| DB00977 | Ethinylestradiol | approved | unknown | inhibitor | Details |
| DB00624 | Testosterone | approved, investigational | unknown | inhibitor | Details |
| DB00396 | Progesterone | approved, vet_approved | unknown | inhibitor | Details |
| DB00286 | Conjugated estrogens | approved | unknown | inhibitor | Details |
| DB00091 | Cyclosporine | approved, investigational, vet_approved | unknown | inhibitor | Details |
| DB02659 | Cholic Acid | approved | unknown | substrateinhibitor | Details |
| DB00887 | Bumetanide | approved | unknown | substrateinhibitor | Details |
| DB01032 | Probenecid | approved, investigational | unknown | inhibitor | Details |
| DB01586 | Ursodeoxycholic acid | approved, investigational | unknown | substrateinhibitor | Details |
| DB04348 | Taurocholic acid | approved, experimental | unknown | substrate | Details |
| DB00279 | Liothyronine | approved, vet_approved | unknown | substrate | Details |
| DB00328 | Indomethacin | approved, investigational | unknown | substrate | Details |
| DB03619 | Deoxycholic acid | approved | unknown | substrate | Details |
| DB02123 | Glycochenodeoxycholic Acid | experimental | unknown | substrate | Details |
| DB01583 | Liotrix | approved | unknown | substrate | Details |
| DB08860 | Pitavastatin | approved | unknown | substrate | Details |
| DB06290 | Simeprevir | approved | unknown | inhibitor | Details |
| DB13943 | Testosterone cypionate | approved | unknown | inhibitor | Details |
| DB13944 | Testosterone enanthate | approved | unknown | inhibitor | Details |
| DB13946 | Testosterone undecanoate | approved, investigational | unknown | inhibitor | Details |
| DB01098 | Rosuvastatin | approved | unknown | | Details |
| DB09100 | Thyroid, porcine | approved | unknown | substrate | Details |
| DB14761 | Remdesivir | approved, investigational | unknown | inhibitor | Details |
| DB15248 | Bulevirtide | approved, investigational | yes | inhibitor | Details |
| DB15688 | Zavegepant | investigational | unknown | substrate | Details |
| DB00412 | Rosiglitazone | approved, investigational | unknown | inhibitor | Details |
| DB00549 | Zafirlukast | approved, investigational | unknown | inhibitor | Details |
| DB03604 | Tiratricol | investigational | unknown | inhibitor | Details |
| DB00795 | Sulfasalazine | approved | unknown | inhibitor | Details |
| DB13215 | Sulfobromophthalein | experimental | unknown | inhibitor | Details |
| DB04574 | Estrone sulfate | approved | unknown | inhibitor | Details |