| DB00361 | Vinorelbine | approved, investigational | yes | antagonistinhibitor | Details |
| DB00541 | Vincristine | approved, investigational | yes | inhibitor | Details |
| DB00570 | Vinblastine | approved | yes | binder | Details |
| DB01394 | Colchicine | approved | yes | inhibitorbinder | Details |
| DB01873 | Epothilone D | investigational | unknown | | Details |
| DB03010 | Patupilone | experimental, investigational | unknown | | Details |
| DB05284 | CA4P | investigational | unknown | | Details |
| DB05147 | CYT997 | investigational | unknown | | Details |
| DB06042 | ZEN-012 | investigational | unknown | | Details |
| DB12334 | Milataxel | investigational | unknown | | Details |
| DB01179 | Podofilox | approved | yes | inhibitor | Details |
| DB11731 | Depatuxizumab mafodotin | investigational | yes | nucleotide exchange blocker | Details |
| DB09130 | Copper | approved, investigational | unknown | | Details |
| DB11638 | Artenimol | approved, experimental, investigational | unknown | ligand | Details |
| DB11641 | Vinflunine | approved, investigational | yes | inhibitor | Details |
| DB15534 | Colchiceine | approved, experimental | unknown | binder | Details |
| DB06137 | Tirbanibulin | approved, investigational | yes | inhibitor | Details |