| DB00206 | Reserpine | approved, investigational, withdrawn | yes | inhibitor | Details |
| DB09363 | Rauwolfia serpentina root | investigational | yes | inhibitor | Details |
| DB04844 | Tetrabenazine | approved, investigational | yes | inhibitor | Details |
| DB01089 | Deserpidine | approved | yes | inhibitor | Details |
| DB00865 | Benzphetamine | approved, illicit | yes | inducer | Details |
| DB00182 | Amphetamine | approved, illicit, investigational | yes | inhibitor | Details |
| DB06714 | Propylhexedrine | approved | yes | | Details |
| DB06706 | Isometheptene | approved | yes | inhibitor | Details |
| DB01454 | Midomafetamine | experimental, illicit, investigational | yes | inhibitor | Details |
| DB01576 | Dextroamphetamine | approved, illicit | yes | inducer | Details |
| DB01472 | 4-Methoxyamphetamine | experimental, illicit | yes | inhibitor | Details |
| DB01577 | Metamfetamine | approved, illicit, withdrawn | yes | inhibitor | Details |
| DB01363 | Ephedra sinica root | nutraceutical | yes | inhibitor | Details |
| DB01442 | MMDA | experimental, illicit | yes | inhibitor | Details |
| DB00368 | Norepinephrine | approved | unknown | binder | Details |
| DB12161 | Deutetrabenazine | approved, investigational | yes | inhibitor | Details |
| DB00988 | Dopamine | approved | unknown | | Details |
| DB00502 | Haloperidol | approved | unknown | | Details |
| DB05381 | Histamine | approved, investigational | unknown | | Details |
| DB08839 | Serotonin | investigational, nutraceutical | unknown | | Details |
| DB00579 | Mazindol | approved, investigational | unknown | | Details |
| DB04821 | Nomifensine | approved, withdrawn | unknown | | Details |
| DB01364 | Ephedrine | approved | unknown | inhibitor | Details |
| DB00714 | Apomorphine | approved, investigational | unknown | inducer | Details |