| DB00790 | Perindopril | approved | yes | inhibitor | Details |
| DB01180 | Rescinnamine | approved | yes | inhibitor | Details |
| DB02032 | Epicaptopril | experimental | unknown | | Details |
| DB03740 | N-acetyl-alpha-D-glucosamine | experimental | unknown | | Details |
| DB00492 | Fosinopril | approved | yes | inhibitor | Details |
| DB00542 | Benazepril | approved, investigational | yes | inhibitor | Details |
| DB01197 | Captopril | approved | yes | inhibitor | Details |
| DB00584 | Enalapril | approved, vet_approved | yes | inhibitor | Details |
| DB00722 | Lisinopril | approved, investigational | yes | inhibitor | Details |
| DB00691 | Moexipril | approved | yes | inhibitor | Details |
| DB00881 | Quinapril | approved, investigational | yes | inhibitor | Details |
| DB00178 | Ramipril | approved | yes | inhibitor | Details |
| DB00519 | Trandolapril | approved | yes | inhibitor | Details |
| DB00886 | Omapatrilat | investigational | unknown | | Details |
| DB01348 | Spirapril | approved | yes | inhibitor | Details |
| DB01340 | Cilazapril | approved | yes | inhibitor | Details |
| DB00616 | Candoxatril | experimental | unknown | inhibitor | Details |
| DB08836 | Temocapril | experimental, investigational | unknown | inhibitor | Details |
| DB09477 | Enalaprilat | approved | yes | inhibitor | Details |
| DB13166 | Zofenopril | approved | yes | inhibitor | Details |
| DB15565 | Cilazaprilat | experimental | yes | | Details |