| DB00338 | Omeprazole | approved, investigational, vet_approved | unknown | inducer | Details |
| DB00515 | Cisplatin | approved | unknown | inducer | Details |
| DB01174 | Phenobarbital | approved, investigational | unknown | inducer | Details |
| DB01045 | Rifampicin | approved | unknown | inducer | Details |
| DB01115 | Nifedipine | approved | unknown | inducer | Details |
| DB01011 | Metyrapone | approved, investigational | unknown | inducer | Details |
| DB01138 | Sulfinpyrazone | approved | unknown | inhibitor | Details |
| DB01032 | Probenecid | approved, investigational | unknown | inhibitor | Details |
| DB00328 | Indomethacin | approved, investigational | unknown | inhibitor | Details |
| DB00541 | Vincristine | approved, investigational | unknown | inhibitor | Details |
| DB00661 | Verapamil | approved | unknown | inhibitor | Details |
| DB04348 | Taurocholic acid | approved, experimental | unknown | substrateinhibitor | Details |
| DB00773 | Etoposide | approved | unknown | substrateinhibitor | Details |
| DB00997 | Doxorubicin | approved, investigational | unknown | inhibitor | Details |
| DB00563 | Methotrexate | approved | unknown | substrateinhibitor | Details |
| DB01016 | Glyburide | approved | unknown | inhibitor | Details |
| DB00286 | Conjugated estrogens | approved | unknown | inhibitor | Details |
| DB02659 | Cholic Acid | approved | unknown | inhibitor | Details |
| DB00143 | Glutathione | approved, investigational, nutraceutical | unknown | substrate | Details |
| DB00158 | Folic acid | approved, nutraceutical, vet_approved | unknown | substrate | Details |
| DB08884 | Gadoxetic acid | approved | unknown | substrate | Details |
| DB00973 | Ezetimibe | approved | unknown | substrate | Details |
| DB00544 | Fluorouracil | approved | unknown | substrate | Details |
| DB00709 | Lamivudine | approved, investigational | unknown | substrate | Details |
| DB05928 | Dovitinib | investigational | unknown | | Details |
| DB00481 | Raloxifene | approved, investigational | unknown | substrate | Details |
| DB00950 | Fexofenadine | approved, investigational | unknown | substrate | Details |
| DB01069 | Promethazine | approved, investigational | unknown | inhibitor | Details |
| DB11936 | Bempedoic acid | approved, investigational | unknown | inhibitor | Details |
| DB15719 | Belantamab mafodotin | approved | unknown | substrate | Details |
| DB06813 | Pralatrexate | approved, investigational | no | substrateinhibitor | Details |