronedaroneA-type voltage-gated potassium channel KCND3target
DronedaronePotassium voltage-gated channel subfamily A member 5target
DronedaroneVoltage gated L-type calcium channeltarget
DronedaroneVoltage-gated sodium channel alpha subunittarget
DronedaroneInward rectifier potassium channel 2target
DuloxetineCytochrome P450 3A4enzyme
DuloxetineCytochrome P450 2C19enzyme
DuloxetineCytochrome P450 2B6enzyme
DuloxetineSodium-dependent serotonin transportertarget
DuloxetineSodium-dependent dopamine transportertarget
DuloxetineSodium-dependent noradrenaline transportertarget
DuloxetineCytochrome P450 1A2enzyme
DuloxetineCytochrome P450 2D6enzyme
DuloxetineCytochrome P450 2C9enzyme
DuloxetineAlbumincarrier
Duloxetinealpha1-acid glycoproteincarrier
DuloxetineATP-dependent translocase ABCB1transporter
EconazoleAromataseenzyme
EconazoleCytochrome P450 2E1enzyme
EconazoleCytochrome P450 3A4enzyme
EconazoleLanosterol 14-alpha demethylasetarget
EconazoleNuclear receptor subfamily 1 group I member 2target
Edetate calcium disodium anhydrousAromataseenzyme
Edetate calcium disodium anhydrousSerum paraoxonase/arylesterase 1enzyme
Edetate calcium disodium anhydrousCytochrome P450 3A4enzyme
Edetate calcium disodium anhydrousManganese cationtarget
Edetate calcium disodium anhydrousIrontarget
Edetate calcium disodium anhydrousLeadtarget
Edetate calcium disodium anhydrousAdenosine deaminaseenzyme
Edetate calcium disodium anhydrousSerum paraoxonase/lactonase 3enzyme
Edetate disodium anhydrousCytochrome P450 3A4enzyme
Edetate disodium anhydrousAromataseenzyme
Edetate disodium anhydrousSerum paraoxonase/lactonase 3enzyme
Edetate disodium anhydrousAdenosine deaminaseenzyme
Edetate disodium anhydrousManganese cationtarget
Edetate disodium anhydrousIrontarget
Edetate disodium anhydrousLeadtarget
Edetate disodium anhydrousSerum paraoxonase/arylesterase 1enzyme
EfavirenzCytochrome P450 3A4enzyme
EfavirenzGag-Pol polyproteintarget
EfavirenzSolute carrier family 22 member 1transporter
EfavirenzBile salt export pumptransporter
EfavirenzUDP-glucuronosyltransferase 1A1enzyme
EfavirenzCytochrome P450 3A7enzyme
EfavirenzCytochrome P450 3A5enzyme
EfavirenzAlbumincarrier
EfavirenzCytochrome P450 2C8enzyme
EfavirenzReverse transcriptase/RNaseHtarget
EfavirenzCytochrome P450 2D6enzyme
EfavirenzCytochrome P450 2B6enzyme
EfavirenzCytochrome P450 1A2enzyme
EfavirenzCytochrome P450 2C19enzyme
EfavirenzCytochrome P450 2C9enzyme
EfonidipineVoltage-dependent calcium channeltarget
EfonidipineVoltage-dependent T-type calcium channel subunit alpha-1Itarget
EfonidipineVoltage-dependent L-type calcium channel subunit alpha-1Ctarget
EfonidipineVoltage-dependent T-type calcium channel subunit alpha-1Htarget
EfonidipineVoltage-dependent T-type calcium channel subunit alpha-1Gtarget
EfonidipineVoltage-dependent T-type calcium channeltarget
EfonidipineVoltage gated L-type calcium channeltarget
EfonidipineCytochrome P450 3A4enzyme
ElagolixATP-dependent translocase ABCB1transporter
ElagolixCytochrome P450 2C8enzyme
ElagolixCytochrome P450 2D6enzyme
ElagolixCytochrome P450 3A Subfamilyenzyme
ElagolixGonadotropin-releasing hormone receptortarget
ElagolixSolute carrier organic anion transporter family member 1B1transporter
ElagolixUDP-glucuronosyltransferases (UGTs)enzyme
ElbasvirNonstructural protein 5Atarget
ElbasvirCytochrome P450 3A43enzyme
ElbasvirCytochrome P450 3A7enzyme
ElbasvirCytochrome P450 3A5enzyme
ElbasvirCytochrome P450 3A4enzyme
ElbasvirATP-dependent translocase ABCB1transporter
ElexacaftorSolute carrier organic anion transporter family member 1B1transporter
ElexacaftorCytochrome P450 2C8enzyme
ElexacaftorCytochrome P450 2C9enzyme
ElexacaftorCytochrome P450 2C19enzyme
ElexacaftorCytochrome P450 2D6enzyme
ElexacaftorCystic fibrosis transmembrane conductance regulatortarget
ElexacaftorCytochrome P450 2B6enzyme
ElexacaftorCytochrome P450 1A2enzyme
ElexacaftorCytochrome P450 3A5enzyme
ElexacaftorCytochrome P450 3A4enzyme
ElexacaftorAlbumincarrier
ElexacaftorATP-dependent translocase ABCB1transporter
ElexacaftorSolute carrier organic anion transporter family member 1B3transporter
EliglustatCeramide glucosyltransferasetarget
EliglustatCytochrome P450 2D6enzyme
EliglustatCytochrome P450 3A4enzyme
EliglustatATP-dependent translocase ABCB1transporter
ElinzanetantATP-dependent translocase ABCB1transporter
ElinzanetantCytochrome P450 3A4enzyme
ElinzanetantSubstance-P receptortarget
ElinzanetantNeuromedin-K receptortarget
Ellagic acidCarbonic anhydrase 4target
Ellagic acidCarbonic anhydrase 3target
Ellagic acidCarbonic anhydrase 2target
Ellagic acidCarbonic anhydrase 1target
Ellagic acidCytochrome P450 2E1enzyme
Ellagic acidCytochrome P450 1A1enzyme
Ellagic acidSolute carrier family 22 member 11transporter
Ellagic acidHeat shock 70 kDa protein 1Btarget
Ellagic acidGlycogen synthase kinase-3 betatarget
Ellagic acidHeat shock 70 kDa protein 1Atarget
Ellagic acidSqualene monooxygenasetarget
Ellagic acidTyrosine-protein kinase SYKtarget
Ellagic acidProtein kinase C beta typetarget
Ellagic acidSolute carrier family 22 member 6transporter
Ellagic acidProtein kinase C alpha typetarget
Ellagic acidcAMP-dependent protein kinase catalytic subunit alphatarget
Ellagic acidCasein kinase II subunit alphatarget
Ellagic acidCarbonic anhydrase 14target
Ellagic acidCarbonic anhydrase 12target
Ellagic acidCarbonic anhydrase 5A, mitochondrialtarget
Ellagic acidCarbonic anhydrase 9target
Ellagic acidCarbonic anhydrase 7target
Ellagic acidCarbonic anhydrase 6target
Ellagic acidCarbonic anhydrase 5B, mitochondrialtarget
EltrombopagUDP-glucuronosyltransferase 1A9enzyme
EltrombopagBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
EltrombopagUDP-glucuronosyltransferase 1A3enzyme
EltrombopagUDP-glucuronosyltransferase 1A1enzyme
EltrombopagCytochrome P450 1A2enzyme
EltrombopagCytochrome P450 2C8enzyme
EltrombopagThrombopoietin receptortarget
EltrombopagSolute carrier organic anion transporter family member 1B1transporter
ElvitegravirGag-Pol polyproteintarget
ElvitegravirCytochrome P450 3A4enzyme
ElvitegravirGag-Pol polyproteintarget
ElvitegravirUDP-glucuronosyltransferase 1A1enzyme
EnasidenibIsocitrate dehydrogenase [NAD] subunit alpha, mitochondrialtarget
EnasidenibIsocitrate dehydrogenase [NADP] cytoplasmictarget
EnasidenibAlbumincarrier
EnasidenibOrganic anion transporter 3transporter
EnasidenibSolute carrier organic anion transporter family member 1B3transporter
EnasidenibSolute carrier family 22 member 2transporter
EnasidenibSolute carrier organic anion transporter family member 1B1transporter
EnasidenibSolute carrier family 22 member 6transporter
EnasidenibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
EnasidenibATP-dependent translocase ABCB1transporter
EnasidenibUDP-glucuronosyltransferase 2B15enzyme
EnasidenibUDP-glucuronosyltransferase 2B7enzyme
EnasidenibUDP-glucuronosyltransferase 1A9enzyme
EnasidenibUDP-glucuronosyltransferase 1A4enzyme
EnasidenibUDP-glucuronosyltransferase 1A3enzyme
EnasidenibUDP-glucuronosyltransferase 1A1enzyme
EnasidenibCytochrome P450 3A4enzyme
EnasidenibCytochrome P450 2D6enzyme
EnasidenibCytochrome P450 2C19enzyme
EnasidenibCytochrome P450 2C9enzyme
EnasidenibIsocitrate dehydrogenase [NAD] subunit beta, mitochondrialtarget
EnasidenibIsocitrate dehydrogenase [NAD] subunit gamma, mitochondrialtarget
EnasidenibCytochrome P450 1A2enzyme
EnasidenibCytochrome P450 2C8enzyme
EnasidenibCytochrome P450 2B6enzyme
EnasidenibIsocitrate dehydrogenase [NADP], mitochondrialtarget
EncorafenibSolute carrier family 22 member 2transporter
EncorafenibCytochrome P450 2B6enzyme
EncorafenibSerine/threonine-protein kinase 36target
EncorafenibDual specificity mitogen-activated protein kinase kinase 4target
EncorafenibLIM domain kinase 2target
EncorafenibLIM domain kinase 1target
EncorafenibMitogen-activated protein kinase 10target
EncorafenibMitogen-activated protein kinase 9target
EncorafenibMitogen-activated protein kinase 8target
EncorafenibRAF proto-oncogene serine/threonine-protein kinasetarget
EncorafenibSolute carrier organic anion transporter family member 1B3transporter
EncorafenibSolute carrier organic anion transporter family member 1B1transporter
EncorafenibOrganic anion transporter 3transporter
EncorafenibSolute carrier family 22 member 6transporter
EncorafenibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
EncorafenibATP-dependent translocase ABCB1transporter
EncorafenibCytochrome P450 3A7enzyme
EncorafenibCytochrome P450 3A5enzyme
EncorafenibCytochrome P450 2C9enzyme
EncorafenibCytochrome P450 2C8enzyme
EncorafenibCytochrome P450 2C19enzyme
EncorafenibCytochrome P450 1A2enzyme
EncorafenibAlbumincarrier
EncorafenibUDP-glucuronosyltransferase 1A1enzyme
EncorafenibG1/S-specific cyclin-D1target
EncorafenibSerine/threonine-protein kinase B-raftarget
EncorafenibCytochrome P450 2D6enzyme
EncorafenibCytochrome P450 3A4enzyme
EnmetazobactamBeta-lactamase TEMtarget
EnmetazobactamBeta-lactamasetarget
EnmetazobactamExtended-spectrum beta-lactamase PER-1target
EnmetazobactamCytochrome P450 2E1enzyme
EnoxacinDNA topoisomerase 2-betatarget
EnoxacinCytochrome P450 1A2enzyme
EnoxacinDNA topoisomerase 2-alphatarget
EnoxacinDNA topoisomerase 4 subunit Atarget
EnoxacinDNA gyrase subunit Atarget
EnrofloxacinDNA gyrase subunit Atarget
EnrofloxacinCytochrome P450 1A2enzyme
EnrofloxacinBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
EnrofloxacinATP-dependent translocase ABCB1transporter
EnrofloxacinDNA topoisomerase 2target
EnsitrelvirATP-dependent translocase ABCB1transporter
EnsitrelvirCytochrome P450 3A4enzyme
EnsitrelvirReplicase polyprotein 1abtarget
EntacaponeCatechol O-methyltransferaseenzyme
EntacaponeCytochrome P450 2D6enzyme
EntacaponeCatechol O-methyltransferasetarget
EntacaponeUDP-glucuronosyltransferase 1A9enzyme
EnzalutamideAndrogen receptortarget
EnzalutamideCytochrome P450 2B6enzyme
EnzalutamideATP-dependent translocase ABCB1transporter
EnzalutamideCytochrome P450 3A5enzyme
EnzalutamideCytochrome P450 2C19enzyme
EnzalutamideCytochrome P450 2C9enzyme
EnzalutamideCytochrome P450 3A4enzyme
EnzalutamideCytochrome P450 2C8enzyme
EnzalutamideAlbumincarrier
EpinastineHistamine H1 receptortarget
EpinastineHistamine H2 receptortarget
EpinastineAlpha-1A adrenergic receptortarget
EpinastineAlpha-2A adrenergic receptortarget
Epinastine5-hydroxytryptamine receptor 2Atarget
Epinastine5-hydroxytryptamine receptor 7target
EpinastineATP-dependent translocase ABCB1transporter
EpinastineCytochrome P450 2B6enzyme
EpinastineCytochrome P450 2D6enzyme
EpinastineCytochrome P450 3A4enzyme
EpinephrineAlpha-2A adrenergic receptortarget
EpinephrineAlpha-2B adrenergic receptortarget
EpinephrineTumor necrosis factortarget
EpinephrineCatechol O-methyltransferaseenzyme
EpinephrineMonoamine oxidaseenzyme
EpinephrineAlpha-1D adrenergic receptortarget
EpinephrineAlpha-1B adrenergic receptortarget
EpinephrineSolute carrier family 22 member 2transporter
EpinephrineCytochrome P450 2C9enzyme
EpinephrineSolute carrier family 22 member 1transporter
EpinephrineAlpha-1A adrenergic receptortarget
EpinephrineBeta-1 adrenergic receptortarget
EpinephrineBeta-2 adrenergic receptortarget
EpinephrineCytochrome P450 3A4enzyme
EpofolateCytochrome P450 3A4enzyme
EpofolateFolate receptor alphatarget
Epothilone DTubulin beta chaintarget
Epothilone DTubulin beta-1 chaintarget
Epothilone DTubulin beta-4B chaintarget
Epothilone DTubulin beta-4A chaintarget
Epothilone DTubulin alpha-4A chaintarget
Epothilone DTubulin beta-3 chaintarget
Epothilone DTubulin alpha-1C chaintarget
Epothilone DTubulin alpha-8 chaintarget
Epothilone DTubulin alpha-1B chaintarget
Epothilone DTubulin alpha-1A chaintarget
Epothilone DCytochrome P450 3A4enzyme
Epothilone DTubulin alpha 3C/D chaintarget
EprinomectinCytochrome P450 3A4enzyme
EprinomectinBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
EprinomectinATP-dependent translocase ABCB1transporter
ErdafitinibProto-oncogene tyrosine-protein kinase receptor Rettarget
ErdafitinibMacrophage colony-stimulating factor 1 receptortarget
ErdafitinibPlatelet-derived growth factor receptor alphatarget
ErdafitinibPlatelet-derived growth factor receptor betatarget
ErdafitinibMast/stem cell growth factor receptor Kittarget
ErdafitinibVascular endothelial growth factor receptor 2target
Erdafitinibalpha1-acid glycoproteincarrier
ErdafitinibFibroblast growth factor receptortarget
ErdafitinibSolute carrier family 22 member 2transporter
ErdafitinibATP-dependent translocase ABCB1transporter
ErdafitinibCytochrome P450 2C9enzyme
ErdafitinibFibroblast growth factor receptor 4target
ErdafitinibFibroblast growth factor receptor 3target
ErdafitinibFibroblast growth factor receptor 2target
ErdafitinibFibroblast growth factor receptor 1target
ErdafitinibCytochrome P450 3A4enzyme
ErgometrineD(2) dopamine receptortarget
ErgometrineAlpha-1A adrenergic receptortarget
ErgometrineATP-dependent translocase ABCB1transporter
ErgometrineCytochrome P450 3A4enzyme
Ergotamine5-hydroxytryptamine receptor 1Ftarget
Ergotamine5-hydroxytryptamine receptor 1Dtarget
ErgotamineAlpha-1A adrenergic receptortarget
ErgotamineAlpha adrenergic receptortarget
ErgotamineAlpha-2C adrenergic receptortarget
Ergotamine5-hydroxytryptamine receptor 2Btarget
Ergotamine5-hydroxytryptamine receptor 2Ctarget
Ergotamine5-hydroxytryptamine receptor 1Btarget
Ergotamine5-hydroxytryptamine receptor 1Atarget
ErgotamineD(1) dopamine receptortarget
ErgotamineATP-dependent translocase ABCB1transporter
ErgotamineAlpha-1D adrenergic receptortarget
ErgotamineAlpha-1B adrenergic receptortarget
ErgotamineCytochrome P450 3A4enzyme
ErgotamineD(2) dopamine receptortarget
ErgotamineAlpha-2A adrenergic receptortarget
Ergotamine5-hydroxytryptamine receptor 2Atarget
ErlotinibEpidermal growth factor receptortarget
ErlotinibCytochrome P450 3A4enzyme
ErlotinibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
ErlotinibATP-dependent translocase ABCB1transporter
ErlotinibNuclear receptor subfamily 1 group I member 2target
ErlotinibEpidermal growth factor receptorenzyme
ErlotinibSolute carrier organic anion transporter family member 2B1transporter
ErlotinibAlpha-1-acid glycoprotein 1carrier
ErlotinibAlbumincarrier
ErlotinibUDP-glucuronosyltransferase 1A1enzyme
ErlotinibCytochrome P450 2C8enzyme
ErlotinibCytochrome P450 2D6enzyme
ErlotinibCytochrome P450 1B1enzyme
ErlotinibCytochrome P450 1A2enzyme
ErlotinibCytochrome P450 1A1enzyme
ErlotinibCytochrome P450 3A5enzyme
ErythromycinCytochrome P450 3A7enzyme
ErythromycinSolute carrier organic anion transporter family member 1A2transporter
ErythromycinATP-binding cassette sub-family C member 2transporter
ErythromycinBile salt export pumptransporter
ErythromycinSolute carrier organic anion transporter family member 1B3transporter
ErythromycinCytochrome P450 3A5enzyme
ErythromycinVoltage-gated inwardly rectifying potassium channel KCNH2target
ErythromycinMotilin receptortarget
ErythromycinSolute carrier organic anion transporter family member 1B1transporter
ErythromycinATP-dependent translocase ABCB1transporter
ErythromycinCytochrome P450 3A4enzyme
Erythromycin23S ribosomal RNAtarget
EscitalopramD(2) dopamine receptortarget
EscitalopramAlpha-2 adrenergic receptorstarget
EscitalopramAlpha-1 adrenergic receptorstarget
Escitalopram5-hydroxytryptamine receptor 2Ctarget
Escitalopram5-hydroxytryptamine receptor 2Atarget
Escitalopram5-hydroxytryptamine receptor 1Atarget
EscitalopramATP-dependent translocase ABCB1transporter
EscitalopramCytochrome P450 2C19enzyme
EscitalopramHistamine H1 receptortarget
EscitalopramMuscarinic acetylcholine receptor M1target
EscitalopramSodium-dependent noradrenaline transportertarget
EscitalopramSodium-dependent dopamine transportertarget
EscitalopramCytochrome P450 2D6enzyme
EscitalopramCytochrome P450 3A4enzyme
EscitalopramSodium-dependent serotonin transportertarget
EscitalopramAmine oxidase [flavin-containing] Aenzyme
EscitalopramAmine oxidase [flavin-containing] Benzyme
EscitalopramAldehyde oxidaseenzyme
EslicarbazepineCytochrome P450 2C19enzyme
EslicarbazepineP2X purinoceptor 4target
EslicarbazepineCytochrome P450 3A4enzyme
EslicarbazepineSodium channel protein type 11 subunit alphatarget
EslicarbazepineVoltage-gated sodium channel alpha subunittarget
EslicarbazepineUDP-glucuronosyltransferase 1A1enzyme
Eslicarbazepine acetateCytochrome P450 3A4enzyme
Eslicarbazepine acetateCytochrome P450 2C19enzyme
Eslicarbazepine acetateP2X purinoceptor 4target
Eslicarbazepine acetateVoltage-gated sodium channel alpha subunittarget
Eslicarbazepine acetateVoltage-dependent T-type calcium channeltarget
Eslicarbazepine acetateUDP-glucuronosyltransferase 1A1enzyme
EsomeprazolePotassium-transporting ATPase subunit betatarget
EsomeprazoleOrganic anion transporter 3transporter
EsomeprazoleATP-dependent translocase ABCB1transporter
EsomeprazoleN(G),N(G)-dimethylarginine dimethylaminohydrolase 1target
EsomeprazoleCytochrome P450 3A4enzyme
EsomeprazoleCytochrome P450 2C19enzyme
EsomeprazolePotassium-transporting ATPase alpha chain 1target
EstradiolEstrogen receptortarget
EstradiolNuclear receptor subfamily 1 group I member 2target
EstradiolSex hormone-binding globulincarrier
EstradiolEstrogen receptor betatarget
EstradiolCytochrome P450 1A2enzyme
EstradiolUDP-glucuronosyltransferase 1A1enzyme
EstradiolAlbumincarrier
EstradiolFatty acid-binding protein, intestinalcarrier
EstradiolCytochrome P450 3A4enzyme
EstradiolCytochrome P450 3A5enzyme
EstradiolCytochrome P450 3A7enzyme
EstradiolSolute carrier family 22 member 2transporter
EstradiolBeclin-1target
EstradiolUDP-glucuronosyltransferase 2B15enzyme
EstradiolCatechol O-methyltransferaseenzyme
EstradiolUDP-glucuronosyltransferases (UGTs)enzyme
EstradiolAromataseenzyme
EstradiolG protein-coupled estrogen receptor 1target
EstradiolATP synthase F(0) complex subunit atarget
EstradiolNeuronal acetylcholine receptor subunit alpha-4target
EstradiolSolute carrier organic anion transporter family member 1C1transporter
EstradiolSolute carrier organic anion transporter family member 1B3transporter
EstradiolOrganic anion transporter 3transporter
EstradiolCytochrome P450 2C9enzyme
EstradiolCytochrome P450 2C8enzyme
EstradiolCytochrome P450 2C19enzyme
EstradiolCytochrome P450 1B1enzyme
EstradiolCytochrome P450 1A1enzyme
EstradiolATP-dependent translocase ABCB1transporter
EstradiolSolute carrier organic anion transporter family member 1B1transporter
EstradiolBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
EstradiolSolute carrier family 22 member 11transporter
EstradiolATP-binding cassette sub-family C member 10transporter
EstradiolSolute carrier family 22 member 3transporter
Estradiol acetateCytochrome P450 3A4enzyme
Estradiol acetateCytochrome P450 3A5enzyme
Estradiol acetateCytochrome P450 3A7enzyme
Estradiol acetateSolute carrier family 22 member 2transporter
Estradiol acetateSolute carrier family 22 member 1transporter
Estradiol acetateSolute carrier family 22 member 3transporter
Estradiol acetateSolute carrier organic anion transporter family member 2B1transporter
Estradiol acetateSolute carrier organic anion transporter family member 1A2transporter
Estradiol acetateATP-binding cassette sub-family C member 10transporter
Estradiol acetateSolute carrier family 22 member 11transporter
Estradiol acetateBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
Estradiol acetateSolute carrier organic anion transporter family member 1B1transporter
Estradiol acetateATP-dependent translocase ABCB1transporter
Estradiol acetateCytochrome P450 1A1enzyme
Estradiol acetateCytochrome P450 1B1enzyme
Estradiol acetateCytochrome P450 2C19enzyme
Estradiol acetateCytochrome P450 2C8enzyme
Estradiol acetateCytochrome P450 2C9enzyme
Estradiol acetateOrganic anion transporter 3transporter
Estradiol acetateSolute carrier organic anion transporter family member 1B3transporter
Estradiol acetateSolute carrier organic anion transporter family member 1C1transporter
Estradiol acetateSolute carrier organic anion transporter family member 4A1transporter
Estradiol acetateNeuronal acetylcholine receptor subunit alpha-4target
Estradiol acetateNuclear receptor coactivator 2target
Estradiol acetateG protein-coupled estrogen receptor 1target
Estradiol acetateATP synthase F(0) complex subunit atarget
Estradiol acetateBeclin-1target
Estradiol acetate17-beta-hydroxysteroid dehydrogenase type 2target
Estradiol acetateEstrogen-related receptor gammatarget
Estradiol acetateFatty acid-binding protein, intestinalcarrier
Estradiol acetateEstrogen receptortarget
Estradiol acetateNuclear receptor subfamily 1 group I member 2target
Estradiol acetateAlbumincarrier
Estradiol acetateUDP-glucuronosyltransferase 1A1enzyme
Estradiol acetateCytochrome P450 1A2enzyme
Estradiol acetateEstrogen receptor betatarget
Estradiol acetateSex hormone-binding globulincarrier
Estradiol benzoateEstrogen receptortarget
Estradiol benzoateNuclear receptor subfamily 1 group I member 2target
Estradiol benzoateSex hormone-binding globulincarrier
Estradiol benzoateEstrogen receptor betatarget
Estradiol benzoateCytochrome P450 1A2enzyme
Estradiol benzoateUDP-glucuronosyltransferase 1A1enzyme
Estradiol benzoateAlbumincarrier
Estradiol benzoateFatty acid-binding protein, intestinalcarrier
Estradiol benzoateCytochrome P450 3A4enzyme
Estradiol benzoateCytochrome P450 3A5enzyme
Estradiol benzoateCytochrome P450 3A7enzyme
Estradiol benzoateSolute carrier family 22 member 2transporter
Estradiol benzoateSolute carrier family 22 member 1transporter
Estradiol benzoateSolute carrier family 22 member 3transporter
Estradiol benzoateSolute carrier organic anion transporter family member 2B1transporter
Estradiol benzoateSolute carrier organic anion transporter family member 1A2transporter
Estradiol benzoateATP-binding cassette sub-family C member 10transporter
Estradiol benzoateSolute carrier family 22 member 11transporter
Estradiol benzoateBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
Estradiol benzoateSolute carrier organic anion transporter family member 1B1transporter
Estradiol benzoateATP-dependent translocase ABCB1transporter
Estradiol benzoateCytochrome P450 1A1enzyme
Estradiol benzoateCytochrome P450 1B1enzyme
Estradiol benzoateCytochrome P450 2C19enzyme
Estradiol benzoateCytochrome P450 2C8enzyme
Estradiol benzoateCytochrome P450 2C9enzyme
Estradiol benzoateOrganic anion transporter 3transporter
Estradiol benzoateSolute carrier organic anion transporter family member 1B3transporter
Estradiol benzoateSolute carrier organic anion transporter family member 1C1transporter
Estradiol benzoateSolute carrier organic anion transporter family member 4A1transporter
Estradiol benzoateNeuronal acetylcholine receptor subunit alpha-4target
Estradiol benzoateNuclear receptor coactivator 2target
Estradiol benzoateG protein-coupled estrogen receptor 1target
Estradiol benzoateATP synthase F(0) complex subunit atarget
Estradiol benzoateBeclin-1target
Estradiol benzoate17-beta-hydroxysteroid dehydrogenase type 2target
Estradiol benzoateEstrogen-related receptor gammatarget
Estradiol cypionateEstrogen receptortarget
Estradiol cypionateNuclear receptor subfamily 1 group I member 2target
Estradiol cypionateSex hormone-binding globulincarrier
Estradiol cypionateEstrogen receptor betatarget
Estradiol cypionateCytochrome P450 1A2enzyme
Estradiol cypionateUDP-glucuronosyltransferase 1A1enzyme
Estradiol cypionateAlbumincarrier
Estradiol cypionateFatty acid-binding protein, intestinalcarrier
Estradiol cypionateCytochrome P450 3A4enzyme
Estradiol cypionateCytochrome P450 3A5enzyme
Estradiol cypionateCytochrome P450 3A7enzyme
Estradiol cypionateSolute carrier family 22 member 2transporter
Estradiol cypionateSolute carrier family 22 member 1transporter
Estradiol cypionateSolute carrier family 22 member 3transporter
Estradiol cypionateSolute carrier organic anion transporter family member 2B1transporter
Estradiol cypionateSolute carrier organic anion transporter family member 1A2transporter
Estradiol cypionateATP-binding cassette sub-family C member 10transporter
Estradiol cypionateSolute carrier family 22 member 11transporter
Estradiol cypionateBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
Estradiol cypionateSolute carrier organic anion transporter family member 1B1transporter
Estradiol cypionateATP-dependent translocase ABCB1transporter
Estradiol cypionateCytochrome P450 1A1enzyme
Estradiol cypionateCytochrome P450 1B1enzyme
Estradiol cypionateCytochrome P450 2C19enzyme
Estradiol cypionateCytochrome P450 2C8enzyme
Estradiol cypionateCytochrome P450 2C9enzyme
Estradiol cypionateOrganic anion transporter 3transporter
Estradiol cypionateSolute carrier organic anion transporter family member 1B3transporter
Estradiol cypionateSolute carrier organic anion transporter family member 1C1transporter
Estradiol cypionateSolute carrier organic anion transporter family member 4A1transporter
Estradiol cypionateNeuronal acetylcholine receptor subunit alpha-4target
Estradiol cypionateNuclear receptor coactivator 2target
Estradiol cypionateG protein-coupled estrogen receptor 1target
Estradiol cypionateATP synthase F(0) complex subunit atarget
Estradiol cypionateBeclin-1target
Estradiol cypionate17-beta-hydroxysteroid dehydrogenase type 2target
Estradiol cypionateEstrogen-related receptor gammatarget
Estradiol dienanthateEstrogen receptortarget
Estradiol dienanthateNuclear receptor subfamily 1 group I member 2target
Estradiol dienanthateSex hormone-binding globulincarrier
Estradiol dienanthateEstrogen receptor betatarget
Estradiol dienanthateCytochrome P450 1A2enzyme
Estradiol dienanthateUDP-glucuronosyltransferase 1A1enzyme
Estradiol dienanthateAlbumincarrier
Estradiol dienanthateFatty acid-binding protein, intestinalcarrier
Estradiol dienanthateCytochrome P450 3A4enzyme
Estradiol dienanthateCytochrome P450 3A5enzyme
Estradiol dienanthateCytochrome P450 3A7enzyme
Estradiol dienanthateSolute carrier family 22 member 2transporter
Estradiol dienanthateSolute carrier family 22 member 1transporter
Estradiol dienanthateSolute carrier family 22 member 3transporter
Estradiol dienanthateSolute carrier organic anion transporter family member 2B1transporter
Estradiol dienanthateSolute carrier organic anion transporter family member 1A2transporter
Estradiol dienanthateATP-binding cassette sub-family C member 10transporter
Estradiol dienanthateSolute carrier family 22 member 11transporter
Estradiol dienanthateBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
Estradiol dienanthateSolute carrier organic anion transporter family member 1B1transporter
Estradiol dienanthateATP-dependent translocase ABCB1transporter
Estradiol dienanthateCytochrome P450 1A1enzyme
Estradiol dienanthateCytochrome P450 1B1enzyme
Estradiol dienanthateCytochrome P450 2C19enzyme
Estradiol dienanthateCytochrome P450 2C8enzyme
Estradiol dienanthateCytochrome P450 2C9enzyme
Estradiol dienanthateOrganic anion transporter 3transporter
Estradiol dienanthateSolute carrier organic anion transporter family member 1B3transporter
Estradiol dienanthateSolute carrier organic anion transporter family member 1C1transporter
Estradiol dienanthateSolute carrier organic anion transporter family member 4A1transporter
Estradiol dienanthateNeuronal acetylcholine receptor subunit alpha-4target
Estradiol dienanthateNuclear receptor coactivator 2target
Estradiol dienanthateG protein-coupled estrogen receptor 1target
Estradiol dienanthateATP synthase F(0) complex subunit atarget
Estradiol dienanthateBeclin-1target
Estradiol dienanthate17-beta-hydroxysteroid dehydrogenase type 2target
Estradiol dienanthateEstrogen-related receptor gammatarget
Estradiol valerateEstrogen receptortarget
Estradiol valerateNuclear receptor subfamily 1 group I member 2target
Estradiol valerateSex hormone-binding globulincarrier
Estradiol valerateEstrogen receptor betatarget
Estradiol valerateCytochrome P450 1A2enzyme
Estradiol valerateUDP-glucuronosyltransferase 1A1enzyme
Estradiol valerateAlbumincarrier
Estradiol valerateFatty acid-binding protein, intestinalcarrier
Estradiol valerateCytochrome P450 3A4enzyme
Estradiol valerateCytochrome P450 3A5enzyme
Estradiol valerateCytochrome P450 3A7enzyme
Estradiol valerateSolute carrier family 22 member 2transporter
Estradiol valerateSolute carrier family 22 member 1transporter
Estradiol valerateSolute carrier family 22 member 3transporter
Estradiol valerateSolute carrier organic anion transporter family member 2B1transporter
Estradiol valerateSolute carrier organic anion transporter family member 1A2transporter
Estradiol valerateATP-binding cassette sub-family C member 10transporter
Estradiol valerateSolute carrier family 22 member 11transporter
Estradiol valerateBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
Estradiol valerateSolute carrier organic anion transporter family member 1B1transporter
Estradiol valerateATP-dependent translocase ABCB1transporter
Estradiol valerateCytochrome P450 1A1enzyme
Estradiol valerateCytochrome P450 1B1enzyme
Estradiol valerateCytochrome P450 2C19enzyme
Estradiol valerateCytochrome P450 2C8enzyme
Estradiol valerateCytochrome P450 2C9enzyme
Estradiol valerateSolute carrier organic anion transporter family member 1B3transporter
Estradiol valerateEstrogen-related receptor gammatarget
Estradiol valerate17-beta-hydroxysteroid dehydrogenase type 2target
Estradiol valerateBeclin-1target
Estradiol valerateATP synthase F(0) complex subunit atarget
Estradiol valerateG protein-coupled estrogen receptor 1target
Estradiol valerateNuclear receptor coactivator 2target
Estradiol valerateNeuronal acetylcholine receptor subunit alpha-4target
Estradiol valerateSolute carrier organic anion transporter family member 4A1transporter
Estradiol valerateSolute carrier organic anion transporter family member 1C1transporter
Estradiol valerateOrganic anion transporter 3transporter
Estrone sulfateCytochrome P450 3A4enzyme
Estrone sulfateEstrogen receptortarget
Estrone sulfateEstrogen receptor betatarget
Estrone sulfateSex hormone-binding globulincarrier
Estrone sulfateCytochrome P450 1A2enzyme
Estrone sulfateAlbumincarrier
Estrone sulfateCytochrome P450 2C9enzyme
Estrone sulfateMultidrug and toxin extrusion protein 1transporter
Estrone sulfateMultidrug and toxin extrusion protein 2transporter
Estrone sulfateHepatic sodium/bile acid cotransportertransporter
EthambutolCytochrome P450 2E1enzyme
EthambutolCytochrome P450 2C19enzyme
EthambutolProbable arabinosyltransferase Ctarget
EthambutolProbable arabinosyltransferase Atarget
EthambutolProbable arabinosyltransferase Btarget
EthambutolCytochrome P450 2D6enzyme
EthambutolCytochrome P450 2A6enzyme
EthambutolCytochrome P450 2C9enzyme
EthambutolCytochrome P450 3A4enzyme
EthambutolCytochrome P450 1A2enzyme
Ethanol5-hydroxytryptamine receptor 3Ctarget
EthanolCytochrome P450 2C9enzyme
EthanolAldo-keto reductase family 1 member A1enzyme
EthanolGamma-aminobutyric acid receptor subunit deltatarget
EthanolGamma-aminobutyric acid receptor subunit thetatarget
EthanolGamma-aminobutyric acid receptor subunit pitarget
EthanolGamma-aminobutyric acid receptor subunit epsilontarget
EthanolGamma-aminobutyric acid receptor subunit gamma-3target
EthanolGamma-aminobutyric acid receptor subunit gamma-1target
EthanolNeuronal acetylcholine receptor subunit beta-3target
EthanolNeuronal acetylcholine receptor subunit alpha-6target
EthanolNeuronal acetylcholine receptor subunit alpha-5target
EthanolNeuronal acetylcholine receptor subunit alpha-3target
EthanolNeuronal acetylcholine receptor subunit beta-4target
EthanolAlcohol dehydrogenase 6enzyme
EthanolVoltage-dependent L-type calcium channel subunit alpha-1Dtarget
EthanolVoltage-dependent L-type calcium channel subunit alpha-1Starget
EthanolGamma-aminobutyric acid receptor subunit beta-2target
EthanolGamma-aminobutyric acid receptor subunit beta-3target
EthanolGamma-aminobutyric acid receptor subunit beta-1target
EthanolNeuronal acetylcholine receptor subunit alpha-9target
EthanolNeuronal acetylcholine receptor subunit alpha-7target
EthanolG protein-activated inward rectifier potassium channel 4target
EthanolEquilibrative nucleoside transporter 1target
EthanolVascular cell adhesion protein 1target
EthanolG protein-activated inward rectifier potassium channel 2target
EthanolG protein-activated inward rectifier potassium channel 1target
EthanolNeuronal acetylcholine receptor subunit beta-2target
Ethanol5-hydroxytryptamine receptor 3Dtarget
EthanolVoltage-dependent calcium channel gamma-2 subunittarget
EthanolG protein-activated inward rectifier potassium channel 3target
EthanolNeural cell adhesion molecule L1target
EthanolAcetylcholinesterasetarget
EthanolAll-trans-retinol dehydrogenase [NAD(+)] ADH7target
EthanolNeuronal acetylcholine receptor subunit alpha-4target
Ethanol5-hydroxytryptamine receptor 3Btarget
EthanolGlutamate receptor 3target
EthanolGlutamate receptor 4target
EthanolGlutamate receptor 2target
EthanolGamma-aminobutyric acid receptor subunit alpha-6target
EthanolNeuronal acetylcholine receptor subunit alpha-2target
EthanolVoltage-dependent calcium channel gamma-1 subunittarget
EthanolGlutamate receptor 1target
EthanolGamma-aminobutyric acid receptor subunit alpha-2target
EthanolGamma-aminobutyric acid receptor subunit alpha-1target
EthanolGlutamate receptor ionotropic, NMDA 3Atarget
EthanolGlycine receptor subunit alpha-1target
EthanolGlycine receptor subunit alpha-2target
EthanolCytochrome P450 2E1enzyme
EthanolCytochrome P450 1A1enzyme
EthanolCytochrome P450 1A2enzyme
EthanolCytochrome P450 2B6enzyme
EthanolCytochrome P450 2C19enzyme
EthanolEquilibrative nucleoside transporter 2target
EthanolCytochrome P450 3A4enzyme
EthanolCytochrome P450 4A11enzyme
EthanolAlcohol dehydrogenase 1Aenzyme
EthanolAll-trans-retinol dehydrogenase [NAD(+)] ADH1Benzyme
EthanolAlcohol dehydrogenase 1Cenzyme
EthanolAlcohol dehydrogenase class-3enzyme
EthanolVoltage-dependent L-type calcium channel subunit beta-1target
Ethanol5-hydroxytryptamine receptor 3Atarget
EthanolAll-trans-retinol dehydrogenase [NAD(+)] ADH4enzyme
Ethanol5-hydroxytryptamine receptor 3Etarget
EthanolNeuronal acetylcholine receptor subunit alpha-10target
EthanolVoltage-dependent L-type calcium channel subunit alpha-1Ctarget
EthanolGamma-aminobutyric acid receptor subunit alpha-5target
EthanolGamma-aminobutyric acid receptor subunit alpha-4target
EthanolAll-trans-retinol dehydrogenase [NAD(+)] ADH7enzyme
EthanolGamma-aminobutyric acid receptor subunit alpha-3target
EthinylestradiolNuclear receptor subfamily 1 group I member 2target
EthinylestradiolCytochrome P450 3A4enzyme
EthinylestradiolCytochrome P450 2C8enzyme
EthinylestradiolBile salt export pumptransporter
EthinylestradiolHepatic sodium/bile acid cotransportertransporter
EthinylestradiolATP-binding cassette sub-family C member 2transporter
EthinylestradiolATP-dependent translocase ABCB1transporter
EthinylestradiolUDP-glucuronosyltransferase 1A1enzyme
EthinylestradiolCytochrome P450 2C19enzyme
EthinylestradiolUDP-glucuronosyltransferase 1A4enzyme
EthinylestradiolUDP-glucuronosyltransferase 1A9enzyme
EthinylestradiolCytochrome P450 2C9enzyme
EthinylestradiolCytochrome P450 1A2enzyme
EthinylestradiolSulfotransferase 1E1enzyme
EthinylestradiolSulfotransferase 1A3enzyme
EthinylestradiolCytochrome P450 3A5enzyme
EthinylestradiolUDP-glucuronosyltransferase 2B7enzyme
EthinylestradiolUDP-glucuronosyltransferase 1A3enzyme
EthinylestradiolCatechol O-methyltransferaseenzyme
EthinylestradiolSolute carrier organic anion transporter family member 1A2transporter
EthinylestradiolAlbumincarrier
EthinylestradiolSex hormone-binding globulincarrier
EthinylestradiolEstrogen receptortarget
EtoposideATP-binding cassette sub-family C member 2transporter
EtoposideDNA topoisomerase 2-alphatarget
EtoposideGlutathione S-transferase theta-1enzyme
EtoposideDNA topoisomerase 2-betatarget
EtoposideDNA topoisomerase 2target
EtoposideUDP-glucuronosyltransferase 1A1enzyme
EtoposideCytochrome P450 3A5enzyme
EtoposideCytochrome P450 2E1enzyme
EtoposideCytochrome P450 1A2enzyme
EtoposideProstaglandin G/H synthase 1enzyme
EtoposideBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
EtoposideProstaglandin G/H synthase 2enzyme
EtoposideATP-binding cassette sub-family C member 10transporter
EtoposideMultidrug resistance-associated protein 1transporter
EtoposideATP-dependent translocase ABCB1transporter
EtoposideATP-binding cassette sub-family C member 6transporter
EtoposideGlutathione S-transferase Penzyme
EtoposideCytochrome P450 3A4enzyme
EtoposideATP-binding cassette sub-family C member 3transporter
EtoricoxibCytochrome P450 2E1enzyme
EtoricoxibCytochrome P450 2C19enzyme
EtoricoxibCytochrome P450 1A2enzyme
EtoricoxibCytochrome P450 2D6enzyme
EtoricoxibCytochrome P450 3A4enzyme
EtoricoxibProstaglandin G/H synthase 2target
EtoricoxibCytochrome P450 2C9enzyme
EtravirineReverse transcriptase/RNaseHtarget
EtravirinePhosphatidylcholine translocator ABCB4transporter
EtravirineATP-dependent translocase ABCB1transporter
EtravirineGag-Pol polyproteintarget
EtravirineGag-Pol polyproteintarget
EtravirineCytochrome P450 2C19enzyme
EtravirineCytochrome P450 2C9enzyme
EtravirineCytochrome P450 3A4enzyme
EtripamilVoltage-dependent L-type calcium channeltarget
EtripamilMultidrug and toxin extrusion protein 1transporter
EtripamilSolute carrier organic anion transporter family member 1B1transporter
EtripamilATP-dependent translocase ABCB1transporter
EtripamilCytochrome P450 2C9enzyme
EtripamilCytochrome P450 2D6enzyme
EtripamilCytochrome P450 3A5enzyme
EtripamilCytochrome P450 3A4enzyme
Evening primrose oilCytochrome P450 2C19enzyme
Evening primrose oilCytochrome P450enzyme
Evening primrose oilAcyl-CoA 6-desaturaseenzyme
Evening primrose oilAcyl-CoA (8-3)-desaturaseenzyme
Evening primrose oilVery long chain fatty acid elongase 5enzyme
EverolimusSerine/threonine-protein kinase mTORtarget
EverolimusSolute carrier organic anion transporter family member 1B1transporter
EverolimusSolute carrier organic anion transporter family member 1B3transporter
EverolimusSolute carrier organic anion transporter family member 1A2transporter
EverolimusCytochrome P450 2D6enzyme
EverolimusATP-dependent translocase ABCB1transporter
EverolimusPeptidyl-prolyl cis-trans isomerase FKBP1Atarget
EverolimusCytochrome P450 3A4enzyme
EzetimibeBile salt export pumptransporter
EzetimibeNPC1-like intracellular cholesterol transporter 1target
EzetimibeAminopeptidase Ntarget
EzetimibeSterol O-acyltransferase 1target
EzetimibeCytochrome P450 2C8enzyme
EzetimibeBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
EzetimibeATP-binding cassette sub-family C member 3transporter
EzetimibeCytochrome P450 3A4enzyme
EzetimibeUDP-glucuronosyltransferase 2B7enzyme
EzetimibeUDP-glucuronosyltransferase 2B15enzyme
EzetimibeUDP-glucuronosyltransferase 1A1enzyme
EzetimibeSolute carrier organic anion transporter family member 1B1transporter
EzetimibeATP-binding cassette sub-family C member 2transporter
EzetimibeATP-dependent translocase ABCB1transporter
EzetimibeUDP-glucuronosyltransferase 1A3enzyme
FamotidineHistamine H2 receptortarget
FamotidineSolute carrier family 22 member 2transporter
FamotidineOrganic anion transporter 3transporter
FamotidineMultidrug and toxin extrusion protein 1transporter
FamotidineCytochrome P450 1A2enzyme
FamotidineSolute carrier family 22 member 6transporter
FavipiravirATP-dependent translocase ABCB1transporter
FavipiravirSolute carrier family 22 member 6transporter
FavipiravirOrganic anion transporter 3transporter
FavipiravirSolute carrier family 22 member 12transporter
FavipiravirCytochrome P450 2E1enzyme
FavipiravirDNA-directed RNA polymerase subunit betatarget
FavipiravirDNA-directed RNA polymerase subunit beta'target
Favipiraviralpha1-acid glycoproteincarrier
FavipiravirAlbumincarrier
FavipiravirCytochrome P450 2C8enzyme
FavipiravirXanthine dehydrogenase/oxidaseenzyme
FavipiravirAldehyde oxidaseenzyme
FavipiravirRNA-directed RNA polymerase catalytic subunittarget
FedratinibCytochrome P450 2D6enzyme
FedratinibTyrosine-protein kinase JAK1target
FedratinibReceptor-type tyrosine-protein kinase FLT3target
FedratinibTyrosine-protein kinase JAK2target
FedratinibFlavin-containing monooxygenase 3enzyme
FedratinibCytochrome P450 2C19enzyme
FedratinibCytochrome P450 3A4enzyme
FedratinibMultidrug and toxin extrusion protein 2transporter
FedratinibMultidrug and toxin extrusion protein 1transporter
FedratinibPOU domain, class 2, transcription factor 2transporter
FedratinibSolute carrier organic anion transporter family member 1B3transporter
FedratinibSolute carrier organic anion transporter family member 1B1transporter
FedratinibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
FedratinibATP-dependent translocase ABCB1transporter
FelbamateCytochrome P450 2C9enzyme
FelbamateCytochrome P450 2E1enzyme
FelbamateCytochrome P450 3A4enzyme
FelbamateCytochrome P450 2C19enzyme
FelbamateGlutamate receptor ionotropic, NMDA 2Atarget
FelbamateGlutamate receptor ionotropic, NMDA 2Btarget
FelodipineVoltage-dependent calcium channel subunit alpha-2/delta-1target
FelodipineCytochrome P450 3A4enzyme
FelodipineVoltage-dependent L-type calcium channel subunit alpha-1Ctarget
FelodipineVoltage-dependent L-type calcium channel subunit beta-2target
FelodipineCytochrome P450 2C8enzyme
FelodipineDual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1Btarget
FelodipineDual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1Atarget
FelodipineVoltage-dependent T-type calcium channel subunit alpha-1Htarget
FelodipineVoltage-dependent calcium channel subunit alpha-2/delta-2target
FelodipineTroponin C, skeletal muscletarget
FelodipineTroponin C, slow skeletal and cardiac musclestarget
FelodipineMineralocorticoid receptortarget
FelodipineVoltage-dependent L-type calcium channel subunit alpha-1Dtarget
FelodipineVoltage-dependent L-type calcium channel subunit alpha-1Starget
FelodipineCytochrome P450 3A5enzyme
FelodipineCytochrome P450 3A7enzyme
FelodipineATP-dependent translocase ABCB1transporter
FelodipineCytochrome P450 2C9enzyme
FelodipineCytochrome P450 2D6enzyme
FelodipineBile salt export pumptransporter
FelodipineCalmodulintarget
FelodipineVoltage gated L-type calcium channeltarget
FenfluramineCytochrome P450 3A5enzyme
FenfluramineCytochrome P450 3A4enzyme
FenfluramineCytochrome P450 2C19enzyme
FenfluramineCytochrome P450 2C9enzyme
FenfluramineCytochrome P450 2B6enzyme
FenfluramineCytochrome P450 1A2enzyme
Fenfluramine5-hydroxytryptamine receptor 1Atarget
FenfluramineSigma non-opioid intracellular receptor 1target
Fenfluramine5-hydroxytryptamine receptor 1Dtarget
Fenfluramine5-hydroxytryptamine receptor 2Atarget
FenfluramineSodium-dependent serotonin transportertarget
FenfluramineCytochrome P450 2D6enzyme
Fenfluramine5-hydroxytryptamine receptor 2Btarget
Fenfluramine5-hydroxytryptamine receptor 2Ctarget
FennelCytochrome P450 2E1enzyme
FennelCytochrome P450 3A4enzyme
FennelCytochrome P450 2D6enzyme
FennelAcetylcholinesterasetarget
FenofibrateAldo-keto reductase family 1 member C3enzyme
FenofibrateAldo-keto reductase family 1 member C2enzyme
FenofibrateAldo-keto reductase family 1 member C1enzyme
FenofibrateAldo-keto reductase family 1 member B1enzyme
FenofibrateCytochrome P450 2C8enzyme
FenofibrateMatrix metalloproteinase-25target
FenofibratePeroxisome proliferator-activated receptor alphatarget
FenofibrateCytochrome P450 2C9enzyme
FenofibrateCarbonyl reductase [NADPH] 1enzyme
FenofibrateLiver carboxylesterase 1enzyme
FenofibrateCytochrome P450 2A6enzyme
FenofibrateCytochrome P450 2C19enzyme
FenofibrateAlbumincarrier
FenofibrateBile salt export pumptransporter
FenofibrateUDP-glucuronosyltransferase 1A9enzyme
FenofibrateNuclear receptor subfamily 1 group I member 2target
FenvalerateProtein phosphatase 3 catalytic subunit alphatarget
FenvalerateCytochrome P450 3A4enzyme
FenvalerateCytochrome P450 2D6enzyme
FerrohemeNitric oxide synthase, inducibletarget
FerrohemeProstaglandin G/H synthase 1target
FerrohemeHeme oxygenase 1target
FerrohemePolyunsaturated fatty acid 5-lipoxygenasetarget
FerrohemeCytochrome P450 3A4target
FerrohemeNitric oxide synthase 1target
FerrohemeHemoglobin subunit alphatarget
FerrohemeNitric oxide synthase 3target
FerrohemeProstaglandin G/H synthase 2target
FerrohemeCystathionine beta-synthasetarget
FexinidazoleCytochrome P450 2C19enzyme
FexinidazoleCytochrome P450 3A4enzyme
FexinidazoleCytochrome P450 3A5enzyme
FexinidazoleFlavin-containing monooxygenase 3enzyme
FexinidazoleCytochrome P450 2D6enzyme
FexinidazoleSolute carrier organic anion transporter family member 1B1transporter
FexinidazoleSolute carrier organic anion transporter family member 1B3transporter
FexinidazoleSolute carrier family 22 member 2transporter
FexinidazoleSolute carrier family 22 member 6transporter
FexinidazoleCytochrome P450 1A2enzyme
FexinidazoleCytochrome P450 2B6enzyme
FexinidazoleOrganic anion transporter 3transporter
FexinidazoleMultidrug and toxin extrusion protein 1transporter
FexinidazoleMultidrug and toxin extrusion protein 2transporter
FexinidazoleCytochrome P450 3A Subfamilyenzyme
FexinidazoleNitroreductasestarget
FidaxomicinATP-dependent translocase ABCB1transporter
FidaxomicinRNA polymerase sigma factor SigAtarget
FidaxomicinCytochrome P450 3A4enzyme
FlecainideRyanodine receptor 2target
FlecainideSodium channel protein type 5 subunit alphatarget
FlecainideCytochrome P450 2D6enzyme
FlecainideSodium channel protein type 4 subunit alphatarget
FlecainideCytochrome P450 2C9enzyme
FlecainideVoltage-gated inwardly rectifying potassium channel KCNH2target
Flecainidealpha1-acid glycoproteincarrier
FlecainideAlbumincarrier
FlecainideMultidrug and toxin extrusion protein 1transporter
FlecainideATP-dependent translocase ABCB1transporter
FlecainideCytochrome P450 1A2enzyme
FloxuridineThyroxine-binding globulincarrier
FloxuridineCytochrome P450 2C9enzyme
FloxuridineThymidine phosphorylaseenzyme
FloxuridineThymidylate synthasetarget
FloxuridineThymidylate synthasetarget
FluconazoleCytochrome P450 3A5enzyme
FluconazoleLanosterol 14-alpha demethylasetarget
FluconazoleATP-dependent translocase ABCB1transporter
FluconazoleCytochrome P450 2C19enzyme
FluconazoleCytochrome P450 2C9enzyme
FluconazoleCytochrome P450 3A4enzyme
FlumequineDNA gyrase subunit Atarget
FlumequineDNA gyrase subunit Btarget
FlumequineCytochrome P450 1A2enzyme
FlunitrazepamCytochrome P450 2E1enzyme
FlunitrazepamCytochrome P450 2C19enzyme
FlunitrazepamUDP-glucuronosyltransferase 2B7enzyme
FlunitrazepamCytochrome P450 2A6enzyme
FlunitrazepamCytochrome P450 2B6enzyme
FlunitrazepamCytochrome P450 2C9enzyme
FlunitrazepamCytochrome P450 3A4enzyme
FlunitrazepamUDP-glucuronosyltransferase 1A1enzyme
FlunitrazepamUDP-glucuronosyltransferase 1A3enzyme
FlunitrazepamGABA(A) Receptortarget
FlunitrazepamGABA(A) Receptor Benzodiazepine Binding Sitetarget
FlunitrazepamTranslocator proteintarget
FluorouracilDNAtarget
FluorouracilRNAtarget
FluorouracilCytochrome P450 2A6enzyme
FluorouracilCytochrome P450 2C8enzyme
FluorouracilMethylenetetrahydrofolate reductase (NADPH)enzyme
FluorouracilThymidylate synthaseenzyme
FluorouracilUridine 5'-monophosphate synthaseenzyme
FluorouracilAmidophosphoribosyltransferaseenzyme
FluorouracilSolute carrier family 22 member 7transporter
FluorouracilEquilibrative nucleoside transporter 1transporter
FluorouracilBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
FluorouracilATP-binding cassette sub-family C member 3transporter
FluorouracilATP-binding cassette sub-family C member 4transporter
FluorouracilATP-binding cassette sub-family C member 5transporter
FluorouracilThyroxine-binding globulincarrier
FluorouracilThymidylate synthasetarget
FluorouracilDihydropyrimidine dehydrogenase [NADP(+)]target
FluorouracilTelomerase reverse transcriptasetarget
FluorouracilUridine phosphorylase 2enzyme
FluorouracilUridine phosphorylase 1enzyme
FluorouracilDihydropyrimidine dehydrogenase [NADP(+)]enzyme
FluorouracilThymidylate synthasetarget
FluorouracilCytochrome P450 1A2enzyme
FluorouracilThymidine phosphorylaseenzyme
FluorouracilAlbumincarrier
FluorouracilCytochrome P450 2C9enzyme
Fluoxetine5-hydroxytryptamine receptor 2Ctarget
FluoxetineVoltage-gated inwardly rectifying potassium channel KCNH2target
FluoxetineCyclin-dependent kinases regulatory subunit 1target
FluoxetineNeuronal acetylcholine receptor subunit alpha-2target
FluoxetineNeuronal acetylcholine receptor subunit alpha-3target
FluoxetineNeuronal acetylcholine receptor subunit beta-4target
FluoxetineCytochrome P450 2C19enzyme
FluoxetineSodium-dependent serotonin transportertarget
FluoxetineCytochrome P450 2C9enzyme
FluoxetineCytochrome P450 2D6enzyme
FluoxetineCytochrome P450enzyme
FluoxetineCytochrome P450 1A2enzyme
FluoxetineCytochrome P450 3A4enzyme
FluoxetineAlpha-1-acid glycoprotein 1carrier
FluoxetineATP-dependent translocase ABCB1transporter
FluoxetineCytochrome P450 2B6enzyme
FluoxetineCytochrome P450 3A5enzyme
FluoxetineAlbumincarrier
FluphenazineCalmodulintarget
Fluphenazine5-hydroxytryptamine receptor 1Btarget
Fluphenazine5-hydroxytryptamine receptor 2Ctarget
Fluphenazine5-hydroxytryptamine receptor 2Atarget
FluphenazineAndrogen receptortarget
FluphenazineCytochrome P450 2E1enzyme
FluphenazineATP-dependent translocase ABCB1transporter
FluphenazineCytochrome P450 2D6enzyme
FluphenazineD(1A) dopamine receptortarget
FluphenazineD(2) dopamine receptortarget
FlurazepamCytochrome P450 2A6enzyme
FlurazepamCytochrome P450 2E1enzyme
FlurazepamATP-dependent translocase ABCB1transporter
FlurazepamCytochrome P450 3A4enzyme
FlurazepamGABA(A) Receptortarget
FlurazepamSolute carrier family 22 member 2transporter
FlurazepamTranslocator proteintarget
FlurazepamGABA(A) Receptor Benzodiazepine Binding Sitetarget
FlurithromycinCytochrome P450 3A4enzyme
FluticasoneProgesterone receptortarget
FluticasoneMineralocorticoid receptortarget
FluticasoneCytosolic phospholipase A2target
FluticasoneCytochrome P450 3A7enzyme
FluticasoneCytochrome P450 3A5enzyme
FluticasoneCorticosteroid-binding globulincarrier
FluticasoneGlucocorticoid receptortarget
FluticasoneSolute carrier organic anion transporter family member 1B1transporter
FluticasoneATP-dependent translocase ABCB1transporter
FluticasoneSolute carrier organic anion transporter family member 1B1carrier
FluticasoneATP-dependent translocase ABCB1carrier
FluticasoneCytochrome P450 2C8enzyme
FluticasoneCytochrome P450 3A4enzyme
Fluticasone furoateAlpha-1-acid glycoprotein 1carrier
Fluticasone furoateAlbumincarrier
Fluticasone furoateMineralocorticoid receptortarget
Fluticasone furoateProgesterone receptortarget
Fluticasone furoateCytochrome P450 3A7enzyme
Fluticasone furoateCytochrome P450 3A4enzyme
Fluticasone furoateGlucocorticoid receptortarget
Fluticasone furoateATP-dependent translocase ABCB1transporter
Fluticasone furoateCytochrome P450 2C8enzyme
Fluticasone furoateSolute carrier organic anion transporter family member 1B1transporter
Fluticasone furoateCorticosteroid-binding globulincarrier
Fluticasone furoateCytochrome P450 3A5enzyme
Fluticasone propionateSolute carrier organic anion transporter family member 1B1transporter
Fluticasone propionateATP-dependent translocase ABCB1transporter
Fluticasone propionateSolute carrier organic anion transporter family member 1B1carrier
Fluticasone propionateCytochrome P450 2C8enzyme
Fluticasone propionateCytochrome P450 3A7enzyme
Fluticasone propionateCytochrome P450 3A5enzyme
Fluticasone propionateMineralocorticoid receptortarget
Fluticasone propionateProgesterone receptortarget
Fluticasone propionateCytochrome P450 3A4enzyme
Fluticasone propionateGlucocorticoid receptortarget
Fluticasone propionateCytosolic phospholipase A2target
Fluticasone propionateCorticosteroid-binding globulincarrier
FluvastatinHistone deacetylase 2target
Fluvastatin3-hydroxy-3-methylglutaryl-coenzyme A reductasetarget
FluvastatinCytochrome P450 2C9enzyme
FluvastatinCytochrome P450 3A4enzyme
FluvastatinCytochrome P450 2C8enzyme
FluvastatinCytochrome P450 2D6enzyme
FluvastatinCytochrome P450 2C19enzyme
FluvastatinCytochrome P450 1A1enzyme
FluvastatinSolute carrier organic anion transporter family member 1B1transporter
FluvastatinSolute carrier organic anion transporter family member 1B3transporter
FluvastatinSolute carrier organic anion transporter family member 2B1transporter
FluvastatinSolute carrier family 15 member 1transporter
FluvastatinCytochrome P450 3A5enzyme
FluvastatinUDP-glucuronosyltransferase 1A1enzyme
FluvastatinUDP-glucuronosyltransferase 1A3enzyme
FluvastatinUDP-glucuronosyltransferase 2B7enzyme
FluvastatinATP-binding cassette sub-family C member 2transporter
FluvastatinCytochrome P450 2B6enzyme
FluvoxamineSodium-dependent serotonin transportertarget
FluvoxamineCytochrome P450 3A Subfamilyenzyme
FluvoxamineCytochrome P450 1A2enzyme
FluvoxamineCytochrome P450 2D6enzyme
FluvoxamineCytochrome P450 2C9enzyme
FluvoxamineCytochrome P450 2C19enzyme
FluvoxamineCytochrome P450 1A1enzyme
FluvoxamineCytochrome P450 3A4enzyme
FluvoxamineATP-dependent translocase ABCB1transporter
FluvoxamineCytochrome P450 2B6enzyme
FluvoxamineVoltage-gated inwardly rectifying potassium channel KCNH2target
FluvoxamineBile salt export pumptransporter
FomepizoleCytochrome P450 2A6enzyme
FomepizoleCytochrome P450 2E1enzyme
FomepizoleCatalasetarget
FomepizoleAlcohol dehydrogenase 1Ctarget
FomepizoleAll-trans-retinol dehydrogenase [NAD(+)] ADH1Btarget
FomepizoleAlcohol dehydrogenase 1Atarget
FosamprenavirGag-Pol polyproteintarget
FosamprenavirCytochrome P450 3A4enzyme
FosamprenavirPol polyproteintarget
FosaprepitantCytochrome P450 3A4enzyme
FosaprepitantSubstance-P receptortarget
FosaprepitantCytochrome P450 2C9enzyme
FosfluconazoleCytochrome P450 3A4enzyme
FosnetupitantCytochrome P450 3A4enzyme
FosnetupitantSubstance-P receptortarget
FostamatinibCalcium/calmodulin-dependent protein kinase type 1Gtarget
FostamatinibSerine/threonine-protein kinase SIK3target
FostamatinibVascular endothelial growth factor receptor 2target
FostamatinibTyrosine-protein kinase JAK3target
FostamatinibTyrosine-protein kinase JAK2target
FostamatinibTyrosine-protein kinase ITK/TSKtarget
FostamatinibInterleukin-1 receptor-associated kinase 4target
FostamatinibInterleukin-1 receptor-associated kinase 3target
FostamatinibInterleukin-1 receptor-associated kinase 1target
FostamatinibAdenosine receptor A3target
FostamatinibSynaptic vesicular amine transportertarget
FostamatinibFatty-acid amide hydrolase 1target
FostamatinibEquilibrative nucleoside transporter 1target
FostamatinibUDP-glucuronosyltransferase 1A1target
FostamatinibcGMP-specific 3',5'-cyclic phosphodiesterasetarget
FostamatinibPolyunsaturated fatty acid 5-lipoxygenasetarget
FostamatinibCathepsin Starget
FostamatinibProcathepsin Ltarget
FostamatinibTyrosine-protein kinase ABL1target
FostamatinibCalcium-dependent protein kinase 1target
FostamatinibSerine/threonine-protein kinase PknBtarget
FostamatinibRibosomal protein S6 kinase alpha-6target
FostamatinibNon-receptor tyrosine-protein kinase TYK2target
FostamatinibAtypical kinase COQ8A, mitochondrialtarget
FostamatinibTyrosine-protein kinase JAK1target
FostamatinibHepatocyte growth factor receptortarget
FostamatinibSerine/threonine-protein kinase NIM1target
FostamatinibSerine/threonine-protein kinase 26target
FostamatinibcAMP-dependent protein kinase catalytic subunit alphatarget
FostamatinibSerine/threonine-protein kinase 24target
FostamatinibSerine/threonine-protein kinase 3target
FostamatinibTyrosine-protein kinase Tectarget
FostamatinibTyrosine-protein kinase SYKtarget
FostamatinibSerine/threonine-protein kinase 33target
FostamatinibSerine/threonine-protein kinase 35target
FostamatinibSerine/threonine-protein kinase 36target
FostamatinibSerine/threonine-protein kinase 38target
FostamatinibSerine/threonine-protein kinase 38-liketarget
FostamatinibSTE20/SPS1-related proline-alanine-rich protein kinasetarget
FostamatinibSerine/threonine-protein kinase TAO1target
FostamatinibSerine/threonine-protein kinase TAO2target
FostamatinibSerine/threonine-protein kinase TAO3target
FostamatinibSerine/threonine-protein kinase TBK1target
FostamatinibAngiopoietin-1 receptortarget
FostamatinibDual specificity testis-specific protein kinase 1target
FostamatinibTGF-beta receptor type-1target
FostamatinibTGF-beta receptor type-2target
FostamatinibTyrosine-protein kinase receptor Tie-1target
FostamatinibSerine/threonine-protein kinase tousled-like 1target
FostamatinibSerine/threonine-protein kinase tousled-like 2target
FostamatinibTRAF2 and NCK-interacting protein kinasetarget
FostamatinibNon-receptor tyrosine-protein kinase TNK1target
FostamatinibActivated CDC42 kinase 1target
FostamatinibSerine/threonine-protein kinase TNNI3Ktarget
FostamatinibTestis-specific serine/threonine-protein kinase 1target
FostamatinibDual specificity protein kinase TTKtarget
FostamatinibTyrosine-protein kinase TXKtarget
FostamatinibTyrosine-protein kinase receptor TYRO3target
FostamatinibSerine/threonine-protein kinase ULK1target
FostamatinibSerine/threonine-protein kinase ULK2target
FostamatinibSerine/threonine-protein kinase ULK3target
FostamatinibWee1-like protein kinasetarget
FostamatinibTyrosine-protein kinase Yestarget
FostamatinibMitogen-activated protein kinase kinase kinase 19target
FostamatinibMitogen-activated protein kinase kinase kinase 20target
FostamatinibTyrosine-protein kinase ZAP-70target
FostamatinibAP2-associated protein kinase 1target
FostamatinibTyrosine-protein kinase ABL2target
FostamatinibActivin receptor type-1target
FostamatinibActivin receptor type-1Btarget
FostamatinibAtypical kinase COQ8B, mitochondrialtarget
FostamatinibALK tyrosine kinase receptortarget
FostamatinibAnkyrin repeat and protein kinase domain-containing protein 1target
FostamatinibAurora kinase Atarget
FostamatinibAurora kinase Btarget
FostamatinibAurora kinase Ctarget
FostamatinibTyrosine-protein kinase receptor UFOtarget
FostamatinibTyrosine-protein kinase Blktarget
FostamatinibBMP-2-inducible protein kinasetarget
FostamatinibBone morphogenetic protein receptor type-1Btarget
FostamatinibBone morphogenetic protein receptor type-2target
FostamatinibCytoplasmic tyrosine-protein kinase BMXtarget
FostamatinibSerine/threonine-protein kinase B-raftarget
FostamatinibTyrosine-protein kinase BTKtarget
FostamatinibCalcium/calmodulin-dependent protein kinase type 1target
FostamatinibCalcium/calmodulin-dependent protein kinase type 1Dtarget
FostamatinibMast/stem cell growth factor receptor Kittarget
FostamatinibCalcium/calmodulin-dependent protein kinase type II subunit alphatarget
FostamatinibCalcium/calmodulin-dependent protein kinase type II subunit betatarget
FostamatinibCalcium/calmodulin-dependent protein kinase type II subunit deltatarget
FostamatinibCalcium/calmodulin-dependent protein kinase type II subunit gammatarget
FostamatinibCalcium/calmodulin-dependent protein kinase kinase 1target
FostamatinibCalcium/calmodulin-dependent protein kinase kinase 2target
FostamatinibPeripheral plasma membrane protein CASKtarget
FostamatinibKappa-caseintarget
FostamatinibCyclin-dependent kinase 1target
FostamatinibSerine/threonine-protein kinase MRCK gammatarget
FostamatinibCyclin-dependent kinase 4target
FostamatinibCyclin-dependent kinase-like 1target
FostamatinibCyclin-dependent kinase-like 2target
FostamatinibSerine/threonine-protein kinase Chk1target
FostamatinibSerine/threonine-protein kinase Chk2target
FostamatinibCitron Rho-interacting kinasetarget
FostamatinibDual specificity protein kinase CLK1target
FostamatinibDual specificity protein kinase CLK2target
FostamatinibDual specificity protein kinase CLK3target
FostamatinibDual specificity protein kinase CLK4target
FostamatinibMacrophage colony-stimulating factor 1 receptortarget
FostamatinibTyrosine-protein kinase CSKtarget
FostamatinibCasein kinase I isoform alphatarget
FostamatinibCasein kinase II subunit alphatarget
FostamatinibCasein kinase II subunit alpha'target
FostamatinibDeath-associated protein kinase 1target
FostamatinibDeath-associated protein kinase 2target
FostamatinibDeath-associated protein kinase 3target
FostamatinibSerine/threonine-protein kinase DCLK1target
FostamatinibSerine/threonine-protein kinase DCLK2target
FostamatinibSerine/threonine-protein kinase DCLK3target
FostamatinibEpithelial discoidin domain-containing receptor 1target
FostamatinibDiscoidin domain-containing receptor 2target
FostamatinibDual specificity tyrosine-phosphorylation-regulated kinase 1Atarget
FostamatinibDual specificity tyrosine-phosphorylation-regulated kinase 1Btarget
FostamatinibEpidermal growth factor receptortarget
FostamatinibEukaryotic translation initiation factor 2-alpha kinase 1target
FostamatinibInterferon-induced, double-stranded RNA-activated protein kinasetarget
FostamatinibeIF-2-alpha kinase GCN2target
FostamatinibEphrin type-A receptor 1target
FostamatinibEphrin type-A receptor 2target
FostamatinibEphrin type-A receptor 3target
FostamatinibEphrin type-A receptor 4target
FostamatinibEphrin type-A receptor 5target
FostamatinibEphrin type-A receptor 6target
FostamatinibEphrin type-A receptor 7target
FostamatinibEphrin type-A receptor 8target
FostamatinibEphrin type-B receptor 1target
FostamatinibEphrin type-B receptor 2target
FostamatinibEphrin type-B receptor 4target
FostamatinibEphrin type-B receptor 6target
FostamatinibReceptor tyrosine-protein kinase erbB-2target
FostamatinibReceptor tyrosine-protein kinase erbB-4target
FostamatinibSerine/threonine-protein kinase/endoribonuclease IRE1target
FostamatinibTyrosine-protein kinase Fertarget
FostamatinibTyrosine-protein kinase Fes/Fpstarget
FostamatinibFibroblast growth factor receptor 1target
FostamatinibFibroblast growth factor receptor 2target
FostamatinibFibroblast growth factor receptor 3target
FostamatinibTyrosine-protein kinase Fgrtarget
FostamatinibVascular endothelial growth factor receptor 1target
FostamatinibReceptor-type tyrosine-protein kinase FLT3target
FostamatinibVascular endothelial growth factor receptor 3target
FostamatinibSerine/threonine-protein kinase mTORtarget
FostamatinibTyrosine-protein kinase FRKtarget
FostamatinibTyrosine-protein kinase Fyntarget
FostamatinibCyclin-G-associated kinasetarget
FostamatinibGlycogen synthase kinase-3 alphatarget
FostamatinibGlycogen synthase kinase-3 betatarget
FostamatinibTyrosine-protein kinase HCKtarget
FostamatinibHomeodomain-interacting protein kinase 2target
FostamatinibHomeodomain-interacting protein kinase 3target
FostamatinibSerine/threonine-protein kinase ICKtarget
FostamatinibInhibitor of nuclear factor kappa-B kinase subunit betatarget
FostamatinibInhibitor of nuclear factor kappa-B kinase subunit epsilontarget
FostamatinibInsulin receptortarget
FostamatinibInsulin receptor-related proteintarget
FostamatinibMitogen-activated protein kinase 14target
FostamatinibMitogen-activated protein kinase 15target
FostamatinibMitogen-activated protein kinase 4target
FostamatinibMitogen-activated protein kinase 7target
FostamatinibMitogen-activated protein kinase 9target
FostamatinibMAP kinase-activated protein kinase 5target
FostamatinibSerine/threonine-protein kinase MARK1target
FostamatinibSerine/threonine-protein kinase MARK2target
FostamatinibMAP/microtubule affinity-regulating kinase 3target
FostamatinibMAP/microtubule affinity-regulating kinase 4target
FostamatinibCLIP-associating protein 1target
FostamatinibMicrotubule-associated serine/threonine-protein kinase 1target
FostamatinibMegakaryocyte-associated tyrosine-protein kinasetarget
FostamatinibMaternal embryonic leucine zipper kinasetarget
FostamatinibTyrosine-protein kinase Mertarget
FostamatinibMisshapen-like kinase 1target
FostamatinibMAP kinase-interacting serine/threonine-protein kinase 1target
FostamatinibMAP kinase-interacting serine/threonine-protein kinase 2target
FostamatinibMacrophage-stimulating protein receptortarget
FostamatinibMuscle, skeletal receptor tyrosine-protein kinasetarget
FostamatinibMyosin light chain kinase, smooth muscletarget
FostamatinibMyosin light chain kinase 2, skeletal/cardiac muscletarget
FostamatinibMyosin light chain kinase 3target
FostamatinibMyosin light chain kinase family member 4target
FostamatinibMyosin-IIIatarget
FostamatinibSerine/threonine-protein kinase Nek1target
FostamatinibSerine/threonine-protein kinase Nek11target
FostamatinibSerine/threonine-protein kinase Nek2target
FostamatinibSerine/threonine-protein kinase Nek3target
FostamatinibSerine/threonine-protein kinase Nek4target
FostamatinibSerine/threonine-protein kinase Nek5target
FostamatinibSerine/threonine-protein kinase Nek9target
FostamatinibHigh affinity nerve growth factor receptortarget
FostamatinibBDNF/NT-3 growth factors receptortarget
FostamatinibNT-3 growth factor receptortarget
FostamatinibNUAK family SNF1-like kinase 1target
FostamatinibNUAK family SNF1-like kinase 2target
FostamatinibSerine/threonine-protein kinase OSR1target
FostamatinibSerine/threonine-protein kinase PAK 1target
FostamatinibSerine/threonine-protein kinase PAK 2target
FostamatinibSerine/threonine-protein kinase PAK 3target
FostamatinibSerine/threonine-protein kinase PAK 4target
FostamatinibSerine/threonine-protein kinase PAK 6target
FostamatinibSerine/threonine-protein kinase PAK 5target
FostamatinibCyclin-dependent kinase 16target
FostamatinibCyclin-dependent kinase 17target
FostamatinibPlatelet-derived growth factor receptor alphatarget
FostamatinibPlatelet-derived growth factor receptor betatarget
Fostamatinib3-phosphoinositide-dependent protein kinase 1target
FostamatinibCyclin-dependent kinase 15target
FostamatinibPhosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoformtarget
FostamatinibPhosphatidylinositol 4-kinase betatarget
FostamatinibPhosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit betatarget
FostamatinibPhosphatidylinositol 3-kinase C2 domain-containing subunit gammatarget
FostamatinibPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoformtarget
FostamatinibSerine/threonine-protein kinase LATS1target
FostamatinibSerine/threonine-protein kinase pim-1target
FostamatinibSerine/threonine-protein kinase pim-3target
FostamatinibPhosphatidylinositol 5-phosphate 4-kinase type-2 betatarget
FostamatinibPhosphatidylinositol 5-phosphate 4-kinase type-2 gammatarget
FostamatinibMembrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinasetarget
FostamatinibSerine/threonine-protein kinase N1target
FostamatinibSerine/threonine-protein kinase N2target
FostamatinibSerine/threonine-protein kinase PLK1target
FostamatinibSerine/threonine-protein kinase PLK2target
FostamatinibSerine/threonine-protein kinase PLK3target
FostamatinibSerine/threonine-protein kinase PLK4target
Fostamatinib5'-AMP-activated protein kinase catalytic subunit alpha-1target
Fostamatinib5'-AMP-activated protein kinasetarget
FostamatinibcAMP-dependent protein kinase catalytic subunit betatarget
FostamatinibProtein kinase C delta typetarget
FostamatinibProtein kinase C epsilon typetarget
FostamatinibProtein kinase C gamma typetarget
FostamatinibProtein kinase C iota typetarget
FostamatinibProtein kinase C theta typetarget
FostamatinibSerine/threonine-protein kinase D1target
FostamatinibcGMP-dependent protein kinase 2target
FostamatinibSerine/threonine-protein kinase PRP4 homologtarget
FostamatinibFocal adhesion kinase 1target
FostamatinibProtein-tyrosine kinase 2-betatarget
FostamatinibProtein-tyrosine kinase 6target
FostamatinibRAF proto-oncogene serine/threonine-protein kinasetarget
FostamatinibProto-oncogene tyrosine-protein kinase receptor Rettarget
FostamatinibSerine/threonine-protein kinase RIO1target
FostamatinibSerine/threonine-protein kinase RIO2target
FostamatinibSerine/threonine-protein kinase RIO3target
FostamatinibReceptor-interacting serine/threonine-protein kinase 1target
FostamatinibReceptor-interacting serine/threonine-protein kinase 2target
FostamatinibReceptor-interacting serine/threonine-protein kinase 4target
FostamatinibRho-associated protein kinase 2target
FostamatinibProto-oncogene tyrosine-protein kinase ROStarget
FostamatinibRibosomal protein S6 kinase alpha-1target
FostamatinibRibosomal protein S6 kinase alpha-3target
FostamatinibSerine/threonine-protein kinase SBK1target
FostamatinibUncharacterized serine/threonine-protein kinase SBK3target
FostamatinibSerine/threonine-protein kinase Sgk3target
FostamatinibSerine/threonine-protein kinase SIK1target
FostamatinibSerine/threonine-protein kinase SIK2target
FostamatinibSTE20-like serine/threonine-protein kinasetarget
FostamatinibSNF-related serine/threonine-protein kinasetarget
FostamatinibProto-oncogene tyrosine-protein kinase Srctarget
FostamatinibTyrosine-protein kinase Srmstarget
FostamatinibSerine/threonine-protein kinase 10target
FostamatinibSerine/threonine-protein kinase 16target
FostamatinibSerine/threonine-protein kinase 17Atarget
FostamatinibSerine/threonine-protein kinase 17Btarget
FostamatinibSerine/threonine-protein kinase 32Atarget
FostamatinibCytochrome P450 3A4enzyme
FostamatinibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
FostamatinibATP-binding cassette sub-family B member 5transporter
FostamatinibUDP-glucuronosyltransferase 1A9enzyme
FostamatinibMitogen-activated protein kinase 13target
FostamatinibMitogen-activated protein kinase 10target
FostamatinibMitogen-activated protein kinase kinase kinase kinase 5target
FostamatinibMitogen-activated protein kinase kinase kinase kinase 4target
FostamatinibMitogen-activated protein kinase kinase kinase kinase 3target
FostamatinibMitogen-activated protein kinase kinase kinase kinase 2target
FostamatinibMitogen-activated protein kinase kinase kinase kinase 1target
FostamatinibMitogen-activated protein kinase kinase kinase 9target
FostamatinibMitogen-activated protein kinase kinase kinase 6target
FostamatinibMitogen-activated protein kinase kinase kinase 4target
FostamatinibMitogen-activated protein kinase kinase kinase 3target
FostamatinibMitogen-activated protein kinase kinase kinase 2target
FostamatinibMitogen-activated protein kinase kinase kinase 15target
FostamatinibMitogen-activated protein kinase kinase kinase 13target
FostamatinibMitogen-activated protein kinase kinase kinase 12target
FostamatinibMitogen-activated protein kinase kinase kinase 11target
FostamatinibMitogen-activated protein kinase kinase kinase 10target
FostamatinibMitogen-activated protein kinase kinase kinase 1target
FostamatinibDual specificity mitogen-activated protein kinase kinase 6target
FostamatinibDual specificity mitogen-activated protein kinase kinase 5target
FostamatinibDual specificity mitogen-activated protein kinase kinase 3target
FostamatinibDual specificity mitogen-activated protein kinase kinase 2target
FostamatinibTyrosine-protein kinase Lyntarget
FostamatinibLeukocyte tyrosine kinase receptortarget
FostamatinibLeucine-rich repeat serine/threonine-protein kinase 2target
FostamatinibLIM domain kinase 2target
FostamatinibLIM domain kinase 1target
FostamatinibTyrosine-protein kinase Lcktarget
FostamatinibPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoformtarget
FurafyllineCytochrome P450 1A2enzyme
Fusidic acidSolute carrier organic anion transporter family member 1B1transporter
Fusidic acidBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
Fusidic acidUDP-glucuronosyltransferase 1A1enzyme
Fusidic acidCytochrome P450 3A4enzyme
Fusidic acidCytochrome P450 2D6enzyme
Fusidic acidElongation factor Gtarget
Fusidic acidATP-binding cassette sub-family C member 2transporter
Fusidic acidBile salt export pumptransporter
Fusidic acidChloramphenicol acetyltransferase 3target
Fusidic acidChloramphenicol acetyltransferasetarget
GarenoxacinDNA topoisomerase 2-alphatarget
GarenoxacinDNA topoisomerase 2-betatarget
GarenoxacinCytochrome P450 1A2enzyme
Garlic oilCytochrome P450 2E1enzyme
Garlic oilCytochrome P450 3A7enzyme
Garlic oilCytochrome P450 3A5enzyme
Garlic oilCytochrome P450 2C19enzyme
Garlic oilCytochrome P450 3A4enzyme
Garlic oilCytochrome P450 2C9enzyme
GatifloxacinDNA gyrase subunit Btarget
GatifloxacinAlbumincarrier
GatifloxacinDNA gyrase subunit Atarget
GatifloxacinDNA gyrase subunit Btarget
GatifloxacinDNA topoisomerase 4 subunit Atarget
GatifloxacinDNA topoisomerase 4 subunit Btarget
GatifloxacinDNA gyrase subunit Atarget
GatifloxacinCytochrome P450 1A2enzyme
GefitinibAlpha-1-acid glycoprotein 1carrier
GefitinibAlbumincarrier
GefitinibCytochrome P450 2C19enzyme
GefitinibCytochrome P450 2C9enzyme
GefitinibCytochrome P450 1A1enzyme
GefitinibCytochrome P450 3A5enzyme
GefitinibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
GefitinibATP-dependent translocase ABCB1transporter
GefitinibCytochrome P450 2D6enzyme
GefitinibCytochrome P450 3A4enzyme
GefitinibEpidermal growth factor receptortarget
GemfibrozilCytochrome P450 2C19enzyme
GemfibrozilCytochrome P450 1A2enzyme
GemfibrozilUDP-glucuronosyltransferase 2B17enzyme
GemfibrozilCytochrome P450 2C9enzyme
GemfibrozilPeroxisome proliferator-activated receptor alphatarget
GemfibrozilUDP-glucuronosyltransferase 1A1enzyme
GemfibrozilCytochrome P450 3A4enzyme
GemfibrozilUDP-glucuronosyltransferase 1A3enzyme
GemfibrozilSolute carrier organic anion transporter family member 1B1target
GemfibrozilUDP-glucuronosyltransferase 2B7enzyme
GemfibrozilUDP-glucuronosyltransferase 1A9enzyme
GemfibrozilUDP-glucuronosyltransferase 2B4enzyme
GemfibrozilLipoprotein lipasetarget
GemfibrozilSolute carrier organic anion transporter family member 1B3target
GemfibrozilSolute carrier organic anion transporter family member 2B1target
GemfibrozilOrganic anion transporter 3target
GemfibrozilAlbumincarrier
GemfibrozilCytochrome P450 2C8enzyme
GemifloxacinDNA gyrase subunit Btarget
GemifloxacinDNA gyrase subunit Atarget
GemifloxacinCytochrome P450 1A2enzyme
GemifloxacinDNA topoisomerase 4 subunit Atarget
GemifloxacinDNA gyrase subunit Atarget
GenisteinCytochrome P450 2C9enzyme
GenisteinCytochrome P450 3A1enzyme
GenisteinCytochrome P450 3A2enzyme
GenisteinCytochrome P450 3A4enzyme
GenisteinCystic fibrosis transmembrane conductance regulatortarget
GenisteinG protein-coupled estrogen receptor 1target
GenisteinCytochrome P450 2C8enzyme
GenisteinSolute carrier organic anion transporter family member 2B1transporter
GenisteinSolute carrier organic anion transporter family member 1B1transporter
GenisteinCytochrome P450 1A1enzyme
GenisteinSex hormone-binding globulintarget
GenisteinRAC-alpha serine/threonine-protein kinasetarget
GenisteinNuclear receptor subfamily 1 group I member 2target
GenisteinSteroid hormone receptor ERR1target
GenisteinSteroid hormone receptor ERR2target
GenisteinTransthyretincarrier
GenisteinCytochrome P450 1B1target
GenisteinNuclear receptor coactivator 2target
GenisteinEstrogen receptortarget
GenisteinNuclear receptor coactivator 1target
GenisteinCytochrome P450 1A2enzyme
GenisteinBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
GenisteinMultidrug resistance-associated protein 1transporter
GenisteinATP-dependent translocase ABCB1transporter
GenisteinProtein-tyrosine kinase 2-betatarget
GenisteinDNA topoisomerase 2-alphatarget
GenisteinEstrogen receptor betatarget
GestodeneCytochrome P450 2C19enzyme
GestodeneCytochrome P450 3A4enzyme
GestodeneProgesterone receptortarget
GestodeneCytochrome P450 3A7enzyme
GestodeneCytochrome P450 3A5enzyme
Ginkgo bilobaCytochrome P450 1A2enzyme
Ginkgo bilobaCytochrome P450 1A1enzyme
Ginkgo bilobaNitric oxide synthase, inducibletarget
Ginkgo bilobaAmine oxidase [flavin-containing] Atarget
Ginkgo bilobaCytochrome P450 3A4enzyme
Ginkgo bilobaGamma-aminobutyric acid receptor subunit gamma-2target
Ginkgo bilobaGamma-aminobutyric acid receptor subunit beta-2target
Ginkgo bilobaGamma-aminobutyric acid receptor subunit alpha-1target
Ginkgo bilobaGlycine receptor subunit alpha-1target
Ginkgo bilobaSodium-dependent noradrenaline transportertarget
Ginkgo bilobaPhospholipase A2, membrane associatedtarget
Ginkgo bilobaCytochrome P450 2C9enzyme
Ginkgo bilobaCytochrome P450 1B1enzyme
Ginsenoside CCytochrome P450 2C19target
Ginsenoside CCytochrome ctarget
Ginsenoside CTransforming growth factor beta-1 proproteintarget
GivinostatCytochrome P450 3A4enzyme
GivinostatTyrosine-protein kinase JAK2target
GivinostatHistone deacetylase 1target
GivinostatHistone deacetylasetarget
GivinostatCytochrome P450 1A2enzyme
GivinostatCytochrome P450 2B6enzyme
GivinostatSolute carrier family 22 member 2transporter
GlecaprevirCytochrome P450 3A Subfamilyenzyme
GlecaprevirUDP-glucuronosyltransferase 1A1enzyme
GlecaprevirATP-dependent translocase ABCB1transporter
GlecaprevirBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
GlecaprevirSolute carrier organic anion transporter family member 1B1transporter
GlecaprevirSolute carrier organic anion transporter family member 1B3transporter
GlecaprevirNS3 proteasetarget
GlecaprevirCytochrome P450 3A4enzyme
GlecaprevirGenome polyproteintarget
GlyburideMultidrug resistance-associated protein 1transporter
GlyburideTransient receptor potential cation channel subfamily M member 4target
GlyburideCytochrome P450 3A5enzyme
GlyburideCytochrome P450 3A7enzyme
GlyburideCarnitine O-palmitoyltransferase 1, liver isoformtarget
GlyburideMitochondrial ATP-sensitive potassium channeltarget
GlyburideAlbumincarrier
GlyburideCytochrome P450 3A4enzyme
GlyburideATP-binding cassette sub-family C member 9target
GlyburideBile salt export pumptarget
GlyburidePhospholipid-transporting ATPase ABCA1target
GlyburideCystic fibrosis transmembrane conductance regulatortarget
GlyburideSulfonylurea receptor 1, Kir6.2target
GlyburideCytochrome P450 2C9enzyme
GlyburideATP-binding cassette sub-family C member 3transporter
GlyburideBile salt export pumptransporter
GlyburideATP-dependent translocase ABCB1transporter
GlyburideATP-binding cassette sub-family C member 8target
GlyburideSolute carrier family 15 member 1transporter
GlyburideSolute carrier organic anion transporter family member 1A2transporter
GlyburideSolute carrier family 15 member 2transporter
GlyburideSolute carrier family 22 member 6transporter
GlyburideATP-binding cassette sub-family C member 2transporter
GlyburideBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
GlyburideSolute carrier family 22 member 7transporter
GlyburideSolute carrier organic anion transporter family member 2B1transporter
GlyburideCytochrome P450 2C19enzyme
Glycerol phenylbutyrate[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrialtarget
Glycerol phenylbutyrate[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrialtarget
Glycerol phenylbutyrate[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrialtarget
Glycerol phenylbutyrateMedium-chain specific acyl-CoA dehydrogenase, mitochondrialenzyme
Glycerol phenylbutyrateBile salt-activated lipaseenzyme
Glycerol phenylbutyratePancreatic lipase-related protein 2enzyme
Glycerol phenylbutyrateCytochrome P450 2D6enzyme
Glycerol phenylbutyrateCytochrome P450 3A4enzyme
Glycerol phenylbutyratePancreatic triacylglycerol lipaseenzyme
Glycerol phenylbutyrate[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 3, mitochondrialtarget
GoldensealCytochrome P450 2D6enzyme
GoldensealCytochrome P450 3A4enzyme
GoldensealCytochrome P450 1A2enzyme
GoldensealCytochrome P450 2E1enzyme
GoldensealCytochrome P450 2C19enzyme
GoldensealCytochrome P450 2C9enzyme
GoldensealThiamine transporter 2transporter
GoldensealThiamine transporter 1transporter
GoldensealCytochrome P450 3A Subfamilyenzyme
GPI-1485Peptidyl-prolyl cis-trans isomerase FKBP1Atarget
GPI-1485Cytochrome P450 3A4enzyme
GrapefruitCytochrome P450 3A4enzyme
GrazoprevirATP-dependent translocase ABCB1transporter
GrazoprevirSolute carrier organic anion transporter family member 1B1transporter
GrazoprevirSolute carrier organic anion transporter family member 1B3transporter
GrazoprevirCytochrome P450 3A4enzyme
GrazoprevirGenome polyproteintarget
GrazoprevirAlbumincarrier
GrazoprevirAlpha-1-acid glycoprotein 1carrier
GrazoprevirGag-Pol polyproteintarget
GrepafloxacinDNA gyrase subunit Btarget
GrepafloxacinDNA gyrase subunit Atarget
GrepafloxacinSolute carrier family 22 member 6transporter
GrepafloxacinMultidrug resistance-associated protein 1transporter
GrepafloxacinDNA gyrase subunit Atarget
GrepafloxacinDNA topoisomerase 4 subunit Atarget
GrepafloxacinCytochrome P450 1A2enzyme
GrepafloxacinSolute carrier family 22 member 2transporter
GrepafloxacinOrganic cation/carnitine transporter 2transporter
GrepafloxacinATP-binding cassette sub-family C member 2transporter
GrepafloxacinATP-dependent translocase ABCB1transporter
GrepafloxacinCytochrome P450 3A4enzyme
GuaiazulenCytochrome P450 2B1enzyme
GuaiazulenCytochrome P450 1A1enzyme
GuaiazulenCytochrome P450 1A2enzyme
HalofantrineCytochrome P450 2D6enzyme
HalofantrinePlasmepsin IItarget
HalofantrineVoltage-gated inwardly rectifying potassium channel KCNH2target
HalofantrineFe(II)-protoporphyrin IXtarget
HalofantrineCytochrome P450 2C8enzyme
HalofantrineCytochrome P450 3A5enzyme
HalofantrineCalmodulin-2target
HalofantrineCalmodulin-3target
HalofantrineCalmodulin-1target
HalofantrineCytochrome P450 3A4enzyme
HaloperidolSynaptic vesicular amine transportertarget
HaloperidolCytochrome P450 2C9enzyme
HaloperidolD(2) dopamine receptortarget
HaloperidolGlutamate receptor ionotropic, NMDA 2Btarget
HaloperidolD(1A) dopamine receptortarget
HaloperidolCytochrome P450 1A2enzyme
HaloperidolCytochrome P450 2D6enzyme
HaloperidolCytochrome P450 1A1enzyme
Haloperidol5-hydroxytryptamine receptor 7target
Haloperidol5-hydroxytryptamine receptor 6target
Haloperidol5-hydroxytryptamine receptor 1Atarget
HaloperidolAlpha-2C adrenergic receptortarget
HaloperidolAlpha-2B adrenergic receptortarget
HaloperidolAlpha-2A adrenergic receptortarget
HaloperidolAlpha-1A adrenergic receptortarget
HaloperidolMuscarinic acetylcholine receptor M3target
HaloperidolHistamine H1 receptortarget
HaloperidolSigma non-opioid intracellular receptor 1target
Haloperidol5-hydroxytryptamine receptor 2Ctarget
Haloperidol5-hydroxytryptamine receptor 2Atarget
HaloperidolMelanin-concentrating hormone receptor 1target
HaloperidolD(3) dopamine receptortarget
HaloperidolCytochrome P450 2C19enzyme
HaloperidolUDP-glucuronosyltransferase 1A9enzyme
HaloperidolCarbonyl reductase [NADPH] 1enzyme
HaloperidolATP-dependent translocase ABCB1transporter
HaloperidolCytochrome P450 3A7enzyme
HaloperidolCytochrome P450 3A5enzyme
HaloperidolCytochrome P450 3A4enzyme
Hippuric acidCarboxypeptidase A4enzyme
Hippuric acidAngiotensin-converting enzymeenzyme
Hippuric acidPeptidyl-glycine alpha-amidating monooxygenaseenzyme
Hippuric acidGlycine N-acyltransferaseenzyme
Hippuric acidAlbumincarrier
Hippuric acidCytochrome P450 3A4enzyme
Hippuric acidBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
Hippuric acidATP-binding cassette sub-family C member 4transporter
Hippuric acidCytochrome P450enzyme
HistamineSynaptic vesicular amine transportertarget
HistamineHistamine H4 receptortarget
HistamineOrganic cation/carnitine transporter 2transporter
HistamineSolute carrier family 22 member 3transporter
HistamineSolute carrier family 22 member 1transporter
HistamineSolute carrier family 22 member 2transporter
HistamineHistamine N-methyltransferaseenzyme
HistamineHistamine H3 receptortarget
HistamineHistamine H2 receptortarget
HistamineHistamine H1 receptortarget
HomochlorcyclizineHistamine H1 receptortarget
HomochlorcyclizineCytochrome P450 2D6enzyme
Human placenta hydrolysateCytochrome P450 2E1target
HydralazineAmine oxidase [copper-containing] 3target
HydralazineProlyl 4-hydroxylase subunit alpha-1target
HydralazineCytochrome P450 3A4enzyme
HydralazineAlbumincarrier
HydralazineHypoxia-inducible factor 1-alphatarget
HydrastineCytochrome P450 2E1enzyme
HydrastineCytochrome P450 2C9enzyme
HydrastineCytochrome P450 3A Subfamilyenzyme
HydrastineCytochrome P450 2D6enzyme
HydrastineCytochrome P450 3A4enzyme
HydrastineCytochrome P450 3A5enzyme
HydrastinineCytochrome P450 2D6enzyme
HydroxychloroquineCytochrome P450 2C8enzyme
HydroxychloroquineAngiotensin-converting enzyme 2target
HydroxychloroquineSolute carrier organic anion transporter family member 1A2transporter
HydroxychloroquineCytochrome P450 3A4enzyme
Hydroxychloroquinealpha1-acid glycoproteincarrier
HydroxychloroquineAlbumincarrier
HydroxychloroquineATP-dependent translocase ABCB1transporter
HydroxychloroquineCytochrome P450 2D6enzyme
HydroxychloroquineToll-like receptor 9target
HydroxychloroquineToll-like receptor 7target
HydroxychloroquineDNAtarget
HydroxyureaRibonucleoside-diphosphate reductase subunit M2target
HydroxyureaUrease subunit alphaenzyme
HydroxyureaAlbumincarrier
HydroxyureaOrganic cation/carnitine transporter 2transporter
HydroxyureaSolute carrier family 22 member 4transporter
HydroxyureaUrea transporter 1transporter
HydroxyureaUrea transporter 2transporter
HydroxyureaSolute carrier organic anion transporter family member 1B3transporter
HydroxyureaSolute carrier organic anion transporter family member 1B1transporter
HydroxyureaSolute carrier organic anion transporter family member 1A2transporter
HydroxyureaRibonucleoside-diphosphate reductase large subunittarget
HydroxyzineATP-dependent translocase ABCB1transporter
HydroxyzineVoltage-gated inwardly rectifying potassium channel KCNH2target
HydroxyzineHistamine H1 receptortarget
HydroxyzineCytochrome P450 2D6enzyme
HydroxyzineCytochrome P450 3A4enzyme
HydroxyzineCytochrome P450 3A5enzyme
HydroxyzineAlbumincarrier
IbrexafungerpUDP-glucuronosyltransferases (UGTs)enzyme
IbrexafungerpCytochrome P450 3A4enzyme
IbrexafungerpSulfotransferaseenzyme
IbrexafungerpCytochrome P450 2C8enzyme
IbrexafungerpATP-dependent translocase ABCB1transporter
IbrexafungerpSolute carrier organic anion transporter family member 1B3transporter
IbrexafungerpAlbumincarrier
Ibrexafungerp1,3-beta-glucan synthase component GSC2target
IbrexafungerpGTP-binding protein RHO1target
IbuprofenSolute carrier family 22 member 11transporter
IbuprofenSolute carrier organic anion transporter family member 2B1transporter
IbuprofenATP-dependent translocase ABCB1transporter
IbuprofenUDP-glucuronosyltransferase 1A3enzyme
IbuprofenUDP-glucuronosyltransferase 1A9enzyme
IbuprofenUDP-glucuronosyltransferase 2B4enzyme
IbuprofenUDP-glucuronosyltransferase 2B7enzyme
IbuprofenCytochrome P450 2C8enzyme
IbuprofenCytochrome P450 2C19enzyme
IbuprofenApoptosis regulator Bcl-2target
IbuprofenThrombomodulintarget
IbuprofenFatty acid-binding protein, intestinaltarget
IbuprofenPeroxisome proliferator-activated receptor gammatarget
IbuprofenCystic fibrosis transmembrane conductance regulatortarget
IbuprofenPeroxisome proliferator-activated receptor alphatarget
IbuprofenPlatelet glycoprotein Ib alpha chaintarget
IbuprofenProtein S100-A7target
IbuprofenAlpha-methylacyl-CoA racemaseenzyme
IbuprofenCytochrome P450 3A4enzyme
IbuprofenC-X-C chemokine receptor type 1target
IbuprofenC-X-C chemokine receptor type 2target
IbuprofenInterleukin-8target
IbuprofenHuman Cyclooxygenasestarget
IbuprofenSolute carrier organic anion transporter family member 1A2transporter
IbuprofenMultidrug resistance-associated protein 1transporter
IbuprofenSolute carrier family 22 member 6transporter
IbuprofenATP-binding cassette sub-family C member 4transporter
IbuprofenAlbumincarrier
IbuprofenCytochrome P450 2C9enzyme
IbuprofenProstaglandin G/H synthase 2target
IbuprofenProstaglandin G/H synthase 1target
IbuprofenOrganic anion transporter 3transporter
IdelalisibUDP-glucuronosyltransferase 1A4enzyme
IdelalisibCytochrome P450 3A4enzyme
IdelalisibCytochrome P450 3A7enzyme
IdelalisibCytochrome P450 3A43enzyme
IdelalisibCytochrome P450 3A5enzyme
IdelalisibSolute carrier organic anion transporter family member 1B1transporter
IdelalisibSolute carrier organic anion transporter family member 1B3transporter
IdelalisibPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoformtarget
IdelalisibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
IdelalisibATP-dependent translocase ABCB1transporter
IdelalisibAldehyde oxidaseenzyme
IdelalisibCytochrome P450 2C8enzyme
IdelalisibCytochrome P450 2C19enzyme
IdelalisibCytochrome P450 2B6enzyme
IfosfamideCytochrome P450 2B6enzyme
IfosfamideDNAtarget
IfosfamideCytochrome P450 3A4enzyme
IfosfamideCytochrome P450 3A5enzyme
IfosfamideCytochrome P450 2C8enzyme
IfosfamideCytochrome P450 2A6enzyme
IfosfamideCytochrome P450 2C19enzyme
IfosfamideCytochrome P450 2C18enzyme
IfosfamideProstaglandin G/H synthase 1enzyme
IfosfamideNuclear receptor subfamily 1 group I member 2target
IfosfamideCytochrome P450 2C9enzyme
ImatinibATP-binding cassette sub-family C member 2transporter
ImatinibBile salt export pumptransporter
ImatinibEpithelial discoidin domain-containing receptor 1target
ImatinibCytochrome P450 3A4enzyme
ImatinibBreakpoint cluster region proteintarget
ImatinibCytochrome P450 1A2enzyme
ImatinibCytochrome P450 2D6enzyme
ImatinibCytochrome P450 2C9enzyme
ImatinibCytochrome P450 2C19enzyme
ImatinibInduced myeloid leukemia cell differentiation protein Mcl-1target
ImatinibDiscoidin domain-containing receptor 2target
ImatinibSolute carrier organic anion transporter family member 1A2transporter
ImatinibATP-binding cassette sub-family C member 4transporter
ImatinibSolute carrier organic anion transporter family member 1B3transporter
ImatinibOrganic cation/carnitine transporter 2transporter
ImatinibMultidrug resistance-associated protein 1transporter
ImatinibCytochrome P450 3A5enzyme
ImatinibCytochrome P450 2C8enzyme
ImatinibPlatelet-derived growth factor receptor alphatarget
ImatinibAlpha-1-acid glycoprotein 1carrier
ImatinibAlbumincarrier
ImatinibPhospholipid-transporting ATPase ABCA3transporter
ImatinibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
ImatinibSolute carrier family 22 member 2transporter
ImatinibATP-dependent translocase ABCB1transporter
ImatinibSolute carrier family 22 member 1transporter
ImatinibCytochrome P450 3A7enzyme
ImatinibMacrophage colony-stimulating factor 1 receptortarget
ImatinibPlatelet-derived growth factor receptor betatarget
ImatinibTyrosine-protein kinase ABL1target
ImatinibMast/stem cell growth factor receptor Kittarget
ImatinibProto-oncogene tyrosine-protein kinase receptor Rettarget
ImipramineCytochrome P450 2B6enzyme
ImipramineCytochrome P450 2C18enzyme
ImipramineCytochrome P450 2E1enzyme
ImipramineCytochrome P450 3A7enzyme
Imipramine5-hydroxytryptamine receptor 2Ctarget
ImipramineAlpha-1B adrenergic receptortarget
Imipramine5-hydroxytryptamine receptor 7target
ImipramineD(1) dopamine receptortarget
ImipramineD(2) dopamine receptortarget
ImipramineVoltage-gated inwardly rectifying potassium channel KCNH2target
ImipramineCytochrome P450 3A4enzyme
ImipramineSodium-dependent dopamine transportertarget
Imipramine5-hydroxytryptamine receptor 1Atarget
Imipramine5-hydroxytryptamine receptor 6target
ImipramineSolute carrier family 22 member 4transporter
ImipramineVoltage-gated delayed rectifier potassium channel KCNH1target
ImipramineAlbumincarrier
ImipramineSolute carrier family 22 member 3transporter
ImipramineSolute carrier family 22 member 2transporter
ImipramineAlpha-1-acid glycoprotein 1carrier
ImipramineAlpha-1D adrenergic receptortarget
ImipramineA-type voltage-gated potassium channel KCND3target
ImipramineA-type voltage-gated potassium channel KCND2target
ImipramineMuscarinic acetylcholine receptor M5target
ImipramineMuscarinic acetylcholine receptor M4target
ImipramineMuscarinic acetylcholine receptor M3target
ImipramineMuscarinic acetylcholine receptor M2target
ImipramineATP-dependent translocase ABCB1transporter
ImipramineMuscarinic acetylcholine receptor M1target
Imipramine5-hydroxytryptamine receptor 2Atarget
ImipramineAlpha-1A adrenergic receptortarget
ImipramineHistamine H1 receptortarget
ImipramineCytochrome P450 2D6enzyme
ImipramineCytochrome P450 2C19enzyme
ImipramineSodium-dependent noradrenaline transportertarget
ImipramineSodium-dependent serotonin transportertarget
ImipramineCytochrome P450 1A2enzyme
ImlunestrantUDP-glucuronosyltransferase 1A9enzyme
ImlunestrantUDP-glucuronosyltransferase 1A10enzyme
ImlunestrantUDP-glucuronosyltransferase 1A3enzyme
ImlunestrantUDP-glucuronosyltransferase 1A1enzyme
ImlunestrantBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
ImlunestrantATP-dependent translocase ABCB1transporter
ImlunestrantCytochrome P450 2C9enzyme
ImlunestrantCytochrome P450 2B6enzyme
ImlunestrantCytochrome P450 3A4enzyme
ImlunestrantEstrogen receptortarget
ImlunestrantUDP-glucuronosyltransferase 1A8enzyme
IndalpineSodium-dependent serotonin transportertarget
IndalpineCytochrome P450 3A4enzyme
IndinavirCytochrome P450 3A4enzyme
IndinavirCytochrome P450 3A5enzyme
IndinavirCytochrome P450 3A7enzyme
IndinavirPol polyproteintarget
IndinavirSolute carrier family 22 member 1transporter
IndinavirMultidrug resistance-associated protein 1transporter
IndinavirSolute carrier organic anion transporter family member 1A2transporter
IndinavirSolute carrier organic anion transporter family member 1B1transporter
IndinavirATP-binding cassette sub-family C member 2transporter
IndinavirCytochrome P450 2D6enzyme
IndinavirUDP-glucuronosyltransferase 1A1enzyme
IndinavirSolute carrier organic anion transporter family member 2B1transporter
IndinavirBile salt export pumptransporter
IndinavirGag-Pol polyproteintarget
IndinavirATP-dependent translocase ABCB1transporter
IndisulamCarbonic anhydrase 9target
IndisulamCytochrome P450 2D6enzyme
IndisulamCytochrome P450 2E1enzyme
IndisulamCytochrome P450 3A4enzyme
IndisulamCytochrome P450 2C9enzyme
IndomethacinUDP-glucuronosyltransferase 2B7enzyme
IndomethacinPeroxisome proliferator-activated receptor alphatarget
IndomethacinAldo-keto reductase family 1 member C3target
IndomethacinSolute carrier organic anion transporter family member 1B1transporter
IndomethacinBile salt export pumptransporter
IndomethacinInterferon-induced, double-stranded RNA-activated protein kinasetarget
IndomethacinHuman Cyclooxygenasestarget
IndomethacinLiver carboxylesterase 1enzyme
IndomethacinUDP-glucuronosyltransferase 1A1enzyme
IndomethacinCytochrome P450 2C9enzyme
IndomethacinSolute carrier family 22 member 7transporter
IndomethacinHepatic sodium/bile acid cotransportertransporter
IndomethacinSolute carrier family 22 member 11transporter
IndomethacinATP-binding cassette sub-family C member 11transporter
IndomethacinATP-binding cassette sub-family C member 2transporter
IndomethacinOrganic anion transporter 3transporter
IndomethacinSolute carrier family 22 member 6transporter
IndomethacinSolute carrier organic anion transporter family member 1A2transporter
IndomethacinMultidrug resistance-associated protein 1transporter
IndomethacinATP-dependent translocase ABCB1transporter
IndomethacinATP-binding cassette sub-family C member 4transporter
IndomethacinATP-binding cassette sub-family C member 6transporter
IndomethacinATP-binding cassette sub-family C member 3transporter
IndomethacinAlbumincarrier
IndomethacinPeroxisome proliferator-activated receptor gammatarget
IndomethacinProstaglandin D2 receptor 2target
IndomethacinLactoylglutathione lyasetarget
IndomethacinProstaglandin reductase 2target
IndomethacinPhospholipase A2, membrane associatedtarget
IndomethacinUDP-glucuronosyltransferase 1A9enzyme
IndomethacinCytochrome P450 2C19enzyme
IndomethacinProstaglandin G/H synthase 2target
IndomethacinProstaglandin G/H synthase 1target
Interferon alfaInterferon alpha/beta receptor 1target
Interferon alfaCytochrome P450 1A2enzyme
Interferon alfa-2aInterferon alpha/beta receptor 1target
Interferon alfa-2aInterferon alpha/beta receptor 2target
Interferon alfa-2aCytochrome P450 1A2enzyme
Interferon alfa-2bInterferon alpha-2target
Interferon alfa-2bCytochrome P450 1A2enzyme
Interferon alfa-2bInterferon alpha/beta receptor 2target
Interferon alfa-2bInterferon alpha/beta receptor 1target
Interferon alfa-2cInterferon alpha/beta receptor (IFNAR)target
Interferon alfa-2cCytochrome P450 1A2enzyme
Interferon alfa-n1Interferon alpha/beta receptor 2target
Interferon alfa-n1Interferon alpha/beta receptor 1target
Interferon alfa-n1Cytochrome P450 1A2enzyme
Interferon alfa-n3Interferon alpha/beta receptor 1target
Interferon alfa-n3Interferon alpha/beta receptor 2target
Interferon alfa-n3Cytochrome P450 1A2enzyme
Interferon alfacon-1Interferon alpha/beta receptor 1target
Interferon alfacon-1Interferon alpha/beta receptor 2target
Interferon alfacon-1Cytochrome P450 1A2enzyme
Interferon beta-1aInterferon alpha/beta receptor 1target
Interferon beta-1aInterferon alpha/beta receptor 2target
Interferon beta-1aCytochrome P450 1A2enzyme
Interferon beta-1aInterferon betatarget
Interferon beta-1bInterferon alpha/beta receptor 1target
Interferon beta-1bInterferon alpha/beta receptor 2target
Interferon beta-1bCytochrome P450 1A2enzyme
Interferon gamma-1bInterferon gamma receptor 1target
Interferon gamma-1bCytochrome P450 1A2enzyme
Interferon gamma-1bInterferon gamma receptor 2target
IpriflavoneAcetylcholinesterasetarget
IpriflavoneCytochrome P450 1A2enzyme
IpriflavoneCytochrome P450 2C8enzyme
IpriflavoneCytochrome P450 2C19enzyme
IpriflavoneCytochrome P450 2C9enzyme
IproniazidMonoamine oxidasetarget
IproniazidAmine oxidase [flavin-containing] Btarget
IproniazidAmine oxidase [flavin-containing] Atarget
IproniazidAmine oxidase [flavin-containing] Aenzyme
IproniazidCytochrome P450 2C9enzyme
IproniazidCytochrome P450 2D6enzyme
IproniazidAmine oxidase [flavin-containing] Benzyme
IrbesartanType-1 angiotensin II receptortarget
IrbesartanTranscription factor Juntarget
IrbesartanCytochrome P450 2C9enzyme
IrbesartanCytochrome P450 2C8enzyme
IrbesartanUDP-glucuronosyltransferase 1A3enzyme
IrbesartanProstaglandin G/H synthase 1enzyme
IrbesartanCytochrome P450 3A4enzyme
IrbesartanAlbumincarrier
Irbesartanalpha1-acid glycoproteincarrier
IrinotecanCytochrome P450 3A7enzyme
IrinotecanDNA topoisomerase I, mitochondrialtarget
IrinotecanDNA topoisomerase 1target
IrinotecanCytochrome P450 3A4enzyme
IrinotecanCytochrome P450 3A5enzyme
IrinotecanUDP-glucuronosyltransferase 1A1enzyme
IrinotecanUDP-glucuronosyltransferase 1A9enzyme
IrinotecanSolute carrier family 22 member 3transporter
IrinotecanSolute carrier organic anion transporter family member 1B1transporter
IrinotecanMultidrug resistance-associated protein 1transporter
IrinotecanBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
IrinotecanAlbumincarrier
IrinotecanATP-dependent translocase ABCB1transporter
IrinotecanATP-binding cassette sub-family C member 2transporter
IrinotecanHuman Carboxylesterasesenzyme
IsavuconazoleSodium channel protein type 5 subunit alphatarget
IsavuconazolePotassium voltage-gated channel subfamily KQT member 1target
IsavuconazoleA-type voltage-gated potassium channel KCND3target
IsavuconazoleCytochrome P450 3A5enzyme
IsavuconazoleCytochrome P450 2C8enzyme
IsavuconazoleCytochrome P450 2C9enzyme
IsavuconazoleCytochrome P450 2C19enzyme
IsavuconazoleCytochrome P450 2D6enzyme
IsavuconazoleCytochrome P450 2B6enzyme
IsavuconazoleUDP-glucuronosyltransferase 1A9enzyme
IsavuconazoleUDP-glucuronosyltransferase 1A8enzyme
IsavuconazoleATP-dependent translocase ABCB1transporter
IsavuconazoleBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
IsavuconazoleSolute carrier family 22 member 2transporter
IsavuconazoleLanosterol 14-alpha demethylasetarget
IsavuconazoleVoltage-gated inwardly rectifying potassium channel KCNH2target
IsavuconazoleVoltage-dependent L-type calcium channel subunit alpha-1Ctarget
IsavuconazoleG protein-activated inward rectifier potassium channel 2target
IsavuconazoleG protein-activated inward rectifier potassium channel 3target
IsavuconazoleATP-sensitive inward rectifier potassium channel 11target
IsavuconazolePotassium voltage-gated channel subfamily A member 5target
IsavuconazoleCytochrome P450 3A4enzyme
IsavuconazoniumAlbumincarrier
IsavuconazoniumCytochrome P450 2C9enzyme
IsavuconazoniumLanosterol 14-alpha demethylasetarget
IsavuconazoniumSolute carrier family 22 member 2transporter
IsavuconazoniumBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
IsavuconazoniumCytochrome P450 2B6enzyme
IsavuconazoniumCytochrome P450 2D6enzyme
IsavuconazoniumCytochrome P450 2C19enzyme
IsavuconazoniumCytochrome P450 2C8enzyme
IsavuconazoniumCholinesteraseenzyme
IsavuconazoniumCytochrome P450 3A5enzyme
IsavuconazoniumATP-dependent translocase ABCB1transporter
IsavuconazoniumCytochrome P450 3A4enzyme
IsoliquiritigeninAldo-keto reductase family 1 member B1target
IsoliquiritigeninCystic fibrosis transmembrane conductance regulatortarget
IsoliquiritigeninCytochrome P450 3A4enzyme
IsoliquiritigeninNACHT, LRR and PYD domains-containing protein 3target
IsoniazidCatalase-peroxidasetarget
IsoniazidCytochrome P450 2A6enzyme
IsoniazidCytochrome P450 3A4enzyme
IsoniazidAlbumincarrier
IsoniazidDihydrofolate reductasetarget
IsoniazidCytochrome P450 2C8enzyme
IsoniazidArylamine N-acetyltransferaseenzyme
IsoniazidArylamine N-acetyltransferase 2enzyme
IsoniazidCytochrome P450 2C19enzyme
IsoniazidCytochrome P450 2D6enzyme
IsoniazidEnoyl-[acyl-carrier-protein] reductase [NADH]target
IsoniazidCytochrome P450 2E1enzyme
IsoniazidCytochrome P450 1A2enzyme
IsoniazidCytochrome P450 2C9enzyme
Isosorbide dinitrateCytochrome P450 2E1enzyme
Isosorbide dinitrateAtrial natriuretic peptide receptor 1target
IsradipineVoltage-dependent calcium channel subunit alpha-2/delta-2target
IsradipineVoltage-dependent L-type calcium channel subunit alpha-1Starget
IsradipineVoltage-dependent T-type calcium channel subunit alpha-1Htarget
IsradipineCytochrome P450 3A4enzyme
IsradipineVoltage-dependent L-type calcium channel subunit alpha-1Ctarget
IsradipineVoltage gated L-type calcium channeltarget
IsradipineBile salt export pumptransporter
IsradipineVoltage-dependent calcium channel subunit alpha-2/delta-1target
IsradipineVoltage-dependent L-type calcium channel subunit alpha-1Dtarget
IsradipineVoltage-dependent L-type calcium channel subunit beta-2target
ItraconazoleCytochrome P450 3A4enzyme
ItraconazoleSolute carrier organic anion transporter family member 2B1transporter
ItraconazoleLanosterol 14-alpha demethylasetarget
ItraconazoleLanosterol 14-alpha demethylasetarget
ItraconazoleAlbumincarrier
ItraconazoleCytochrome P450 2E1enzyme
ItraconazoleBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
ItraconazoleCytochrome P450 3A Subfamilyenzyme
ItraconazoleCytochrome P450 1A1enzyme
ItraconazoleATP-dependent translocase ABCB1transporter
ItraconazoleCytochrome P450 2B6enzyme
ItraconazoleCytochrome P450 3A7enzyme
ItraconazoleCytochrome P450 3A5enzyme
IvacaftorCytochrome P450 2C9enzyme
IvacaftorCytochrome P450 3A5enzyme
IvacaftorATP-dependent translocase ABCB1transporter
IvacaftorAlpha-1-acid glycoprotein 1carrier
IvacaftorAlbumincarrier
IvacaftorCytochrome P450 3A4enzyme
IvacaftorCystic fibrosis transmembrane conductance regulatortarget
JPC-3210Cytochrome P450 3A4enzyme
JPC-3210Cytochrome P450 2D6enzyme
KavaCytochrome P450 2C9enzyme
KavaATP-dependent translocase ABCB1transporter
KavaLiver carboxylesterase 1enzyme
KavaNuclear receptor subfamily 1 group I member 2target
KavaNuclear factor NF-kappa-B complextarget
KavaCytochrome P450 2C19enzyme
KavaCytochrome P450 3A4enzyme
KavaCytochrome P450 2D6enzyme
KavaCytochrome P450 1A2enzyme
KavaCytochrome P450 2E1enzyme
KavaAmine oxidase [flavin-containing] Atarget
KavaAmine oxidase [flavin-containing] Btarget
KetazolamGABA(A) Receptor Benzodiazepine Binding Sitetarget
KetazolamGABA(A) Receptortarget
KetazolamAlbumincarrier
KetazolamATP-dependent translocase ABCB1transporter
KetazolamCytochrome P450 3A4enzyme
KetoconazoleCytochrome P450 3A4enzyme
KetoconazoleCytochrome P450 11B1, mitochondrialenzyme
KetoconazoleATP-dependent translocase ABCB1transporter
KetoconazoleBile salt export pumptransporter
KetoconazoleCytochrome P450 2D6enzyme
KetoconazoleCytochrome P450 1A1enzyme
KetoconazoleCytochrome P450 2C8enzyme
KetoconazoleCytochrome P450 1A2enzyme
KetoconazoleCytochrome P450 3A5enzyme
KetoconazoleCytochrome P450 2C19enzyme
KetoconazoleCytochrome P450 2C9enzyme
KetoconazoleCytochrome P450 1B1enzyme
KetoconazoleCytochrome P450 2A6enzyme
KetoconazoleCytochrome P450 2B6enzyme
KetoconazoleLanosterol 14-alpha demethylasetarget
KetoconazoleAndrogen receptortarget
KetoconazoleSteroid 17-alpha-hydroxylase/17,20 lyasetarget
KetoconazoleSteroid 21-hydroxylasetarget
KetoconazoleVoltage-gated inwardly rectifying potassium channel KCNH2target
KetoconazoleNuclear receptor subfamily 1 group I member 2target
KetoconazoleNuclear receptor subfamily 1 group I member 3target
KetoconazoleUDP-glucuronosyltransferase 1A1enzyme
KetoconazoleUDP-glucuronosyltransferase 2B7enzyme
KetoconazoleSolute carrier organic anion transporter family member 1B1transporter
KetoconazoleCytochrome P450 4F12enzyme
KetoconazoleCytochrome P450 4F2enzyme
KetoconazoleAlbumincarrier
KetoconazoleSex hormone-binding globulincarrier
KetoconazoleAromataseenzyme
KetoconazoleUDP-glucuronosyltransferase 1A7enzyme
KetoconazoleLanosterol 14-alpha demethylasetarget
KetoprofenProstaglandin G/H synthase 2target
KetoprofenProstaglandin G/H synthase 1target
KetoprofenC-X-C chemokine receptor type 1target
KetoprofenAlbumincarrier
KetoprofenATP-binding cassette sub-family C member 4transporter
KetoprofenSolute carrier organic anion transporter family member 1A2transporter
KetoprofenSolute carrier family 22 member 6transporter
KetoprofenOrganic anion transporter 3transporter
KetoprofenSolute carrier family 22 member 11transporter
KetoprofenSolute carrier family 22 member 7transporter
KetoprofenCytochrome P450 2C9enzyme
KetoprofenCytochrome P450 2C8enzyme
KetoprofenUDP-glucuronosyltransferase 1A1enzyme
KetoprofenHuman Cyclooxygenasestarget
KitasamycinCytochrome P450 3A4enzyme
KitasamycinE3 ubiquitin-protein ligase HUWE1target
KOS-1584Cytochrome P450 3A4enzyme
LabetalolAlpha-1 adrenergic receptorstarget
LabetalolBeta-1 adrenergic receptortarget
LabetalolBeta-2 adrenergic receptortarget
LabetalolCytochrome P450 2D6enzyme
LabetalolCytochrome P450 2C19enzyme
LabetalolAlbumincarrier
Labetalolalpha1-acid glycoproteincarrier
LabetalolATP-binding cassette sub-family B member 5transporter
LabetalolUDP-glucuronosyltransferase 1A1enzyme
LabetalolUDP-glucuronosyltransferase 2B7enzyme
LabetalolUDP-glucuronosyltransferase 1A9enzyme
LandiololCytochrome P450 2D6enzyme
LandiololBeta-1 adrenergic receptortarget
LandiololBeta-2 adrenergic receptortarget
LandiololCholinesteraseenzyme
LandiololHuman Carboxylesterasesenzyme
LanreotideCytochrome P450 3A4enzyme
LanreotideSomatostatin receptor type 5target
LanreotideSomatostatin receptor type 2target
LansoprazolePotassium-transporting ATPase alpha chain 1target
LansoprazoleCytochrome P450 2C19enzyme
LansoprazoleCytochrome P450 2C9enzyme
LansoprazoleCytochrome P450 3A4enzyme
LansoprazoleATP-dependent translocase ABCB1transporter
LansoprazoleBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
LansoprazoleCytochrome P450 1A1enzyme
LansoprazoleCytochrome P450 1B1enzyme
LansoprazoleCytochrome P450 2C18enzyme
LansoprazoleCytochrome P450 2C8enzyme
LansoprazoleCytochrome P450 2D6enzyme
LansoprazoleMicrotubule-associated protein tautarget
LansoprazoleOrganic anion transporter 3transporter
LansoprazoleSolute carrier family 22 member 1transporter
LansoprazoleSolute carrier family 22 member 2transporter
LansoprazoleSolute carrier family 22 member 3transporter
LapatinibEukaryotic elongation factor 2 kinasetarget
LapatinibEpidermal growth factor receptortarget
LapatinibReceptor tyrosine-protein kinase erbB-2target
LapatinibCytochrome P450 3A4enzyme
LapatinibCytochrome P450 2C8enzyme
LapatinibATP-dependent translocase ABCB1transporter
LapatinibAntigen peptide transporter 1transporter
LapatinibCytochrome P450 3A5enzyme
LapatinibCytochrome P450 2C19enzyme
LaromustineCytochrome P450 2B6enzyme
LaromustineMethylated-DNA--protein-cysteine methyltransferasetarget
LaromustineCytochrome P450 3A4enzyme
LaromustineCytochrome P450 2C19enzyme
LaromustineGlutathione reductase, mitochondrialtarget
LaromustineDNA polymerase betatarget
LasmiditanCytochrome P450 2D6enzyme
LasmiditanMultidrug and toxin extrusion protein 2transporter
LasmiditanMultidrug and toxin extrusion protein 1transporter
LasmiditanSolute carrier family 22 member 1transporter
LasmiditanBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
LasmiditanATP-dependent translocase ABCB1transporter
Lasmiditan5-hydroxytryptamine receptor 1Ftarget
LazertinibGlutathione S-transferase Mu 1enzyme
LazertinibCytochrome P450 3A4enzyme
LazertinibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
LazertinibUDP-glucuronosyltransferase 1A1enzyme
LazertinibEpidermal growth factor receptortarget
LazertinibSolute carrier family 22 member 1transporter
LeflunomideCytochrome P450 1A2enzyme
LeflunomideDihydroorotate dehydrogenase (quinone), mitochondrialtarget
LeflunomideCytochrome P450 2C9enzyme
LeflunomideAryl hydrocarbon receptortarget
LeflunomideProtein-tyrosine kinase 2-betatarget
LeflunomideBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
LeflunomideDihydroorotate dehydrogenase (quinone), mitochondrialtarget
LemborexantATP-dependent translocase ABCB1transporter
LemborexantCytochrome P450 2B6enzyme
LemborexantCytochrome P450 3A Subfamilyenzyme
LemborexantCytochrome P450 3A5enzyme
LemborexantCytochrome P450 3A4enzyme
LemborexantOrexin receptor type 2target
LemborexantOrexin/Hypocretin receptor type 1target
LenacapavirGag-Pol polyproteintarget
LenacapavirATP-dependent translocase ABCB1transporter
LenacapavirUDP-glucuronosyltransferase 1A1enzyme
LenacapavirCytochrome P450 3A4enzyme
LenacapavirGag-Pol polyproteintarget
LeniolisibCytochrome P450 1A2enzyme
LeniolisibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
LeniolisibSolute carrier organic anion transporter family member 1B1transporter
LeniolisibCytochrome P450 2D6enzyme
LeniolisibCytochrome P450 1A1enzyme
LeniolisibCytochrome P450 3A5enzyme
LeniolisibCytochrome P450 3A4enzyme
LeniolisibPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoformtarget
LeniolisibATP-dependent translocase ABCB1transporter
LeniolisibSolute carrier organic anion transporter family member 1B3transporter
LenvatinibCytochrome P450 2B6enzyme
LenvatinibCytochrome P450 1A2enzyme
LenvatinibCytochrome P450 2C9enzyme
LenvatinibCytochrome P450 2C8enzyme
LenvatinibAldehyde oxidaseenzyme
LenvatinibCytochrome P450 3A4enzyme
LenvatinibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
LenvatinibATP-dependent translocase ABCB1transporter
LenvatinibMast/stem cell growth factor receptor Kittarget
LenvatinibProto-oncogene tyrosine-protein kinase receptor Rettarget
LenvatinibPlatelet-derived growth factor receptor alphatarget
LenvatinibFibroblast growth factor receptor 4target
LenvatinibFibroblast growth factor receptor 3target
LenvatinibFibroblast growth factor receptor 2target
LenvatinibFibroblast growth factor receptor 1target
LenvatinibVascular endothelial growth factor receptor 3target
LenvatinibVascular endothelial growth factor receptor 2target
LenvatinibVascular endothelial growth factor receptor 1target
LenvatinibVascular endothelial growth factor receptortarget
LenvatinibSolute carrier organic anion transporter family member 1B3transporter
LenvatinibCytochrome P450 2D6enzyme
LenvatinibBile salt export pumptransporter
LenvatinibSolute carrier organic anion transporter family member 1B1transporter
LenvatinibSolute carrier family 22 member 2transporter
LenvatinibOrganic anion transporter 3transporter
LenvatinibSolute carrier family 22 member 6transporter
LenvatinibCytochrome P450 2C19enzyme
LercanidipineVoltage-dependent calcium channel gamma-1 subunittarget
LercanidipineCytochrome P450 3A4enzyme
LercanidipineCytochrome P450 3A5enzyme
LercanidipineCytochrome P450 3A7enzyme
LercanidipineCytochrome P450 2D6enzyme
LercanidipineVoltage-dependent calcium channel subunit alpha-2/delta-1target
LercanidipineVoltage gated L-type calcium channeltarget
LestaurtinibProto-oncogene tyrosine-protein kinase receptor Rettarget
LestaurtinibNT-3 growth factor receptortarget
LestaurtinibBDNF/NT-3 growth factors receptortarget
LestaurtinibHigh affinity nerve growth factor receptortarget
LestaurtinibTyrosine-protein kinase JAK2target
LestaurtinibCytochrome P450 3A4enzyme
LestaurtinibReceptor-type tyrosine-protein kinase FLT3target
LetermovirUDP-glucuronosyltransferase 1A1enzyme
LetermovirUDP-glucuronosyltransferase 1A3enzyme
LetermovirSolute carrier organic anion transporter family member 1B1transporter
LetermovirSolute carrier organic anion transporter family member 1B3transporter
LetermovirCytochrome P450 2D6enzyme
LetermovirCytochrome P450 2C8enzyme
LetermovirCytochrome P450 2C19enzyme
LetermovirCytochrome P450 2C9enzyme
LetermovirCytochrome P450 2B6enzyme
LetermovirATP-dependent translocase ABCB1transporter
LetermovirBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
LetermovirBile salt export pumptransporter
LetermovirOrganic anion transporter 3transporter
LetermovirATP-binding cassette sub-family C member 2transporter
LetermovirCMV DNA Terminase Complextarget
LetermovirCytochrome P450 3A Subfamilyenzyme
LetrozoleUDP-glucuronosyltransferase 2B7enzyme
LetrozoleAromatasetarget
LetrozoleCytochrome P450 3A4enzyme
LetrozoleCytochrome P450 2A6enzyme
LetrozoleAromataseenzyme
LetrozoleCytochrome P450 2C19enzyme
LetrozoleAlbumincarrier
LetrozoleATP-dependent translocase ABCB1transporter
LevofloxacinMultidrug and toxin extrusion protein 1transporter
LevofloxacinMultidrug and toxin extrusion protein 2transporter
LevofloxacinCytochrome P450 2C9enzyme
LevofloxacinAlbumincarrier
LevofloxacinSolute carrier organic anion transporter family member 4C1transporter
LevofloxacinSolute carrier family 22 member 1transporter
LevofloxacinSolute carrier organic anion transporter family member 1A2transporter
LevofloxacinDNA gyrase subunit Atarget
LevofloxacinDNA gyrase subunit Btarget
LevofloxacinATP-dependent translocase ABCB1transporter
LevofloxacinSolute carrier family 22 member 2transporter
LevofloxacinDNA topoisomerase 4 subunit Atarget
LevofloxacinDNA gyrase subunit Atarget
LevofloxacinSolute carrier family 22 member 4transporter
LevoketoconazoleCytochrome P450 7A1enzyme
LevoketoconazoleCytochrome P450 1A2enzyme
LevoketoconazoleCytochrome P450 2C8enzyme
LevoketoconazoleCytochrome P450 2B6enzyme
LevoketoconazoleMultidrug and toxin extrusion protein 1transporter
LevoketoconazoleSolute carrier family 22 member 2transporter
LevoketoconazoleCholesterol side-chain cleavage enzyme, mitochondrialtarget
LevoketoconazoleAromataseenzyme
LevoketoconazoleSteroid 17-alpha-hydroxylase/17,20 lyasetarget
LevoketoconazoleATP-dependent translocase ABCB1transporter
LevoketoconazoleSteroid 21-hydroxylaseenzyme
LevoketoconazoleCytochrome P450 3A5enzyme
LevoketoconazoleCytochrome P450 3A4enzyme
LevoketoconazoleLanosterol 14-alpha demethylasetarget
LevoketoconazoleCytochrome P450 11B1, mitochondrialtarget
LevoketoconazoleCytochrome P450 11B2, mitochondrialtarget
LevosalbutamolBeta-2 adrenergic receptortarget
LevosalbutamolSolute carrier organic anion transporter family member 1B1transporter
LevosalbutamolSolute carrier organic anion transporter family member 1B3transporter
LevothyroxineThyroid hormone receptor alphatarget
LevothyroxineLarge neutral amino acids transporter small subunit 1transporter
LevothyroxineThyroid hormone receptor betatarget
LevothyroxineCytochrome P450 2C8enzyme
LevothyroxineTransthyretincarrier
LevothyroxineAlbumincarrier
LevothyroxineThyroxine-binding globulincarrier
LevothyroxineATP-dependent translocase ABCB1transporter
LevothyroxineMonocarboxylate transporter 8transporter
LevothyroxineSolute carrier organic anion transporter family member 1C1transporter
LevothyroxineSolute carrier organic anion transporter family member 1A2transporter
LevothyroxineSolute carrier organic anion transporter family member 1B1transporter
LevothyroxineSolute carrier organic anion transporter family member 4A1transporter
LevothyroxineATP-dependent translocase ABCB1enzyme
LevothyroxineIntegrin beta-3target
LevothyroxineIntegrin alpha-Vtarget
LevothyroxineSolute carrier organic anion transporter family member 2B1transporter
LevothyroxineUDP-glucuronosyltransferase 1A1enzyme
LicofelonePolyunsaturated fatty acid 5-lipoxygenasetarget
LicofeloneProstaglandin G/H synthase 2target
LicofeloneGroup IIE secretory phospholipase A2target
LicofeloneCytochrome P450 2C9enzyme
LicofeloneCytochrome P450 2C8enzyme
LicofeloneCytochrome P450 2J2enzyme
LicofeloneUDP-glucuronosyltransferase 1A3enzyme
LidocaineAlpha-1-acid glycoprotein 2target
LidocaineSodium channel protein type 5 subunit alphatarget
LidocaineVoltage-gated sodium channel alpha subunittarget
LidocaineSodium channel protein type 11 subunit alphatarget
LidocaineAlpha-1-acid glycoprotein 1target
LidocaineSodium channel protein type 10 subunit alphatarget
LidocaineEpidermal growth factor receptortarget
LidocaineSodium channel protein type 9 subunit alphatarget
LidocaineCytochrome P450 1A2enzyme
LidocaineCytochrome P450 2D6enzyme
LidocaineCytochrome P450 3A4enzyme
LidocaineCytochrome P450 3A5enzyme
LidocaineCytochrome P450 3A7enzyme
LidocaineOrganic cation/carnitine transporter 2transporter
LidocaineATP-dependent translocase ABCB1transporter
LidocaineCytochrome P450 2A6enzyme
LidocaineCytochrome P450 2B6enzyme
LidocaineCytochrome P450 2C8enzyme
LidocaineCytochrome P450 2C9enzyme
LidocaineSodium channel protein type 4 subunit alphatarget
LifitegrastSolute carrier organic anion transporter family member 2B1transporter
LifitegrastIntercellular adhesion molecule 1target
LifitegrastIntegrin alpha-Ltarget
LifitegrastCytochrome P450 2C9enzyme
LifitegrastSolute carrier organic anion transporter family member 1A2transporter
LimnetrelvirCytochrome P450 3A4enzyme
LimnetrelvirReplicase polyprotein 1abtarget
LinagliptinDipeptidyl peptidase 4target
LinagliptinCytochrome P450 3A4enzyme
LinagliptinSolute carrier family 22 member 3transporter
LinagliptinSolute carrier family 22 member 2transporter
LinagliptinSolute carrier family 22 member 1transporter
LinagliptinATP-dependent translocase ABCB1transporter
LinerixibatIleal sodium/bile acid cotransportertarget
LinerixibatCytochrome P450 3A4enzyme
LinerixibatSolute carrier organic anion transporter family member 1B1transporter
LinerixibatSolute carrier organic anion transporter family member 1B3transporter
LinzagolixSolute carrier family 22 member 6transporter
LinzagolixBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
LinzagolixOrganic anion transporter 3transporter
LinzagolixSolute carrier organic anion transporter family member 1B3transporter
LinzagolixSolute carrier organic anion transporter family member 1B1transporter
LinzagolixCytochrome P450 3A4enzyme
LinzagolixCytochrome P450 2C9enzyme
LinzagolixAlbumincarrier
LinzagolixGonadotropin-releasing hormone receptortarget
LinzagolixCytochrome P450 2C8enzyme
LiotrixThyroid hormone receptor alphatarget
LiotrixThyroid hormone receptor betatarget
LiotrixCytochrome P450 2C8enzyme
LiotrixSolute carrier organic anion transporter family member 1A2transporter
LiotrixSolute carrier organic anion transporter family member 1B1transporter
LiotrixSolute carrier organic anion transporter family member 1B3transporter
LiotrixSolute carrier organic anion transporter family member 4C1transporter
LiotrixHepatic sodium/bile acid cotransportertransporter
LiotrixSolute carrier organic anion transporter family member 1C1transporter
LiotrixSolute carrier organic anion transporter family member 4A1transporter
LiotrixOrganic anion transporter 3transporter
LiotrixMonocarboxylate transporter 8transporter
LiotrixMonocarboxylate transporter 10transporter
LiotrixTransthyretincarrier
LiotrixThyroxine-binding globulincarrier
LiotrixAlbumincarrier
LiotrixCytochrome P450 3A4enzyme
LiotrixATP-dependent translocase ABCB1transporter
LobeglitazoneCytochrome P450 1A2enzyme
LobeglitazoneATP-dependent translocase ABCB1transporter
LobeglitazoneSolute carrier organic anion transporter family member 3A1transporter
LobeglitazoneSolute carrier organic anion transporter family member 1B1transporter
LobeglitazoneCytochrome P450 2C9enzyme
LobeglitazoneCytochrome P450 2C19enzyme
LobeglitazonePeroxisome proliferator-activated receptor gammatarget
LobeglitazoneCytochrome P450 3A4enzyme
LobeglitazoneCytochrome P450 2C8enzyme
LobeglitazonePeroxisome proliferator-activated receptor alphatarget
LomefloxacinDNA topoisomerase 4 subunit Atarget
LomefloxacinDNA gyrase subunit Atarget
LomefloxacinDNA topoisomerase 2-alphatarget
LomefloxacinCytochrome P450 1A2enzyme
LomefloxacinOrganic cation/carnitine transporter 2transporter
LomefloxacinATP-binding cassette sub-family C member 2transporter
LomefloxacinDNA topoisomerase 2-betatarget
LomitapideATP-dependent translocase ABCB1transporter
LomitapideCytochrome P450 3A4enzyme
LomitapideMicrosomal triglyceride transfer protein large subunittarget
LomustineDNAtarget
LomustineCytochrome P450 3A4enzyme
LomustineCytochrome P450 2D6enzyme
LomustineStathmin-4target
LonafarnibCytochrome P450 1A2enzyme
LonafarnibCytochrome P450 2E1enzyme
LonafarnibCytochrome P450 2C19enzyme
LonafarnibCytochrome P450 2C8enzyme
LonafarnibCytochrome P450 3A Subfamilyenzyme
LonafarnibProtein farnesyltransferase subunit betatarget
LonafarnibATP-dependent translocase ABCB1transporter
LonafarnibProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alphatarget
LonafarnibCytochrome P450 2A6enzyme
LonafarnibCytochrome P450 2C9enzyme
LonafarnibSolute carrier organic anion transporter family member 1B1transporter
LonafarnibSolute carrier organic anion transporter family member 1B3transporter
LonafarnibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
LonafarnibATP-binding cassette sub-family C member 2transporter
LonafarnibCytochrome P450 3A5enzyme
LonafarnibCytochrome P450 3A4enzyme
Lonapegsomatropin11-beta-hydroxysteroid dehydrogenase 1enzyme
LonapegsomatropinGrowth hormone receptortarget
LonapegsomatropinProlactin receptortarget
LonapegsomatropinCytochrome P450 1A2enzyme
LonapegsomatropinCytochrome P450 2C19enzyme
LonapegsomatropinATP-dependent translocase ABCB1transporter
LoperamideCalmodulintarget
LoperamideVoltage-gated inwardly rectifying potassium channel KCNH2target
LoperamideCytochrome P450 2D6enzyme
LoperamideCytochrome P450 2B6enzyme
LoperamideCytochrome P450 2C8enzyme
LoperamideKappa-type opioid receptortarget
LoperamideATP-dependent translocase ABCB1transporter
LoperamideCytochrome P450 3A4enzyme
LoperamideDelta-type opioid receptortarget
LoperamidePro-opiomelanocortintarget
LoperamideMu-type opioid receptortarget
LoperamideVoltage-dependent P/Q-type calcium channel subunit alpha-1Atarget
LopinavirAlbumincarrier
LopinavirAlpha-1-acid glycoprotein 1carrier
LopinavirCytochrome P450 1A2enzyme
LopinavirBile salt export pumptransporter
LopinavirSolute carrier organic anion transporter family member 1B3transporter
LopinavirSolute carrier organic anion transporter family member 1B1transporter
LopinavirCytochrome P450 3A Subfamilyenzyme
LopinavirCytochrome P450 2C9enzyme
LopinavirCytochrome P450 2B6enzyme
LopinavirATP-dependent translocase ABCB1transporter
LopinavirCytochrome P450 2C19enzyme
LopinavirCytochrome P450 2D6enzyme
LopinavirCytochrome P450 3A4enzyme
LopinavirPol polyproteintarget
LoratadineUDP-glucuronosyltransferase 2B15enzyme
LoratadineUDP-glucuronosyltransferase 1A3enzyme
LoratadineUDP-glucuronosyltransferase 1A1enzyme
LoratadineUDP-glucuronosyltransferase 2B10enzyme
LoratadineCytochrome P450 3A5enzyme
LoratadineCytochrome P450 2C9enzyme
LoratadineCytochrome P450 1A2enzyme
LoratadineCytochrome P450 1A1enzyme
LoratadineBile salt export pumptransporter
LoratadineVoltage-gated inwardly rectifying potassium channel KCNH2target
LoratadineATP-dependent translocase ABCB1transporter
LoratadineCytochrome P450 2C8enzyme
LoratadineCytochrome P450 2D6enzyme
LoratadineCytochrome P450 2C19enzyme
LoratadineCytochrome P450 3A4enzyme
LoratadineHistamine H1 receptortarget
LoratadineCytochrome P450 2B6enzyme
LorcaserinCytochrome P450 2C19enzyme
LorcaserinCytochrome P450 2D6enzyme
LorcaserinCytochrome P450 3A4enzyme
LorcaserinCytochrome P450 2B6enzyme
LorcaserinCytochrome P450 1A1enzyme
LorcaserinCytochrome P450 2A6enzyme
LorcaserinCytochrome P450 1A2enzyme
Lorcaserin5-hydroxytryptamine receptor 2Ctarget
LorcaserinFlavin-containing monooxygenase 1enzyme
LorlatinibTyrosine-protein kinase Fertarget
LorlatinibTyrosine-protein kinase STYK1target
LorlatinibProto-oncogene tyrosine-protein kinase ROStarget
LorlatinibCytochrome P450 3A4enzyme
LorlatinibUDP-glucuronosyltransferase 1A3enzyme
LorlatinibCytochrome P450 2C19enzyme
LorlatinibCytochrome P450 2C8enzyme
LorlatinibCytochrome P450 2B6enzyme
LorlatinibCytochrome P450 3A5enzyme
LorlatinibCytochrome P450 3A Subfamilyenzyme
LorlatinibALK tyrosine kinase receptortarget
LorlatinibTyrosine-protein kinase Fes/Fpstarget
LorlatinibHigh affinity nerve growth factor receptortarget
LorlatinibBDNF/NT-3 growth factors receptortarget
LorlatinibNT-3 growth factor receptortarget
LorlatinibFocal adhesion kinase 1target
LorlatinibProtein-tyrosine kinase 2-betatarget
LorlatinibActivated CDC42 kinase 1target
Lorvotuzumab mertansineCytochrome P450 3A4enzyme
Lorvotuzumab mertansineNeural cell adhesion molecule 1target
LosartanUDP-glucuronosyltransferase 1A1enzyme
LosartanUDP-glucuronosyltransferase 1A3enzyme
LosartanSolute carrier family 22 member 6transporter
LosartanATP-dependent translocase ABCB1transporter
LosartanCytochrome P450 2C9enzyme
LosartanCytochrome P450 3A4enzyme
LosartanType-1 angiotensin II receptortarget
LosartanUDP-glucuronosyltransferase 1A10enzyme
LosartanUDP-glucuronosyltransferase 2B7enzyme
LosartanUDP-glucuronosyltransferase 2B17enzyme
LosartanCytochrome P450 2C19enzyme
LosartanAlbumincarrier
LosartanSolute carrier family 22 member 12transporter
LosartanSolute carrier family 2, facilitated glucose transporter member 9transporter
LosartanBile salt export pumptransporter
LosartanErythropoietin receptortarget
LosartanCytochrome P450 2C8enzyme
LuliconazoleLanosterol 14-alpha demethylasetarget
LuliconazoleCytochrome P450 2C19enzyme
LuliconazoleCytochrome P450 3A4enzyme
LumacaftorCytochrome P450 2B6enzyme
LumacaftorCytochrome P450 2C9enzyme
LumacaftorCytochrome P450 2C19enzyme
LumacaftorAlbumincarrier
LumacaftorCystic fibrosis transmembrane conductance regulatortarget
LumacaftorCytochrome P450 3A4enzyme
LumacaftorATP-dependent translocase ABCB1transporter
LumacaftorCytochrome P450 2C8enzyme
LumasiranHydroxyacid oxidase 1 mRNAtarget
LumasiranCytochrome P450 2C8enzyme
LumasiranAlbumincarrier
LumefantrineSodium/potassium-transporting ATPase subunit alpha-1target
LumefantrineCytochrome P450 3A4enzyme
LumefantrineCytochrome P450 2D6enzyme
LynestrenolCytochrome P450 3A4enzyme
LynestrenolCytochrome P450 2C9enzyme
LynestrenolEstrogen receptortarget
LynestrenolCytochrome P450 2C19enzyme
LynestrenolProgesterone receptortarget
Madecassic acidCytochrome P450 3A4enzyme
Madecassic acidCytochrome P450 2D6enzyme
Madecassic acidCytochrome P450 2C9enzyme
Madecassic acidPeroxisome proliferator-activated receptor gammatarget
Madecassic acidAcetylcholinesterasetarget
MafosfamideCytochrome P450 3A4enzyme
MafosfamideAldehyde dehydrogenase 1A1enzyme
MafosfamideAldehyde dehydrogenase, dimeric NADP-preferringenzyme
ManidipineVoltage-dependent L-type calcium channeltarget
ManidipineVoltage-dependent T-type calcium channeltarget
ManidipineCytochrome P450 2C9enzyme
ManidipineCytochrome P450 2D6enzyme
ManidipineCytochrome P450 1A1enzyme
ManidipineCytochrome P450 2B6enzyme
ManidipineCytochrome P450 2C19enzyme
ManidipineCytochrome P450 3A4enzyme
ManidipineVoltage-dependent T-type calcium channel subunit alpha-1Gtarget
ManidipineVoltage-dependent T-type calcium channel subunit alpha-1Htarget
ManidipineVoltage-dependent T-type calcium channel subunit alpha-1Itarget
ManidipineVoltage-dependent L-type calcium channel subunit alpha-1Dtarget
ManidipineVoltage-dependent L-type calcium channel subunit alpha-1Ctarget
ManidipineCruzipaintarget
ManidipineVoltage gated L-type calcium channeltarget
MaralixibatIleal sodium/bile acid cotransportertarget
MaralixibatSolute carrier organic anion transporter family member 2B1transporter
MaralixibatCytochrome P450 3A4enzyme
MaralixibatHepatic sodium/bile acid cotransportertarget
MavorixaforCytochrome P450 2C19enzyme
MavorixaforCytochrome P450 3A5enzyme
MavorixaforCytochrome P450 2D6enzyme
MavorixaforCytochrome P450 3A4enzyme
MavorixaforC-X-C chemokine receptor type 4target
MavorixaforCytochrome P450 1A2enzyme
MavorixaforCytochrome P450 2B6enzyme
MavorixaforCytochrome P450 2C8enzyme
MavorixaforCytochrome P450 2C9enzyme
MavorixaforATP-dependent translocase ABCB1transporter
MavorixaforMultidrug and toxin extrusion protein 1transporter
MavorixaforSolute carrier family 22 member 2transporter
Medical CannabisDelta-type opioid receptortarget
Medical CannabisNeuronal acetylcholine receptor subunit alpha-7target
Medical Cannabis5-hydroxytryptamine receptor 2Atarget
Medical Cannabis5-hydroxytryptamine receptor 1Atarget
Medical CannabisG protein-coupled receptor 55target
Medical CannabisN-arachidonyl glycine receptortarget
Medical CannabisGlycine receptor subunit alpha-3target
Medical CannabisGlycine receptor (alpha-1/beta)target
Medical CannabisGlycine receptor subunit alpha-1target
Medical CannabisG protein-coupled receptor 12target
Medical CannabisCytochrome P450 3A4enzyme
Medical CannabisCytochrome P450 2D6enzyme
Medical CannabisCytochrome P450 2C19enzyme
Medical CannabisCytochrome P450 2C9enzyme
Medical CannabisCannabinoid receptor 2target
Medical CannabisCannabinoid receptor 1target
Medical CannabisMu-type opioid receptortarget
Medical CannabisPeroxisome proliferator-activated receptor gammatarget
Medical CannabisCytochrome P450 3A5enzyme
Medical CannabisCytochrome P450 3A7enzyme
Medical CannabisCytochrome P450 1A1enzyme
Medical CannabisCytochrome P450 1A2enzyme
Medical CannabisCytochrome P450 1B1enzyme
Medical CannabisPolyunsaturated fatty acid 5-lipoxygenaseenzyme
Medical CannabisPolyunsaturated fatty acid lipoxygenase ALOX15enzyme
Medical CannabisSuperoxide dismutase [Cu-Zn]enzyme
Medical CannabisMultidrug resistance-associated protein 1transporter
Medical CannabisBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
Medical CannabisEquilibrative nucleoside transporter 1transporter
Medical CannabisTransient receptor potential cation channel subfamily V member 1target
Medical CannabisVoltage-dependent T-type calcium channel subunit alpha-1Gtarget
Medical CannabisVoltage-dependent T-type calcium channel subunit alpha-1Htarget
Medical CannabisVoltage-dependent T-type calcium channel subunit alpha-1Itarget
Medical CannabisTransient receptor potential cation channel subfamily A member 1target
Medical CannabisTransient receptor potential cation channel subfamily M member 8target
Medical CannabisTransient receptor potential cation channel subfamily V member 2target
Medical CannabisTransient receptor potential cation channel subfamily V member 3target
Medical CannabisTransient receptor potential cation channel subfamily V member 4target
Medical CannabisNon-selective voltage-gated ion channel VDAC1target
Medical CannabisN-acyl-phosphatidylethanolamine-hydrolyzing phospholipase Dtarget
Medical CannabisN-acylethanolamine-hydrolyzing acid amidasetarget
Medical CannabisSerotonin N-acetyltransferasetarget
Medical CannabisPhospholipase A2target
Medical CannabisSuperoxide dismutase [Cu-Zn]target
Medical CannabisFatty-acid amide hydrolase 1target
Medical CannabisCatalasetarget
Medical CannabisZeta-crystallintarget
Medical CannabisSphingomyelin phosphodiesterasetarget
Medical CannabisGlutathione peroxidase 1target
Medical CannabisGlutathione reductase, mitochondrialtarget
Medical Cannabis3-hydroxy-3-methylglutaryl-coenzyme A reductasetarget
Medical CannabisIndoleamine 2,3-dioxygenase 1target
Medical CannabisProstaglandin G/H synthase 1target
Medical CannabisProstaglandin G/H synthase 2target
Medical CannabisSteroid 17-alpha-hydroxylase/17,20 lyasetarget
Medical CannabisAcetyl-CoA acetyltransferase, mitochondrialtarget
Medical CannabisCytochrome P450 2A6enzyme
Medical CannabisCytochrome P450 2B6enzyme
Medical CannabisCytochrome P450 2C8enzyme
Medical CannabisCytochrome P450 2E1enzyme
Medical CannabisUDP-glucuronosyltransferase 2B7enzyme
Medical CannabisATP-dependent translocase ABCB1transporter
Medical CannabisLiver carboxylesterase 1enzyme
Medical CannabisUDP-glucuronosyltransferase 2B17enzyme
Medical CannabisUDP-glucuronosyltransferase 1A10enzyme
Medical CannabisUDP-glucuronosyltransferase 1A9enzyme
Medical CannabisUDP-glucuronosyltransferase 1A8enzyme
Medical CannabisUDP-glucuronosyltransferase 1A7enzyme
Medical CannabisCytochrome P450 2J2enzyme
Medroxyprogesterone acetateATP-dependent translocase ABCB1transporter
Medroxyprogesterone acetateGABA(A) Receptortarget
Medroxyprogesterone acetateATP-dependent translocase ABCB1target
Medroxyprogesterone acetateAlbumincarrier
Medroxyprogesterone acetateCytochrome P450 3A1enzyme
Medroxyprogesterone acetateCytochrome P450 2C9enzyme
Medroxyprogesterone acetate3 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 2enzyme
Medroxyprogesterone acetateCytochrome P450 2C8enzyme
Medroxyprogesterone acetateCytochrome P450 3A4enzyme
Medroxyprogesterone acetateEstrogen receptortarget
Medroxyprogesterone acetateProgesterone receptortarget
Mefenamic acidProstaglandin G/H synthase 2target
Mefenamic acidProstaglandin G/H synthase 1target
Mefenamic acidCytochrome P450 2C9enzyme
Mefenamic acidCytochrome P450 2C8enzyme
Mefenamic acidAlbumincarrier
Mefenamic acidUDP-glucuronosyltransferase 1A9enzyme
Mefenamic acidCytochrome P450 1A2enzyme
Mefenamic acidUDP-glucuronosyltransferase 2B7enzyme
Mefenamic acidHuman Cyclooxygenasestarget
MefloquineCholinesteraseenzyme
MefloquineCytochrome P450 3A4enzyme
MefloquineAdenosine receptor A2atarget
MefloquineFe(II)-protoporphyrin IXtarget
MefloquineATP-dependent translocase ABCB1transporter
MefloquineAromataseenzyme
MefloquineAcetylcholinesteraseenzyme
Mefloquine80S ribosomal subunittarget
MelperoneCytochrome P450 2D6enzyme
MelperoneD(2) dopamine receptortarget
Memantine5-hydroxytryptamine receptor 3Atarget
MemantineNeuronal acetylcholine receptor subunit alpha-7target
MemantineCytochrome P450 2A6enzyme
MemantineCytochrome P450 2C19enzyme
MemantineD(2) dopamine receptortarget
MemantineGlutamate receptor ionotropic, NMDA 1target
MemantineSodium/hydrogen exchanger 1transporter
MemantineSolute carrier family 22 member 2transporter
MemantineCytochrome P450 2B6enzyme
MemantineSolute carrier family 22 member 4transporter
MemantineMultidrug and toxin extrusion protein 1transporter
MemantineGlutamate (NMDA) receptortarget
MemantineGABA(A) Receptortarget
MenadioneCytochrome P450 3A7enzyme
MenadioneCytochrome P450 3A5enzyme
MenadioneCytochrome P450 3A4enzyme
MenadioneCytochrome P450 2E1enzyme
MenadioneCytochrome P450 2D6enzyme
MenadioneCytochrome P450 2C19enzyme
MenadioneCytochrome P450 2C9enzyme
MenadioneProthrombintarget
MenadioneVitamin K epoxide reductase complex subunit 1target
MenadioneCoagulation factor IXtarget
MenadioneVitamin K-dependent gamma-carboxylasetarget
MenadioneVitamin K-dependent protein Ctarget
MenadioneVitamin K-dependent protein Starget
MenadioneNAD(P)H dehydrogenase [quinone] 1target
MenadioneRibosyldihydronicotinamide dehydrogenase [quinone]target
MenadioneCytochrome P450 2C8enzyme
MenadioneCytochrome P450 2B6enzyme
MenadioneCytochrome P450 1B1enzyme
MenadioneCytochrome P450 2A6enzyme
MenadioneCytochrome P450 1A2enzyme
MenadioneOsteocalcintarget
MenadioneCytochrome P450 1A1enzyme
MenadioneVitamin K epoxide reductase complex subunit 1-like protein 1target
MenadioneAldehyde oxidasetarget
MenadioneXanthine dehydrogenase/oxidaseenzyme
MenadioneAldehyde oxidaseenzyme
MenadioneMethylenetetrahydrofolate reductase (NADPH)enzyme
MephenytoinCytochrome P450 2C9enzyme
MephenytoinCytochrome P450 2C19enzyme
MephenytoinCytochrome P450 1A2enzyme
MephenytoinCytochrome P450 2D6enzyme
MephenytoinCytochrome P450 2C8enzyme
MephenytoinNuclear receptor subfamily 1 group I member 2target
MephenytoinThyroxine-binding globulincarrier
MephenytoinVoltage-gated sodium channel alpha subunittarget
MephenytoinSodium channel protein type 5 subunit alphatarget
MephenytoinCytochrome P450 2B6enzyme
MepyramineCytochrome P450 2D6enzyme
MepyramineHistamine H1 receptortarget
MepyramineSolute carrier family 22 member 4transporter
MepyramineOrganic cation/carnitine transporter 2transporter
MequitazineHistamine H1 receptortarget
MequitazineCytochrome P450 2D6enzyme
MequitazineCytochrome P450 3A4enzyme
MetacetamolCytochrome P450 2E1enzyme
MetacetamolGlyceraldehyde-3-phosphate dehydrogenasetarget
MethadoneCytochrome P450 2C9enzyme
MethadoneCytochrome P450 2C18enzyme
MethadoneCytochrome P450 1A2enzyme
MethadoneAromataseenzyme
MethadoneCytochrome P450 2C8enzyme
MethadoneATP-dependent translocase ABCB1transporter
MethadoneCytochrome P450 2D6enzyme
MethadoneCytochrome P450 3A7enzyme
MethadoneDelta-type opioid receptortarget
MethadoneCytochrome P450 2C19enzyme
MethadoneCytochrome P450 3A4enzyme
MethadoneCytochrome P450 2B6enzyme
MethadoneMu-type opioid receptortarget
MethadoneNMDA receptortarget
MethadoneNeuronal acetylcholine receptor subunit alpha-7target
MethadoneNeuronal acetylcholine receptor subunit alpha-3target
MethadoneAlbumincarrier
MethadoneNeuronal acetylcholine receptor subunit alpha-4target
MethadoneNeuronal acetylcholine receptor subunit beta-2target
MethadoneCytochrome P450 3A Subfamilyenzyme
MethadoneUDP-glucuronosyltransferase 2B4enzyme
MethadoneAlpha-1-acid glycoprotein 1carrier
Methadone5-hydroxytryptamine receptor 3Atarget
MethimazoleThyroid peroxidasetarget
MethimazoleCytochrome P450 1A2enzyme
MethimazoleCytochrome P450 2A6enzyme
MethimazoleCytochrome P450 2B6enzyme
MethimazoleCytochrome P450 2C19enzyme
MethimazoleCytochrome P450 2C9enzyme
MethimazoleCytochrome P450 2D6enzyme
MethimazoleCytochrome P450 2E1enzyme
MethimazoleCytochrome P450 3A4enzyme
MethimazoleFlavin-containing monooxygenase 3enzyme
MethotrimeprazineMuscarinic acetylcholine receptor M1target
MethotrimeprazineD(1A) dopamine receptortarget
Methotrimeprazine5-hydroxytryptamine receptor 2Atarget
MethotrimeprazineAlpha-2C adrenergic receptortarget
MethotrimeprazineAlpha-2B adrenergic receptortarget
MethotrimeprazineAlpha-2A adrenergic receptortarget
MethotrimeprazineD(4) dopamine receptortarget
MethotrimeprazineD(1B) dopamine receptortarget
MethotrimeprazineCytochrome P450 2E1enzyme
MethotrimeprazineD(2) dopamine receptortarget
MethotrimeprazineCytochrome P450 2D6enzyme
MethotrimeprazineAlpha-1D adrenergic receptortarget
MethotrimeprazineAlpha-1B adrenergic receptortarget
MethotrimeprazineAlpha-1A adrenergic receptortarget
MethotrimeprazineMuscarinic acetylcholine receptor M5target
MethotrimeprazineMuscarinic acetylcholine receptor M4target
MethotrimeprazineMuscarinic acetylcholine receptor M3target
MethotrimeprazineMuscarinic acetylcholine receptor M2target
MethotrimeprazineHistamine H1 receptortarget
MethotrimeprazineD(3) dopamine receptortarget
Methotrimeprazine5-hydroxytryptamine receptor 2Ctarget
MethoxsalenDNAtarget
MethoxsalenCytochrome P450 2A6enzyme
MethoxsalenCytochrome P450 1A2enzyme
MethoxsalenCytochrome P450 1A1enzyme
MethoxsalenCytochrome P450 2A13enzyme
MethoxsalenCytochrome P450 2A6target
MethsuximideCytochrome P450 2C19enzyme
MethsuximideVoltage-dependent T-type calcium channeltarget
MethsuximideVoltage-dependent T-type calcium channel subunit alpha-1Gtarget
Methylene blueCytochrome P450 2C8enzyme
Methylene blueCytochrome P450 2C9enzyme
Methylene blueCytochrome P450 2C19enzyme
Methylene blueCytochrome P450 3A4enzyme
Methylene blueCytochrome P450 3A5enzyme
Methylene blueAlbumincarrier
Methylene blueATP-dependent translocase ABCB1transporter
Methylene blueSolute carrier family 22 member 2transporter
Methylene blueMultidrug and toxin extrusion protein 2transporter
Methylene blueMultidrug and toxin extrusion protein 1transporter
Methylene blueFlavin reductase (NADPH)enzyme
Methylene blueCytochrome P450 2D6enzyme
Methylene blueAmine oxidase [flavin-containing] Atarget
Methylene blueGuanylate cyclase soluble subunit alpha-2target
Methylene blueNitric oxide synthase 1target
Methylene blueUDP-glucuronosyltransferase 1A4enzyme
Methylene blueUDP-glucuronosyltransferase 1A9enzyme
Methylene blueCytochrome P450 1A2enzyme
Methylene blueCytochrome P450 2B6enzyme
MethylergometrineD(1A) dopamine receptortarget
MethylergometrineCytochrome P450 3A4enzyme
Methylergometrine5-hydroxytryptamine receptor 2Btarget
MethyloneSodium-dependent dopamine transportertarget
MethyloneCytochrome P450 2C19enzyme
MethyloneCytochrome P450 2B6enzyme
MethyloneCytochrome P450 1A2enzyme
MethyloneCytochrome P450 2D6enzyme
MethyloneSodium-dependent serotonin transportertarget
MethyloneSodium-dependent noradrenaline transportertarget
MetoclopramideD(2) dopamine receptortarget
MetoclopramideMuscarinic acetylcholine receptor M1target
MetoclopramideCytochrome P450 2D6enzyme
Metoclopramide5-hydroxytryptamine receptor 4target
Metoclopramide5-hydroxytryptamine receptor 3Atarget
MetoclopramideCytochrome P450 3A4enzyme
MetoclopramideCytochrome P450 1A2enzyme
MetoclopramideATP-dependent translocase ABCB1transporter
MetoclopramideAlpha-1-acid glycoprotein 1carrier
MetoprololBeta-2 adrenergic receptortarget
MetoprololSolute carrier family 22 member 2transporter
MetoprololBeta adrenergic receptortarget
MetoprololCytochrome P450 3A4enzyme
MetoprololAlbumincarrier
MetoprololCytochrome P450 2D6enzyme
MetoprololBeta-1 adrenergic receptortarget
MetronidazoleAnaerobic bacterial DNAtarget
MetronidazoleUDP-glucuronosyltransferase 1A1enzyme
MetronidazoleCytochrome P450 2C8enzyme
MetronidazoleCytochrome P450 3A4enzyme
MetronidazoleCytochrome P450 2C9enzyme
MetronidazoleOxygen-insensitive NADPH nitroreductasetarget
MetronidazoleProtozoal DNAtarget
MetronidazoleATP-dependent translocase ABCB1transporter
MetronidazoleCytochrome P450 2A6enzyme
MetronidazoleCytochrome P450 3A5enzyme
MetronidazoleCytochrome P450 3A7enzyme
MetyraponeCamphor 5-monooxygenasetarget
MetyraponeCytochrome P450 11B2, mitochondrialenzyme
MetyraponeCytochrome P450 2A6enzyme
MetyraponeCytochrome P450 3A4enzyme
MetyraponeATP-binding cassette sub-family C member 3transporter
MetyraponeCytochrome P450 11B1, mitochondrialtarget
MetyraponeCytochrome P450 11B1, mitochondrialenzyme
MetyraponeCytochrome P450 2E1enzyme
MexiletineCytochrome P450 1A2enzyme
MexiletineCytochrome P450 2D6enzyme
MexiletineCytochrome P450 2B6enzyme
MexiletineSodium channel protein type 5 subunit alphatarget
MexiletineCytochrome P450 3A4enzyme
MexiletineAryl hydrocarbon receptortarget
MexiletineVoltage-gated sodium channel alpha subunittarget
MexiletineCytochrome P450 2E1enzyme
MibefradilVoltage-dependent T-type calcium channeltarget
MibefradilCytochrome P450 11B2, mitochondrialenzyme
MibefradilCytochrome P450 11B1, mitochondrialenzyme
MibefradilVoltage-dependent L-type calcium channel subunit beta-4target
MibefradilVoltage-dependent L-type calcium channel subunit beta-3target
MibefradilVoltage-dependent T-type calcium channel subunit alpha-1Gtarget
MibefradilVoltage-dependent T-type calcium channel subunit alpha-1Htarget
MibefradilVoltage-dependent L-type calcium channel subunit alpha-1Ctarget
MibefradilVoltage-dependent L-type calcium channel subunit beta-1target
MibefradilCytochrome P450 3A4enzyme
MibefradilCytochrome P450 1A2enzyme
MibefradilCytochrome P450 2D6enzyme
MibefradilVoltage-dependent L-type calcium channel subunit beta-2target
MibefradilVoltage-dependent L-type calcium channel subunit alpha-1Dtarget
MibefradilVoltage-dependent L-type calcium channel subunit alpha-1Ftarget
MibefradilVoltage-dependent L-type calcium channel subunit alpha-1Starget
MibefradilVoltage-dependent T-type calcium channel subunit alpha-1Itarget
MibefradilATP-dependent translocase ABCB1transporter
MibefradilCytochrome P450 3A7enzyme
MibefradilCytochrome P450 3A5enzyme
MiconazoleATP-dependent translocase ABCB1transporter
MiconazoleCytochrome P450 2C8enzyme
MiconazoleAlbumincarrier
MiconazoleVoltage gated L-type calcium channeltarget
MiconazoleInward rectifier potassium channeltarget
MiconazoleVoltage-gated Potassium Channelstarget
MiconazoleCalcium-activated potassium channeltarget
MiconazoleLanosterol 14-alpha demethylasetarget
MiconazoleNitric oxide synthase 3target
MiconazoleNitric oxide synthase, inducibletarget
MiconazoleCytochrome P450 11B1, mitochondrialenzyme
MiconazoleCytochrome P450 2A6enzyme
MiconazoleCytochrome P450 2B6enzyme
MiconazoleCytochrome P450 2C19enzyme
MiconazoleCytochrome P450 2E1enzyme
MiconazoleNuclear receptor subfamily 1 group I member 2target
MiconazoleLanosterol 14-alpha demethylaseenzyme
MiconazoleAromataseenzyme
MiconazoleCytochrome P450 3A4enzyme
MiconazoleCytochrome P450 2D6enzyme
MiconazoleCytochrome P450 2C9enzyme
MidazolamTranslocator proteintarget
MidazolamUDP-glucuronosyltransferase 2B4enzyme
MidazolamUDP-glucuronosyltransferase 2B7enzyme
MidazolamExcitatory amino acid transporter 2transporter
MidazolamAdenosine receptor A2atarget
MidazolamAlpha-1-acid glycoprotein 1carrier
MidazolamAlbumincarrier
MidazolamATP-dependent translocase ABCB1transporter
MidazolamGABA(A) Receptor Benzodiazepine Binding Sitetarget
MidazolamGABA(A) Receptortarget
MidazolamCytochrome P450 3A7enzyme
MidazolamUDP-glucuronosyltransferase 1A4enzyme
MidazolamCytochrome P450 3A5enzyme
MidazolamCytochrome P450 3A4enzyme
MidecamycinCytochrome P450 3A4enzyme
MidecamycinBacterial 50S ribosomal proteintarget
MidostaurinCytochrome P450 2B6enzyme
MidostaurinCytochrome P450 2C8enzyme
MidostaurinCytochrome P450 2C9enzyme
MidostaurinCytochrome P450 2C19enzyme
MidostaurinCytochrome P450 2D6enzyme
MidostaurinCytochrome P450 2E1enzyme
MidostaurinCytochrome P450 3A4enzyme
MidostaurinCytochrome P450 3A5enzyme
MidostaurinCytochrome P450 3A7enzyme
MidostaurinProtein kinase C alpha typetarget
MidostaurinVascular endothelial growth factor receptor 2target
MidostaurinMast/stem cell growth factor receptor Kittarget
MidostaurinPlatelet-derived growth factor receptor alphatarget
MidostaurinPlatelet-derived growth factor receptor betatarget
MidostaurinReceptor-type tyrosine-protein kinase FLT3target
MidostaurinCytochrome P450 3A Subfamilyenzyme
MidostaurinCytochrome P450 1A2enzyme
MidostaurinProtein kinase Ctarget
MidostaurinProtein kinase C gamma typetarget
MidostaurinCytochrome P450 3A43enzyme
MifentidineCytochrome P450 1A2enzyme
MifentidineHistamine H2 receptortarget
MifepristoneMultidrug resistance-associated protein 1transporter
MifepristoneCytochrome P450 2D6enzyme
MifepristoneNuclear receptor subfamily 1 group I member 2target
MifepristoneBile salt export pumptransporter
MifepristoneCytochrome P450 2C8enzyme
MifepristoneCytochrome P450 2C9enzyme
MifepristoneSolute carrier organic anion transporter family member 1B1transporter
MifepristoneSolute carrier organic anion transporter family member 1B3transporter
MifepristoneATP-dependent translocase ABCB1transporter
MifepristoneCytochrome P450 3A5enzyme
MifepristoneCytochrome P450 3A4enzyme
MifepristoneGlucocorticoid receptortarget
MifepristoneProgesterone receptortarget
MilnacipranSodium-dependent serotonin transportertarget
MilnacipranCytochrome P450 3A4enzyme
MilnacipranNMDA receptortarget
MilnacipranSodium-dependent noradrenaline transportertarget
MiocamycinCytochrome P450 3A4enzyme
MiocamycinBacterial 50S ribosomal proteintarget
MirabegronCholinesteraseenzyme
MirabegronBeta-3 adrenergic receptortarget
MirabegronUDP-glucuronosyltransferase 2B7enzyme
MirabegronUDP-glucuronosyltransferase 1A3enzyme
MirabegronUDP-glucuronosyltransferase 1A8enzyme
MirabegronSolute carrier family 22 member 1transporter
MirabegronSolute carrier family 22 member 2transporter
MirabegronSolute carrier family 22 member 3transporter
MirabegronBeta-1 adrenergic receptortarget
MirabegronAlpha-1-acid glycoprotein 1carrier
MirabegronAlbumincarrier
MirabegronSolute carrier organic anion transporter family member 1A2transporter
MirabegronATP-dependent translocase ABCB1transporter
MirabegronCytochrome P450 2D6enzyme
MirabegronCytochrome P450 3A4enzyme
MiricorilantBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
MiricorilantCytochrome P450 2C8enzyme
MiricorilantCytochrome P450 2C19enzyme
MiricorilantMineralocorticoid receptortarget
MiricorilantGlucocorticoid receptortarget
MirtazapineAlpha-2 adrenergic receptorstarget
MirtazapineSodium-dependent serotonin transportertransporter
MirtazapineAlpha-1 adrenergic receptorstarget
MirtazapineCytochrome P450 2D6enzyme
MirtazapineCytochrome P450 3A4enzyme
MirtazapineCytochrome P450 1A2enzyme
MirtazapineHistamine H1 receptortarget
MirtazapineKappa-type opioid receptortarget
Mirtazapine5-hydroxytryptamine receptor 2Ctarget
MirtazapineAlpha-2A adrenergic receptortarget
Mirtazapine5HT3 serotonin receptortarget
Mirtazapine5-hydroxytryptamine receptor 2Atarget
MitemcinalCytochrome P450 3A4enzyme
MitemcinalMotilin receptortarget
MitoxantroneCytochrome P450 2E1enzyme
MitoxantroneDNA topoisomerase 2-betatarget
MitoxantroneCytochrome P450 3A4enzyme
MitoxantroneCytochrome P450 1B1enzyme
MitoxantroneDNAtarget
MitoxantroneBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
MitoxantroneMultidrug resistance-associated protein 1transporter
MitoxantroneDNA topoisomerase 2-alphatarget
MitoxantroneATP-dependent translocase ABCB1transporter
MizolastineHistamine H1 receptortarget
MizolastineCytochrome P450 2D6enzyme
MoclobemideAmine oxidase [flavin-containing] Atarget
MoclobemideAmine oxidase [flavin-containing] Btarget
MoclobemideMonoamine oxidasetarget
MoclobemideCytochrome P450 2C9enzyme
MoclobemideAmine oxidase [flavin-containing] Benzyme
MoclobemideAmine oxidase [flavin-containing] Aenzyme
MoclobemideCytochrome P450 2D6enzyme
MoclobemideCytochrome P450 2C19enzyme
ModafinilSodium-dependent dopamine transportertarget
ModafinilCytochrome P450 2D6enzyme
ModafinilCytochrome P450 3A5enzyme
ModafinilCytochrome P450 2C9enzyme
ModafinilCytochrome P450 2B6enzyme
ModafinilCytochrome P450 1A2enzyme
ModafinilCytochrome P450 2C19enzyme
ModafinilCytochrome P450 3A4enzyme
ModafinilAlpha-1B adrenergic receptortarget
MomelotinibCytochrome P450 2C19enzyme
MomelotinibATP-dependent translocase ABCB1transporter
MomelotinibCytochrome P450 3A4enzyme
MomelotinibCytochrome P450 2C8enzyme
MomelotinibCytochrome P450 2C9enzyme
MomelotinibCytochrome P450 1A2enzyme
MomelotinibCytochrome P450 2B6enzyme
MomelotinibUDP-glucuronosyltransferase 1A1enzyme
MomelotinibUDP-glucuronosyltransferase 1A9enzyme
MomelotinibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
MomelotinibSolute carrier organic anion transporter family member 1B1transporter
MomelotinibReceptor-type tyrosine-protein kinase FLT3target
MomelotinibActivin receptor type-1target
MomelotinibNon-receptor tyrosine-protein kinase TYK2target
MomelotinibTyrosine-protein kinase JAK3target
MomelotinibTyrosine-protein kinase JAK2target
MomelotinibTyrosine-protein kinase JAK1target
MomelotinibSolute carrier organic anion transporter family member 1B3transporter
MometasoneGlucocorticoid receptortarget
MometasoneCytochrome P450 2C8enzyme
MometasoneProgesterone receptortarget
MometasoneCytochrome P450 3A4enzyme
MometasoneCytochrome P450 3A5enzyme
Mometasone furoateGlucocorticoid receptortarget
Mometasone furoateCytochrome P450 2C8enzyme
Mometasone furoateProgesterone receptortarget
Mometasone furoateCytochrome P450 3A4enzyme
Mometasone furoateCytochrome P450 3A5enzyme
MontelukastProstaglandin G/H synthase 1enzyme
MontelukastCytochrome P450 2A6enzyme
MontelukastCytochrome P450 2C8enzyme
MontelukastCytochrome P450 2C9enzyme
MontelukastCytochrome P450 3A4enzyme
MontelukastPolyunsaturated fatty acid 5-lipoxygenasetarget
MontelukastCysteinyl leukotriene receptor 1target
MontelukastSolute carrier organic anion transporter family member 2B1transporter
MoxifloxacinDNA gyrase subunit Btarget
MoxifloxacinDNA gyrase subunit Atarget
MoxifloxacinSerum paraoxonase/arylesterase 1target
MoxifloxacinCytochrome P450 1A2enzyme
MoxifloxacinDNA topoisomerase 2-alphatarget
MoxifloxacinDNA topoisomerase 4 subunit Atarget
MoxifloxacinDNA gyrase subunit Atarget
NabiloneCannabinoid receptor 2target
NabiloneCannabinoid receptor 1target
NabiloneCytochrome P450 2E1enzyme
NabiloneCytochrome P450 2C8enzyme
NabiloneCytochrome P450 2C9enzyme
NabiloneCytochrome P450 3A4enzyme
NabiloneCytochrome P450 2J2enzyme
NabiximolsCannabinoid receptor 1target
NabiximolsCannabinoid receptor 2target
NabiximolsG protein-coupled receptor 12target
NabiximolsCytochrome P450 2C9enzyme
NabiximolsCytochrome P450 2C19enzyme
NabiximolsCytochrome P450 2D6enzyme
NabiximolsCytochrome P450 3A4enzyme
NabiximolsGlycine receptor subunit alpha-1target
NabiximolsGlycine receptor (alpha-1/beta)target
NabiximolsGlycine receptor subunit alpha-3target
NabiximolsN-arachidonyl glycine receptortarget
NabiximolsG protein-coupled receptor 55target
Nabiximols5-hydroxytryptamine receptor 1Atarget
Nabiximols5-hydroxytryptamine receptor 2Atarget
NabiximolsNeuronal acetylcholine receptor subunit alpha-7target
NabiximolsDelta-type opioid receptortarget
NabiximolsMu-type opioid receptortarget
NabiximolsPeroxisome proliferator-activated receptor gammatarget
NabiximolsCytochrome P450 3A5enzyme
NabiximolsPolyunsaturated fatty acid 5-lipoxygenaseenzyme
NabiximolsPolyunsaturated fatty acid lipoxygenase ALOX15enzyme
NabiximolsMultidrug resistance-associated protein 1transporter
NabiximolsBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
NabiximolsEquilibrative nucleoside transporter 1transporter
NabiximolsN-acylethanolamine-hydrolyzing acid amidasetarget
NabiximolsSuperoxide dismutase [Cu-Zn]target
NabiximolsFatty-acid amide hydrolase 1target
NabiximolsCatalasetarget
NabiximolsZeta-crystallintarget
NabiximolsCytochrome P450 3A7target
NabiximolsCytochrome P450 1A1target
NabiximolsCytochrome P450 1A2target
NabiximolsCytochrome P450 2D6target
NabiximolsCytochrome P450 3A5target
NabiximolsCytochrome P450 1B1target
NabiximolsSerotonin N-acetyltransferasetarget
NabiximolsIndoleamine 2,3-dioxygenase 1target
NabiximolsVoltage-dependent T-type calcium channel subunit alpha-1Gtarget
NabiximolsGlutathione peroxidase 1target
NabiximolsTransient receptor potential cation channel subfamily V member 1target
NabiximolsGlutathione reductase, mitochondrialtarget
Nabiximols3-hydroxy-3-methylglutaryl-coenzyme A reductasetarget
NabiximolsSteroid 17-alpha-hydroxylase/17,20 lyasetarget
NabiximolsAcetyl-CoA acetyltransferase, mitochondrialtarget
NabiximolsProstaglandin G/H synthase 2target
NabiximolsProstaglandin G/H synthase 1target
NabiximolsNon-selective voltage-gated ion channel VDAC1target
NabiximolsTransient receptor potential cation channel subfamily V member 4target
NabiximolsTransient receptor potential cation channel subfamily V member 3target
NabiximolsTransient receptor potential cation channel subfamily V member 2target
NabiximolsTransient receptor potential cation channel subfamily M member 8target
NabiximolsTransient receptor potential cation channel subfamily A member 1target
NabiximolsVoltage-dependent T-type calcium channel subunit alpha-1Itarget
NabiximolsVoltage-dependent T-type calcium channel subunit alpha-1Htarget
NafimidoneCytochrome P450 2D6enzyme
NafimidoneCytochrome P450 1A2enzyme
NafithromycinCytochrome P450 3A Subfamilyenzyme
NafithromycinCytochrome P450 3A5enzyme
NafithromycinCytochrome P450 3A4enzyme
Nalidixic acidSolute carrier family 22 member 6transporter
Nalidixic acidTryptophan 2,3-dioxygenaseenzyme
Nalidixic acidCytochrome P450 1A2enzyme
Nalidixic acidAerobic bacterial DNAtarget
Nalidixic acidDNA gyrase subunit Atarget
Nalidixic acidDNA gyrase subunit Btarget
Nalidixic acidDNA topoisomerase 2-alphatarget
Nalidixic acidDNA topoisomerase 2-betatarget
NaloxegolCytochrome P450 3A4enzyme
NaloxegolCytochrome P450 2D6enzyme
NaloxegolCytochrome P450 2C19enzyme
NaloxegolMu-type opioid receptortarget
NaloxoneUDP-glucuronosyltransferase 1A1enzyme
NaloxoneCytochrome P450 2C18enzyme
NaloxoneCytochrome P450 2C19enzyme
NaloxoneLiver carboxylesterase 1target
NaloxoneToll-like receptor 4target
NaloxoneAlbumincarrier
NaloxoneCytochrome P450 3A4enzyme
NaloxoneKappa-type opioid receptortarget
NaloxoneATP-dependent translocase ABCB1transporter
NaloxoneSolute carrier organic anion transporter family member 1A2transporter
NaloxoneDelta-type opioid receptortarget
NaloxoneEstrogen receptortarget
NaloxoneMu-type opioid receptortarget
NaringinSolute carrier organic anion transporter family member 1A2transporter
NaringinCytochrome P450 3A4enzyme
NaringinSolute carrier organic anion transporter family member 2B1transporter
NaringinGrowth hormone secretagogue receptor type 1target
NaringinCarbonic anhydrase 2target
NaringinAcetylcholinesterasetarget
Nefazodone5-hydroxytryptamine receptor 1Atarget
NefazodoneCytochrome P450enzyme
NefazodoneATP-dependent translocase ABCB1transporter
Nefazodone5-hydroxytryptamine receptor 2Ctarget
NefazodoneVoltage-gated inwardly rectifying potassium channel KCNH2target
NefazodoneCytochrome P450 3A Subfamilyenzyme
NefazodoneSolute carrier organic anion transporter family member 1B3transporter
NefazodoneSolute carrier organic anion transporter family member 2B1transporter
NefazodoneBile salt export pumptransporter
NefazodoneAlpha-2A adrenergic receptortarget
NefazodoneSodium-dependent dopamine transportertarget
NefazodoneCytochrome P450 2D6enzyme
NefazodoneCytochrome P450 3A4enzyme
NefazodoneAlpha-1B adrenergic receptortarget
NefazodoneAlpha-1A adrenergic receptortarget
NefazodoneSodium-dependent noradrenaline transportertarget
NefazodoneSodium-dependent serotonin transportertarget
Nefazodone5-hydroxytryptamine receptor 2Atarget
NelfinavirCytochrome P450 3A7enzyme
NelfinavirATP-dependent translocase ABCB1transporter
NelfinavirCytochrome P450 2C19enzyme
NelfinavirCytochrome P450 3A4enzyme
NelfinavirPol polyproteintarget
NelfinavirGag-Pol polyproteintarget
NelfinavirAlpha-1-acid glycoprotein 1carrier
NelfinavirCytochrome P450 2C9enzyme
NelfinavirBile salt export pumptransporter
NelfinavirSolute carrier organic anion transporter family member 2B1transporter
NelfinavirSolute carrier organic anion transporter family member 1B3transporter
NelfinavirUDP-glucuronosyltransferase 1A1enzyme
NelfinavirAlbumincarrier
NelfinavirCytochrome P450 2D6enzyme
NelfinavirSolute carrier organic anion transporter family member 1B1transporter
NelfinavirCytochrome P450 2B6enzyme
NelfinavirCytochrome P450 3A5enzyme
NelfinavirSolute carrier family 22 member 1transporter
NelfinavirSolute carrier organic anion transporter family member 1A2transporter
NelfinavirBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
NemonoxacinDNA gyrase subunit Atarget
NemonoxacinCytochrome P450 1A2enzyme
NemonoxacinDNA gyrase subunit Btarget
NetoglitazoneCytochrome P450 2C8enzyme
NetoglitazoneCytochrome P450 3A4enzyme
NetoglitazonePeroxisome proliferator-activated receptor gammatarget
NetupitantCytochrome P450 3A4enzyme
NetupitantCytochrome P450 2D6enzyme
NetupitantATP-dependent translocase ABCB1transporter
NetupitantCytochrome P450 2C9enzyme
NetupitantCytochrome P450 3A43enzyme
NetupitantSubstance-P receptortarget
NevirapineGag-Pol polyproteintarget
NevirapineCytochrome P450 3A7enzyme
NevirapineSolute carrier family 22 member 1transporter
NevirapineCytochrome P450 1A2enzyme
NevirapineCytochrome P450 3A4enzyme
NevirapineAlbumincarrier
NevirapineReverse transcriptase/RNaseHtarget
NevirapineCytochrome P450 2D6enzyme
NevirapineCytochrome P450 2A6enzyme
NevirapineCytochrome P450 2C9enzyme
NevirapineCytochrome P450 3A5enzyme
NevirapineCytochrome P450 2B6enzyme
NiacinCytochrome P450 2E1enzyme
NiacinDiacylglycerol O-acyltransferase 2target
NiacinNicotinamide N-methyltransferasetarget
NiacinNicotinate-nucleotide pyrophosphorylase [carboxylating]target
NiacinHydroxycarboxylic acid receptor 3target
NiacinOrganic cation/carnitine transporter 2transporter
NiacinSolute carrier organic anion transporter family member 2B1transporter
NiacinMonocarboxylate transporter 1transporter
NiacinCytochrome P450 2D6enzyme
NiacinHydroxycarboxylic acid receptor 2target
NiacinSodium-coupled monocarboxylate transporter 1transporter
NiacinMonocarboxylate transporter 4transporter
NiacinThyroxine-binding globulincarrier
NiacinCytochrome P450 3A4enzyme
NicardipineBile salt export pumptransporter
NicardipineSolute carrier organic anion transporter family member 1B1transporter
NicardipineCytochrome P450 3A5enzyme
NicardipineCytochrome P450 2C9enzyme
NicardipineVoltage-dependent calcium channeltarget
NicardipineVoltage-dependent T-type calcium channel subunit alpha-1Gtarget
NicardipineCytochrome P450 2D6enzyme
NicardipineCytochrome P450 2E1enzyme
NicardipineVoltage-dependent T-type calcium channel subunit alpha-1Htarget
NicardipineVoltage-dependent T-type calcium channel subunit alpha-1Itarget
NicardipineCalmodulintarget
NicardipineVoltage gated L-type calcium channeltarget
NicardipineVoltage-dependent L-type calcium channel subunit alpha-1Ctarget
NicardipineCytochrome P450 3A4enzyme
NicardipineCytochrome P450 2C19enzyme
NicardipineCytochrome P450 2C8enzyme
NicardipineCytochrome P450 2B6enzyme
NicardipineDual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1Btarget
NicardipineDual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1Atarget
NicardipineAlpha-1A adrenergic receptortarget
NicardipineAlpha-1D adrenergic receptortarget
NicardipineAlpha-1B adrenergic receptortarget
NicardipineMuscarinic acetylcholine receptor M1target
NicardipineMuscarinic acetylcholine receptor M2target
NicardipineMuscarinic acetylcholine receptor M3target
NicardipineMuscarinic acetylcholine receptor M4target
NicardipineMuscarinic acetylcholine receptor M5target
NicardipineVoltage-dependent calcium channel subunit alpha-2/delta-1target
NicardipineVoltage-dependent L-type calcium channel subunit beta-2target
NicardipineVoltage-dependent L-type calcium channel subunit alpha-1Dtarget
NicardipineATP-dependent translocase ABCB1transporter
NiclosamideCytochrome P450 1A2enzyme
NiclosamideCytochrome P450 2C9enzyme
NiclosamideDNAtarget
NicotinamideCytochrome P450 3A4enzyme
NicotinamideNAD-dependent protein deacylase sirtuin-5, mitochondrialtarget
NicotinamideADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 2target
NicotinamideExotoxin Atarget
NicotinamideL-lactate dehydrogenase A chaintarget
NicotinamidePoly [ADP-ribose] polymerase 1target
NicotinamideCytochrome P450 2D6enzyme
NicotinamideCytochrome P450 2E1enzyme
NicotineSolute carrier family 22 member 2transporter
NicotineCholine O-acetyltransferasetarget
NicotineAromatasetarget
NicotineAmine oxidase [flavin-containing] Benzyme
NicotineAmine oxidase [flavin-containing] Aenzyme
NicotineCytochrome P450 3A4enzyme
NicotineCytochrome P450 2D6enzyme
NicotineCytochrome P450 2C9enzyme
NicotineCytochrome P450 2C8enzyme
NicotineCytochrome P450 2C19enzyme
NicotineCytochrome P450 1A2enzyme
NicotineCytochrome P450 1A1enzyme
NicotineSolute carrier family 22 member 4transporter
NicotineOrganic cation/carnitine transporter 2transporter
NicotineSolute carrier family 22 member 3transporter
NicotineSolute carrier family 22 member 1transporter
NicotineNeuronal acetylcholine receptor subunit beta-3target
NicotineNeuronal acetylcholine receptor subunit alpha-6target
NicotineNeuronal acetylcholine receptor subunit alpha-5target
NicotineNeuronal acetylcholine receptor subunit alpha-3target
NicotineNeuronal acetylcholine receptor subunit beta-4target
NicotineCytochrome P450 2B6enzyme
NicotineCytochrome P450 2A13enzyme
NicotineCytochrome P450 2E1enzyme
NicotineCytochrome P450 2A6enzyme
NicotineNeuronal acetylcholine receptor subunit alpha-9target
NicotineNeuronal acetylcholine receptor subunit alpha-10target
NicotineNeuronal acetylcholine receptor subunit alpha-4target
NicotineNeuronal acetylcholine receptor subunit alpha-7target
NicotineNeuronal acetylcholine receptor subunit beta-2target
NicotineNeuronal acetylcholine receptor subunit alpha-2target
NifedipineSolute carrier organic anion transporter family member 1B1transporter
NifedipineNuclear receptor subfamily 1 group I member 2target
NifedipineCytochrome P450 2B6enzyme
NifedipineBile salt export pumptransporter
NifedipineATP-binding cassette sub-family C member 2transporter
NifedipineATP-dependent translocase ABCB1transporter
NifedipineCytochrome P450 2C9enzyme
NifedipineAlbumincarrier
NifedipineCytochrome P450 3A4enzyme
Nifedipinealpha1-acid glycoproteincarrier
NifedipineCytochrome P450 3A5enzyme
NifedipineCalmodulintarget
NifedipineVoltage gated L-type calcium channeltarget
NifedipineCytochrome P450 2E1enzyme
NifedipineCytochrome P450 2D6enzyme
NifedipineVoltage-dependent L-type calcium channel subunit alpha-1Dtarget
NifedipineVoltage-dependent L-type calcium channel subunit alpha-1Starget
NifedipineVoltage-dependent L-type calcium channel subunit alpha-1Ctarget
NifedipineVoltage-dependent L-type calcium channel subunit beta-2target
NifedipineA-type voltage-gated potassium channel KCND3target
NifedipineVoltage-dependent T-type calcium channeltarget
NifedipineCytochrome P450 1A2enzyme
NifedipineCytochrome P450 2A6enzyme
NifedipineCytochrome P450 2C8enzyme
NifedipineATP-binding cassette sub-family C member 3transporter
NifedipineCytochrome P450 1A1enzyme
NilotinibDiscoidin domain receptortarget
NilotinibTyrosine-protein kinase ABL1target
NilotinibMast/stem cell growth factor receptor Kittarget
NilotinibCytochrome P450 2D6enzyme
NilotinibCytochrome P450 2C8enzyme
NilotinibCytochrome P450 2C9enzyme
NilotinibCytochrome P450 3A4enzyme
NilotinibATP-dependent translocase ABCB1transporter
NilotinibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
NilotinibGranulocyte colony-stimulating factor receptortarget
NilotinibPlatelet-derived growth factor receptortarget
NilotinibSolute carrier organic anion transporter family member 1B1transporter
NilotinibCytochrome P450 2B6enzyme
NilotinibUDP-glucuronosyltransferase 1A1transporter
NilutamideNADPH--cytochrome P450 reductaseenzyme
NilutamideCytochrome P450 2C19enzyme
NilutamideAndrogen receptortarget
NilvadipineCytochrome P450 2C19enzyme
NilvadipineCytochrome P450 3A4enzyme
NilvadipineVoltage-dependent T-type calcium channeltarget
NilvadipineVoltage gated L-type calcium channeltarget
NilvadipineVoltage-dependent T-type calcium channel subunit alpha-1Itarget
NilvadipineCytochrome P450 2A6enzyme
NilvadipineVoltage-dependent calcium channel subunit alpha-2/delta-3target
NilvadipineVoltage-dependent L-type calcium channel subunit alpha-1Starget
NilvadipineVoltage-dependent L-type calcium channel subunit alpha-1Dtarget
NilvadipineVoltage-dependent L-type calcium channel subunit beta-2target
NilvadipineVoltage-dependent calcium channel subunit alpha-2/delta-1target
NilvadipineVoltage-dependent L-type calcium channel subunit alpha-1Ctarget
NilvadipineCytochrome P450 2E1enzyme
NilvadipineCytochrome P450 2C8enzyme
NilvadipineVoltage-dependent T-type calcium channel subunit alpha-1Htarget
NirmatrelvirReplicase polyprotein 1abtarget
NirmatrelvirCytochrome P450 3A4enzyme
NirmatrelvirATP-dependent translocase ABCB1transporter
NirmatrelvirReplicase polyprotein 1atarget
NitisinoneCytochrome P450 3A4enzyme
Nitisinone4-hydroxyphenylpyruvate dioxygenasetarget
NitrazepamGamma-aminobutyric acid receptor subunit alpha-1target
NitrazepamGABA(A) Receptor Benzodiazepine Binding Sitetarget
NitrazepamSodium channel protein type 1 subunit alphatarget
NitrazepamCytochrome P450 3A4enzyme
NitrazepamCytochrome P450 2E1enzyme
NitrazepamGABA(A) Receptortarget
Nitric OxideGuanylate cyclase soluble subunit beta-1target
Nitric OxideGuanylate cyclase soluble subunit alpha-1target
Nitric OxideNitric oxide synthase 3target
Nitric OxideIndoleamine 2,3-dioxygenase 1target
Nitric OxideMetallothionein-1Atarget
Nitric OxideCytochrome P450 3A4enzyme
Nitric OxideGuanylate cyclase soluble subunit alpha-2target
Nitric OxideAldehyde dehydrogenase, mitochondrialenzyme
Nitric OxideCytochrome P450 1A2enzyme
Nitric OxideCytochrome P450 2B6enzyme
NivasorexantOrexin/Hypocretin receptor type 1target
NivasorexantCytochrome P450 2C19enzyme
NivasorexantCytochrome P450 3A4enzyme
NivasorexantCytochrome P450 2C9enzyme
Nix-0699Cytochrome P450 3A4enzyme
NorfloxacinDNA topoisomerase 4 subunit Atarget
NorfloxacinDNA gyrase subunit Atarget
NorfloxacinCytochrome P450 1A2enzyme
NorfloxacinCytochrome P450 3A4enzyme
NorfloxacinDNA gyrase subunit Btarget
NorfloxacinDNA topoisomerase 4 subunit Atarget
NorfloxacinDNA topoisomerase 2target
NorfloxacinDNA gyrase subunit Atarget
NorfloxacinCytochrome P450 3A7enzyme
NorfloxacinCytochrome P450 1A1enzyme
NorfloxacinSolute carrier family 22 member 6transporter
NorfloxacinOrganic cation/carnitine transporter 2transporter
NorfloxacinDNA topoisomerase 2-alphatarget
NortriptylineATP-dependent translocase ABCB1transporter
NortriptylineMuscarinic acetylcholine receptortarget
NortriptylineSodium-dependent noradrenaline transportertransporter
Nortriptyline5-hydroxytryptamine receptor 2Ctarget
NortriptylineSigma receptortarget
NortriptylineD(2) dopamine receptortarget
NortriptylineBeta adrenergic receptortarget
NortriptylineAlpha-2 adrenergic receptorstarget
NortriptylineAlpha-1B adrenergic receptortarget
Nortriptyline5-hydroxytryptamine receptor 2Ctarget
NortriptylineCytochrome P450 2E1enzyme
NortriptylineCytochrome P450 2C19enzyme
NortriptylineAlpha-1D adrenergic receptortarget
NortriptylineCytochrome P450 3A5enzyme
NortriptylineCytochrome P450 3A4enzyme
NortriptylineAlpha-1A adrenergic receptortarget
Nortriptyline5-hydroxytryptamine receptor 2Atarget
NortriptylineHistamine H1 receptortarget
NortriptylineAlpha-1-acid glycoprotein 1carrier
NortriptylineAlbumincarrier
NortriptylineCytochrome P450 2D6enzyme
NortriptylineCytochrome P450 1A2enzyme
NortriptylineSodium-dependent noradrenaline transportertarget
NortriptylineSodium-dependent serotonin transportertarget
Nortriptyline5-hydroxytryptamine receptor 1Atarget
NoscapineCytochrome P450 2C9enzyme
NoscapineSigma non-opioid intracellular receptor 1target
NoscapineCytochrome P450 3A4enzyme
Obeticholic acidBile salt export pumptransporter
Obeticholic acidBile acid receptortarget
Obeticholic acidCytochrome P450 1A2enzyme
OctreotideATP-binding cassette sub-family C member 2transporter
OctreotideSomatostatin receptortarget
OctreotideSomatostatin receptor type 2target
OctreotideATP-dependent translocase ABCB1transporter
OctreotideAlbumincarrier
OctreotideSomatostatin receptortarget
OctreotideCytochrome P450 3A4enzyme
OctreotideMyeloperoxidaseenzyme
OfloxacinATP-binding cassette sub-family C member 2transporter
OfloxacinSolute carrier family 22 member 4transporter
OfloxacinBile salt export pumptransporter
OfloxacinDNA gyrase subunit Atarget
OfloxacinDNA gyrase subunit Btarget
OfloxacinMultidrug resistance-associated protein 1transporter
OfloxacinOrganic cation/carnitine transporter 2transporter
OfloxacinCytochrome P450 1A2enzyme
OfloxacinDNA topoisomerase 2-alphatarget
OfloxacinDNA topoisomerase 4 subunit Atarget
OfloxacinDNA gyrase subunit Atarget
OfloxacinSolute carrier family 22 member 6transporter
Olanzapine5-hydroxytryptamine receptor 1target
OlanzapineBeta adrenergic receptortarget
OlanzapineD(1) dopamine receptortarget
OlanzapineCytochrome P450 2C19enzyme
OlanzapineATP-dependent translocase ABCB1transporter
OlanzapineCytochrome P450 2D6enzyme
OlanzapineFlavin-containing monooxygenase 3enzyme
OlanzapineD(1B) dopamine receptortarget
OlanzapineAlpha-1-acid glycoprotein 1carrier
OlanzapineAlbumincarrier
OlanzapineCytochrome P450 3A4enzyme
OlanzapineAlpha-1A adrenergic receptortarget
Olanzapine5-hydroxytryptamine receptor 6target
Olanzapine5-hydroxytryptamine receptor 3Atarget
OlanzapineCytochrome P450 1A2enzyme
OlanzapineAlpha-1B adrenergic receptortarget
OlanzapineD(3) dopamine receptortarget
Olanzapine5-hydroxytryptamine receptor 2Ctarget
OlanzapineD(2) dopamine receptortarget
OlanzapineMuscarinic acetylcholine receptor M2target
OlanzapineMuscarinic acetylcholine receptor M4target
OlanzapineHistamine H1 receptortarget
OlanzapineD(4) dopamine receptortarget
Olanzapine5-hydroxytryptamine receptor 2Atarget
OlanzapineMuscarinic acetylcholine receptor M3target
OlanzapineMuscarinic acetylcholine receptor M1target
OlanzapineD(1A) dopamine receptortarget
OlanzapineGABA(A) Receptor Benzodiazepine Binding Sitetarget
OlanzapineCytochrome P450 2C9enzyme
OlanzapineUDP-glucuronosyltransferase 1A4enzyme
OlanzapineCytochrome P450 3A Subfamilyenzyme
OlaparibAlpha-1-acid glycoprotein 1carrier
OlaparibAlbumincarrier
OlaparibUDP-glucuronosyltransferase 1A1enzyme
OlaparibAldo-keto reductase family 1 member C3target
OlaparibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
OlaparibATP-dependent translocase ABCB1transporter
OlaparibCytochrome P450 3A5enzyme
OlaparibProtein mono-ADP-ribosyltransferase PARP3target
OlaparibPoly [ADP-ribose] polymerase 2target
OlaparibCytochrome P450 2B6enzyme
OlaparibCytochrome P450 3A4enzyme
OlaparibPoly [ADP-ribose] polymerase 1target
OlaparibPoly [ADP-ribose] polymerasestarget
OleandomycinCytochrome P450 3A1enzyme
OleandomycinCytochrome P450 3A4enzyme
OlorofimApolipoprotein A-Ienzyme
OlorofimCytochrome P450 3A4enzyme
OlorofimCytochrome P450 2C8enzyme
OlorofimCytochrome P450 2C9enzyme
OlorofimCytochrome P450 2D6enzyme
OlorofimDihydroorotate dehydrogenase (quinone), mitochondrialtarget
OlorofimCytochrome P450 1A2enzyme
OlorofimCytochrome P450 2B6enzyme
OmeprazoleAryl hydrocarbon receptortarget
OmeprazolePotassium-transporting ATPase subunit betatarget
OmeprazoleCytochrome P450 2D6enzyme
OmeprazoleCytochrome P450 2C8enzyme
OmeprazoleCytochrome P450 2C18enzyme
OmeprazoleCytochrome P450 1B1enzyme
OmeprazoleCytochrome P450 1A1enzyme
OmeprazoleATP-dependent translocase ABCB1transporter
OmeprazoleATP-binding cassette sub-family C member 3transporter
OmeprazoleCytochrome P450 1A2enzyme
OmeprazoleCytochrome P450 2C9enzyme
OmeprazoleCytochrome P450 3A4enzyme
OmeprazoleCytochrome P450 2C19enzyme
OmeprazolePotassium-transporting ATPase alpha chain 1target
OmeprazoleBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
OndansetronCytochrome P450 2E1enzyme
OndansetronCytochrome P450 2D6enzyme
OndansetronCytochrome P450 2C9enzyme
OndansetronMu-type opioid receptortarget
Ondansetron5-hydroxytryptamine receptor 1Btarget
Ondansetron5-hydroxytryptamine receptor 1Atarget
Ondansetron5-hydroxytryptamine receptor 4target
OndansetronCytochrome P450 3A7enzyme
OndansetronCytochrome P450 3A5enzyme
OndansetronCytochrome P450 1A2enzyme
OndansetronCytochrome P450 3A4enzyme
Ondansetron5-hydroxytryptamine receptor 3Atarget
OpelconazoleLanosterol 14-alpha demethylasetarget
OpelconazoleCytochrome P450 1A2enzyme
OpelconazoleCytochrome P450 3A4enzyme
OpicaponeCytochrome P450 2B6enzyme
OpicaponeCytochrome P450 1A2enzyme
OpicaponeCytochrome P450 2C9enzyme
OpicaponeSolute carrier organic anion transporter family member 2B1transporter
OpicaponeSolute carrier organic anion transporter family member 1B3transporter
OpicaponeBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
OpicaponeATP-dependent translocase ABCB1transporter
OpicaponeSolute carrier organic anion transporter family member 1B1transporter
OpicaponeCatechol O-methyltransferasetarget
OpicaponeCytochrome P450 2C8enzyme
OpicaponeCytochrome P450 2C19enzyme
OrbifloxacinCytochrome P450 1A2enzyme
OritavancinPentaglycyl bridging segmenttarget
OritavancinBacterial cell wall peptide bridging segmentstarget
OritavancinPeptidoglycan precursorstarget
OritavancinAlbumincarrier
OritavancinCytochrome P450 2C19enzyme
OritavancinCytochrome P450 2C9enzyme
OritavancinCytochrome P450 2D6enzyme
OritavancinCytochrome P450 3A4enzyme
OritavancinDihydropteroate synthasetarget
OrphenadrineCytochrome P450 2D6enzyme
OrphenadrineAlbumincarrier
OrphenadrineVoltage-gated sodium channel alpha subunittarget
OrphenadrineCytochrome P450 1A2enzyme
OrphenadrineSodium channel protein type 10 subunit alphatarget
OrphenadrineSodium-dependent noradrenaline transportertarget
OrphenadrineCytochrome P450 3A4enzyme
OrphenadrineCytochrome P450 2E1enzyme
OrphenadrineCytochrome P450 2B6enzyme
OrphenadrineHistamine H1 receptortarget
OrphenadrineGlutamate receptor ionotropic, NMDA 3Atarget
OrphenadrineGlutamate receptor ionotropic, NMDA 3Btarget
OrphenadrineGlutamate receptor ionotropic, NMDA 2Dtarget
OrphenadrineGlutamate receptor ionotropic, NMDA 1target
OsilodrostatUDP-glucuronosyltransferase 1A1enzyme
OsilodrostatMultidrug and toxin extrusion protein 1transporter
OsilodrostatOrganic anion transporter 3transporter
OsilodrostatSolute carrier family 22 member 6transporter
OsilodrostatSolute carrier family 22 member 2transporter
OsilodrostatSolute carrier family 22 member 1transporter
OsilodrostatSolute carrier organic anion transporter family member 1B1transporter
OsilodrostatCytochrome P450 2E1enzyme
OsilodrostatCytochrome P450 2C19enzyme
OsilodrostatCytochrome P450 1A2enzyme
OsilodrostatCytochrome P450 3A5enzyme
OsilodrostatUDP-glucuronosyltransferase 2B10enzyme
OsilodrostatUDP-glucuronosyltransferase 2B7enzyme
OsilodrostatUDP-glucuronosyltransferase 1A4enzyme
OsilodrostatCytochrome P450 2D6enzyme
OsilodrostatCytochrome P450 2B6enzyme
OsilodrostatCytochrome P450 3A4enzyme
OsilodrostatCytochrome P450 11B2, mitochondrialtarget
OsilodrostatCytochrome P450 11B1, mitochondrialtarget
OsimertinibEpidermal growth factor receptortarget
OsimertinibATP-dependent translocase ABCB1transporter
OsimertinibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
OsimertinibCytochrome P450 3A4enzyme
OsimertinibCytochrome P450 1A2enzyme
OspemifeneEstrogen receptortarget
OspemifeneCytochrome P450 2D6enzyme
OspemifeneCytochrome P450 2B6enzyme
OspemifeneCytochrome P450 2C19enzyme
OspemifeneCytochrome P450 2C9enzyme
OspemifeneCytochrome P450 3A4enzyme
OspemifeneEstrogen receptortarget
OSU-6162D(2) dopamine receptortarget
OSU-6162Cytochrome P450 2D6enzyme
OxamniquineDNAtarget
OxamniquineCytochrome P450 2D6enzyme
OxandroloneCytochrome P450 2C9enzyme
OxandroloneAndrogen receptortarget
OxcarbazepineAlbumincarrier
OxcarbazepineATP-dependent translocase ABCB1transporter
OxcarbazepineAldo-keto reductase family 1 member C1enzyme
OxcarbazepineAldo-keto reductase family 1 member C2enzyme
OxcarbazepineAldo-keto reductase family 1 member C3enzyme
OxcarbazepineAldo-keto reductase family 1 member C4enzyme
OxcarbazepineCarbonyl reductase [NADPH] 1enzyme
OxcarbazepineCytochrome P450 3A5enzyme
OxcarbazepineSodium channel proteintarget
OxcarbazepineSodium channel protein type 11 subunit alphatarget
OxcarbazepineVoltage-gated sodium channel alpha subunittarget
OxcarbazepineCytochrome P450 3A4enzyme
OxcarbazepineCytochrome P450 2C19enzyme
OxcarbazepineCarbonyl reductase [NADPH] 3enzyme
OxethazaineCytochrome P450 3A4enzyme
OxethazaineGastrintarget
OxprenololCytochrome P450 2D6enzyme
OxprenololBeta-3 adrenergic receptortarget
OxprenololSolute carrier family 22 member 2transporter
OxprenololBeta-2 adrenergic receptortarget
OxprenololBeta-1 adrenergic receptortarget
OxybutyninAlpha-1-acid glycoprotein 1carrier
OxybutyninCytochrome P450 3A5enzyme
OxybutyninCytochrome P450 2D6enzyme
OxybutyninCytochrome P450 2C8enzyme
OxybutyninCytochrome P450 3A4enzyme
OxybutyninMuscarinic acetylcholine receptor M3target
OxybutyninMuscarinic acetylcholine receptor M2target
OxybutyninMuscarinic acetylcholine receptor M1target
OxybutyninAlbumincarrier
OxymetholoneAndrogen receptortarget
OxymetholoneSex hormone-binding globulincarrier
OxymetholoneAmine oxidase [flavin-containing] Aenzyme
OxymetholoneCytochrome P450 2D6enzyme
Oxymetholone3-oxo-5-alpha-steroid 4-dehydrogenase 1enzyme
OxymetholoneCytochrome P450 3A4enzyme
OxymetholoneCytochrome P450 3A5enzyme
OxymetholoneCytochrome P450 3A7enzyme
OxymetholoneCytochrome P450 3A43enzyme
OxymetholoneAlbumincarrier
P-57AS3Multidrug resistance-associated protein 1transporter
P-57AS3ATP-dependent translocase ABCB1transporter
P-57AS3Cytochrome P450 3A4enzyme
P-57AS3ATP-binding cassette sub-family C member 2transporter
PacritinibReceptor-type tyrosine-protein kinase FLT3target
PacritinibTyrosine-protein kinase JAK3target
PacritinibSolute carrier family 22 member 2transporter
PacritinibCytochrome P450 2C19enzyme
PacritinibSolute carrier family 22 member 1transporter
PacritinibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
PacritinibATP-dependent translocase ABCB1transporter
PacritinibActivin receptor type-1target
PacritinibTyrosine-protein kinase JAK2target
PacritinibCytochrome P450 1A2enzyme
PacritinibCytochrome P450 3A4enzyme
PacritinibInterleukin-1 receptor-associated kinase 1target
PalbociclibCyclin-dependent kinase 4target
PalbociclibCyclin-dependent kinase 6target
PalbociclibCytochrome P450 3A4enzyme
PalbociclibSulfotransferase 2A1enzyme
PalbociclibATP-dependent translocase ABCB1transporter
PalbociclibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
PalbociclibAlbumincarrier
PalbociclibSolute carrier family 22 member 1transporter
PaltusotineSomatostatin receptor type 2target
PaltusotineUDP-glucuronosyltransferase 1A1enzyme
PaltusotineUDP-glucuronosyltransferase 1A9enzyme
PaltusotineCytochrome P450 3A4enzyme
PaltusotineCytochrome P450 3A5enzyme
PaltusotineBile salt export pumptransporter
PaltusotineMultidrug and toxin extrusion protein 2transporter
PaltusotineMultidrug and toxin extrusion protein 1transporter
PaltusotineBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
PaltusotineATP-dependent translocase ABCB1transporter
PaltusotineCytochrome P450 2C19enzyme
PaltusotineUDP-glucuronosyltransferase 1A3enzyme
PaltusotineCytochrome P450 2D6enzyme
PanobinostatATP-dependent translocase ABCB1transporter
PanobinostatHistone deacetylase 1target
PanobinostatHistone deacetylasetarget
PanobinostatCytochrome P450 3A4enzyme
PanobinostatCytochrome P450 2D6enzyme
PantoprazoleN(G),N(G)-dimethylarginine dimethylaminohydrolase 1target
PantoprazolePotassium-transporting ATPase alpha chain 1target
PantoprazoleOrganic anion transporter 3transporter
PantoprazoleBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
PantoprazoleATP-dependent translocase ABCB1transporter
PantoprazoleCytochrome P450 3A4enzyme
PantoprazoleCytochrome P450 2C19enzyme
PantoprazolePotassium-transporting ATPase subunit betatarget
ParamethasoneGlucocorticoid receptortarget
ParamethasoneCorticosteroid-binding globulintarget
ParamethasoneCytochrome P450 3A5enzyme
ParamethasoneCytochrome P450 3A4enzyme
ParamethasoneCorticosteroid-binding globulincarrier
ParoxetineCytochrome P450 2B6enzyme
ParoxetineATP-dependent translocase ABCB1transporter
ParoxetineCytochrome P450 2C9enzyme
ParoxetineCytochrome P450 1A2enzyme
Paroxetine5-hydroxytryptamine receptor 2Atarget
ParoxetineSodium-dependent noradrenaline transportertarget
ParoxetineSodium-dependent serotonin transportertarget
ParoxetineCytochrome P450 3A4enzyme
ParoxetineAlpha-1 adrenergic receptorstarget
ParoxetineAlpha-2 adrenergic receptorstarget
ParoxetineBeta adrenergic receptortarget
ParoxetineD(2) dopamine receptortarget
ParoxetineHistamine H1 receptortarget
ParoxetineMuscarinic acetylcholine receptortarget
Paroxetine5-hydroxytryptamine receptor 2Btarget
ParoxetineD(1) dopamine receptortarget
ParoxetineCytochrome P450 2C19enzyme
ParoxetineCytochrome P450 2D6enzyme
PasireotideSomatostatin receptor type 3target
PasireotideSomatostatin receptor type 2target
PasireotideSomatostatin receptor type 1target
PasireotideCytochrome P450 3A4enzyme
PasireotideSomatostatin receptor type 5target
PatupiloneTubulin beta chaintarget
PatupiloneTubulin beta-1 chaintarget
PatupiloneTubulin beta-4B chaintarget
PatupiloneTubulin beta-4A chaintarget
PatupiloneTubulin alpha-4A chaintarget
PatupiloneTubulin beta-3 chaintarget
PatupiloneTubulin alpha-8 chaintarget
PatupiloneTubulin alpha-1B chaintarget
PatupiloneTubulin alpha-1A chaintarget
PatupiloneCytochrome P450 3A4enzyme
PatupiloneTubulin alpha 3C/D chaintarget
PatupiloneTubulin alpha-1C chaintarget
PazopanibTyrosine-protein kinase ITK/TSKtarget
PazopanibVascular endothelial growth factor receptor 1target
PazopanibVascular endothelial growth factor receptor 2target
PazopanibVascular endothelial growth factor receptor 3target
PazopanibPlatelet-derived growth factor receptor alphatarget
PazopanibVascular endothelial growth factor receptortarget
PazopanibFibroblast growth factor receptor 1target
PazopanibCytochrome P450 3A4enzyme
PazopanibCytochrome P450 2D6enzyme
PazopanibCytochrome P450 2C8enzyme
PazopanibCytochrome P450 1A2enzyme
PazopanibATP-dependent translocase ABCB1transporter
PazopanibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
PazopanibSolute carrier organic anion transporter family member 1B1transporter
PazopanibPlatelet-derived growth factor receptor betatarget
PazopanibUDP-glucuronosyltransferase 1A1transporter
PazopanibFibroblast growth factor receptor 3target
PazopanibTyrosine-protein kinase Lcktarget
PazopanibMacrophage colony-stimulating factor 1 receptortarget
PazopanibSH2B adapter protein 3target
PazopanibMast/stem cell growth factor receptor Kittarget
PazopanibFibroblast growth factor 1target
PazufloxacinCytochrome P450 1A2enzyme
PazufloxacinDNA gyrase subunit Atarget
PazufloxacinDNA gyrase subunit Btarget
PazufloxacinDNA topoisomerase 4 subunit Atarget
PazufloxacinDNA topoisomerase 2target
PefloxacinDNA gyrase subunit Atarget
PefloxacinDNA topoisomerase 4 subunit Atarget
PefloxacinDNA topoisomerase 2-alphatarget
PefloxacinCytochrome P450 1A2enzyme
PefloxacinDNA topoisomerase 1target
PefloxacinDNA topoisomerase 2-betatarget
Peginterferon alfa-2aInterferon alpha-2target
Peginterferon alfa-2aCytochrome P450 1A2enzyme
Peginterferon alfa-2aInterferon alpha/beta receptor 2target
Peginterferon alfa-2aInterferon alpha/beta receptor 1target
Peginterferon alfa-2bCytochrome P450 1A2enzyme
Peginterferon alfa-2bCytochrome P450 2D6enzyme
Peginterferon alfa-2bCytochrome P450 2C9enzyme
Peginterferon alfa-2bInterferon alpha-2target
Peginterferon alfa-2bInterferon alpha/beta receptor 2target
Peginterferon alfa-2bInterferon alpha/beta receptor 1target
Peppermint oilVoltage-dependent L-type calcium channeltarget
Peppermint oil5-hydroxytryptamine receptor 3target
Peppermint oilCytochrome P450 3A4enzyme
Peppermint oilCytochrome P450 1A2enzyme
PerampanelCytochrome P450 3A5enzyme
PerampanelGlutamate receptor 1target
PerampanelCytochrome P450 1A2enzyme
PerampanelGlutamate receptor 4target
PerampanelGlutamate receptor 3target
PerampanelCytochrome P450 3A4enzyme
PerampanelGlutamate receptor 2target
PerampanelCytochrome P450 2B6enzyme
Pergolide5-hydroxytryptamine receptor 2Atarget
PergolideDopamine receptortarget
PergolideCytochrome P450 3A4enzyme
Pergolide5-hydroxytryptamine receptor 2Ctarget
Pergolide5-hydroxytryptamine receptor 2Btarget
PergolideD(2) dopamine receptortarget
PergolideD(1A) dopamine receptortarget
PergolideD(3) dopamine receptortarget
Pergolide5-hydroxytryptamine receptor 1Atarget
PergolideAlpha-1A adrenergic receptortarget
PergolideAlpha-2 adrenergic receptorstarget
PergolideAlpha-1B adrenergic receptortarget
PergolideAlpha-1D adrenergic receptortarget
PergolideD(4) dopamine receptortarget
PergolideD(1B) dopamine receptortarget
Pergolide5-hydroxytryptamine receptor 1Btarget
Pergolide5-hydroxytryptamine receptor 1Dtarget
PerhexilineSerine/threonine-protein kinase mTORtarget
PerhexilineCarnitine O-palmitoyltransferase 1, muscle isoformtarget
PerhexilineVoltage-gated inwardly rectifying potassium channel KCNH2target
PerhexilineCytochrome P450 3A4enzyme
PerhexilineCytochrome P450 2B6enzyme
PerhexilineCytochrome P450 2D6enzyme
PerhexilineCarnitine O-palmitoyltransferase 2, mitochondrialtarget
PerhexilineCarnitine O-palmitoyltransferase 1, liver isoformtarget
PerphenazineCytochrome P450 1A2enzyme
PerphenazineCytochrome P450 2C18enzyme
PerphenazineCytochrome P450 2C19enzyme
PerphenazineCytochrome P450 2C8enzyme
PerphenazineCytochrome P450 2C9enzyme
PerphenazineCytochrome P450 3A4enzyme
PerphenazineAlbumincarrier
PerphenazineCalmodulintarget
PerphenazineCytochrome P450 2D6enzyme
PerphenazineD(2) dopamine receptortarget
PerphenazineD(1A) dopamine receptortarget
PexidartinibSolute carrier organic anion transporter family member 1B3transporter
PexidartinibSolute carrier organic anion transporter family member 2B1transporter
PexidartinibAlbumincarrier
PexidartinibAlpha-1-acid glycoprotein 1carrier
PexidartinibMast/stem cell growth factor receptor Kittarget
PexidartinibReceptor-type tyrosine-protein kinase FLT3target
PexidartinibPlatelet-derived growth factor receptor betatarget
PexidartinibCytochrome P450 3A4enzyme
PexidartinibUDP-glucuronosyltransferase 1A4enzyme
PexidartinibMacrophage colony-stimulating factor 1 receptortarget
PexidartinibCytochrome P450 2B6enzyme
PexidartinibCytochrome P450 2C9enzyme
PexidartinibSolute carrier organic anion transporter family member 1B1transporter
PexidartinibMultidrug and toxin extrusion protein 2transporter
PexidartinibMultidrug and toxin extrusion protein 1transporter
PexidartinibUDP-glucuronosyltransferase 1A1enzyme
PhencyclidineGlutamate receptor ionotropic, NMDA 3Atarget
PhencyclidineSigma non-opioid intracellular receptor 1target
PhencyclidineCytochrome P450 2B6enzyme
PhencyclidineGlutamate receptor ionotropic, NMDA 1target
PhencyclidineGlutamate receptor ionotropic, NMDA 2Btarget
PhencyclidineGlutamate receptor ionotropic, NMDA 2Atarget
PhenelzineGlutamate decarboxylase 2target
PhenelzineAmine oxidase [copper-containing] 3target
PhenelzineAmine oxidase [flavin-containing] Btarget
PhenelzineAmine oxidase [flavin-containing] Atarget
PhenelzineAmine oxidase [flavin-containing] Aenzyme
PhenelzineAmine oxidase [flavin-containing] Benzyme
PhenelzineCytochrome P450 2E1enzyme
Phenelzine4-aminobutyrate aminotransferase, mitochondrialtarget
PhenelzineAlanine aminotransferase 1target
PhenelzineAlanine aminotransferase 2target
PhenelzineCytochrome P450 2C19enzyme
PhenelzineCytochrome P450 2C8enzyme
PhenelzineCytochrome P450 3A4enzyme
PhenelzineCytochrome P450 3A5enzyme
PhenelzineCytochrome P450 3A7enzyme
PhenelzineCytochrome P450 2D6enzyme
PhenelzineCytochrome P450 3A Subfamilyenzyme
PhenelzineMonoamine oxidasetarget
PhenylbutazoneProstaglandin G/H synthase 2target
PhenylbutazoneProstacyclin synthasetarget
PhenylbutazoneCytochrome P450 2C9enzyme
PhenylbutazoneSolute carrier family 22 member 6transporter
PhenylbutazoneOrganic anion transporter 3transporter
PhenylbutazoneSolute carrier family 22 member 11transporter
PhenylbutazoneCytochrome P450 3A4enzyme
PhenylbutazoneHuman Cyclooxygenasestarget
PhenylbutazoneProstaglandin G/H synthase 1target
Phenylbutyric acidAromatic-amino-acid aminotransferasetarget
Phenylbutyric acidProtein kinase C alpha typetarget
Phenylbutyric acidHistone deacetylase 1target
Phenylbutyric acidHistone deacetylasetarget
PhenytoinCytochrome P450 2D6enzyme
PhenytoinCytochrome P450 2E1enzyme
PhenytoinEpoxide hydrolase 1enzyme
PhenytoinUDP-glucuronosyltransferase 1A4enzyme
PhenytoinCatechol O-methyltransferaseenzyme
PhenytoinNAD(P)H dehydrogenase [quinone] 1enzyme
PhenytoinCytochrome P450 2C18enzyme
PhenytoinVoltage-gated sodium channel alpha subunittarget
PhenytoinCytochrome P450 2A6enzyme
PhenytoinCytochrome P450 1A2enzyme
PhenytoinSodium channel protein type 8 subunit alphatarget
PhenytoinSodium channel protein type 2 subunit alphatarget
PhenytoinVoltage-dependent L-type calcium channeltarget
PhenytoinVoltage-gated inwardly rectifying potassium channel KCNH2target
PhenytoinThyroxine-binding globulincarrier
PhenytoinUDP-glucuronosyltransferase 1A9enzyme
PhenytoinUDP-glucuronosyltransferase 1A6enzyme
PhenytoinUDP-glucuronosyltransferase 1A1enzyme
PhenytoinSodium channel protein type 3 subunit alphatarget
PhenytoinSodium channel regulatory subunit beta-1target
PhenytoinCytochrome P450 3A7enzyme
PhenytoinCytochrome P450 11B1, mitochondrialenzyme
PhenytoinATP-binding cassette sub-family C member 2transporter
PhenytoinATP-dependent translocase ABCB1transporter
PhenytoinSolute carrier organic anion transporter family member 1C1transporter
PhenytoinCytochrome P450 3A4enzyme
PhenytoinAlbumincarrier
PhenytoinCytochrome P450 3A5enzyme
PhenytoinCytochrome P450 2B6enzyme
PhenytoinCytochrome P450 2C9enzyme
PhenytoinCytochrome P450 2C19enzyme
PhenytoinCytochrome P450 2C8enzyme
PhenytoinSodium channel protein type 1 subunit alphatarget
PhenytoinSodium channel protein type 5 subunit alphatarget
PhenytoinNuclear receptor subfamily 1 group I member 2target
Phloxine BCystic fibrosis transmembrane conductance regulatortarget
Phloxine BATP-sensitive potassium channeltarget
Phloxine BPoly(ADP-ribose) glycohydrolasetarget
Phloxine BCytochrome P450 3A4enzyme
Phloxine BATP-dependent translocase ABCB1transporter
Phloxine BIodotyrosine deiodinase 1target
PibrentasvirCytochrome P450 3A Subfamilyenzyme
PibrentasvirUDP-glucuronosyltransferase 1A1enzyme
PibrentasvirATP-dependent translocase ABCB1transporter
PibrentasvirBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
PibrentasvirSolute carrier organic anion transporter family member 1B1transporter
PibrentasvirSolute carrier organic anion transporter family member 1B3transporter
PibrentasvirNonstructural protein 5Atarget
PilocarpineMuscarinic acetylcholine receptor M5target
PilocarpineCytochrome P450 3A4enzyme
PilocarpineSerum paraoxonase/arylesterase 1enzyme
PilocarpineMuscarinic acetylcholine receptor M4target
PilocarpineMuscarinic acetylcholine receptor M1target
PilocarpineMuscarinic acetylcholine receptor M3target
PilocarpineCytochrome P450 2A6enzyme
PilocarpineMuscarinic acetylcholine receptor M2target
PimozideD(2) dopamine receptortarget
PimozideVoltage-gated inwardly rectifying potassium channel KCNH2target
PimozideCytochrome P450 3A4enzyme
PimozideCytochrome P450 1A2enzyme
PimozideCytochrome P450 3A5enzyme
PimozideCytochrome P450 3A7enzyme
PimozideATP-dependent translocase ABCB1transporter
PimozideD(3) dopamine receptortarget
PimozideCytochrome P450 2D6enzyme
PimozideCalmodulintarget
Pimozide5-hydroxytryptamine receptor 2Atarget
PimozideDopamine receptortarget
Pindolol5-hydroxytryptamine receptor 1Atarget
Pindolol5-hydroxytryptamine receptor 1Btarget
PindololCytochrome P450 2D6enzyme
PindololBeta-3 adrenergic receptortarget
PindololUDP-glucuronosyltransferases (UGTs)enzyme
PindololSulfotransferaseenzyme
PindololSolute carrier family 22 member 2transporter
Pindololalpha1-acid glycoproteincarrier
PindololBeta-2 adrenergic receptortarget
PindololBeta-1 adrenergic receptortarget
PioglitazonePeroxisome proliferator-activated receptor gammatarget
PioglitazoneCytochrome P450 2C8enzyme
PioglitazoneCytochrome P450 3A4enzyme
PioglitazoneSolute carrier organic anion transporter family member 1B3transporter
PioglitazoneSolute carrier organic anion transporter family member 1B1transporter
PioglitazoneAmine oxidase [flavin-containing] Btarget
PioglitazoneAlbumincarrier
PioglitazoneCytochrome P450 1A1enzyme
Pipemidic acidCytochrome P450 1A2enzyme
Pipemidic acidDNA topoisomerase 4 subunit Atarget
Pipemidic acidDNA topoisomerase 4 subunit Btarget
Pipemidic acidDNA gyrase subunit Atarget
Pipemidic acidDNA gyrase subunit Btarget
PiperaquineCytochrome P450 3A4enzyme
PiperaquineCytochrome P450 2C19enzyme
PiperaquineCytochrome P450 2C9enzyme
PiperaquineCytochrome P450 2B6enzyme
PiperaquineCytochrome P450 2E1enzyme
PiperaquineCytochrome P450 2D6enzyme
PiperaquineCytochrome P450 2C8enzyme
PiperaquineCytochrome P450 3A Subfamilyenzyme
PiperaquineMultidrug resistance protein 1transporter
PiperaquineVoltage-gated inwardly rectifying potassium channel KCNH2target
PiperineNuclear receptor subfamily 1 group I member 2target
PiperineCytochrome P450 3A4enzyme
PiperineATP-dependent translocase ABCB1transporter
PiperineAmine oxidase [flavin-containing] Atarget
PiperineAmine oxidase [flavin-containing] Btarget
Piperonyl butoxideCytochrome P450target
Piperonyl butoxideCytochrome P450 2B1target
Piperonyl butoxideCytochrome P450 3A5target
Piperonyl butoxideCytochrome P450 1A2target
PipotiazineCytochrome P450 2C19enzyme
PipotiazineAlbumincarrier
PipotiazineSolute carrier family 22 member 1transporter
Pipotiazine5-hydroxytryptamine receptor 1Atarget
Pipotiazine5-hydroxytryptamine receptor 2Atarget
PipotiazineD(2) dopamine receptortarget
PipotiazineCytochrome P450 3A4enzyme
PipotiazineCytochrome P450 2D6enzyme
PipotiazineD(1A) dopamine receptortarget
PirfenidoneCytochrome P450 2D6enzyme
PirfenidoneCytochrome P450 1A2enzyme
PirfenidoneCytochrome P450 2C9enzyme
PirfenidoneCytochrome P450 2C19enzyme
PirfenidoneTransforming growth factor beta-1 proproteintarget
PirfenidoneCytochrome P450 2E1enzyme
PirfenidoneAlbumincarrier
PirfenidoneCytochrome P450 3A4enzyme
PirfenidoneATP-dependent translocase ABCB1transporter
PiroxicamHuman Cyclooxygenasestarget
PiroxicamProstaglandin G/H synthase 1target
PiroxicamProstaglandin G/H synthase 2target
PiroxicamAlbumincarrier
PiroxicamCytochrome P450 2C9enzyme
PiroxicamSolute carrier family 22 member 6transporter
PiroxicamOrganic anion transporter 3transporter
PiroxicamSolute carrier family 22 member 11transporter
PiroxicamCytochrome P450 2C8enzyme
PiroxicamSolute carrier organic anion transporter family member 2B1transporter
PirtobrutinibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
PirtobrutinibATP-dependent translocase ABCB1transporter
PirtobrutinibTyrosine-protein kinase BTKtarget
PirtobrutinibCytochrome P450 3A5enzyme
PirtobrutinibCytochrome P450 2D6enzyme
PirtobrutinibCytochrome P450 2C19enzyme
PirtobrutinibCytochrome P450 2B6enzyme
PirtobrutinibCytochrome P450 1A2enzyme
PirtobrutinibCytochrome P450 2C9enzyme
PirtobrutinibCytochrome P450 2C8enzyme
PirtobrutinibUDP-glucuronosyltransferase 1A9enzyme
PirtobrutinibUDP-glucuronosyltransferase 1A8enzyme
PirtobrutinibCytochrome P450 3A4enzyme
PitolisantAlpha-1-acid glycoprotein 1carrier
PitolisantAlbumincarrier
PitolisantVoltage-gated inwardly rectifying potassium channel KCNH2target
PitolisantSolute carrier family 22 member 1transporter
PitolisantCytochrome P450 2B6enzyme
PitolisantCytochrome P450 1A2enzyme
PitolisantCytochrome P450 2D6enzyme
PitolisantCytochrome P450 3A4enzyme
PitolisantHistamine H3 receptortarget
Poloxamer 188NADH-ubiquinone oxidoreductase chain 1target
Poloxamer 188Albumincarrier
Poloxamer 188Fibrinogentarget
Poloxamer 188Cytochrome c oxidase subunit 8A, mitochondrialtarget
Poloxamer 188ATP-dependent translocase ABCB1transporter
Poloxamer 188Cytochrome P450 3A4enzyme
Poloxamer 188Cytochrome P450 3A Subfamilyenzyme
Poloxamer 188Multidrug resistance-associated protein 1transporter
Polysorbate 80ATP-dependent translocase ABCB1target
Polysorbate 80Cytosolic phospholipase A2enzyme
Polysorbate 80Lysosomal acid lipase/cholesteryl ester hydrolaseenzyme
Polysorbate 80Cytochrome P450 3A Subfamilyenzyme
Polysorbate 80Multidrug resistance-associated protein 1target
Polysorbate 80ATP-dependent translocase ABCB1transporter
Polysorbate 80Multidrug resistance-associated protein 1transporter
Polysorbate 80Cytochrome P450 3A4enzyme
Polysorbate 80Human Carboxylesterasesenzyme
PosaconazoleCytochrome P450 3A4enzyme
PosaconazoleATP-dependent translocase ABCB1transporter
PosaconazoleLanosterol 14-alpha demethylasetarget
PralsetinibCytochrome P450 2D6enzyme
PralsetinibCytochrome P450 3A5enzyme
PralsetinibCytochrome P450 3A4enzyme
PralsetinibFibroblast growth factor receptor 2target
PralsetinibFibroblast growth factor receptor 1target
PralsetinibPlatelet-derived growth factor receptor betatarget
PralsetinibVascular endothelial growth factor receptor 2target
PralsetinibCytochrome P450 1A2enzyme
PralsetinibCytochrome P450 2C8enzyme
PralsetinibCytochrome P450 2C9enzyme
PralsetinibATP-dependent translocase ABCB1transporter
PralsetinibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
PralsetinibSolute carrier organic anion transporter family member 1B1transporter
PralsetinibSolute carrier organic anion transporter family member 1B3transporter
PralsetinibSolute carrier family 22 member 6transporter
PralsetinibMultidrug and toxin extrusion protein 1transporter
PralsetinibHigh affinity nerve growth factor receptortarget
PralsetinibMultidrug and toxin extrusion protein 2transporter
PralsetinibBile salt export pumptransporter
PralsetinibProto-oncogene tyrosine-protein kinase receptor Rettarget
PralsetinibEpithelial discoidin domain-containing receptor 1target
PralsetinibNT-3 growth factor receptortarget
PralsetinibReceptor-type tyrosine-protein kinase FLT3target
PralsetinibTyrosine-protein kinase JAK1target
PralsetinibTyrosine-protein kinase JAK2target
PranlukastNuclear factor NF-kappa-Btarget
PranlukastCytochrome P450 2C9enzyme
PranlukastATP-binding cassette sub-family C member 2transporter
PranlukastCytochrome P450 3A4enzyme
PranlukastCysteinyl leukotriene receptor 1target
PranlukastMucin-2target
PranlukastNuclear factor NF-kappa-B p105 subunittarget
PranlukastEosinophil cationic proteintarget
PranlukastInterleukin-5target
PranlukastTumor necrosis factortarget
PrasteroneATP-binding cassette sub-family C member 4transporter
PrasteroneGABA(A) Receptortarget
PrasteroneBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
PrasteroneMultidrug resistance-associated protein 1transporter
PrasteroneSolute carrier organic anion transporter family member 1A2transporter
PrasteroneSolute carrier organic anion transporter family member 1B1transporter
PrasteroneSolute carrier organic anion transporter family member 2B1transporter
PrasteroneSolute carrier organic anion transporter family member 1B3transporter
PrasteroneSteroid 17-alpha-hydroxylase/17,20 lyaseenzyme
PrasteroneCholesterol oxidaseenzyme
PrasteroneCytochrome P450 3A7enzyme
PrasteronePeroxisome proliferator-activated receptor alphatarget
PrasteroneEstrogen receptortarget
PrasteroneSigma non-opioid intracellular receptor 1target
PrasteroneEstrogen receptor betatarget
PrasteroneNuclear receptor subfamily 1 group I member 2target
PrasteroneNuclear receptor subfamily 1 group I member 3target
PrasteroneGlucose-6-phosphate 1-dehydrogenasetarget
PrasteroneNMDA receptortarget
PrasteroneAndrogen receptortarget
Prasterone17-beta-hydroxysteroid dehydrogenase type 1enzyme
PrasteroneSulfotransferase 2A1enzyme
PrasteroneSulfotransferase 2B1enzyme
Prasterone3 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 1enzyme
PrimaquineCytochrome P450 1A1enzyme
PrimaquineCytochrome P450 1A2enzyme
PrimaquineCytochrome P450 3A4enzyme
PrimaquineKeratin, type II cytoskeletal 7target
PrimaquineCytochrome P450 1B1enzyme
PrimaquineCytochrome P450 2D6enzyme
PrimaquineRibosyldihydronicotinamide dehydrogenase [quinone]target
PrimaquineFe(II)-protoporphyrin IXtarget
PrimaquineATP-dependent translocase ABCB1transporter
ProbenecidATP-binding cassette sub-family C member 11transporter
ProbenecidATP-binding cassette sub-family C member 2transporter
ProbenecidSolute carrier family 22 member 11transporter
ProbenecidSolute carrier organic anion transporter family member 1C1transporter
ProbenecidSolute carrier family 22 member 7transporter
ProbenecidSolute carrier family 22 member 6target
ProbenecidSolute carrier family 22 member 1transporter
ProbenecidATP-binding cassette sub-family C member 3transporter
ProbenecidATP-binding cassette sub-family C member 4transporter
ProbenecidATP-binding cassette sub-family C member 5transporter
ProbenecidMonocarboxylate transporter 2transporter
ProbenecidOrganic cation/carnitine transporter 2transporter
ProbenecidATP-binding cassette sub-family C member 6transporter
ProbenecidMultidrug resistance-associated protein 1transporter
ProbenecidSolute carrier organic anion transporter family member 1A2transporter
ProbenecidMonocarboxylate transporter 1transporter
ProbenecidPannexin-1target
ProbenecidHepatic sodium/bile acid cotransportertransporter
ProbenecidSolute carrier family 22 member 6transporter
ProbenecidSolute carrier family 22 member 10transporter
ProbenecidOrganic anion transporter 3transporter
ProbenecidSolute carrier family 22 member 2transporter
ProbenecidCytochrome P450 2C8enzyme
ProbenecidCytochrome P450 2C9enzyme
ProbenecidUDP-glucuronosyltransferase 1A1enzyme
ProbenecidTaste receptor type 2 member 16target
ProbenecidSolute carrier family 2, facilitated glucose transporter member 9transporter
ProbenecidSolute carrier family 22 member 12transporter
ProbenecidCytochrome P450 3A4enzyme
ProbenecidAlbumincarrier
ProbenecidOrganic anion transporter 3target
ProbenecidSolute carrier family 22 member 11target
ProgesteroneSex hormone-binding globulintarget
ProgesteroneSolute carrier organic anion transporter family member 1B1transporter
ProgesteroneBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
ProgesteroneEstrogen receptor betatarget
ProgesteroneSolute carrier organic anion transporter family member 1B3transporter
ProgesteroneSolute carrier family 22 member 1transporter
ProgesteroneSolute carrier family 22 member 2transporter
ProgesteroneATP-dependent translocase ABCB1transporter
ProgesteroneCytochrome P450 3A7enzyme
ProgesteroneSolute carrier family 22 member 3transporter
ProgesteroneCytochrome P450 3A4enzyme
ProgesteroneCytochrome P450 2C9enzyme
ProgesteroneCytochrome P450 2C19enzyme
ProgesteroneSteroid 17-alpha-hydroxylase/17,20 lyasetarget
ProgesteroneEstrogen receptortarget
ProgesteroneProgesterone receptortarget
ProgesteroneBile salt export pumptransporter
ProgesteroneMultidrug resistance-associated protein 1transporter
ProgesteroneHepatic sodium/bile acid cotransportertransporter
ProgesteroneSteroid 17-alpha-hydroxylase/17,20 lyaseenzyme
ProgesteroneCytochrome P450 1A1enzyme
ProgesteroneCytochrome P450 1B1enzyme
ProgesteroneCytochrome P450 3A5enzyme
ProgesteroneCytochrome P450 2A6enzyme
ProgesteroneCytochrome P450 2D6enzyme
ProgesteroneMineralocorticoid receptortarget
ProgesteroneKappa-type opioid receptortarget
ProgesteroneAlpha-1-acid glycoprotein 1target
ProgesteroneGlucocorticoid receptortarget
ProgesteroneAndrogen receptortarget
ProguanilPeptide deformylase, mitochondrialtarget
ProguanilBifunctional dihydrofolate reductase-thymidylate synthasetarget
ProguanilCytochrome P450 2C19enzyme
ProguanilCytochrome P450 2D6enzyme
ProguanilCytochrome P450 2C9enzyme
PromazineMuscarinic acetylcholine receptor M5target
PromazineD(2) dopamine receptortarget
Promazine5-hydroxytryptamine receptor 2Atarget
Promazine5-hydroxytryptamine receptor 2Ctarget
PromazineAlpha-1A adrenergic receptortarget
PromazineMuscarinic acetylcholine receptor M1target
PromazineHistamine H1 receptortarget
PromazineCytochrome P450 2C19enzyme
PromazineCytochrome P450 1A2enzyme
PromazineCytochrome P450 3A4enzyme
PromazineCytochrome P450 2C9enzyme
PromazineCytochrome P450 2D6enzyme
PromethazineP2 Purinoceptorstarget
PromethazineCytochrome P450 2B6enzyme
PromethazineVoltage-gated sodium channel alpha subunittarget
PromethazineVoltage-gated Potassium Channelstarget
PromethazineATP-binding cassette sub-family C member 3transporter
PromethazineATP-binding cassette sub-family C member 4transporter
PromethazineAlbumincarrier
PromethazineCalmodulintarget
PromethazineNMDA receptortarget
PromethazineAlpha adrenergic receptortarget
PromethazineHistamine H2 receptortarget
PromethazineCytochrome P450 2C9enzyme
PromethazineATP-dependent translocase ABCB1transporter
PromethazineD(2) dopamine receptortarget
PromethazineHistamine H1 receptortarget
PromethazineMuscarinic acetylcholine receptor M4target
PromethazineMuscarinic acetylcholine receptor M1target
PromethazineMuscarinic acetylcholine receptor M5target
PromethazineMuscarinic acetylcholine receptor M2target
PromethazineMuscarinic acetylcholine receptor M3target
PromethazineCytochrome P450 2D6enzyme
PropacetamolSulfotransferase 1E1enzyme
PropacetamolSulfotransferase 1A3enzyme
PropacetamolSulfotransferase 1A1enzyme
PropacetamolUDP-glucuronosyltransferase 1A10enzyme
PropacetamolUDP-glucuronosyltransferase 2B15enzyme
PropacetamolUDP-glucuronosyltransferase 1A9enzyme
PropacetamolUDP-glucuronosyltransferase 1A6enzyme
PropacetamolUDP-glucuronosyltransferase 1A1enzyme
PropacetamolCytochrome P450 2D6enzyme
PropacetamolCytochrome P450 1A2enzyme
PropacetamolCytochrome P450 2E1enzyme
PropacetamolCannabinoid receptor 1target
PropacetamolTransient receptor potential cation channel subfamily V member 1target
PropacetamolProstaglandin G/H synthase 2target
PropacetamolSulfotransferase 2A1enzyme
PropacetamolArylamine N-acetyltransferase 2enzyme
PropacetamolCytochrome P450 2C9enzyme
PropacetamolProstaglandin G/H synthase 1target
PropacetamolCholinesteraseenzyme
PropacetamolCytochrome P450 3A4enzyme
PropafenoneVoltage-gated sodium channel alpha subunittarget
PropafenoneBeta-2 adrenergic receptortarget
PropafenoneBeta-1 adrenergic receptortarget
PropafenoneATP-dependent translocase ABCB1transporter
PropafenoneCytochrome P450 3A4enzyme
PropafenoneCytochrome P450 2D6enzyme
PropafenoneCytochrome P450 1A2enzyme
PropafenoneVoltage-gated inwardly rectifying potassium channel KCNH2target
PropafenoneSodium channel protein type 5 subunit alphatarget
PropofolCytochrome P450 2B6enzyme
PropofolUDP-glucuronosyltransferase 1A1enzyme
PropofolUDP-glucuronosyltransferase 1A9enzyme
PropofolGamma-aminobutyric acid receptor subunit beta-2target
PropofolGamma-aminobutyric acid receptor subunit beta-3target
PropofolAlbumincarrier
PropofolSodium channel protein type 4 subunit alphatarget
PropofolSodium channel protein type 2 subunit alphatarget
PropofolFatty-acid amide hydrolase 1enzyme
PropofolCytochrome P450 2C9enzyme
PropofolUDP-glucuronosyltransferase 1A8enzyme
PropofolCytochrome P450 2E1enzyme
PropofolCytochrome P450 1B1enzyme
PropofolCytochrome P450 1A1enzyme
PropofolCytochrome P450 1A2enzyme
PropofolCytochrome P450 2C18enzyme
PropofolCytochrome P450 2C19enzyme
PropofolCytochrome P450 2C8enzyme
PropofolUDP-glucuronosyltransferase 1A6enzyme
PropofolGABA(A) Receptortarget
PropofolATP-dependent translocase ABCB1transporter
PropranololAlbumincarrier
PropranololAmine oxidase [flavin-containing] Aenzyme
PropranololCytochrome P450 1A1enzyme
PropranololATP-dependent translocase ABCB1transporter
PropranololBeta-1 adrenergic receptortarget
PropranololBeta-2 adrenergic receptortarget
PropranololBeta-3 adrenergic receptortarget
Propranolol5-hydroxytryptamine receptor 1Atarget
Propranolol5-hydroxytryptamine receptor 1Btarget
PropranololCytochrome P450 1A2enzyme
PropranololCytochrome P450 2D6enzyme
PropranololAlpha-1-acid glycoprotein 1carrier
PropranololCytochrome P450 2C19enzyme
PropranololCytochrome P450 3A4enzyme
PropranololSolute carrier family 22 member 2transporter
PropranololCytochrome P450 3A7enzyme
PropranololCytochrome P450 3A5enzyme
PrulifloxacinCytochrome P450 1A2enzyme
PrulifloxacinDNA topoisomerase 4 subunit Atarget
PrulifloxacinDNA gyrase subunit Atarget
PrulifloxacinDNA gyrase subunit Btarget
PyrimethamineFolate receptor alphatarget
PyrimethamineBifunctional dihydrofolate reductase-thymidylate synthasetarget
PyrimethamineDihydrofolate reductasetarget
PyrimethamineCytochrome P450 2C8enzyme
PyrimethamineMultidrug and toxin extrusion protein 2transporter
PyrimethamineBeta-hexosaminidase subunit betatarget
PyrimethamineMultidrug and toxin extrusion protein 1transporter
QuazepamCytochrome P450 2C9enzyme
QuazepamTranslocator proteintarget
QuazepamGABA(A) Receptor Benzodiazepine Binding Sitetarget
QuazepamCytochrome P450 2C19enzyme
QuazepamCytochrome P450 3A4enzyme
QuazepamGABA(A) Receptortarget
QuercetinSolute carrier organic anion transporter family member 1B1transporter
QuercetinAlbumincarrier
QuercetinCarbonyl reductase [NADPH] 1target
QuercetinLysophosphatidylcholine acyltransferase 2target
QuercetinLysophosphatidylcholine acyltransferase 1target
QuercetinSignal transducer and activator of transcription 3target
QuercetinCytochrome P450 2D6enzyme
QuercetinCytochrome P450 3A Subfamilyenzyme
QuercetinCytochrome P450 2C19enzyme
QuercetinCytochrome P450 2E1enzyme
QuercetinCytochrome P450 1A2enzyme
QuercetinCytochrome P450 2C9enzyme
QuercetinAryl hydrocarbon receptortarget
QuercetinNuclear receptor subfamily 1 group I member 2target
QuercetinCCAAT/enhancer-binding protein betatarget
QuercetinRibosyldihydronicotinamide dehydrogenase [quinone]target
QuercetinSex hormone-binding globulintarget
QuercetinUbiquitin-like modifier-activating enzyme 1target
QuercetinSplicing factor 3B subunit 3target
QuercetinRuvB-like 2target
QuercetinHeat shock-related 70 kDa protein 2target
QuercetinHeat shock protein HSP 90-alphatarget
QuercetinEukaryotic translation initiation factor 3 subunit Ftarget
QuercetinCasein kinase II subunit betatarget
QuercetinCasein kinase II subunit alphatarget
QuercetinActin, cytoplasmic 1target
QuercetinCytochrome P450 1B1target
QuercetinEstrogen receptor betatarget
QuercetinTyrosine-protein kinase HCKtarget
QuercetinEstrogen receptortarget
QuercetinSerine/threonine-protein kinase 17Btarget
Quercetin3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZtarget
Quercetin3-hydroxyisobutyryl-CoA hydrolase, mitochondrialtarget
QuercetinHTH-type transcriptional regulator TtgRtarget
QuercetinSerine/threonine-protein kinase pim-1target
QuercetinATP synthase F(1) complex subunit gamma, mitochondrialtarget
QuercetinATP synthase F(1) complex subunit beta, mitochondrialtarget
QuercetinATP synthase F(1) complex subunit alpha, mitochondrialtarget
QuercetinUDP-glycosyltransferase 3A1target
QuercetinPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoformtarget
QuercetinBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
QuercetinMonocarboxylate transporter 1transporter
QuercetinATP-dependent translocase ABCB1transporter
QuercetinSolute carrier organic anion transporter family member 2B1transporter
QuercetinMonocarboxylate transporter 2transporter
QuercetinATP-binding cassette sub-family C member 2transporter
QuercetinMultidrug resistance-associated protein 1transporter
QuercetinCytochrome P450 2C8enzyme
QuinidineCytochrome P450 2D6enzyme
QuinidineSolute carrier family 22 member 2transporter
QuinidineSodium channel protein type 5 subunit alphatarget
QuinidineAlpha-1-acid glycoprotein 1carrier
QuinidineVoltage-gated inwardly rectifying potassium channel KCNH2target
QuinidinePotassium channel subfamily K member 1target
QuinidineVoltage-gated sodium channel alpha subunittarget
QuinidineAlbumincarrier
QuinidineCytochrome P450 2C8enzyme
QuinidineBile salt export pumptransporter
QuinidineAlpha-1D adrenergic receptortarget
QuinidineAlpha-1B adrenergic receptortarget
QuinidineAlpha-1A adrenergic receptortarget
QuinidineCytochrome P450 2C9enzyme
QuinidineCytochrome P450 2B6enzyme
QuinidineSolute carrier organic anion transporter family member 1B1transporter
QuinidineSolute carrier family 22 member 4transporter
QuinidineATP-binding cassette sub-family C member 2transporter
QuinidineOrganic anion transporter 3transporter
QuinidineSolute carrier organic anion transporter family member 1A2transporter
QuinidineATP-dependent translocase ABCB1transporter
QuinidineOrganic cation/carnitine transporter 2transporter
QuinidineSolute carrier family 22 member 1transporter
QuinidinePotassium channel subfamily K member 6target
QuinidineCytochrome P450 3A7enzyme
QuinidineCytochrome P450 3A4enzyme
QuinidineCytochrome P450 1A2enzyme
QuinidineCytochrome P450 1A1enzyme
QuinidineCytochrome P450 2E1enzyme
QuinineCytochrome P450 2D6enzyme
QuininePlatelet glycoprotein IXtarget
QuinineIntermediate conductance calcium-activated potassium channel protein 4target
QuinineCytochrome P450 3A4enzyme
QuinineCytochrome P450 3A5enzyme
QuinineCytochrome P450 1A1enzyme
QuinineCytochrome P450 1A2enzyme
QuinineFe(II)-protoporphyrin IXtarget
QuinineCytochrome P450 2C8enzyme
QuinineCytochrome P450 2C9enzyme
QuinineCytochrome P450 2C19enzyme
QuinineCytochrome P450 2E1enzyme
QuinineCytochrome P450 3A7enzyme
QuinineSolute carrier family 22 member 2transporter
QuinineSolute carrier family 22 member 1transporter
QuinineOrganic cation/carnitine transporter 2transporter
QuinineATP-dependent translocase ABCB1transporter
QuinineSolute carrier organic anion transporter family member 1A2transporter
QuinineSolute carrier family 22 member 4transporter
QuinineSolute carrier organic anion transporter family member 1B1transporter
QuinupristinCytochrome P450 3A4enzyme
QuinupristinLarge ribosomal subunit protein uL22target
QuinupristinLarge ribosomal subunit protein uL10target
Quinupristin23S ribosomal RNAtarget
RabeprazoleCytochrome P450 2D6enzyme
RabeprazoleCytochrome P450 2C9enzyme
RabeprazoleCytochrome P450 1A2enzyme
RabeprazoleCytochrome P450 2C8enzyme
RabeprazoleBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
RabeprazoleCytochrome P450 2C19enzyme
RabeprazoleCytochrome P450 3A4enzyme
RabeprazolePotassium-transporting ATPase alpha chain 1target
RabeprazoleCytochrome P450 1A1enzyme
RaloxifeneUDP-glucuronosyltransferase 1A10enzyme
RaloxifeneATP-dependent translocase ABCB1transporter
RaloxifeneBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
RaloxifeneATP-binding cassette sub-family C member 2transporter
RaloxifeneATP-binding cassette sub-family C member 3transporter
RaloxifeneUDP-glucuronosyltransferase 1A8enzyme
RaloxifeneATP-binding cassette sub-family C member 4transporter
RaloxifeneSolute carrier organic anion transporter family member 1B3transporter
RaloxifeneSolute carrier organic anion transporter family member 1B1transporter
RaloxifeneAlpha-1-acid glycoprotein 1carrier
RaloxifeneAlbumincarrier
RaloxifeneUDP-glucuronosyltransferase 1A1enzyme
RaloxifeneTrefoil factor 1target
RaloxifeneSerpin B9target
RaloxifeneCytochrome P450 3A4enzyme
RaloxifeneAromataseenzyme
RaloxifeneCytochrome P450 2B6enzyme
RaloxifeneCytochrome P450 2C8enzyme
RaloxifeneAldehyde oxidaseenzyme
RaloxifeneEstrogen receptor betatarget
RaloxifeneEstrogen receptortarget
RanitidineSolute carrier family 22 member 1transporter
RanitidineHistamine H2 receptortarget
RanitidineCytochrome P450 1A2enzyme
RanitidineCytochrome P450 2D6enzyme
RanitidineATP-dependent translocase ABCB1transporter
RanitidineOrganic anion transporter 3transporter
RanitidineCytochrome P450 3A4enzyme
RanitidineAcetylcholinesterasetarget
RanitidineSolute carrier family 22 member 2transporter
RanitidineAcetylcholinesteraseenzyme
RanolazineMultidrug and toxin extrusion protein 1transporter
RanolazineAlpha-1-acid glycoprotein 1carrier
RanolazineFatty acidtarget
RanolazineBeta-1 adrenergic receptortarget
RanolazineMultidrug and toxin extrusion protein 2transporter
RanolazinePlasminogentarget
RanolazineSodium channel protein type 5 subunit alphatarget
RanolazineSodium channel protein type 4 subunit alphatarget
RanolazineAlpha-1 adrenergic receptorstarget
RanolazineVoltage gated L-type calcium channeltarget
RanolazineInward rectifier potassium channeltarget
RanolazineSodium channel proteintarget
RanolazineATP-dependent translocase ABCB1transporter
RanolazineBile salt export pumptransporter
RanolazineCytochrome P450 2D6enzyme
RanolazineCytochrome P450 3A4enzyme
ReboxetineCytochrome P450 2D6enzyme
ReboxetineCytochrome P450 3A4enzyme
ReboxetineSodium-dependent noradrenaline transportertarget
ReboxetineATP-dependent translocase ABCB1transporter
RegorafenibHigh affinity nerve growth factor receptortarget
RegorafenibEphrin type-A receptor 2target
RegorafenibRAF proto-oncogene serine/threonine-protein kinasetarget
RegorafenibSerine/threonine-protein kinase B-raftarget
RegorafenibCytochrome P450 2C8enzyme
RegorafenibCytochrome P450 2C9enzyme
RegorafenibCytochrome P450 2B6enzyme
RegorafenibMitogen-activated protein kinase 11target
RegorafenibTyrosine-protein kinase FRKtarget
RegorafenibTyrosine-protein kinase ABL1target
RegorafenibATP-dependent translocase ABCB1transporter
RegorafenibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
RegorafenibUDP-glucuronosyltransferase 1A1enzyme
RegorafenibCytochrome P450 2C19enzyme
RegorafenibMacrophage colony-stimulating factor 1 receptortarget
RegorafenibVascular endothelial growth factor receptortarget
RegorafenibDiscoidin domain-containing receptor 2target
RegorafenibAngiopoietin-1 receptortarget
RegorafenibFibroblast growth factor receptor 2target
RegorafenibFibroblast growth factor receptor 1target
RegorafenibPlatelet-derived growth factor receptor betatarget
RegorafenibPlatelet-derived growth factor receptor alphatarget
RegorafenibMast/stem cell growth factor receptor Kittarget
RegorafenibVascular endothelial growth factor receptor 3target
RegorafenibVascular endothelial growth factor receptor 2target
RegorafenibVascular endothelial growth factor receptor 1target
RegorafenibProto-oncogene tyrosine-protein kinase receptor Rettarget
RegorafenibUDP-glucuronosyltransferase 1A9enzyme
RegorafenibCytochrome P450 3A4enzyme
RelacorilantCytochrome P450 2C9enzyme
RelacorilantCytochrome P450 3A7enzyme
RelacorilantCytochrome P450 3A5enzyme
RelacorilantCytochrome P450 3A4enzyme
RelacorilantBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
RelacorilantCytochrome P450 1A2enzyme
RelacorilantCytochrome P450 2C8enzyme
RelacorilantGlucocorticoid receptortarget
RemacemideVoltage-gated sodium channel alpha subunittarget
RemacemideNMDA receptortarget
RemacemideCytochrome P450 3A4enzyme
RemdesivirCytochrome P450 2C8enzyme
RemdesivirReplicase polyprotein 1abtarget
RemdesivirRNA-directed RNA polymerase Ltarget
RemdesivirCytochrome P450 2D6enzyme
RemdesivirCytochrome P450 3A4enzyme
RemdesivirSolute carrier organic anion transporter family member 1B1transporter
RemdesivirATP-dependent translocase ABCB1transporter
RemdesivirSolute carrier organic anion transporter family member 1B3transporter
RemdesivirBile salt export pumptransporter
RemdesivirATP-binding cassette sub-family C member 4transporter
RemdesivirHepatic sodium/bile acid cotransportertransporter
RemdesivirLiver carboxylesterase 1enzyme
RemdesivirLysosomal protective proteinenzyme
RemdesivirReplicase polyprotein 1abtarget
RemdesivirReplicase polyprotein 1abtarget
RemdesivirMultidrug and toxin extrusion protein 1transporter
RemibrutinibCytochrome P450 3A4enzyme
RemibrutinibATP-dependent translocase ABCB1transporter
RemibrutinibTyrosine-protein kinase BTKtarget
RemibrutinibCytochrome P450 1A2enzyme
RemibrutinibCytochrome P450 2B6enzyme
RemibrutinibCytochrome P450 2C8enzyme
RemibrutinibCytochrome P450 2C9enzyme
RemibrutinibCytochrome P450 2C19enzyme
RemibrutinibSolute carrier family 22 member 1transporter
RemibrutinibSolute carrier family 22 member 2transporter
RemibrutinibOrganic anion transporter 3transporter
RemibrutinibMultidrug and toxin extrusion protein 1transporter
RemibrutinibSolute carrier family 22 member 6transporter
RemibrutinibSolute carrier organic anion transporter family member 1B3transporter
RemibrutinibSolute carrier organic anion transporter family member 1B1transporter
RemibrutinibBile salt export pumptransporter
RemibrutinibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
RemibrutinibCytochrome P450 3A5enzyme
RemibrutinibCytochrome P450 2D6enzyme
RemoxiprideSigma non-opioid intracellular receptor 1target
RemoxiprideCytochrome P450 3A Subfamilyenzyme
RemoxiprideCytochrome P450 2B1enzyme
RemoxiprideCytochrome P450 1A2enzyme
Remoxipridealpha1-acid glycoproteincarrier
RemoxiprideCytochrome P450 2D6enzyme
RemoxiprideD(3) dopamine receptortarget
Remoxipride5-hydroxytryptamine receptor 2Atarget
RemoxiprideD(4) dopamine receptortarget
RemoxiprideD(2) dopamine receptortarget
RepotrectinibUDP-glucuronosyltransferase 1A1enzyme
RepotrectinibProto-oncogene tyrosine-protein kinase ROStarget
RepotrectinibCytochrome P450 3A5enzyme
RepotrectinibCytochrome P450 2C9enzyme
RepotrectinibCytochrome P450 2C19enzyme
RepotrectinibCytochrome P450 2C8enzyme
RepotrectinibHigh affinity nerve growth factor receptortarget
RepotrectinibBDNF/NT-3 growth factors receptortarget
RepotrectinibNT-3 growth factor receptortarget
RepotrectinibCytochrome P450 3A4enzyme
RepotrectinibATP-dependent translocase ABCB1transporter
RepotrectinibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
RepotrectinibSolute carrier organic anion transporter family member 1B1transporter
RepotrectinibMultidrug and toxin extrusion protein 2transporter
RepotrectinibCytochrome P450 2B6enzyme
ResmetiromCytochrome P450 2C8enzyme
ResmetiromUDP-glucuronosyltransferase 1A4enzyme
ResmetiromUDP-glucuronosyltransferase 1A9enzyme
ResmetiromSolute carrier organic anion transporter family member 1B1transporter
ResmetiromSolute carrier organic anion transporter family member 1B3transporter
ResmetiromBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
ResmetiromOrganic anion transporter 3transporter
ResmetiromBile salt export pumptransporter
ResmetiromThyroid hormone receptor betatarget
ResveratrolPolyunsaturated fatty acid lipoxygenase ALOX15target
ResveratrolCytochrome P450 2C9enzyme
ResveratrolCytochrome P450 2C19enzyme
ResveratrolCytochrome P450 2B6enzyme
ResveratrolCytochrome P450 2D6enzyme
ResveratrolTyrosine--tRNA ligase, cytoplasmictarget
ResveratrolFar upstream element-binding protein 2target
ResveratrolRAC-alpha serine/threonine-protein kinasetarget
ResveratrolPeroxisome proliferator-activated receptor gammatarget
ResveratrolPeroxisome proliferator-activated receptor alphatarget
ResveratrolCarbonyl reductase [NADPH] 1target
ResveratrolSolute carrier family 2, facilitated glucose transporter member 1target
ResveratrolNuclear receptor subfamily 1 group I member 3target
ResveratrolNuclear receptor subfamily 1 group I member 2target
ResveratrolC-type lectin domain family 14 member Atarget
ResveratrolMelatonin receptor type 1Btarget
ResveratrolMelatonin receptor type 1Atarget
ResveratrolEstrogen receptortarget
ResveratrolAlpha-synucleintarget
ResveratrolAmyloid-beta precursor proteintarget
ResveratrolAlbumincarrier
ResveratrolIntegrin beta-3target
ResveratrolIntegrin alpha-5target
ResveratrolPhosphatidylinositol 4-kinase type 2-betatarget
ResveratrolAryl hydrocarbon receptortarget
ResveratrolPolyunsaturated fatty acid 5-lipoxygenasetarget
ResveratrolCytochrome P450 1B1enzyme
ResveratrolTransthyretincarrier
ResveratrolRibosyldihydronicotinamide dehydrogenase [quinone]target
ResveratrolProstaglandin G/H synthase 1target
ResveratrolCasein kinase II subunit alphatarget
ResveratrolProstaglandin G/H synthase 2target
ResveratrolNAD-dependent protein deacetylase sirtuin-1target
ResveratrolCytochrome P450 1A1enzyme
ResveratrolCytochrome P450 3A4enzyme
ResveratrolCytochrome P450 1A2enzyme
RevumenibAlbumincarrier
RevumenibCytochrome P450 2C8enzyme
RevumenibMultidrug and toxin extrusion protein 1transporter
RevumenibOrganic anion transporter 3transporter
RevumenibSolute carrier family 22 member 6transporter
RevumenibSolute carrier family 22 member 2transporter
RevumenibSolute carrier family 22 member 1transporter
RevumenibCytochrome P450 3A4enzyme
RevumenibMenintarget
RheinCytochrome P450 2E1enzyme
RheinCytochrome P450 1A2enzyme
RheinPolyunsaturated fatty acid 5-lipoxygenasetarget
RheinCytochrome P450 2C9enzyme
RheinCytochrome P450 2D6enzyme
RheinHeat shock protein HSP 90-alphatarget
RheinArylamine N-acetyltransferasetarget
RheinOxysterols receptor LXR-betatarget
RheinOxysterols receptor LXR-alphatarget
RheinCytochrome P450 3A Subfamilyenzyme
RibociclibCyclin-dependent kinase 6target
RibociclibCytochrome P450 3A4enzyme
RibociclibCyclin-dependent kinase 4target
RidaforolimusSerine/threonine-protein kinase mTORtarget
RidaforolimusCytochrome P450 3A4enzyme
RifampinDNA-directed RNA polymerase subunit betatarget
Rifampinalpha1-acid glycoproteincarrier
RifampinAlbumincarrier
RifampinCytochrome P450 3A5enzyme
RifampinUDP-glucuronosyltransferase 1A9enzyme
RifampinOrganic anion transporter 3transporter
RifampinSolute carrier family 22 member 6transporter
RifampinCytochrome P450 2C8enzyme
RifampinNuclear receptor subfamily 1 group I member 2target
RifampinCytochrome P450 3A4enzyme
RifampinCytochrome P450 1A2enzyme
RifampinUDP-glucuronosyltransferase 1A1enzyme
RifampinCytochrome P450 2C9enzyme
RifampinCytochrome P450 2B6enzyme
RifampinCytochrome P450 2C19enzyme
RifampinATP-binding cassette sub-family C member 3transporter
RifampinATP-binding cassette sub-family C member 5transporter
RifampinATP-dependent translocase ABCB1transporter
RifampinATP-binding cassette sub-family C member 2transporter
RifampinSolute carrier organic anion transporter family member 2B1transporter
RifampinBile salt export pumptransporter
RifampinMultidrug resistance-associated protein 1transporter
RifampinSolute carrier organic anion transporter family member 1A2transporter
RifampinSolute carrier organic anion transporter family member 1B3transporter
RifampinSolute carrier family 22 member 7transporter
RifampinSolute carrier organic anion transporter family member 1B1transporter
RifampinCytochrome P450 2A6enzyme
RifampinCytochrome P450 2E1enzyme
RifampinCytochrome P450 3A43enzyme
RifampinCytochrome P450 3A7enzyme
RifamycinMultidrug and toxin extrusion protein 1transporter
RifamycinCytochrome P450 2B6enzyme
RifamycinCytochrome P450 1A2enzyme
RifamycinATP-dependent translocase ABCB1transporter
RifamycinCytochrome P450 2D6enzyme
RifamycinDNA-directed RNA polymerase subunit beta'target
RifamycinDNA-directed RNA polymerase subunit alphatarget
RifamycinDNA-directed RNA polymerase subunit betatarget
RifamycinDNA-directed RNA polymerase subunit betatarget
RifamycinDNA-directed RNA polymerase subunit beta'target
RifamycinAlbumincarrier
RifamycinSolute carrier organic anion transporter family member 2B1transporter
RifamycinSolute carrier organic anion transporter family member 2A1transporter
RifamycinSolute carrier organic anion transporter family member 1B3transporter
RifamycinSolute carrier organic anion transporter family member 1B1transporter
RifamycinCytochrome P450 3A4enzyme
RifamycinCytochrome P450 2C19enzyme
RifamycinSolute carrier organic anion transporter family member 1A2transporter
RifamycinCytochrome P450 2C8enzyme
RifamycinCytochrome P450 2C9enzyme
RilpivirineSodium channel protein type 10 subunit alphatarget
RilpivirineGag-Pol polyproteintarget
RilpivirineCytochrome P450 2E1enzyme
RilpivirineCytochrome P450 2C8enzyme
RilpivirineCytochrome P450 2C9enzyme
RilpivirineCytochrome P450 2D6enzyme
RilpivirineAlbumincarrier
RilpivirineSolute carrier organic anion transporter family member 1B3transporter
RilpivirineSolute carrier organic anion transporter family member 1B1transporter
RilpivirineBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
RilpivirineATP-dependent translocase ABCB1transporter
RilpivirineCytochrome P450 2B6enzyme
RilpivirineCytochrome P450 2C19enzyme
RilpivirineNuclear receptor subfamily 1 group I member 2target
RilpivirineReverse transcriptase/RNaseHtarget
RilpivirineCytochrome P450 3A4enzyme
RilzabrutinibTyrosine-protein kinase BTKtarget
RilzabrutinibATP-dependent translocase ABCB1transporter
RilzabrutinibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
RilzabrutinibSolute carrier organic anion transporter family member 1B1transporter
RilzabrutinibSolute carrier organic anion transporter family member 1B3transporter
RilzabrutinibBile salt export pumptransporter
RilzabrutinibCytochrome P450 3A4enzyme
RimegepantCytochrome P450 3A4enzyme
RimegepantCytochrome P450 2C9enzyme
RimegepantMultidrug and toxin extrusion protein 1transporter
RimegepantSolute carrier family 22 member 2transporter
RimegepantSolute carrier organic anion transporter family member 1B3transporter
RimegepantOrganic anion transporter 3transporter
RimegepantSolute carrier organic anion transporter family member 1B1transporter
RimegepantBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
RimegepantATP-dependent translocase ABCB1transporter
RimegepantCalcitonin gene-related peptide type 1 receptortarget
RipretinibMast/stem cell growth factor receptor Kittarget
RipretinibPlatelet-derived growth factor receptor betatarget
RipretinibAngiopoietin-1 receptortarget
RipretinibVascular endothelial growth factor receptor 2target
RipretinibSerine/threonine-protein kinase B-raftarget
RipretinibPlatelet-derived growth factor receptor alphatarget
RipretinibCytochrome P450 2E1enzyme
RipretinibCytochrome P450 2C8enzyme
RipretinibPlatelet-derived growth factor receptor alphaenzyme
RipretinibAlbumincarrier
Ripretinibalpha1-acid glycoproteincarrier
RipretinibATP-dependent translocase ABCB1transporter
RipretinibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
RipretinibMultidrug and toxin extrusion protein 1transporter
RipretinibCytochrome P450 3A4enzyme
RipretinibCytochrome P450 2D6enzyme
RisperidoneCytochrome P450 3A4enzyme
RisperidoneATP-dependent translocase ABCB1transporter
RisperidoneAlbumincarrier
RisperidoneAlpha-1-acid glycoprotein 1carrier
Risperidone5-hydroxytryptamine receptor 2Atarget
RisperidoneCytochrome P450 2D6enzyme
RisperidoneD(1A) dopamine receptortarget
Risperidone5-hydroxytryptamine receptor 7target
Risperidone5-hydroxytryptamine receptor 1Atarget
Risperidone5-hydroxytryptamine receptor 1Dtarget
Risperidone5-hydroxytryptamine receptor 2Ctarget
RisperidoneHistamine H1 receptortarget
RisperidoneAlpha-2C adrenergic receptortarget
RisperidoneAlpha-1A adrenergic receptortarget
RisperidoneAlpha-2B adrenergic receptortarget
RisperidoneAlpha-1B adrenergic receptortarget
RisperidoneD(2) dopamine receptortarget
Ritanserin5-hydroxytryptamine receptor 2Ctarget
Ritanserin5-hydroxytryptamine receptor 2Btarget
RitanserinCytochrome P450 2D6enzyme
Ritanserin5-hydroxytryptamine receptor 2Atarget
RitanserinVoltage-dependent N-type calcium channel subunit alpha-1Btarget
RitlecitinibMicrosomal glutathione S-transferase 1enzyme
RitlecitinibGlutathione S-transferase Mu 3enzyme
RitlecitinibGlutathione S-transferase Mu 5enzyme
RitlecitinibMaleylacetoacetate isomeraseenzyme
RitlecitinibGlutathione S-transferase Penzyme
RitlecitinibGlutathione S-transferase Mu 1enzyme
RitlecitinibGlutathione S-transferase A3enzyme
RitlecitinibGlutathione S-transferase A1enzyme
RitlecitinibCytochrome P450 2C9enzyme
RitlecitinibCytochrome P450 1A2enzyme
RitlecitinibCytochrome P450 2C8enzyme
RitlecitinibTyrosine-protein kinase JAK3target
RitlecitinibTyrosine-protein kinase Tectarget
RitlecitinibTyrosine-protein kinase ITK/TSKtarget
RitlecitinibTyrosine-protein kinase TXKtarget
RitlecitinibTyrosine-protein kinase BTKtarget
RitlecitinibGlutathione S-transferase theta-2enzyme
RitlecitinibCytoplasmic tyrosine-protein kinase BMXtarget
RitlecitinibGlutathione S-transferase 3, mitochondrialenzyme
RitlecitinibMicrosomal glutathione S-transferase 2enzyme
RitlecitinibCytochrome P450 3A4enzyme
RitonavirCytochrome P450 3A Subfamilytarget
RitonavirGag-Pol polyproteintarget
RitonavirCytochrome P450 2C9enzyme
RitonavirSolute carrier organic anion transporter family member 1B3transporter
RitonavirAlpha-1-acid glycoprotein 1carrier
RitonavirBile salt export pumptransporter
RitonavirSolute carrier organic anion transporter family member 2B1transporter
RitonavirUDP-glucuronosyltransferases (UGTs)enzyme
RitonavirCytochrome P450 3A7enzyme
RitonavirCytochrome P450 3A5enzyme
RitonavirCytochrome P450 3A4enzyme
RitonavirAlbumincarrier
RitonavirNuclear receptor subfamily 1 group I member 2target
RitonavirCytochrome P450 1A2enzyme
RitonavirSolute carrier organic anion transporter family member 1B1transporter
RitonavirBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
RitonavirSolute carrier organic anion transporter family member 1A2transporter
RitonavirATP-binding cassette sub-family C member 2transporter
RitonavirMultidrug resistance-associated protein 1transporter
RitonavirATP-dependent translocase ABCB1transporter
RitonavirCytochrome P450 2C8enzyme
RitonavirCytochrome P450 2B6enzyme
RitonavirPol polyproteintarget
RitonavirCytochrome P450 2D6enzyme
RitonavirCytochrome P450 2C19enzyme
RivoglitazonePeroxisome proliferator-activated receptor gammatarget
RivoglitazoneCytochrome P450 2C8enzyme
RivoglitazoneCytochrome P450 3A4enzyme
Rizatriptan5-hydroxytryptamine receptor 1Dtarget
Rizatriptan5-hydroxytryptamine receptor 7target
Rizatriptan5-hydroxytryptamine receptor 1Etarget
Rizatriptan5-hydroxytryptamine receptor 1Btarget
Rizatriptan5-hydroxytryptamine receptor 1Ftarget
RizatriptanAmine oxidase [flavin-containing] Aenzyme
RizatriptanCytochrome P450 2D6enzyme
Rizatriptan5-hydroxytryptamine receptor 1Atarget
RofecoxibProstaglandin G/H synthase 2target
RofecoxibElastintarget
RofecoxibCytochrome P450 3A4enzyme
RofecoxibCytochrome P450 2C9enzyme
RofecoxibCytochrome P450 2C8enzyme
RofecoxibProstaglandin G/H synthase 1enzyme
RofecoxibATP-binding cassette sub-family C member 4transporter
RofecoxibCytochrome P450 1A2enzyme
RokitamycinCytochrome P450 3A4enzyme
RokitamycinCholinesteraseenzyme
RolapitantATP-dependent translocase ABCB1transporter
RolapitantBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
RolapitantCytochrome P450 3A4enzyme
RolapitantCytochrome P450 2D6enzyme
RolapitantSubstance-P receptortarget
Ropeginterferon alfa-2bCytochrome P450 1A2enzyme
Ropeginterferon alfa-2bCytochrome P450 2D6enzyme
Ropeginterferon alfa-2bInterferon alpha/beta receptor (IFNAR)target
Ropeginterferon alfa-2bCytochrome P450 2A6enzyme
RosiglitazonePeroxisome proliferator-activated receptor gammatarget
RosiglitazoneCytochrome P450 2C8enzyme
RosiglitazoneCytochrome P450 2C9enzyme
RosiglitazoneLong-chain-fatty-acid--CoA ligase 4target
RosiglitazoneSolute carrier organic anion transporter family member 1B1transporter
RosiglitazoneProstaglandin G/H synthase 1enzyme
RosiglitazoneCytochrome P450 1A2enzyme
RosiglitazoneCytochrome P450 2D6enzyme
RosiglitazoneAlbumincarrier
RosiglitazoneRetinoic acid receptor RXR-alphatarget
RosiglitazoneCytochrome P450 3A4enzyme
RosiglitazoneBile salt export pumptransporter
RosiglitazoneCytochrome P450 2B6enzyme
RosiglitazoneCytochrome P450 2E1enzyme
RosiglitazoneHepatic sodium/bile acid cotransportertransporter
RosoxacinCytochrome P450 1A2enzyme
RosoxacinDNA topoisomerase 2-betatarget
RosoxacinDNA topoisomerase 2-alphatarget
RosoxacinDNA gyrase subunit Btarget
RosoxacinDNA topoisomerase 4 subunit Atarget
RosuvastatinAlbumincarrier
RosuvastatinATP-binding cassette sub-family C member 2transporter
RosuvastatinOrganic anion transporter 3transporter
RosuvastatinHepatic sodium/bile acid cotransportertransporter
RosuvastatinIntegrin alpha-Ltarget
RosuvastatinBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
RosuvastatinBile salt export pumptransporter
RosuvastatinSolute carrier organic anion transporter family member 1B1transporter
RosuvastatinCystine/glutamate transportertransporter
RosuvastatinSolute carrier organic anion transporter family member 2B1transporter
RosuvastatinSolute carrier organic anion transporter family member 1B3transporter
RosuvastatinSolute carrier organic anion transporter family member 1A2transporter
RosuvastatinATP-binding cassette sub-family C member 4transporter
RosuvastatinCytochrome P450 2C9enzyme
Rosuvastatin3-hydroxy-3-methylglutaryl-coenzyme A reductasetarget
RotigotineCytochrome P450 2C19enzyme
RotigotineAlpha-2B adrenergic receptortarget
RotigotineCytochrome P450 3A4enzyme
RotigotineCytochrome P450 2D6enzyme
RotigotineD(1A) dopamine receptortarget
Rotigotine5-hydroxytryptamine receptor 1Atarget
RotigotineD(2) dopamine receptortarget
RotigotineD(4) dopamine receptortarget
RotigotineD(1B) dopamine receptortarget
RotigotineD(3) dopamine receptortarget
RoxithromycinLarge ribosomal subunit protein uL10target
RoxithromycinATP-dependent translocase ABCB1target
RoxithromycinCytochrome P450 3A4enzyme
RoxithromycinCytochrome P450 2B6enzyme
RucaparibPoly [ADP-ribose] polymerasestarget
RucaparibUDP-glucuronosyltransferase 1A1enzyme
RucaparibCytochrome P450 2C8enzyme
RucaparibCytochrome P450 2C9enzyme
RucaparibCytochrome P450 2C19enzyme
RucaparibCytochrome P450 3A43enzyme
RucaparibCytochrome P450 3A7enzyme
RucaparibCytochrome P450 3A5enzyme
RucaparibOrganic anion transporter 3transporter
RucaparibSolute carrier family 22 member 6transporter
RucaparibSolute carrier organic anion transporter family member 1B3transporter
RucaparibSolute carrier organic anion transporter family member 1B1transporter
RucaparibATP-binding cassette sub-family C member 4transporter
RucaparibSolute carrier family 22 member 1transporter
RucaparibMultidrug and toxin extrusion protein 2transporter
RucaparibMultidrug and toxin extrusion protein 1transporter
RucaparibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
RucaparibATP-dependent translocase ABCB1transporter
RucaparibCytochrome P450 3A4enzyme
RucaparibCytochrome P450 1A2enzyme
RucaparibCytochrome P450 2D6enzyme
RucaparibProtein mono-ADP-ribosyltransferase PARP3target
RucaparibPoly [ADP-ribose] polymerase 2target
RucaparibPoly [ADP-ribose] polymerase 1target
RufinamideCytochrome P450 3A4enzyme
RufinamideMetabotropic glutamate receptor 5target
RufinamideLiver carboxylesterase 1enzyme
RufinamideSodium channel protein type 9 subunit alphatarget
RufinamideAlbumincarrier
RufinamideVoltage-gated sodium channel alpha subunittarget
RufinamideCytochrome P450 2E1enzyme
RufloxacinDNA gyrase subunit Atarget
RufloxacinCytochrome P450 1A2enzyme
RutinAldo-keto reductase family 1 member C3target
RutinCytochrome P450 3A4enzyme
RutinCarbonyl reductase [NADPH] 1target
SafinamideCytochrome P450 3A5enzyme
SafinamideCytochrome P450 2C19enzyme
SafinamideCytochrome P450 2D6enzyme
SafinamideCytochrome P450 1A2enzyme
SafinamideCytochrome P450 1A1enzyme
SafinamideCytochrome P450 3A4enzyme
SafinamideSolute carrier organic anion transporter family member 3A1transporter
SafinamideBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
SafinamideAmine oxidase [flavin-containing] Btarget
SafinamideAmine oxidase [flavin-containing] Aenzyme
SagopiloneCytochrome P450 3A4enzyme
SagopiloneTubulintarget
SalmeterolSolute carrier family 22 member 2transporter
SalmeterolBeta-2 adrenergic receptortarget
SalmeterolCytochrome P450 3A4enzyme
SalmeterolCytochrome P450 2C8enzyme
SalmeterolCytochrome P450 3A5enzyme
SalmeterolCytochrome P450 3A7enzyme
SalmeterolSolute carrier family 22 member 1transporter
SalmeterolBeta-3 adrenergic receptortarget
SalmeterolAlbumincarrier
Salmeterolalpha1-acid glycoproteincarrier
SalmeterolSolute carrier family 22 member 3transporter
SalmeterolBeta-1 adrenergic receptortarget
SaquinavirPol polyproteintarget
SaquinavirCytochrome P450 3A4enzyme
SaquinavirCytochrome P450 3A5enzyme
SaquinavirAlpha-1-acid glycoprotein 1carrier
SaquinavirAlbumincarrier
SaquinavirCytochrome P450 3A7enzyme
SaquinavirATP-dependent translocase ABCB1transporter
SaquinavirSolute carrier family 22 member 1transporter
SaquinavirSolute carrier organic anion transporter family member 1A2transporter
SaquinavirBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
SaquinavirSolute carrier organic anion transporter family member 1B1transporter
SaquinavirMultidrug resistance-associated protein 1transporter
SaquinavirATP-binding cassette sub-family C member 2transporter
SaquinavirCytochrome P450 2C8enzyme
SaquinavirCytochrome P450 2D6enzyme
SaquinavirSolute carrier organic anion transporter family member 2B1transporter
SaquinavirBile salt export pumptransporter
SaquinavirGag-Pol polyproteintarget
SaracatinibCytochrome P450 3A4enzyme
SaracatinibProto-oncogene tyrosine-protein kinase Srctarget
SaracatinibTyrosine-protein kinase ABL1target
SarafloxacinDNA gyrase subunit Atarget
SarafloxacinCytochrome P450 1A2enzyme
SarafloxacinCatalaseenzyme
SarilumabCytochrome P450 3A4enzyme
SarilumabInterleukin-6 receptor subunit alphatarget
SarilumabHigh affinity immunoglobulin gamma Fc receptor Itarget
SarilumabLow affinity immunoglobulin gamma Fc region receptor II-atarget
SarilumabLow affinity immunoglobulin gamma Fc region receptor II-btarget
SarilumabLow affinity immunoglobulin gamma Fc region receptor III-Atarget
SarilumabLow affinity immunoglobulin gamma Fc region receptor III-Btarget
SarilumabInterleukin-6 receptor subunit betatarget
Saw palmetto3-oxo-5-alpha-steroid 4-dehydrogenase 1target
Saw palmetto3-oxo-5-alpha-steroid 4-dehydrogenase 2target
Saw palmettoAndrogen receptortarget
Saw palmetto3-oxo-5-alpha-steroid 4-dehydrogenasetarget
Saw palmettoCytochrome P450 2C8enzyme
SebetralstatCytochrome P450 3A4enzyme
SebetralstatCytochrome P450 2C8enzyme
SebetralstatCytochrome P450 2C9enzyme
SebetralstatPlasma kallikreintarget
SebetralstatATP-dependent translocase ABCB1transporter
SebetralstatBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
SebetralstatSolute carrier organic anion transporter family member 1B1transporter
SebetralstatSolute carrier organic anion transporter family member 1B3transporter
SebetralstatOrganic anion transporter 3transporter
SebetralstatSolute carrier family 22 member 2transporter
SebetralstatMultidrug and toxin extrusion protein 1transporter
SebetralstatMultidrug and toxin extrusion protein 2transporter
SebetralstatBile salt export pumptransporter
SecnidazoleCytochrome P450 3A5enzyme
SecnidazoleCytochrome P450 2C19enzyme
SecnidazoleCytochrome P450 3A4enzyme
SelamectinAnoctamin-1target
SelamectinATP-dependent translocase ABCB1transporter
SelamectinCytochrome P450 3A4enzyme
SelegilineAmine oxidase [flavin-containing] Btarget
SelegilineCytochrome P450 2B6enzyme
SelegilineAmine oxidase [flavin-containing] Atarget
SelegilineCytochrome P450 2A6enzyme
SelegilineCytochrome P450 3A4enzyme
SelegilineATP-dependent translocase ABCB1transporter
SelegilineCytochrome P450 1A2enzyme
SelegilineCytochrome P450 2C19enzyme
SelegilineCytochrome P450 2C8enzyme
SelegilineCytochrome P450 2C9enzyme
SelegilineCytochrome P450 2D6enzyme
SelegilineSubstance-P receptortarget
SelpercatinibProto-oncogene tyrosine-protein kinase receptor Rettarget
SelpercatinibVascular endothelial growth factor receptor 1target
SelpercatinibMultidrug and toxin extrusion protein 1transporter
SelpercatinibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
SelpercatinibATP-dependent translocase ABCB1transporter
SelpercatinibCytochrome P450 3A Subfamilyenzyme
SelpercatinibCytochrome P450 2C8enzyme
SelpercatinibCytochrome P450 3A4enzyme
SelpercatinibFibroblast growth factor receptor 3target
SelpercatinibFibroblast growth factor receptor 2target
SelpercatinibFibroblast growth factor receptor 1target
SelpercatinibVascular endothelial growth factor receptor 3target
SeproxetineSodium-dependent dopamine transportertarget
SeproxetineSodium-dependent serotonin transportertarget
SeproxetineSodium-dependent noradrenaline transportertarget
SeproxetineCytochrome P450 3A4enzyme
SeproxetineCytochrome P450 2C19enzyme
SeproxetineCytochrome P450 2C9enzyme
SeproxetineCytochrome P450 3A7enzyme
SeproxetineCytochrome P450 3A5enzyme
SeratrodastThromboxane A2 receptortarget
SeratrodastCytochrome P450 2A6enzyme
SeratrodastProstaglandin G/H synthase 1enzyme
SeratrodastUDP-glucuronosyltransferase 1A9enzyme
SeratrodastCytochrome P450 2B6enzyme
SeratrodastCytochrome P450 2C19enzyme
SeratrodastCytochrome P450 2C8enzyme
SeratrodastCytochrome P450 3A4enzyme
SeratrodastCytochrome P450 2C9enzyme
SertralineCytochrome P450 2E1enzyme
SertralineEquilibrative nucleoside transporter 4target
SertralineSodium-dependent noradrenaline transportertarget
SertralineSigma receptortarget
SertralineAlbumincarrier
SertralineATP-dependent translocase ABCB1transporter
SertralineAmine oxidase [flavin-containing] Aenzyme
SertralineAmine oxidase [flavin-containing] Benzyme
SertralineCytochrome P450 3A4enzyme
SertralineCytochrome P450enzyme
SertralineSodium-dependent dopamine transportertarget
SertralineCytochrome P450 2D6enzyme
SertralineCytochrome P450 2C9enzyme
SertralineCytochrome P450 2C19enzyme
SertralineCytochrome P450 2B6enzyme
SertralineSodium-dependent serotonin transportertarget
SevabertinibCytochrome P450 3A Subfamilyenzyme
SevabertinibCytochrome P450 1A1enzyme
SevabertinibCytochrome P450 2C8enzyme
SevabertinibReceptor tyrosine-protein kinase erbB-2target
SevabertinibEpidermal growth factor receptortarget
SevabertinibATP-dependent translocase ABCB1transporter
SevabertinibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
SevabertinibMultidrug and toxin extrusion protein 1transporter
SevabertinibMultidrug and toxin extrusion protein 2transporter
SeviteronelAndrogen receptortarget
SeviteronelSteroid 17-alpha-hydroxylase/17,20 lyasetarget
SildenafilProgrammed cell death 1 ligand 1target
SildenafilOrnithine decarboxylasetarget
SildenafilPlasma protease C1 inhibitortarget
SildenafilSolute carrier organic anion transporter family member 1B1transporter
SildenafilCytochrome P450 2E1enzyme
SildenafilCytochrome P450 2D6enzyme
SildenafilCytochrome P450 2C19enzyme
SildenafilATP-binding cassette sub-family C member 10transporter
SildenafilATP-binding cassette sub-family C member 5transporter
SildenafilATP-binding cassette sub-family C member 4transporter
SildenafilCytochrome P450 3A7enzyme
SildenafilCytochrome P450 3A5enzyme
SildenafilCytochrome P450 3A4enzyme
SildenafilRetinal cone rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit gammatarget
SildenafilRod cGMP 3',5'-cyclic phosphodiesterase subunit gammatarget
SildenafilCytochrome P450 2C9enzyme
SildenafilcGMP-specific 3',5'-cyclic phosphodiesterasetarget
SildenafilATP-dependent translocase ABCB1transporter
SiltuximabInterleukin-6target
SiltuximabCytochrome P450 3A4enzyme
SimeprevirBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
SimeprevirNS3 proteasetarget
SimeprevirAlbumincarrier
SimeprevirCytochrome P450 1A2enzyme
SimeprevirATP-dependent translocase ABCB1transporter
SimeprevirSolute carrier organic anion transporter family member 1B1transporter
SimeprevirSolute carrier organic anion transporter family member 1B3transporter
SimeprevirCytochrome P450 3A4enzyme
SimeprevirATP-binding cassette sub-family C member 2transporter
SimeprevirGenome polyproteintarget
SimeprevirSolute carrier organic anion transporter family member 2B1transporter
SimeprevirGenome polyproteintarget
SimeprevirBile salt export pumptransporter
SimeprevirHepatic sodium/bile acid cotransportertransporter
Simvastatin3-hydroxy-3-methylglutaryl-coenzyme A reductasetarget
SimvastatinCytochrome P450 3A4enzyme
SimvastatinCytochrome P450 2C8enzyme
SimvastatinCytochrome P450 2C9enzyme
SimvastatinCytochrome P450 3A5enzyme
SimvastatinATP-dependent translocase ABCB1transporter
SimvastatinSolute carrier organic anion transporter family member 1A2transporter
SimvastatinSolute carrier organic anion transporter family member 1B1transporter
SimvastatinCytochrome P450 2B6enzyme
SimvastatinCytochrome P450 2D6enzyme
SimvastatinUDP-glucuronosyltransferase 1A1enzyme
SimvastatinUDP-glucuronosyltransferase 1A3enzyme
SimvastatinLiver carboxylesterase 1enzyme
SimvastatinUDP-glucuronosyltransferase 2B7enzyme
SimvastatinATP-binding cassette sub-family C member 2transporter
SimvastatinIntegrin alpha-Ltarget
SimvastatinBile salt export pumptransporter
SimvastatinCytochrome P450 2C19enzyme
SimvastatinSolute carrier organic anion transporter family member 2B1transporter
SimvastatinSolute carrier organic anion transporter family member 1B3transporter
SimvastatinHistone deacetylase 2target
SimvastatinCocaine esteraseenzyme
SitafloxacinCytochrome P450 1A2enzyme
SitafloxacinDNA gyrase subunit Atarget
SitafloxacinDNA topoisomerase 4 subunit Atarget
SitafloxacinDNA gyrase subunit Btarget
SitaxentanEndothelin receptor type Btarget
SitaxentanCytochrome P450 2C19enzyme
SitaxentanCytochrome P450 2C9enzyme
SitaxentanCytochrome P450 3A4enzyme
SitaxentanEndothelin-1 receptortarget
SN-38Cytochrome P450 3A4enzyme
SN-38DNA topoisomerase 1target
SofpironiumMultidrug and toxin extrusion protein 1transporter
SofpironiumSolute carrier family 22 member 2transporter
SofpironiumSolute carrier family 22 member 1transporter
SofpironiumMuscarinic acetylcholine receptortarget
SofpironiumCytochrome P450 3A4enzyme
SofpironiumCytochrome P450 2D6enzyme
SofpironiumMuscarinic acetylcholine receptor M3target
SolithromycinArylamine N-acetyltransferase 2enzyme
SolithromycinArylamine N-acetyltransferase 1enzyme
SolithromycinATP-dependent translocase ABCB1transporter
SolithromycinCytochrome P450 3A7enzyme
SolithromycinCytochrome P450 3A5enzyme
SolithromycinBacterial 50S ribosomal proteintarget
SolithromycinCytochrome P450 3A4enzyme
SomapacitanAlbumincarrier
SomapacitanCytochrome P450 2C19enzyme
SomapacitanCytochrome P450 1A2enzyme
SomapacitanCytochrome P450 2C12, female-specificenzyme
Somapacitan11-beta-hydroxysteroid dehydrogenase 1enzyme
SomapacitanGrowth hormone receptortarget
SomatostatinSomatostatin receptortarget
SomatostatinDelta-type opioid receptortarget
SomatostatinMu-type opioid receptortarget
SomatostatinCytochrome P450 3A4enzyme
SomatostatinATP-dependent translocase ABCB1transporter
SomatostatinSomatostatin receptor type 5target
SomatostatinSomatostatin receptor type 4target
SomatostatinSomatostatin receptor type 3target
SomatostatinSomatostatin receptor type 2target
SomatostatinSomatostatin receptor type 1target
SomatotropinGrowth hormone receptortarget
SomatotropinProlactin receptortarget
SomatotropinCytochrome P450 1A2enzyme
SomatotropinCytochrome P450 2C19enzyme
SomatotropinATP-dependent translocase ABCB1transporter
SonrotoclaxBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
SonrotoclaxATP-dependent translocase ABCB1transporter
SonrotoclaxApoptosis regulator Bcl-2target
SonrotoclaxCytochrome P450 2C8enzyme
SonrotoclaxCytochrome P450 3A7enzyme
SonrotoclaxCytochrome P450 3A5enzyme
SonrotoclaxCytochrome P450 3A4enzyme
Sophora flavescens rootCytochrome P450 3A4enzyme
Sophora flavescens rootCytochrome P450 3A4target
SorafenibCytochrome P450 2C8enzyme
SorafenibFibroblast growth factor receptor 1target
SorafenibATP-dependent translocase ABCB1transporter
SorafenibATP-binding cassette sub-family C member 4transporter
SorafenibCytochrome P450 2C9enzyme
SorafenibCytochrome P450 3A7enzyme
SorafenibCytochrome P450 3A5enzyme
SorafenibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
SorafenibCytochrome P450 2B6enzyme
SorafenibUDP-glucuronosyltransferase 1A9enzyme
SorafenibCytochrome P450 3A4enzyme
SorafenibVascular endothelial growth factor receptor 2target
SorafenibMast/stem cell growth factor receptor Kittarget
SorafenibPlatelet-derived growth factor receptor betatarget
SorafenibVascular endothelial growth factor receptor 3target
SorafenibRAF proto-oncogene serine/threonine-protein kinasetarget
SorafenibReceptor-type tyrosine-protein kinase FLT3target
SorafenibSerine/threonine-protein kinase B-raftarget
SorafenibATP-binding cassette sub-family C member 2transporter
SorafenibVascular endothelial growth factor receptortarget
SorafenibEpidermal growth factor receptortarget
SorafenibSolute carrier organic anion transporter family member 1B1transporter
SorafenibVascular endothelial growth factor receptor 1target
SorafenibProto-oncogene tyrosine-protein kinase receptor Rettarget
SorafenibCytochrome P450 1A2enzyme
SorafenibRalA-binding protein 1transporter
SorafenibUDP-glucuronosyltransferase 1A1enzyme
SorafenibCytochrome P450 2D6enzyme
SorafenibCytochrome P450 2C19enzyme
SotagliflozinSolute carrier organic anion transporter family member 1B1transporter
SotagliflozinSolute carrier organic anion transporter family member 1B3transporter
SotagliflozinATP-binding cassette sub-family C member 2transporter
SotagliflozinATP-dependent translocase ABCB1transporter
SotagliflozinBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
SotagliflozinCytochrome P450 2D6enzyme
SotagliflozinSodium/glucose cotransporter 1target
SotagliflozinSodium/glucose cotransporter 2target
SotagliflozinUDP-glucuronosyltransferase 2B7enzyme
SotagliflozinUDP-glucuronosyltransferase 1A1enzyme
SotagliflozinUDP-glucuronosyltransferase 1A9enzyme
SotagliflozinCytochrome P450 3A4enzyme
SparfloxacinATP-binding cassette sub-family C member 2transporter
SparfloxacinDNA gyrase subunit Atarget
SparfloxacinDNA topoisomerase 4 subunit Atarget
SparfloxacinDNA topoisomerase 2-alphatarget
SparfloxacinOrganic cation/carnitine transporter 2transporter
SparfloxacinATP-dependent translocase ABCB1transporter
SparfloxacinCytochrome P450 1A2enzyme
SparfloxacinDNA gyrase subunit Atarget
SparfloxacinDNA gyrase subunit Btarget
SparsentanCytochrome P450 3A4enzyme
SparsentanBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
SparsentanEndothelin-1 receptortarget
SparsentanType-2 angiotensin II receptortarget
SparsentanCytochrome P450 2B6enzyme
SparsentanCytochrome P450 2C9enzyme
SparsentanCytochrome P450 2C19enzyme
SparsentanATP-dependent translocase ABCB1transporter
SparsentanSolute carrier organic anion transporter family member 1B3transporter
SparsentanOrganic anion transporter 3transporter
SparsentanType-1 angiotensin II receptortarget
SparteineCytochrome P450 2D6enzyme
SpiramycinLarge ribosomal subunit protein uL3target
SpironolactoneVoltage-dependent L-type calcium channeltarget
SpironolactoneMineralocorticoid receptortarget
SpironolactoneCytochrome P450 2C8enzyme
SpironolactoneATP-binding cassette sub-family C member 2transporter
SpironolactoneATP-dependent translocase ABCB1transporter
SpironolactoneSolute carrier organic anion transporter family member 1A2transporter
SpironolactoneCytochrome P450 11B1, mitochondrialenzyme
SpironolactoneAndrogen receptortarget
SpironolactoneProgesterone receptortarget
SpironolactoneGlucocorticoid receptortarget
SpironolactoneNuclear receptor subfamily 1 group I member 2target
SpironolactoneBile salt export pumptransporter
SpironolactoneAlbumincarrier
Spironolactonealpha1-acid glycoproteincarrier
SpironolactoneEstrogen receptortarget
SpironolactoneCytochrome P450 11B2, mitochondrialenzyme
St. John's WortCytochrome P450 2C19enzyme
St. John's WortSodium-dependent noradrenaline transportertarget
St. John's WortCytochrome P450 2D6enzyme
St. John's WortCytochrome P450 3A4enzyme
St. John's WortATP-dependent translocase ABCB1transporter
StiripentolCytochrome P450 2C19enzyme
StiripentolCytochrome P450 2D6enzyme
StiripentolCytochrome P450 3A4enzyme
StiripentolCytochrome P450 1A2enzyme
StiripentolCytochrome P450 2C9enzyme
StiripentolGABA(A) Receptortarget
StiripentolL-lactate dehydrogenase A chaintarget
StiripentolL-lactate dehydrogenase B chaintarget
StiripentolCytochrome P450 2B6enzyme
StiripentolCytochrome P450 2C8enzyme
StiripentolATP-dependent translocase ABCB1transporter
StiripentolBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
StiripentolGamma-aminobutyric acid receptor subunit gamma-3target
SulconazoleLanosterol 14-alpha demethylasetarget
SulconazoleCytochrome P450 1A2enzyme
SulconazoleCytochrome P450 2C9enzyme
SulconazoleCytochrome P450 2D6enzyme
SulconazoleLanosterol 14-alpha demethylasetarget
SulfadiazineCytochrome P450 2C9enzyme
Sulfadiazinedihydropteroate synthasetarget
SulfadiazineDihydropteroate synthasetarget
SulfadiazineCytochrome P450 3A4enzyme
SulfadiazineCytochrome P450 2C8enzyme
SulfadimethoxineDihydropteroate synthasetarget
SulfadimethoxineAlbumincarrier
SulfadimethoxineCytochrome P450 2C9enzyme
SulfamethizoleCytochrome P450 2C9enzyme
SulfamethizoleAlbumincarrier
SulfamethizoleDihydropteroate synthasetarget
SulfamethoxazoleCytochrome P450 2C9enzyme
SulfamethoxazoleArylamine N-acetyltransferase 1enzyme
SulfamethoxazoleArylamine N-acetyltransferase 2enzyme
SulfamethoxazoleAlbumincarrier
SulfamethoxazoleDihydropteroate synthasetarget
SulfamethoxazoleCytochrome P450 3A4enzyme
SulfamethoxazoleBile salt export pumptransporter
Sulfamoxoledihydropteroate synthasetarget
SulfamoxoleCytochrome P450 2C9enzyme
SulfanilamideDihydropteroate synthasetarget
SulfaphenazoleCytochrome P450 2C9target
SulfaphenazoleDihydropteroate synthasetarget
SulfaphenazoleCytochrome P450 2D6enzyme
SulfaphenazoleCytochrome P450 2C8enzyme
SulfaphenazoleCytochrome P450 2B6enzyme
SulfaphenazoleCytochrome P450 2C9enzyme
SulfapyridineDihydropteroate synthasetarget
SulfapyridineCytochrome P450 2C9enzyme
SulfapyridineDihydropteroate synthase type-1target
SulfinpyrazoneBile salt export pumptransporter
SulfinpyrazoneSolute carrier family 22 member 12target
SulfinpyrazoneCytochrome P450 2C8enzyme
SulfinpyrazoneCytochrome P450 2B6enzyme
SulfinpyrazoneCytochrome P450 3A4enzyme
SulfinpyrazoneATP-binding cassette sub-family C member 2transporter
SulfinpyrazoneMultidrug resistance-associated protein 1transporter
SulfinpyrazoneATP-binding cassette sub-family C member 6transporter
SulfinpyrazoneATP-binding cassette sub-family C member 5transporter
SulfinpyrazoneATP-binding cassette sub-family C member 4transporter
SulfinpyrazoneATP-binding cassette sub-family C member 3transporter
SulfinpyrazoneCytochrome P450 2C9enzyme
SulfinpyrazoneFatty acid-binding protein, intestinalcarrier
SulfinpyrazoneATP-binding cassette sub-family C member 2target
SulfinpyrazoneMultidrug resistance-associated protein 1target
SulfinpyrazoneNuclear receptor subfamily 1 group I member 2target
SulfisoxazoleDihydropteroate synthasetarget
SulfisoxazoleCytochrome P450 2C9enzyme
Sulforaphane3-phosphoinositide-dependent protein kinase 1target
SulforaphaneKelch-like ECH-associated protein 1target
SulforaphaneNuclear factor erythroid 2-related factor 2target
SulforaphaneHistone deacetylasetarget
SulforaphaneCytochrome P450 2E1target
SulforaphaneTubulintarget
SulforaphaneMacrophage migration inhibitory factortarget
SulforaphaneNuclear receptor subfamily 1 group I member 2target
SunitinibVascular endothelial growth factor receptor 3target
SunitinibVascular endothelial growth factor receptor 2target
SunitinibVascular endothelial growth factor receptor 1target
SunitinibPlatelet-derived growth factor receptor betatarget
SunitinibPlatelet-derived growth factor receptor alphatarget
SunitinibCytochrome P450 3A4enzyme
SunitinibCytochrome P450 3A5enzyme
SunitinibCytochrome P450 3A7enzyme
SunitinibATP-binding cassette sub-family C member 4transporter
SunitinibATP-dependent translocase ABCB1transporter
SunitinibATP-binding cassette sub-family C member 2transporter
SunitinibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
SunitinibHepatocyte growth factor receptortarget
SunitinibVascular endothelial growth factor receptortarget
SunitinibProto-oncogene tyrosine-protein kinase receptor Rettarget
SunitinibMast/stem cell growth factor receptor Kittarget
SunitinibReceptor-type tyrosine-protein kinase FLT3target
SunitinibMacrophage colony-stimulating factor 1 receptortarget
SuprofenHuman Cyclooxygenasestarget
SuprofenAlbumincarrier
SuprofenUDP-glucuronosyltransferase 2B7enzyme
SuprofenSolute carrier family 22 member 12transporter
SuprofenUDP-glucuronosyltransferase 1A1enzyme
SuprofenCytochrome P450 2C9enzyme
SuprofenProstaglandin G/H synthase 2target
SuprofenProstaglandin G/H synthase 1target
SuvorexantOrexin receptor type 2target
SuvorexantATP-dependent translocase ABCB1transporter
SuvorexantCytochrome P450 3A4enzyme
SuvorexantOrexin/Hypocretin receptor type 1target
SuzetrigineATP-dependent translocase ABCB1transporter
SuzetrigineCytochrome P450 3A4enzyme
SuzetrigineOrganic anion transporter 3transporter
SuzetrigineSolute carrier organic anion transporter family member 1B3transporter
SuzetrigineSolute carrier organic anion transporter family member 1B1transporter
SuzetrigineCytochrome P450 2C19enzyme
SuzetrigineCytochrome P450 2B6enzyme
SuzetrigineCytochrome P450 2C9enzyme
SuzetrigineCytochrome P450 2C8enzyme
SuzetrigineSodium channel protein type 10 subunit alphatarget
TabimorelinGrowth hormone secretagogue receptor type 1target
TabimorelinCytochrome P450 3A4target
TacrolimusPeptidyl-prolyl cis-trans isomerase FKBP1Atarget
TacrolimusCytochrome P450 3A4enzyme
TacrolimusCytochrome P450 3A5enzyme
TacrolimusATP-dependent translocase ABCB1transporter
TacrolimusCholesterol transporter ABCA5transporter
TacrolimusAlbumincarrier
TacrolimusAlpha-1-acid glycoprotein 1carrier
TacrolimusSolute carrier organic anion transporter family member 1B1transporter
TacrolimusProtein phosphatase 3 catalytic subunit alphatarget
TalarozoleCytochrome P450 26A1target
TalarozoleSubstance-K receptortarget
TaletrectinibBDNF/NT-3 growth factors receptortarget
TaletrectinibMultidrug and toxin extrusion protein 2transporter
TaletrectinibMultidrug and toxin extrusion protein 1transporter
TaletrectinibSolute carrier organic anion transporter family member 1B1transporter
TaletrectinibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
TaletrectinibATP-dependent translocase ABCB1transporter
TaletrectinibCytochrome P450 3A4enzyme
TaletrectinibCytochrome P450 1A2enzyme
TaletrectinibCytochrome P450 2D6enzyme
TaletrectinibProto-oncogene tyrosine-protein kinase ROStarget
TaletrectinibHigh affinity nerve growth factor receptortarget
TaletrectinibCytochrome P450 2C9enzyme
TaletrectinibNT-3 growth factor receptortarget
TaletrectinibCytochrome P450 3A Subfamilyenzyme
TaletrectinibCytochrome P450 2C8enzyme
TamoxifenCytochrome P450 2C8enzyme
TamoxifenVoltage-gated inwardly rectifying potassium channel KCNH2target
TamoxifenCytochrome P450 2B6enzyme
TamoxifenUDP-glucuronosyltransferase 2B17enzyme
TamoxifenLiver carboxylesterase 1enzyme
TamoxifenCytochrome P450 3A5enzyme
TamoxifenCytochrome P450 1A1enzyme
TamoxifenCytochrome P450 1B1enzyme
TamoxifenCytochrome P450 2C19enzyme
TamoxifenFlavin-containing monooxygenase 1enzyme
TamoxifenAlbumincarrier
TamoxifenMitogen-activated protein kinase 8target
TamoxifenPhospholipid-transporting ATPase ABCA1transporter
TamoxifenSulfotransferase 1E1enzyme
TamoxifenFlavin-containing monooxygenase 3enzyme
TamoxifenUDP-glucuronosyltransferase 2B7enzyme
TamoxifenCytochrome P450 1A2enzyme
TamoxifenSulfotransferase 2A1enzyme
TamoxifenThyroxine-binding globulincarrier
TamoxifenBile salt export pumptransporter
TamoxifenSex hormone-binding globulintarget
TamoxifenEstrogen-related receptor gammatarget
TamoxifenNuclear receptor subfamily 1 group I member 2target
TamoxifenCytochrome P450 3A7enzyme
TamoxifenAndrogen receptortarget
TamoxifenProtein kinase Ctarget
Tamoxifen3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerasetarget
TamoxifenATP-binding cassette sub-family C member 2transporter
TamoxifenSulfotransferase 1A1enzyme
TamoxifenUDP-glucuronosyltransferase 1A10enzyme
TamoxifenCytochrome P450 2E1enzyme
TamoxifenCytochrome P450 2A6enzyme
TamoxifenAromataseenzyme
TamoxifenBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
TamoxifenATP-dependent translocase ABCB1transporter
TamoxifenEstrogen receptortarget
TamoxifenEstrogen receptor betatarget
TamoxifenCytochrome P450 2C9enzyme
TamoxifenCytochrome P450 3A4enzyme
TamoxifenCytochrome P450 2D6enzyme
Tanshinone ICytochrome P450 1A2enzyme
Tanshinone IReplicase polyprotein 1abtarget
Tanshinone ICytochrome P450 3A4enzyme
Tanshinone ICytochrome P450 2E1enzyme
Tanshinone ICytochrome P450 2C9enzyme
Tanshinone ICytochrome P450 2D6enzyme
TasisulamCytochrome P450 2C9enzyme
TasisulamRNA-binding protein 39target
Technetium Tc-99m ciprofloxacinDNA gyrase subunit Btarget
Technetium Tc-99m ciprofloxacinDNA topoisomerase 2-betatarget
Technetium Tc-99m ciprofloxacinCytochrome P450 1A2enzyme
TecovirimatEnvelope phospholipase OPG057target
TecovirimatCytochrome P450 2B6enzyme
TecovirimatBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
TecovirimatUDP-glucuronosyltransferase 1A3enzyme
TecovirimatCytochrome P450 2C19enzyme
TecovirimatCytochrome P450 2C8enzyme
TecovirimatCytochrome P450 3A4enzyme
TecovirimatUDP-glucuronosyltransferase 1A4enzyme
TecovirimatUDP-glucuronosyltransferase 1A1enzyme
TegaserodBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
TegaserodCytochrome P450 2E1enzyme
TegaserodCytochrome P450 2D6enzyme
TegaserodCytochrome P450 2C8enzyme
TegaserodCytochrome P450 1A2enzyme
TegaserodSodium-dependent serotonin transportertransporter
Tegaserod5-hydroxytryptamine receptor 2Atarget
Tegaserod5-hydroxytryptamine receptor 2Ctarget
Tegaserod5-hydroxytryptamine receptor 2Btarget
Tegaserod5-hydroxytryptamine receptor 4target
TegaserodATP-dependent translocase ABCB1transporter
TelaprevirGenome polyproteintarget
TelaprevirATP-dependent translocase ABCB1transporter
TelaprevirAlbumincarrier
TelaprevirAlpha-1-acid glycoprotein 1carrier
TelaprevirSolute carrier organic anion transporter family member 1B1target
TelaprevirSolute carrier organic anion transporter family member 2B1target
TelaprevirGenome polyproteintarget
TelaprevirCytochrome P450 3A4enzyme
Telisotuzumab vedotinHepatocyte growth factor receptortarget
Telisotuzumab vedotinCytochrome P450 3A4enzyme
Telisotuzumab vedotinCytochrome P450 3A5enzyme
Telisotuzumab vedotinATP-binding cassette sub-family B member 5transporter
TelithromycinSolute carrier organic anion transporter family member 1B3transporter
Telithromycin23S ribosomal RNAtarget
TelithromycinCytochrome P450 3A4enzyme
TelithromycinSolute carrier organic anion transporter family member 1B1transporter
TelmisartanUDP-glucuronosyltransferase 1A3enzyme
TelmisartanBile salt export pumptransporter
TelmisartanCytochrome P450 2C19enzyme
TelmisartanBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
TelmisartanATP-binding cassette sub-family C member 2transporter
TelmisartanATP-dependent translocase ABCB1transporter
TelmisartanPeroxisome proliferator-activated receptor gammatarget
TelmisartanType-1 angiotensin II receptortarget
Telotristat ethylBroad substrate specificity ATP-binding cassette transporter ABCG2carrier
Telotristat ethylCytochrome P450 2C8enzyme
Telotristat ethylCytochrome P450 2D6enzyme
Telotristat ethylCytochrome P450 2C19enzyme
Telotristat ethylCytochrome P450 2C9enzyme
Telotristat ethylTryptophan 5-hydroxylase 2target
Telotristat ethylTryptophan 5-hydroxylase 1target
Telotristat ethylATP-dependent translocase ABCB1transporter
Telotristat ethylCytochrome P450 3A4enzyme
Telotristat ethylCytochrome P450 2B6enzyme
Telotristat ethylLiver carboxylesterase 1enzyme
Telotristat ethylUDP-glucuronosyltransferase 2B7enzyme
Telotristat ethylCocaine esteraseenzyme
Telotristat ethylUDP-glucuronosyltransferase 2B4enzyme
TemafloxacinDNA gyrase subunit Btarget
TemafloxacinDNA gyrase subunit Atarget
TemafloxacinCytochrome P450 1A2enzyme
TemafloxacinDNA topoisomerase 4 subunit Atarget
TemafloxacinDNA gyrase subunit Atarget
TemsirolimusPeptidyl-prolyl cis-trans isomerase FKBP1Atarget
TemsirolimusATP-dependent translocase ABCB1transporter
TemsirolimusCytochrome P450 2D6enzyme
TemsirolimusCytochrome P450 3A7enzyme
TemsirolimusCytochrome P450 3A5enzyme
TemsirolimusCytochrome P450 3A4enzyme
TemsirolimusSerine/threonine-protein kinase mTORtarget
TeniposideCytochrome P450 3A4enzyme
TeniposideDNA topoisomerase 2target
TeniposideDNA topoisomerase 2-betatarget
TeniposideCytochrome P450 3A5enzyme
TeniposideBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
TeniposideATP-binding cassette sub-family C member 6transporter
TeniposideCytochrome P450 2C9enzyme
TeniposideCytochrome P450 2C19enzyme
TeniposideDNA topoisomerase 2-alphatarget
TepotinibCytochrome P450 2C9enzyme
TepotinibAlpha-1-acid glycoprotein 1carrier
TepotinibSolute carrier family 22 member 1transporter
TepotinibSolute carrier family 22 member 2transporter
TepotinibMultidrug and toxin extrusion protein 1transporter
TepotinibAlbumincarrier
TepotinibMelatonin receptor type 1Btarget
TepotinibNischarintarget
TepotinibHepatocyte growth factor receptortarget
TepotinibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
TepotinibCytochrome P450 2C8enzyme
TepotinibCytochrome P450 3A4enzyme
TepotinibATP-dependent translocase ABCB1transporter
TepotinibMultidrug and toxin extrusion protein 2transporter
TepotinibBile salt export pumptransporter
TerbinafineSqualene monooxygenasetarget
TerbinafineCytochrome P450 2D6enzyme
TerbinafineCytochrome P450 2C9enzyme
TerbinafineCytochrome P450 1A2enzyme
TerbinafineCytochrome P450 3A4enzyme
TerbinafineAlbumincarrier
TerbinafineCytochrome P450 2C19enzyme
TerbinafineSqualene epoxidase ERG1target
TerbinafineABC multidrug transporter MDR2transporter
Terbinafinealpha1-acid glycoproteincarrier
TerbinafineProstaglandin G/H synthase 1enzyme
TerbinafineCytochrome P450 2C8enzyme
TerfenadineHistamine H1 receptortarget
TerfenadineAlbumincarrier
Terfenadinealpha1-acid glycoproteincarrier
TerfenadineBile salt export pumptransporter
TerfenadineMuscarinic acetylcholine receptor M2target
TerfenadineMuscarinic acetylcholine receptor M4target
TerfenadineMuscarinic acetylcholine receptor M5target
TerfenadineMuscarinic acetylcholine receptor M1target
TerfenadineCytochrome P450 2J2enzyme
TerfenadineCytochrome P450 2C8enzyme
TerfenadineATP-dependent translocase ABCB1transporter
TerfenadineCytochrome P450 3A7enzyme
TerfenadineCytochrome P450 3A5enzyme
TerfenadineMuscarinic acetylcholine receptor M3target
TerfenadineCytochrome P450 2D6enzyme
TerfenadineCytochrome P450 3A4enzyme
TerfenadineVoltage-gated inwardly rectifying potassium channel KCNH2target
TeriflunomideDihydroorotate dehydrogenase (quinone), mitochondrialtarget
Teriflunomide3-hydroxy-3-methylglutaryl-coenzyme A reductasetarget
TeriflunomideCytochrome P450 1A2enzyme
TeriflunomideSolute carrier organic anion transporter family member 1B1transporter
TeriflunomideCytochrome P450 2C8enzyme
TeriflunomideDihydroorotate dehydrogenase (quinone), mitochondrialtarget
TeriflunomideBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
TesmilifeneHistamine H1 receptortarget
TesmilifeneATP-dependent translocase ABCB1target
TesmilifeneCytochrome P450 3A4enzyme
TesmilifeneCytochrome P450 2D6enzyme
TesmilifeneCytochrome P450 1A1enzyme
Testosterone cypionateCytochrome P450 3A5enzyme
Testosterone cypionateSex hormone-binding globulincarrier
Testosterone cypionateAlbumincarrier
Testosterone cypionateCholesterol side-chain cleavage enzyme, mitochondrialenzyme
Testosterone cypionateAmine oxidase [flavin-containing] Aenzyme
Testosterone cypionateCytochrome P450 3A4enzyme
Testosterone cypionateAndrogen receptortarget
Testosterone cypionateCytochrome P450 3A7enzyme
Testosterone cypionateSolute carrier organic anion transporter family member 1A2transporter
Testosterone cypionateOrganic anion transporter 3transporter
Testosterone cypionateSolute carrier family 22 member 7transporter
Testosterone cypionateAromataseenzyme
Testosterone cypionate3-oxo-5-alpha-steroid 4-dehydrogenaseenzyme
Testosterone cypionateMineralocorticoid receptortarget
Testosterone cypionateEstrogen receptortarget
Testosterone cypionateCytochrome P450 3A43enzyme
Testosterone cypionateCytochrome P450 2C9enzyme
Testosterone cypionateCytochrome P450 2C8enzyme
Testosterone cypionateCytochrome P450 2C19enzyme
Testosterone cypionateCytochrome P450 2B6enzyme
Testosterone cypionateATP-dependent translocase ABCB1transporter
Testosterone cypionateCytochrome P450 1A1enzyme
Testosterone cypionateBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
Testosterone cypionateSolute carrier family 22 member 4transporter
Testosterone cypionateSolute carrier family 22 member 3transporter
Testosterone cypionateHepatic sodium/bile acid cotransportertransporter
Testosterone cypionateCytochrome P450 2A13enzyme
Testosterone enanthateCytochrome P450 2C19enzyme
Testosterone enanthate3-oxo-5-alpha-steroid 4-dehydrogenaseenzyme
Testosterone enanthateAndrogen receptortarget
Testosterone enanthateCytochrome P450 3A4enzyme
Testosterone enanthateAmine oxidase [flavin-containing] Aenzyme
Testosterone enanthateCholesterol side-chain cleavage enzyme, mitochondrialenzyme
Testosterone enanthateAlbumincarrier
Testosterone enanthateSex hormone-binding globulincarrier
Testosterone enanthateCytochrome P450 3A5enzyme
Testosterone enanthateCytochrome P450 3A7enzyme
Testosterone enanthateSolute carrier organic anion transporter family member 1A2transporter
Testosterone enanthateOrganic anion transporter 3transporter
Testosterone enanthateSolute carrier family 22 member 7transporter
Testosterone enanthateATP-dependent translocase ABCB1transporter
Testosterone enanthateHepatic sodium/bile acid cotransportertransporter
Testosterone enanthateSolute carrier family 22 member 3transporter
Testosterone enanthateSolute carrier family 22 member 4transporter
Testosterone enanthateBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
Testosterone enanthateCytochrome P450 1A1enzyme
Testosterone enanthateCytochrome P450 2A13enzyme
Testosterone enanthateCytochrome P450 2B6enzyme
Testosterone enanthateCytochrome P450 2C8enzyme
Testosterone enanthateCytochrome P450 2C9enzyme
Testosterone enanthateCytochrome P450 3A43enzyme
Testosterone enanthateEstrogen receptortarget
Testosterone enanthateMineralocorticoid receptortarget
Testosterone enanthateAromataseenzyme
Testosterone undecanoateAndrogen receptortarget
Testosterone undecanoateCytochrome P450 3A4enzyme
Testosterone undecanoateSex hormone-binding globulincarrier
Testosterone undecanoateAmine oxidase [flavin-containing] Aenzyme
Testosterone undecanoateCholesterol side-chain cleavage enzyme, mitochondrialenzyme
Testosterone undecanoateAromataseenzyme
Testosterone undecanoateSolute carrier organic anion transporter family member 1B3transporter
Testosterone undecanoateMultidrug and toxin extrusion protein 1transporter
Testosterone undecanoateAlbumincarrier
Testosterone undecanoateSolute carrier family 22 member 2transporter
Testosterone undecanoate3-oxo-5-alpha-steroid 4-dehydrogenaseenzyme
Testosterone undecanoateCytochrome P450 3A43enzyme
Testosterone undecanoateCytochrome P450 2C9enzyme
Testosterone undecanoateCytochrome P450 2C8enzyme
Testosterone undecanoateCytochrome P450 2C19enzyme
Testosterone undecanoateCytochrome P450 2B6enzyme
Testosterone undecanoateCytochrome P450 2A13enzyme
Testosterone undecanoateCytochrome P450 1B1enzyme
Testosterone undecanoateCytochrome P450 1A1enzyme
Testosterone undecanoateBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
Testosterone undecanoateSolute carrier family 22 member 4transporter
Testosterone undecanoateHepatic sodium/bile acid cotransportertransporter
Testosterone undecanoateATP-dependent translocase ABCB1transporter
Testosterone undecanoateSolute carrier family 22 member 7transporter
Testosterone undecanoateOrganic anion transporter 3transporter
Testosterone undecanoateSolute carrier organic anion transporter family member 1A2transporter
Testosterone undecanoateCytochrome P450 3A7enzyme
Testosterone undecanoateCytochrome P450 3A5enzyme
TetracyclineCytochrome P450 3A4enzyme
TetracyclineSolute carrier family 22 member 6transporter
TetracyclineOrganic anion transporter 3transporter
TetracyclineSolute carrier family 22 member 11transporter
TetracyclineSolute carrier family 22 member 7transporter
TetracyclineSmall ribosomal subunit protein uS3target
TetracyclineSmall ribosomal subunit protein uS8target
TetracyclineSmall ribosomal subunit protein uS19target
TetracyclineSmall ribosomal subunit protein uS14target
TetracyclineSmall ribosomal subunit protein uS7target
TetracyclineSolute carrier organic anion transporter family member 2B1transporter
TetracyclineAlbumincarrier
Tetracycline16S ribosomal RNAtarget
TetracyclineMajor prion proteintarget
TezacaftorSolute carrier family 22 member 2transporter
TezacaftorSolute carrier family 22 member 6transporter
TezacaftorOrganic anion transporter 3transporter
TezacaftorBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
TezacaftorATP-dependent translocase ABCB1transporter
TezacaftorCystic fibrosis transmembrane conductance regulatortarget
TezacaftorSolute carrier organic anion transporter family member 1B3transporter
TezacaftorCytochrome P450 3A5enzyme
TezacaftorCytochrome P450 3A4enzyme
TezacaftorSolute carrier organic anion transporter family member 1B1transporter
TezacaftorCytochrome P450 1A2enzyme
TezacaftorCytochrome P450 2B6enzyme
TezacaftorCytochrome P450 2C8enzyme
TezacaftorCytochrome P450 2C9enzyme
TezacaftorCytochrome P450 2C19enzyme
TezacaftorCytochrome P450 2D6enzyme
ThalidomideTumor necrosis factortarget
ThalidomideCytochrome P450 2B6enzyme
ThalidomideCytochrome P450 1A1enzyme
ThalidomideCytochrome P450 3A4enzyme
Thalidomidealpha1-acid glycoproteintarget
ThalidomideProtein cereblontarget
ThalidomideDNAtarget
ThalidomideCytochrome P450 3A5enzyme
ThalidomideProstaglandin G/H synthase 2enzyme
ThalidomideCytochrome P450 2C9enzyme
ThalidomideCytochrome P450 2C19enzyme
ThalidomideProstaglandin G/H synthase 1enzyme
ThiabendazoleCytochrome P450 1A1enzyme
ThiabendazoleCytochrome P450 1A2enzyme
ThiabendazoleFumarate reductase flavoprotein subunittarget
ThiopentalNeuronal acetylcholine receptor subunit alpha-7target
ThiopentalCytochrome P450 2C19enzyme
ThiopentalMuscarinic acetylcholine receptor M3target
ThiopentalCytochrome P450 3A Subfamilyenzyme
ThiopentalGlutamate receptor ionotropic, kainate 2target
ThiopentalGlutamate receptor 2target
ThiopentalNeuronal acetylcholine receptor subunit alpha-4target
ThiopentalGamma-aminobutyric acid receptor subunit alpha-6target
ThiopentalGamma-aminobutyric acid receptor subunit alpha-5target
ThiopentalGamma-aminobutyric acid receptor subunit alpha-4target
ThiopentalGamma-aminobutyric acid receptor subunit alpha-3target
ThiopentalGamma-aminobutyric acid receptor subunit alpha-2target
ThiopentalFatty-acid amide hydrolase 1target
ThiopentalGamma-aminobutyric acid receptor subunit alpha-1target
ThioridazineCytochrome P450 2E1enzyme
Thioridazine5-hydroxytryptamine receptor 2Ctarget
ThioridazineAlpha-1A adrenergic receptortarget
ThioridazineD(2) dopamine receptortarget
Thioridazine5-hydroxytryptamine receptor 2Atarget
ThioridazineD(1A) dopamine receptortarget
ThioridazineCytochrome P450 2C19enzyme
ThioridazineCytochrome P450 2D6enzyme
ThioridazineVoltage-gated inwardly rectifying potassium channel KCNH2target
ThioridazineAlpha-1B adrenergic receptortarget
ThiotepaCytochrome P450 2B6enzyme
ThiotepaCytochrome P450 3A4enzyme
ThiotepaDNAtarget
ThiotepaCholinesteraseenzyme
ThiothixeneD(1A) dopamine receptortarget
Thiothixene5-hydroxytryptamine receptor 2Atarget
ThiothixeneSolute carrier family 22 member 1transporter
ThiothixeneAlbumincarrier
ThiothixeneD(2) dopamine receptortarget
ThiothixeneCytochrome P450 2D6enzyme
ThiothixeneCytochrome P450 1A2enzyme
TiamulinTumor necrosis factortarget
TiamulinATP-dependent translocase ABCB1transporter
TiamulinCytochrome P450 2E1enzyme
TiamulinCytochrome P450 3A4enzyme
TicagrelorCytochrome P450 2B6enzyme
TicagrelorCytochrome P450 3A5enzyme
TicagrelorAlbumincarrier
TicagrelorCytochrome P450 2C9enzyme
TicagrelorATP-dependent translocase ABCB1transporter
TicagrelorP2Y purinoceptor 12target
TicagrelorCytochrome P450 3A4enzyme
TiclopidineCytochrome P450 2E1enzyme
TiclopidinePlatelet-activating factor receptortarget
TiclopidineP2Y purinoceptor 12target
TiclopidineCytochrome P450 2C19enzyme
TiclopidineCytochrome P450 2B6enzyme
TiclopidineCytochrome P450 2C9enzyme
TiclopidineCytochrome P450 2D6enzyme
TiclopidineMyeloperoxidaseenzyme
TiclopidineCytochrome P450 1A2enzyme
TiclopidineCytochrome P450 2C8enzyme
Tienilic acidCytochrome P450 2C9enzyme
TildipirosinCytochrome P450 3A4enzyme
TilidineATP-dependent translocase ABCB1transporter
TilidineMu-type opioid receptortarget
TilidineCytochrome P450 3A4enzyme
TilidineCytochrome P450 2C19enzyme
TilidineCytochrome P450 2D6enzyme
TilidineCytochrome P450 2B6enzyme
TioconazoleLanosterol 14-alpha demethylasetarget
TioconazoleLanosterol 14-alpha demethylasetarget
TioconazoleAromataseenzyme
TioconazoleCytochrome P450 2C19enzyme
TioconazoleCytochrome P450 2E1enzyme
TioconazoleCytochrome P450 3A4enzyme
TipranavirCytochrome P450 3A4enzyme
TipranavirCytochrome P450 2D6enzyme
TipranavirCytochrome P450 2C19enzyme
TipranavirBile salt export pumptransporter
TipranavirUDP-glucuronosyltransferase 1A1enzyme
TipranavirSolute carrier organic anion transporter family member 2B1transporter
TipranavirSolute carrier organic anion transporter family member 1B1transporter
TipranavirSolute carrier organic anion transporter family member 1B3transporter
TipranavirATP-dependent translocase ABCB1transporter
TipranavirGag-Pol polyproteintarget
TipranavirPol polyproteintarget
TirbanibulinProto-oncogene tyrosine-protein kinase Srctarget
TirbanibulinTubulin beta chaintarget
TirbanibulinCytochrome P450 3A4enzyme
TirbanibulinCytochrome P450 2C8enzyme
TirbanibulinCytochrome P450 1A2enzyme
TirbanibulinCytochrome P450 2B6enzyme
TirbanibulinCytochrome P450 2C9enzyme
TirbanibulinCytochrome P450 2C19enzyme
TirbanibulinCytochrome P450 2D6enzyme
TirbanibulinMultidrug and toxin extrusion protein 1transporter
TirbanibulinMultidrug and toxin extrusion protein 2transporter
TirbanibulinSolute carrier organic anion transporter family member 1B1transporter
TirbanibulinSolute carrier organic anion transporter family member 1B3transporter
TirbanibulinSolute carrier family 22 member 1transporter
TirbanibulinSolute carrier family 22 member 2transporter
TocainideVoltage-gated sodium channel alpha subunittarget
TocainideCytochrome P450 1A2enzyme
TocainideAlbumincarrier
TocainideSodium channel protein type 5 subunit alphatarget
TofisopamCytochrome P450 3A4enzyme
TofisopamcGMP-dependent 3',5'-cyclic phosphodiesterasetarget
TofisopamcGMP-inhibited 3',5'-cyclic phosphodiesterase 3Atarget
TofisopamcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10Atarget
Tofisopam3',5'-cyclic-AMP phosphodiesterase 4Atarget
TolbutamideSolute carrier family 22 member 6transporter
TolbutamideSolute carrier organic anion transporter family member 2B1transporter
TolbutamideCytochrome P450 2C18enzyme
TolbutamideAlbumincarrier
TolbutamideATP-binding cassette sub-family C member 9target
TolbutamideSolute carrier family 15 member 2transporter
TolbutamideSolute carrier organic anion transporter family member 1A2transporter
TolbutamideSolute carrier family 15 member 1transporter
TolbutamideATP-binding cassette sub-family C member 8target
TolbutamideCytochrome P450 2C8enzyme
TolbutamideCytochrome P450 2C9enzyme
TolbutamideCytochrome P450 2C19enzyme
TolbutamideATP-sensitive inward rectifier potassium channel 1target
TolcaponeCytochrome P450 2C9enzyme
TolcaponeCatechol O-methyltransferasetarget
TopiramateVoltage-gated sodium channel alpha subunittarget
TopiramateGamma-aminobutyric acid receptor subunit alpha-1target
TopiramateCarbonic anhydrase 4target
TopiramateKainate receptorstarget
TopiramateCytochrome P450 2C19enzyme
TopiramateCytochrome P450 3A4enzyme
TopiramateCarbonic anhydrase 1target
TopiramateCarbonic anhydrase 3target
TopiramateVoltage gated L-type calcium channeltarget
TopiramateVoltage-dependent R-type calcium channeltarget
TopiramateAlbumincarrier
TopiramateATP-dependent translocase ABCB1transporter
Topiramate5'-AMP-activated protein kinasetransporter
TopiramateGlutamate receptor ionotropic, kainate 1target
TopiramateCarbonic anhydrase 2target
TopiroxostatBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
TopiroxostatAlbumincarrier
TopiroxostatAlpha-1-acid glycoprotein 1carrier
TopiroxostatCytochrome P450 2C8enzyme
TopiroxostatCytochrome P450 2C9enzyme
TopiroxostatCytochrome P450 1A1enzyme
TopiroxostatCytochrome P450 3A4enzyme
TopiroxostatCytochrome P450 2C19enzyme
TopiroxostatOrganic anion transporter 3transporter
TopiroxostatSolute carrier family 22 member 6transporter
TopiroxostatUDP-glucuronosyltransferase 1A9enzyme
TopiroxostatXanthine dehydrogenase/oxidasetarget
TopotecanMultidrug and toxin extrusion protein 1transporter
TopotecanDNAtarget
TopotecanATP-dependent translocase ABCB1transporter
TopotecanBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
TopotecanDNA topoisomerase 1target
TopotecanDNA topoisomerase I, mitochondrialtarget
TopotecanMultidrug and toxin extrusion protein 2transporter
TorasemideSolute carrier family 12 member 1target
TorasemideAlbumincarrier
TorasemideSolute carrier family 12 member 2target
TorasemideSolute carrier organic anion transporter family member 1B1transporter
TorasemideCytochrome P450 2C9enzyme
TorasemideCytochrome P450 2C8enzyme
ToremifeneEstrogen receptortarget
ToremifeneCytochrome P450 3A4enzyme
ToremifeneATP-dependent translocase ABCB1transporter
ToremifeneCytochrome P450 1A1enzyme
ToremifeneSex hormone-binding globulintarget
ToremifeneEstrogen receptortarget
TovorafenibSerine/threonine-protein kinase A-Raftarget
TovorafenibSerine/threonine-protein kinase B-raftarget
TovorafenibCytochrome P450 2C8enzyme
TovorafenibCytochrome P450 3A4enzyme
TovorafenibCytochrome P450 2C9enzyme
TovorafenibCytochrome P450 2C19enzyme
TovorafenibCytochrome P450 1A2enzyme
TovorafenibCytochrome P450 2B6enzyme
TovorafenibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
TovorafenibRAF proto-oncogene serine/threonine-protein kinasetarget
TradipitantCytochrome P450 3A4enzyme
TradipitantCytochrome P450 2C8enzyme
TradipitantUDP-glucuronosyltransferase 1A4enzyme
TradipitantSubstance-P receptortarget
TradipitantCytochrome P450 2C19enzyme
TradipitantUDP-glucuronosyltransferase 2B7enzyme
TradipitantATP-dependent translocase ABCB1transporter
TrametinibMitogen-activated protein kinase kinase (MAPKK)target
TrametinibDual specificity mitogen-activated protein kinase kinase 2target
TrametinibDual specificity mitogen-activated protein kinase kinase 1target
TrametinibCytochrome P450 3A4enzyme
TrametinibCytochrome P450 2C8enzyme
TranylcypromineMonoamine oxidasetarget
TranylcypromineCytochrome P450 2C9enzyme
TranylcypromineCytochrome P450 3A4enzyme
TranylcypromineAmine oxidase [flavin-containing] Btarget
TranylcypromineAmine oxidase [flavin-containing] Atarget
TranylcypromineCytochrome P450 2C19enzyme
TranylcypromineCytochrome P450 2A6enzyme
TranylcypromineCytochrome P450 2D6enzyme
TranylcypromineCytochrome P450 1A2enzyme
TrazodoneCytochrome P450 3A7enzyme
TrazodoneCytochrome P450 3A5enzyme
Trazodone5-hydroxytryptamine receptor 2Ctarget
TrazodoneCytochrome P450 3A4enzyme
TrazodoneCytochrome P450 2D6enzyme
Trazodone5-hydroxytryptamine receptor 1Atarget
TrazodoneHistamine H1 receptortarget
TrazodoneATP-dependent translocase ABCB1transporter
TrazodoneAlpha-1A adrenergic receptortarget
TrazodoneSodium-dependent serotonin transportertarget
Trazodone5-hydroxytryptamine receptor 2Atarget
Trazodone5-hydroxytryptamine receptor 2Ctarget
TrazodoneAlpha-2A adrenergic receptortarget
TreosulfanCytochrome P450 3A4enzyme
TreosulfanDNAtarget
TreosulfanCytochrome P450 2D6enzyme
TreosulfanCytochrome P450 2C8enzyme
TreosulfanCytochrome P450 2C19enzyme
TriazolamCytochrome P450 2C8enzyme
TriazolamGABA(A) Receptor Benzodiazepine Binding Sitetarget
TriazolamCytochrome P450 3A7enzyme
TriazolamTranslocator proteintarget
TriazolamCytochrome P450 3A5enzyme
TriazolamCytochrome P450 3A4enzyme
TriazolamGABA(A) Receptortarget
TrichloroethyleneCytochrome P450 2E1enzyme
TrichloroethyleneAcetylcholinesterasetarget
TrichloroethyleneGlutathione S-transferases (Cytosolic)enzyme
TriclabendazoleCruzipaintarget
TriclabendazoleCytochrome P450 2B6enzyme
TriclabendazoleCytochrome P450 2C8enzyme
TriclabendazoleCytochrome P450 2A6enzyme
TriclabendazoleCytochrome P450 2D6enzyme
TriclabendazoleCytochrome P450 2C19enzyme
TriclabendazoleCytochrome P450 1B1enzyme
TriclabendazoleCytochrome P450 1A1enzyme
TriclabendazoleCytochrome P450 3A4enzyme
TriclabendazoleExcretory Secretory (ES) proteinstarget
TriclabendazoleCytochrome P450 2C9enzyme
TriclabendazoleCytochrome P450 1A2enzyme
TrilaciclibCyclin-dependent kinase 7target
TrilaciclibCyclin-dependent kinase 5target
TrilaciclibCyclin-dependent kinase 2target
TrilaciclibCyclin-dependent kinase 9target
TrilaciclibCyclin-dependent kinase 6target
TrilaciclibCyclin-dependent kinase 4target
TrilaciclibATP-dependent translocase ABCB1transporter
TrilaciclibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
TrilaciclibCytochrome P450 1A2enzyme
TrilaciclibSolute carrier family 22 member 2transporter
TrilaciclibMultidrug and toxin extrusion protein 1transporter
TrilaciclibMultidrug and toxin extrusion protein 2transporter
TrimethoprimSolute carrier family 22 member 1transporter
TrimethoprimDihydrofolate reductasetarget
TrimethoprimMultidrug and toxin extrusion protein 2transporter
TrimethoprimMultidrug and toxin extrusion protein 1transporter
TrimethoprimCytochrome P450 1A2enzyme
TrimethoprimCytochrome P450 2C9enzyme
TrimethoprimATP-dependent translocase ABCB1transporter
TrimethoprimCytochrome P450 3A4enzyme
TrimethoprimCytochrome P450 2C8enzyme
TrimethoprimDihydrofolate reductasetarget
TrimethoprimSolute carrier family 22 member 2transporter
TripelennamineCytochrome P450 2D6enzyme
TripelennamineHistamine H1 receptortarget
TripelennamineAlbumincarrier
TrofinetideCytochrome P450 3A4enzyme
TrofinetideUDP-glucuronosyltransferase 1A9enzyme
TrofinetideSolute carrier organic anion transporter family member 1B3transporter
TrofinetideUDP-glucuronosyltransferase 2B7enzyme
TrofinetideUDP-glucuronosyltransferase 2B15enzyme
TrofinetideSolute carrier organic anion transporter family member 1B1transporter
TroglitazoneUDP-glucuronosyltransferase 1A9enzyme
TroglitazoneUDP-glucuronosyltransferase 1A10enzyme
TroglitazoneUDP-glucuronosyltransferase 2B7enzyme
TroglitazoneUDP-glucuronosyltransferase 2B15enzyme
TroglitazoneGlutathione S-transferase Ptarget
TroglitazonePeroxisome proliferator-activated receptor deltatarget
TroglitazoneUDP-glucuronosyltransferase 1A8enzyme
TroglitazoneUDP-glucuronosyltransferase 1A7enzyme
TroglitazoneUDP-glucuronosyltransferase 1A6enzyme
TroglitazoneUDP-glucuronosyltransferase 1A4enzyme
TroglitazoneUDP-glucuronosyltransferase 1A3enzyme
TroglitazoneCytochrome P450 3A7enzyme
TroglitazoneEstrogen-related receptor gammatarget
TroglitazoneCytochrome P450 3A5enzyme
TroglitazoneCytochrome P450 2C9enzyme
TroglitazoneCytochrome P450 2B6enzyme
TroglitazoneCytochrome P450 1A1enzyme
TroglitazoneAromataseenzyme
TroglitazoneSteroid hormone receptor ERR1target
TroglitazonePeroxisome proliferator-activated receptor gammatarget
TroglitazoneLong-chain-fatty-acid--CoA ligase 4target
TroglitazonePlasminogen activator inhibitor 1target
TroglitazoneEquilibrative nucleoside transporter 1target
TroglitazoneCytochrome P450 3A4enzyme
TroglitazoneCytochrome P450 2C19enzyme
TroglitazoneUDP-glucuronosyltransferase 1A1enzyme
TroglitazoneCytochrome P450 2C8enzyme
TroglitazoneBile salt export pumptransporter
TroglitazoneSolute carrier organic anion transporter family member 1B1transporter
TroglitazonePeroxisome proliferator-activated receptor alphatarget
TroleandomycinCytochrome P450 3A7enzyme
TroleandomycinNuclear receptor subfamily 1 group I member 2target
TroleandomycinCytochrome P450 3A4enzyme
TroleandomycinCytochrome P450 2C8enzyme
TroleandomycinATP-dependent translocase ABCB1transporter
TroleandomycinLarge ribosomal subunit protein bL32target
TroleandomycinLarge ribosomal subunit protein uL4target
TroleandomycinCytochrome P450 3A43enzyme
TroleandomycinCytochrome P450 3A5enzyme
TrospiumMuscarinic acetylcholine receptor M1target
TrospiumCytochrome P450 2D6enzyme
TrospiumMuscarinic acetylcholine receptor M3target
TrospiumMuscarinic acetylcholine receptor M5target
TrospiumMuscarinic acetylcholine receptor M2target
TrovafloxacinDNA gyrase subunit Atarget
TrovafloxacinDNA topoisomerase 4 subunit Atarget
TrovafloxacinDNA topoisomerase 2-alphatarget
TrovafloxacinCytochrome P450 1A2enzyme
TrovafloxacinDNA gyrase subunit Atarget
TrovafloxacinDNA gyrase subunit Btarget
TucatinibCytochrome P450 2C8enzyme
TucatinibCytochrome P450 3A Subfamilyenzyme
TucatinibMultidrug and toxin extrusion protein 2transporter
TucatinibMultidrug and toxin extrusion protein 1transporter
TucatinibSolute carrier family 22 member 2transporter
TucatinibATP-dependent translocase ABCB1transporter
TucatinibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
TucatinibReceptor tyrosine-protein kinase erbB-2target
TucatinibReceptor tyrosine-protein kinase erbB-3target
TucatinibReceptor tyrosine-protein kinase erbB-2enzyme
UbrogepantCalcitonin gene-related peptide type 1 receptortarget
UbrogepantSolute carrier family 22 member 6transporter
UbrogepantSolute carrier organic anion transporter family member 1B3transporter
UbrogepantSolute carrier organic anion transporter family member 1B1transporter
UbrogepantUDP-glucuronosyltransferase 1A1enzyme
UbrogepantAmine oxidase [flavin-containing] Aenzyme
UbrogepantCytochrome P450 2C19enzyme
UbrogepantCytochrome P450 2D6enzyme
UbrogepantCytochrome P450 2C9enzyme
UbrogepantCytochrome P450 2C8enzyme
UbrogepantCytochrome P450 3A4enzyme
UbrogepantBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
UbrogepantSolute carrier family 22 member 2transporter
UbrogepantATP-dependent translocase ABCB1transporter
VadadustatCytochrome P450 2C9enzyme
VadadustatAlbumincarrier
VadadustatSolute carrier family 22 member 6transporter
VadadustatOrganic anion transporter 3transporter
VadadustatBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
VadadustatCytochrome P450 3A4enzyme
VadadustatCytochrome P450 2C8enzyme
VadadustatCytochrome P450 2B6enzyme
VadadustatUDP-glucuronosyltransferase 2B7enzyme
VadadustatUDP-glucuronosyltransferase 1A9enzyme
VadadustatUDP-glucuronosyltransferase 1A8enzyme
VadadustatUDP-glucuronosyltransferase 1A7enzyme
VadadustatUDP-glucuronosyltransferase 1A1enzyme
VadadustatEndothelial PAS domain-containing protein 1target
VadadustatHypoxia-inducible factor 1-alphatarget
VadadustatEgl nine homolog 1target
VadadustatProlyl hydroxylase EGLN3target
VadadustatProlyl hydroxylase EGLN2target
ValdecoxibCarbonic anhydrase 3target
ValdecoxibCarbonic anhydrase 2target
ValdecoxibUDP-glucuronosyltransferase 1A9enzyme
ValdecoxibCytochrome P450 3A4enzyme
ValdecoxibProstaglandin G/H synthase 2target
ValdecoxibCytochrome P450 2C9enzyme
Valproic acidPeroxisome proliferator-activated receptor alphatarget
Valproic acidPeroxisome proliferator-activated receptor deltatarget
Valproic acidPeroxisome proliferator-activated receptor gammatarget
Valproic acidAlbumincarrier
Valproic acidUDP-glucuronosyltransferase 1A1enzyme
Valproic acidSolute carrier organic anion transporter family member 2B1transporter
Valproic acidHistone deacetylasetarget
Valproic acidCyclin-dependent kinase inhibitor 1target
Valproic acidHepatocyte growth factortarget
Valproic acidOrnithine decarboxylasetarget
Valproic acidProgrammed cell death 1 ligand 1target
Valproic acid4-aminobutyrate aminotransferase, mitochondrialtarget
Valproic acidGlycogen synthase kinase-3 alphatarget
Valproic acidHistone deacetylase 2target
Valproic acidHistone deacetylase 9target
Valproic acidShort/branched chain specific acyl-CoA dehydrogenase, mitochondrialtarget
Valproic acidCytochrome P450 2A6enzyme
Valproic acidCytochrome P450 2B6enzyme
Valproic acidCytochrome P450 2C9enzyme
Valproic acidOrganic cation/carnitine transporter 2transporter
Valproic acidSolute carrier family 22 member 6transporter
Valproic acidOrganic anion transporter 3transporter
Valproic acidMonocarboxylate transporter 1transporter
Valproic acidSolute carrier family 22 member 7transporter
Valproic acidCytochrome P450 3A5enzyme
Valproic acidUDP-glucuronosyltransferase 1A9enzyme
Valproic acidProstaglandin G/H synthase 1enzyme
Valproic acidCytochrome P450 1A2enzyme
Valproic acidCytochrome P450 2C19enzyme
Valproic acidCytochrome P450 3A4enzyme
Valproic acidUDP-glucuronosyltransferase 1A4enzyme
Valproic acidUDP-glucuronosyltransferase 1A8enzyme
Valproic acidUDP-glucuronosyltransferase 1A10enzyme
Valproic acidUDP-glucuronosyltransferase 1A6enzyme
Valproic acidUDP-glucuronosyltransferase 1A3enzyme
Valproic acidUDP-glucuronosyltransferase 2B7enzyme
Valproic acidUDP-glucuronosyltransferase 2B15enzyme
Valproic acid2-oxoglutarate dehydrogenase complex component E1target
Valproic acidSuccinate-semialdehyde dehydrogenase, mitochondrialtarget
Valproic acidSodium channel proteintarget
ValsartanATP-binding cassette sub-family C member 2transporter
ValsartanSolute carrier organic anion transporter family member 1B3transporter
ValsartanCytochrome P450 2C9enzyme
ValsartanType-1 angiotensin II receptortarget
ValsartanSolute carrier organic anion transporter family member 1B1transporter
VapreotideSomatostatin receptor type 2target
VapreotideCytochrome P450 3A4enzyme
VapreotideSomatostatin receptor type 3target
VapreotideSubstance-P receptortarget
VapreotideSomatostatin receptor type 5target
VardenafilCytochrome P450 2D6enzyme
VardenafilCytochrome P450 2C19enzyme
VardenafilCytochrome P450 2C8enzyme
VardenafilCytochrome P450 2C9enzyme
VardenafilATP-dependent translocase ABCB1transporter
VardenafilCytochrome P450 3A5enzyme
VardenafilRetinal cone rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit gammatarget
VardenafilRod cGMP 3',5'-cyclic phosphodiesterase subunit gammatarget
VardenafilCytochrome P450 3A4enzyme
VardenafilcGMP-specific 3',5'-cyclic phosphodiesterasetarget
VayarinPeroxisomal acyl-coenzyme A oxidase 1enzyme
VayarinVery long chain fatty acid elongase 4enzyme
VayarinAcyl-CoA (8-3)-desaturaseenzyme
VayarinCytochrome P450 2E1enzyme
VemurafenibCytochrome P450 3A4enzyme
VemurafenibSerine/threonine-protein kinase B-raftarget
VemurafenibMultidrug resistance-associated protein 1transporter
VemurafenibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
VemurafenibCytochrome P450 2C9enzyme
VemurafenibCytochrome P450 2C8enzyme
VemurafenibCytochrome P450 2B6enzyme
VemurafenibATP-dependent translocase ABCB1transporter
VemurafenibAlbumincarrier
VemurafenibAlpha-1-acid glycoprotein 1carrier
VemurafenibCytochrome P450 1A2enzyme
VemurafenibCytochrome P450 2D6enzyme
VenetoclaxSolute carrier organic anion transporter family member 1B1transporter
VenetoclaxBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
VenetoclaxATP-dependent translocase ABCB1transporter
VenetoclaxCytochrome P450 3A4enzyme
VenetoclaxApoptosis regulator Bcl-2target
VenlafaxineCytochrome P450 2C9enzyme
VenlafaxineBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
VenlafaxineATP-dependent translocase ABCB1transporter
VenlafaxineSodium-dependent dopamine transportertarget
VenlafaxineCytochrome P450 3A4enzyme
VenlafaxineCytochrome P450 2D6enzyme
VenlafaxineSodium-dependent noradrenaline transportertarget
VenlafaxineSodium-dependent serotonin transportertarget
VenlafaxineCytochrome P450 2C19enzyme
VepdegestrantEstrogen receptortarget
VepdegestrantCytochrome P450 2C8enzyme
VepdegestrantCytochrome P450 2C9enzyme
VepdegestrantCytochrome P450 3A5enzyme
VepdegestrantCytochrome P450 2B6enzyme
VepdegestrantUDP-glucuronosyltransferase 1A9enzyme
VepdegestrantATP-dependent translocase ABCB1transporter
VepdegestrantCytochrome P450 3A4enzyme
VerapamilAlpha-1B adrenergic receptortarget
VerapamilAlpha-1D adrenergic receptortarget
VerapamilAlbumincarrier
VerapamilAlpha-1-acid glycoprotein 1carrier
VerapamilCytochrome P450 2C18enzyme
VerapamilCytochrome P450 2E1enzyme
VerapamilMultidrug resistance-associated protein 1transporter
VerapamilMultidrug and toxin extrusion protein 1transporter
VerapamilMultidrug and toxin extrusion protein 2transporter
VerapamilVoltage-dependent N-type calcium channel subunit alpha-1Btarget
VerapamilVoltage-dependent calcium channeltarget
VerapamilATP-dependent translocase ABCB1target
VerapamilVoltage gated L-type calcium channeltarget
VerapamilCytochrome P450 1A2enzyme
VerapamilVoltage-dependent L-type calcium channel subunit alpha-1Ctarget
VerapamilVoltage-gated inwardly rectifying potassium channel KCNH2target
VerapamilVoltage-dependent T-type calcium channel subunit alpha-1Gtarget
VerapamilATP-sensitive inward rectifier potassium channel 11target
VerapamilAlpha-1A adrenergic receptortarget
VerapamilCytochrome P450 2D6enzyme
VerapamilCytochrome P450 2C19enzyme
VerapamilCytochrome P450 2B6enzyme
VerapamilCytochrome P450 2C9enzyme
VerapamilCytochrome P450 2C8enzyme
VerapamilCytochrome P450 3A5enzyme
VerapamilSolute carrier organic anion transporter family member 1B1transporter
VerapamilSolute carrier family 22 member 4transporter
VerapamilATP-binding cassette sub-family C member 10transporter
VerapamilSolute carrier organic anion transporter family member 1A2transporter
VerapamilOrganic cation/carnitine transporter 2transporter
VerapamilATP-binding cassette sub-family C member 4transporter
VerapamilATP-binding cassette sub-family C member 3transporter
VerapamilSolute carrier family 22 member 1transporter
VerapamilATP-dependent translocase ABCB1transporter
VerapamilCytochrome P450 3A4enzyme
VerapamilSodium-dependent serotonin transportertarget
VerapamilVoltage-dependent P/Q-type calcium channel subunit alpha-1Atarget
VerapamilVoltage-dependent T-type calcium channel subunit alpha-1Htarget
VernakalantCytochrome P450 2D6enzyme
VernakalantSodium channel protein type 5 subunit alphatarget
VernakalantPotassium voltage-gated channel subfamily A member 5target
VernakalantVoltage-gated inwardly rectifying potassium channel KCNH2target
VernakalantA-type voltage-gated potassium channel KCND3target
Vilazodone5-hydroxytryptamine receptor 1Atarget
VilazodoneCytochrome P450 3A4enzyme
VilazodoneCytochrome P450 2D6enzyme
VilazodoneSodium-dependent serotonin transportertarget
VilazodoneCytochrome P450 2C19enzyme
ViloxazineMuscarinic acetylcholine receptor M3target
ViloxazineMuscarinic acetylcholine receptor M4target
ViloxazineMuscarinic acetylcholine receptor M1target
ViloxazineHistamine H2 receptortarget
ViloxazineHistamine H1 receptortarget
ViloxazineAmine oxidase [flavin-containing] Btarget
ViloxazineAmine oxidase [flavin-containing] Atarget
ViloxazineBeta-2 adrenergic receptortarget
ViloxazineAlpha-1B adrenergic receptortarget
Viloxazine5-hydroxytryptamine receptor 2Ctarget
Viloxazine5-hydroxytryptamine receptor 2Btarget
ViloxazineMultidrug and toxin extrusion protein 1transporter
ViloxazineCytochrome P450 3A5enzyme
ViloxazineCytochrome P450 3A4enzyme
ViloxazineCytochrome P450 2B6enzyme
ViloxazineUDP-glucuronosyltransferase 2B15enzyme
ViloxazineUDP-glucuronosyltransferase 1A9enzyme
ViloxazineCytochrome P450 2D6enzyme
ViloxazineCytochrome P450 1A2enzyme
ViloxazineSodium-dependent noradrenaline transportertarget
ViloxazineMuscarinic acetylcholine receptor M2target
VinblastineTubulin gamma-1 chaintarget
VinblastineTubulin beta chaintarget
VinblastineTranscription factor Juntarget
VinblastineCytochrome P450 3A4enzyme
VinblastineATP-dependent translocase ABCB1transporter
VinblastineMultidrug resistance-associated protein 1transporter
VinblastineATP-binding cassette sub-family C member 2transporter
VinblastineTubulin beta-2A chaintarget
VinblastineSolute carrier organic anion transporter family member 1B1transporter
VinblastineCytochrome P450 2D6enzyme
VinblastineATP-binding cassette sub-family C member 6transporter
VinblastineTubulin epsilon chaintarget
VinblastineTubulin delta chaintarget
VinblastineTubulin alpha-1A chaintarget
VinblastineBile salt export pumptransporter
VinorelbineMicrotubule-associated protein 4target
VinorelbineTubulin beta chaintarget
VinorelbineCytochrome P450 3A4enzyme
VinorelbineCytochrome P450 2D6enzyme
VinorelbineMitogen-activated protein kinase 1target
VinorelbineApoptosis regulator Bcl-2target
VismodegibAlpha-1-acid glycoprotein 1carrier
VismodegibAlbumincarrier
VismodegibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
VismodegibCytochrome P450 2C19enzyme
VismodegibCytochrome P450 2C8enzyme
VismodegibATP-dependent translocase ABCB1transporter
VismodegibCytochrome P450 3A4enzyme
VismodegibCytochrome P450 2C9enzyme
VismodegibProtein smoothenedtarget
Vitis vinifera seedDihydrofolate reductasetarget
Vitis vinifera seedCytochrome P450 3A4enzyme
VoclosporinProtein phosphatase 3 catalytic subunit alphatarget
VoclosporinGuided entry of tail-anchored proteins factor CAMLGtarget
VoclosporinCytochrome P450 3A4enzyme
VoclosporinATP-dependent translocase ABCB1transporter
VoclosporinCalcineurin subunit B type 2target
VoclosporinCalcineurin subunit B type 1target
VonoprazanHydrogen potassium ATPasetarget
VonoprazanCytochrome P450 3A4enzyme
VonoprazanCytochrome P450 3A5enzyme
VonoprazanCytochrome P450 2B6enzyme
VonoprazanPotassium-transporting ATPase subunit betatarget
VonoprazanPotassium-transporting ATPase alpha chain 1target
VonoprazanAlpha-1-acid glycoprotein 1carrier
VonoprazanAlbumincarrier
VonoprazanATP-dependent translocase ABCB1transporter
VonoprazanCytochrome P450 2D6enzyme
VonoprazanCytochrome P450 2C9enzyme
VonoprazanCytochrome P450 2C19enzyme
VoriconazoleCytochrome P450 2B6enzyme
VoriconazoleLanosterol 14-alpha demethylasetarget
VoriconazoleProstaglandin G/H synthase 1enzyme
VoriconazoleCytochrome P450 3A7enzyme
VoriconazoleCytochrome P450 3A5enzyme
VoriconazoleFlavin-containing monooxygenase 3enzyme
VoriconazoleFlavin-containing monooxygenase 1enzyme
VoriconazoleCytochrome P450 2C9enzyme
VoriconazoleCytochrome P450 3A4enzyme
VoriconazoleCytochrome P450 2C19enzyme
WarfarinNuclear receptor subfamily 1 group I member 2target
WarfarinCytochrome P450 2C18enzyme
WarfarinCytochrome P450 3A4enzyme
WarfarinCytochrome P450 2C19enzyme
WarfarinAlbumincarrier
WarfarinAlpha-1-acid glycoprotein 1carrier
WarfarinCytochrome P450 2C9enzyme
WarfarinCytochrome P450 1A2enzyme
WarfarinCytochrome P450 2C8enzyme
WarfarinVitamin K epoxide reductase complex subunit 1target
WIN 55212-2Cannabinoid receptor 1target
WIN 55212-2Cytochrome P450 3A4enzyme
WIN 55212-2Cannabinoid receptor 2target
XanomelineFlavin-containing monooxygenase 1enzyme
XanomelineFlavin-containing monooxygenase 3enzyme
XanomelineCytochrome P450 3A4enzyme
XanomelineATP-dependent translocase ABCB1transporter
XanomelineCytochrome P450 2C19enzyme
XanomelineCytochrome P450 2C9enzyme
XanomelineCytochrome P450 1A2enzyme
XanomelineCytochrome P450 2B6enzyme
XanomelineCytochrome P450 2D6enzyme
XanomelineMuscarinic acetylcholine receptor M5target
XanomelineMuscarinic acetylcholine receptor M4target
XanomelineMuscarinic acetylcholine receptor M3target
XanomelineMuscarinic acetylcholine receptor M2target
XanomelineMuscarinic acetylcholine receptor M1target
ZafirlukastCysteinyl leukotriene receptor 1target
ZafirlukastCytochrome P450 2C9enzyme
ZafirlukastCytochrome P450 2C8enzyme
ZafirlukastProstaglandin G/H synthase 1enzyme
ZafirlukastCytochrome P450 3A4enzyme
ZafirlukastCytochrome P450 1A2enzyme
ZafirlukastCytochrome P450 2C19enzyme
ZafirlukastBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
ZafirlukastCytochrome P450 2D6enzyme
ZafirlukastHepatic sodium/bile acid cotransportertransporter
ZileutonPolyunsaturated fatty acid 5-lipoxygenasetarget
ZileutonCytochrome P450 2C9enzyme
ZileutonCytochrome P450 1A2enzyme
ZileutonCytochrome P450 3A4enzyme
ZileutonProstaglandin G/H synthase 1enzyme
ZileutonUDP-glucuronosyltransferase 1A9enzyme
ZileutonAlbumincarrier
ZimelidineSodium-dependent serotonin transportertarget
ZimelidineATP-dependent translocase ABCB1transporter
ZimelidineAmine oxidase [flavin-containing] Btarget
ZimelidineAmine oxidase [flavin-containing] Atarget
ZimelidineCytochrome P450 3A4enzyme
ZimelidineSerotonin Receptorstarget
Ziprasidone5-hydroxytryptamine receptor 1Etarget
Ziprasidone5-hydroxytryptamine receptor 1Btarget
ZiprasidoneMuscarinic acetylcholine receptor M5target
ZiprasidoneMuscarinic acetylcholine receptor M4target
ZiprasidoneMuscarinic acetylcholine receptor M3target
ZiprasidoneNeuronal acetylcholine receptor subunit alpha-7target
ZiprasidoneMuscarinic acetylcholine receptor M1target
ZiprasidoneD(1B) dopamine receptortarget
ZiprasidoneD(1A) dopamine receptortarget
ZiprasidoneAlpha-2C adrenergic receptortarget
ZiprasidoneAlpha-2B adrenergic receptortarget
ZiprasidoneAlpha-1B adrenergic receptortarget
ZiprasidoneAlpha-2A adrenergic receptortarget
ZiprasidoneCytochrome P450 3A4enzyme
Ziprasidone5-hydroxytryptamine receptor 7target
ZiprasidoneD(4) dopamine receptortarget
Ziprasidone5-hydroxytryptamine receptor 2Atarget
ZiprasidoneHistamine H1 receptortarget
Ziprasidone5-hydroxytryptamine receptor 1Dtarget
Ziprasidone5-hydroxytryptamine receptor 1Atarget
ZiprasidoneD(3) dopamine receptortarget
Ziprasidone5-hydroxytryptamine receptor 2Ctarget
ZiprasidoneD(2) dopamine receptortarget
ZiprasidoneAlpha-1A adrenergic receptortarget
Ziprasidone5-hydroxytryptamine receptor 6target
ZiprasidoneAldehyde oxidaseenzyme
ZiprasidoneAlbumincarrier
ZiprasidoneATP-dependent translocase ABCB1transporter
ZiprasidoneAlpha-1-acid glycoprotein 1carrier
Ziprasidone5-hydroxytryptamine 3 receptortarget
Ziprasidone5-hydroxytryptamine receptor 5Atarget
ZiprasidoneMuscarinic acetylcholine receptor M2target
ZonisamideVoltage-dependent T-type calcium channel subunit alpha-1Gtarget
ZonisamideCytochrome P450 3A4enzyme
ZonisamideAldehyde oxidaseenzyme
ZonisamideAmine oxidase [flavin-containing] Btarget
ZonisamideCarbonic anhydrase 2target
ZonisamideCarbonic anhydrase 3target
ZonisamideCarbonic anhydrase 4target
ZonisamideCarbonic anhydrase 5A, mitochondrialtarget
ZonisamideCarbonic anhydrase 5B, mitochondrialtarget
ZonisamideCarbonic anhydrase 6target
ZonisamideCarbonic anhydrase 7target
ZonisamideCarbonic anhydrase-related proteintarget
ZonisamideCarbonic anhydrase 9target
ZonisamideCarbonic anhydrase-related protein 10target
ZonisamideCarbonic anhydrase 1target
ZonisamideCarbonic anhydrase 12target
ZonisamideCarbonic anhydrase 13target
ZonisamideCarbonic anhydrase 14target
ZonisamideVoltage-dependent T-type calcium channel subunit alpha-1Htarget
ZonisamideVoltage-dependent T-type calcium channel subunit alpha-1Itarget
ZonisamideSodium channel protein type 2 subunit alphatarget
ZonisamideSodium channel protein type 3 subunit alphatarget
ZonisamideSodium channel protein type 4 subunit alphatarget
ZonisamideSodium channel protein type 5 subunit alphatarget
ZonisamideSodium channel protein type 9 subunit alphatarget
ZonisamideSodium channel protein type 11 subunit alphatarget
ZonisamideSodium channel regulatory subunit beta-1target
ZonisamideSodium channel regulatory subunit beta-2target
ZonisamideSodium channel regulatory subunit beta-3target
ZonisamideSodium channel regulatory subunit beta-4target
ZonisamideAmine oxidase [flavin-containing] Atarget
ZonisamideCytochrome P450 2C19enzyme
ZonisamideUDP-glucuronosyltransferase 1A1enzyme
ZonisamideCytochrome P450 3A5enzyme
ZonisamideATP-dependent translocase ABCB1transporter
ZonisamideGABA(A) Receptor Benzodiazepine Binding Sitetarget
ZonisamideVoltage-gated sodium channel alpha subunittarget
ZonisamideSodium channel protein type 1 subunit alphatarget
ZonisamideCarbonic anhydrase-related protein 11target
ZucapsaicinTransient receptor potential cation channel subfamily V member 1target
ZucapsaicinCytochrome P450 1A2enzyme
ZucapsaicinCytochrome P450 2C19enzyme
ZucapsaicinCytochrome P450 2C9enzyme
ZucapsaicinCytochrome P450 2E1enzyme