| DB00232 | Methyclothiazide | withdrawn | unknown | inhibitor | Details |
| DB00273 | Topiramate | approved | yes | inhibitor | Details |
| DB00436 | Bendroflumethiazide | approved | unknown | inhibitor | Details |
| DB00562 | Benzthiazide | approved | unknown | inhibitor | Details |
| DB00774 | Hydroflumethiazide | approved, investigational, withdrawn | unknown | inhibitor | Details |
| DB01021 | Trichlormethiazide | approved, vet_approved | unknown | inhibitor | Details |
| DB00869 | Dorzolamide | approved | yes | inhibitor | Details |
| DB00909 | Zonisamide | approved, investigational | unknown | inhibitor | Details |
| DB00819 | Acetazolamide | approved, vet_approved | yes | inhibitor | Details |
| DB00311 | Ethoxzolamide | withdrawn | yes | inhibitor | Details |
| DB00703 | Methazolamide | approved | yes | inhibitor | Details |
| DB01144 | Diclofenamide | approved, investigational | yes | inhibitor | Details |
| DB01194 | Brinzolamide | approved | unknown | inhibitor | Details |
| DB08846 | Ellagic acid | investigational | unknown | inhibitor | Details |
| DB09460 | Sodium carbonate | approved | unknown | inhibitor | Details |