| DB00836 | Loperamide | approved | unknown | inhibitor | Details |
| DB00527 | Cinchocaine | approved, vet_approved | unknown | inhibitor | Details |
| DB00623 | Fluphenazine | approved | unknown | inhibitor | Details |
| DB00753 | Isoflurane | approved, vet_approved | unknown | other/unknown | Details |
| DB00850 | Perphenazine | approved | unknown | inhibitor | Details |
| DB00925 | Phenoxybenzamine | approved | unknown | inhibitor | Details |
| DB01023 | Felodipine | approved, investigational | unknown | other | Details |
| DB01069 | Promethazine | approved, investigational | unknown | inhibitor | Details |
| DB01100 | Pimozide | approved | unknown | inhibitor | Details |
| DB01373 | Calcium | nutraceutical | unknown | | Details |
| DB01429 | Aprindine | experimental | unknown | inhibitor | Details |
| DB02868 | Deacetoxyvinzolidine | experimental | unknown | | Details |
| DB03977 | Trimethyllysine | experimental | unknown | | Details |
| DB03900 | tert-butanol | experimental | unknown | | Details |
| DB04841 | Flunarizine | approved | yes | antagonist | Details |
| DB01244 | Bepridil | approved, withdrawn | unknown | binder | Details |
| DB01065 | Melatonin | approved, nutraceutical, vet_approved | unknown | | Details |
| DB04825 | Prenylamine | approved, withdrawn | unknown | | Details |
| DB01115 | Nifedipine | approved | unknown | inhibitor | Details |
| DB00622 | Nicardipine | approved, investigational | unknown | other/unknown | Details |
| DB08039 | (3Z)-N,N-DIMETHYL-2-OXO-3-(4,5,6,7-TETRAHYDRO-1H-INDOL-2-YLMETHYLIDENE)-2,3-DIHYDRO-1H-INDOLE-5-SULFONAMIDE | experimental | unknown | | Details |
| DB08231 | Myristic acid | experimental | unknown | | Details |
| DB04513 | N-(6-Aminohexyl)-5-Chloro-1-Naphthalenesulfonamide | experimental | unknown | | Details |
| DB00831 | Trifluoperazine | approved, investigational | unknown | inhibitor | Details |
| DB00477 | Chlorpromazine | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB11093 | Calcium citrate | approved, investigational | unknown | agonist | Details |
| DB11348 | Calcium Phosphate | approved | unknown | agonist | Details |
| DB13800 | Calcium levulinate | approved, experimental | unknown | agonist | Details |
| DB14481 | Calcium phosphate dihydrate | approved | unknown | | Details |
| DB04209 | Dequalinium | approved, investigational | unknown | antagonist | Details |