| DB00390 | Digoxin | approved | yes | inhibitor | Details |
| DB00511 | Acetyldigitoxin | approved | yes | inhibitor | Details |
| DB01078 | Deslanoside | approved | yes | inhibitor | Details |
| DB01092 | Ouabain | approved | yes | inhibitor | Details |
| DB00774 | Hydroflumethiazide | approved, investigational, withdrawn | unknown | inducer | Details |
| DB01021 | Trichlormethiazide | approved, vet_approved | yes | inhibitor | Details |
| DB01396 | Digitoxin | approved, investigational | yes | inhibitor | Details |
| DB00903 | Etacrynic acid | approved, investigational | yes | inhibitor | Details |
| DB01119 | Diazoxide | approved | unknown | other | Details |
| DB01158 | Bretylium | approved | yes | inhibitor | Details |
| DB01244 | Bepridil | approved, withdrawn | unknown | inhibitor | Details |
| DB01345 | Potassium cation | approved, investigational | unknown | | Details |
| DB01370 | Aluminium | approved, investigational | unknown | binder | Details |
| DB01378 | Magnesium cation | approved, nutraceutical | unknown | | Details |
| DB01430 | Almitrine | approved | yes | binder | Details |
| DB06157 | Istaroxime | investigational | unknown | | Details |
| DB01188 | Ciclopirox | approved, investigational | yes | binder | Details |
| DB09479 | Rubidium Rb-82 | approved, investigational | yes | substrate | Details |
| DB13996 | Magnesium acetate | approved | unknown | | Details |
| DB13749 | Magnesium gluconate | approved, investigational | yes | inducer | Details |
| DB13620 | Potassium gluconate | approved | yes | substrate | Details |
| DB14498 | Potassium acetate | approved, investigational | unknown | | Details |
| DB14499 | Potassium sulfate | approved, investigational | unknown | | Details |
| DB14514 | Magnesium levulinate | nutraceutical | unknown | | Details |
| DB14515 | Magnesium lactate | nutraceutical | unknown | | Details |
| DB14517 | Aluminium phosphate | approved, investigational | unknown | | Details |
| DB14518 | Aluminum acetate | approved, investigational | unknown | | Details |
| DB14500 | Potassium | approved, experimental | unknown | regulator | Details |
| DB14500 | Potassium | approved, experimental | unknown | substrate | Details |