Anti-Allergic Agents

Name
Anti-Allergic Agents
Accession Number
DBCAT000133
Description

Agents that are used to treat allergic reactions. Most of these drugs act by preventing the release of inflammatory mediators or inhibiting the actions of released mediators on their target cells. (From AMA Drug Evaluations Annual, 1994, p475)

Drugs
DrugDrug Description
AmlexanoxUsed as a paste in the mouth to treat aphthous ulcers (canker sores).
AntazolineAn antihistamine agent used for the symptomatic treatment of nasal congestion and allergic conjunctivitis.
AstemizoleA second generation antihistamine used to treat allergy symptoms.
AzelastineA histamine H1-receptor antagonist used intranasally to treat allergic and vasomotor rhinitis and in an ophthalmic solution to treat allergic conjunctivitis.
BepotastineAn ophthalmic H1 antagonist used to treat itchiness associated with allergic conjunctivitis.
BrompheniramineA histamine H1 antagonist used to treat coughs, upper respiratory symptoms, and nasal congestion associated with allergies and the common cold.
CetirizineA selective Histamine-1 antagonist drug used in allergic rhinitis and chronic urticaria.
ChlorpheniramineA histamine-H1 receptor antagonist indicated for the management of symptoms associated with upper respiratory allergies.
CiclesonideA glucocorticoid used in the symptomatic relief of nasal symptoms associated with seasonal and perennial allergic rhinitis in adults and adolescents.
ClemastineAn antihistamine with sedative and anticholinergic effects used to treat the symptoms of allergic rhinitis.
Cromoglicic acidA medication used to treat asthma, allergic reactions of the eyes and nose, as well as other mast cell reactions.
CyproheptadineA combined serotonin and histamine antagonist used in the treatment of allergic symptoms, for appetite stimulation, and off-label in the treatment of serotonin syndrome.
Dexamethasone isonicotinateDexamethasone isonicotinate is an anti-inflammatory, anti-allergic glucocorticoid that can be administered orally, by inhalation, topically, and parenterally. Its unintended mineralocorticoid action may cause salt and water retention.
DimetindeneA 1st generation selective H1 antagonist used topically as an antipruritic and orally to treat allergies.
DiphenhydramineA H1 receptor antihistamine used in the treatment of seasonal allergies, and various allergic reactions including sneezing, runny nose, itchy/watery eyes, itching of nose or throat, pruritus, urticaria, insect bites/stings, and allergic rashes.
EmedastineA selective H1-receptor antagonist used topically to manage symptoms of allergic conjunctivitis.
FexofenadineA selective H1-antagonist for the symptomatic treatment of seasonal allergic rhinitis and chronic idiopathic urticaria.
FluocinonideA high potency corticosteroid commonly used topically for a number of inflammatory skin conditions.
FluorometholoneAn ophthalmic corticosteroid used for the relief of inflammation located in both the palpebral and bulbar conjunctiva, the cornea, and the anterior segment of the globe of the eye.
FluticasoneA corticosteroid indicated in the treatment of corticosteroid responsive dermatoses, asthma, and COPD.
Fluticasone propionateA glucocorticoid used to treat asthma, inflammatory pruritic dermatoses, and nonallergic rhinitis.
HonokiolHonokiol is under investigation in clinical trial NCT00966953 (Development of Clinical Method to Determination Triclosan Retention in Plaque Following Brushing.).
Isospaglumic acidIsospaglumic acid is a small molecule drug. Isospaglumic acid is under investigation in clinical trial NCT06800274 (Clinical and Biological Evaluation of NAAGA Versus Azelastine Eye Drops in Allergic Subjects With...
KetotifenA histamine H1 receptor blocker and mast cell stabilizer used to treat mild atopic asthma and allergic conjunctivitis.
LevocabastineA selective histamine H1 receptor antagonist indicated for the management of seasonal allergic conjunctivitis symptoms.
LodoxamideAn ophthalmic agent used for the treatment of the ocular disorders referred to by the terms vernal keratoconjunctivitis, vernal conjunctivitis, and vernal keratitis.
LoratadineA second generation antihistamine used to manage the symptoms of allergic rhinitis.
LoteprednolA corticosteroid indicated in the treatment of pain and inflammation after cataract surgery.
Loteprednol etabonateA corticosteroid used to treat allergic conjunctivitis as well as inflammation and pain after ocular surgery.
MeclizineA histamine H1 antagonist used to treat nausea, vomiting, and dizziness associated with motion sickness.
MepyramineAn antihistamine agent used for the symptomatic treatment of allergy, hypersensitivity reactions, and pruritic skin disorders.
MequitazineFor the treatment of Hay fever, urticaria (hives) and allergic rhinitis
MethapyrileneMethapyrilene, formerly marketed in many drug products, was shown to be a potent carcinogen. Manufacturers voluntarily withdrew methapyriline drug products from the market in May and June 1979.
MometasoneA corticosteroid with no indications.
Mometasone furoateA corticosteroid used to treat asthma, allergic rhinitis, nasal congestion, nasal polyps, dermatitis, and pruritus.
NedocromilA pyrano quinoline used to treat allergic conjunctivitis.
OlopatadineA histamine H1 antagonist used to treat allergic conjunctivitis and rhinitis.
OmalizumabA monoclonal anti-immunoglobulin E (IgE) antibody used to treat asthma, chronic idiopathic urticaria, chronic rhinosinusitis with nasal polyps, and IgE-mediated food allergy.
OxatomideAn antihistamine indicated in the treatment and prevention of allergic symptoms.
PheniramineAn antihistamine used to treat allergic rhinitis and pruritus.
PromethazineA first-generation antihistamine used for the treatment of allergic conditions, nausea and vomiting, and motion sickness.
SuplatastSuplatast is under investigation in clinical trial NCT05983471 (Efficacy and Safety of ME-015 (Suplatast Tosilate) in Cough Related to Idiopathic Pulmonary Fibrosis (COSMIC-IPF)).
TixocortolA corticosteroid used for the symptomatic treatment of rhinitis, pharyngitis, and ulcerative colitis.
TranilastFor the treatment of bronchial asthma, keloid and hypertrophic scar, and allergic disorders such as asthma, allergic rhinitis and atopic dermatitis.
TripelennamineA histamine H1 antagonist used to treat hypersensitivity reactions, coughs, and the common cold.
TriprolidineA sedating antihistamine combined with pseudoephedrine and guaifenesin in various types of cold and allergy medications to relieve allergy symptoms, hay fever and common cold symptoms, and to aid in sleep.
Drugs & Drug Targets
DrugTargetType
AmlexanoxPhosphodiesterase 4target
AmlexanoxHeat shock protein HSP 90-alphatarget
AmlexanoxFibroblast growth factor 1target
AmlexanoxProtein S100-A13target
AmlexanoxProtein S100-A12target
AmlexanoxInterleukin-3target
AntazolineHistamine H1 receptortarget
AstemizoleCytochrome P450 2D6enzyme
AstemizoleBile salt export pumptransporter
AstemizoleMicrotubule-associated protein tautarget
AstemizoleVoltage-gated delayed rectifier potassium channel KCNH1target
AstemizoleCytochrome P450 2J2enzyme
AstemizoleATP-dependent translocase ABCB1transporter
AstemizoleCytochrome P450 3A7enzyme
AstemizoleCytochrome P450 3A5enzyme
AstemizoleCytochrome P450 3A4enzyme
AstemizoleVoltage-gated inwardly rectifying potassium channel KCNH2target
AstemizoleHistamine H1 receptortarget
AzelastineCytochrome P450 1A1enzyme
AzelastineCytochrome P450 2C8enzyme
AzelastineCytochrome P450 2C19enzyme
AzelastineCytochrome P450 3A4enzyme
AzelastineCytochrome P450 2D6enzyme
AzelastineCytochrome P450 1A2enzyme
AzelastineHistamine H1 receptortarget
AzelastinePhospholipase A2target
AzelastineHistamine H2 receptortarget
AzelastineCytochrome P450 3A5enzyme
AzelastineCytochrome P450 2A6enzyme
AzelastineCytochrome P450 2C9enzyme
AzelastineATP-dependent translocase ABCB1transporter
AzelastineCytochrome P450 2B6enzyme
AzelastineLeukotriene C4 synthasetarget
AzelastineCytochrome P450 2E1enzyme
BepotastineHistamine H1 receptortarget
BrompheniramineMuscarinic acetylcholine receptor M5target
BrompheniramineHistamine H1 receptortarget
BrompheniramineMuscarinic acetylcholine receptor M1target
BrompheniramineMuscarinic acetylcholine receptor M2target
BrompheniramineMuscarinic acetylcholine receptor M3target
BrompheniramineMuscarinic acetylcholine receptor M4target
CetirizineHistamine H1 receptortarget
CetirizineATP-dependent translocase ABCB1transporter
ChlorpheniramineCytochrome P450 3A7enzyme
ChlorpheniramineSolute carrier family 22 member 2transporter
ChlorpheniramineSolute carrier family 22 member 1transporter
ChlorpheniramineCytochrome P450 3A5enzyme
ChlorpheniramineSodium-dependent dopamine transportertarget
ChlorpheniramineSodium-dependent noradrenaline transportertarget
ChlorpheniramineSodium-dependent serotonin transportertarget
ChlorpheniramineCytochrome P450 2D6enzyme
ChlorpheniramineCytochrome P450 3A4enzyme
ChlorpheniramineHistamine H1 receptortarget
CiclesonideCorticosteroid-binding globulincarrier
CiclesonideCytochrome P450 3A4enzyme
CiclesonideCytochrome P450 2D6enzyme
CiclesonideGlucocorticoid receptortarget
CiclesonideLiver carboxylesterase 1enzyme
CiclesonideCorticosteroid-binding globulintarget
ClemastineCytochrome P450 2D6enzyme
ClemastineHistamine H1 receptortarget
Cromoglicic acidProtein S100-Ptarget
Cromoglicic acidHeat shock protein HSP 90-alphatarget
Cyproheptadine5-hydroxytryptamine receptor 2Atarget
CyproheptadineMuscarinic acetylcholine receptor M1target
CyproheptadineMuscarinic acetylcholine receptor M2target
CyproheptadineMuscarinic acetylcholine receptor M3target
Cyproheptadine5-hydroxytryptamine receptor 2Ctarget
CyproheptadineUDP-glucuronosyltransferase 1A3enzyme
Cyproheptadine5-hydroxytryptamine receptor 7target
CyproheptadineUDP-glucuronosyltransferase 2B10enzyme
CyproheptadineUDP-glucuronosyltransferase 1A4enzyme
Cyproheptadine5-hydroxytryptamine receptor 2Btarget
CyproheptadineHistamine H2 receptortarget
CyproheptadineSolute carrier family 22 member 1transporter
CyproheptadineAlbumincarrier
CyproheptadineHistamine H1 receptortarget
Dexamethasone isonicotinateCytochrome P450 3A4enzyme
Dexamethasone isonicotinateCytochrome P450 3A5enzyme
DimetindeneHistamine H1 receptortarget
DimetindeneMuscarinic acetylcholine receptor M2target
DiphenhydramineSolute carrier family 22 member 2transporter
DiphenhydramineOrganic cation/carnitine transporter 2transporter
DiphenhydramineProstaglandin G/H synthase 1enzyme
DiphenhydramineMuscarinic acetylcholine receptor M2target
DiphenhydramineHistamine N-methyltransferasetarget
DiphenhydramineCytochrome P450 2C19enzyme
DiphenhydramineCytochrome P450 2C9enzyme
DiphenhydramineCytochrome P450 2D6enzyme
DiphenhydramineHistamine H1 receptortarget
EmedastineHistamine H1 receptortarget
FexofenadineSolute carrier organic anion transporter family member 1A2transporter
FexofenadineSolute carrier organic anion transporter family member 2B1transporter
FexofenadineATP-dependent translocase ABCB1transporter
FexofenadineHistamine H1 receptortarget
FexofenadineSolute carrier organic anion transporter family member 1B1transporter
FexofenadineSolute carrier organic anion transporter family member 1B3transporter
FexofenadineOrganic anion transporter 3transporter
FexofenadineATP-binding cassette sub-family C member 2transporter
FexofenadineATP-binding cassette sub-family C member 3transporter
FexofenadineAlbumincarrier
Fexofenadinealpha1-acid glycoproteincarrier
FluocinonideEstrogen-related receptor gammatarget
FluocinonideSteroid hormone receptor ERR2target
FluocinonideSteroid hormone receptor ERR1target
FluocinonideCytochrome P450 3A5enzyme
FluocinonideCytochrome P450 3A4enzyme
FluocinonideProtein smoothenedtarget
FluocinonideGlucocorticoid receptortarget
FluocinonideCorticosteroid-binding globulincarrier
FluorometholoneCorticosteroid-binding globulincarrier
FluorometholoneCytochrome P450 3A4enzyme
FluorometholoneGlucocorticoid receptortarget
FluorometholoneCytochrome P450 3A5enzyme
FluticasoneCytosolic phospholipase A2target
FluticasoneProgesterone receptortarget
FluticasoneCytochrome P450 3A7enzyme
FluticasoneCytochrome P450 3A5enzyme
FluticasoneCorticosteroid-binding globulincarrier
FluticasoneGlucocorticoid receptortarget
FluticasoneSolute carrier organic anion transporter family member 1B1transporter
FluticasoneATP-dependent translocase ABCB1transporter
FluticasoneCytochrome P450 3A4enzyme
FluticasoneSolute carrier organic anion transporter family member 1B1carrier
FluticasoneATP-dependent translocase ABCB1carrier
FluticasoneMineralocorticoid receptortarget
FluticasoneCytochrome P450 2C8enzyme
Fluticasone propionateSolute carrier organic anion transporter family member 1B1transporter
Fluticasone propionateATP-dependent translocase ABCB1transporter
Fluticasone propionateSolute carrier organic anion transporter family member 1B1carrier
Fluticasone propionateCytochrome P450 2C8enzyme
Fluticasone propionateCytochrome P450 3A5enzyme
Fluticasone propionateMineralocorticoid receptortarget
Fluticasone propionateProgesterone receptortarget
Fluticasone propionateCytochrome P450 3A4enzyme
Fluticasone propionateGlucocorticoid receptortarget
Fluticasone propionateCytosolic phospholipase A2target
Fluticasone propionateCorticosteroid-binding globulincarrier
Fluticasone propionateCytochrome P450 3A7enzyme
HonokiolProstaglandin G/H synthase 1target
HonokiolProstaglandin G/H synthase 2target
HonokiolPolyunsaturated fatty acid 5-lipoxygenasetarget
Isospaglumic acidMetabotropic glutamate receptor 3target
Ketotifen6-phosphogluconate dehydrogenase, decarboxylatingtarget
KetotifenUDP-glucuronosyltransferase 1A3enzyme
KetotifenUDP-glucuronosyltransferase 1A4enzyme
KetotifenUDP-glucuronosyltransferase 2B10enzyme
KetotifenHistamine H1 receptortarget
LevocabastineNeurotensin receptor type 2target
LevocabastineHistamine H1 receptortarget
LodoxamideG protein-coupled receptor 35target
LodoxamideXanthine dehydrogenase/oxidasetarget
LoratadineUDP-glucuronosyltransferase 1A3enzyme
LoratadineHistamine H1 receptortarget
LoratadineCytochrome P450 3A4enzyme
LoratadineCytochrome P450 2C19enzyme
LoratadineUDP-glucuronosyltransferase 2B15enzyme
LoratadineUDP-glucuronosyltransferase 1A1enzyme
LoratadineUDP-glucuronosyltransferase 2B10enzyme
LoratadineCytochrome P450 3A5enzyme
LoratadineCytochrome P450 2C9enzyme
LoratadineCytochrome P450 2D6enzyme
LoratadineCytochrome P450 2C8enzyme
LoratadineATP-dependent translocase ABCB1transporter
LoratadineVoltage-gated inwardly rectifying potassium channel KCNH2target
LoratadineBile salt export pumptransporter
LoratadineCytochrome P450 1A1enzyme
LoratadineCytochrome P450 2B6enzyme
LoratadineCytochrome P450 1A2enzyme
LoteprednolGlucocorticoid receptortarget
Loteprednol etabonateEstrogen-related receptor gammatarget
Loteprednol etabonateSteroid hormone receptor ERR2target
Loteprednol etabonateSteroid hormone receptor ERR1target
Loteprednol etabonateSerum paraoxonase/arylesterase 1enzyme
Loteprednol etabonateCytochrome P450 3A4enzyme
Loteprednol etabonateGlucocorticoid receptortarget
MeclizineCytochrome P450 2D6enzyme
MeclizineHistamine H1 receptortarget
MeclizineNuclear receptor subfamily 1 group I member 3target
MeclizineAlbumincarrier
MepyramineOrganic cation/carnitine transporter 2transporter
MepyramineSolute carrier family 22 member 4transporter
MepyramineHistamine H1 receptortarget
MepyramineCytochrome P450 2D6enzyme
MequitazineCytochrome P450 3A4enzyme
MequitazineCytochrome P450 2D6enzyme
MequitazineHistamine H1 receptortarget
MethapyrileneHistamine H1 receptortarget
MometasoneCytochrome P450 3A5enzyme
MometasoneCytochrome P450 3A4enzyme
MometasoneProgesterone receptortarget
MometasoneCytochrome P450 2C8enzyme
MometasoneGlucocorticoid receptortarget
Mometasone furoateGlucocorticoid receptortarget
Mometasone furoateCytochrome P450 3A5enzyme
Mometasone furoateCytochrome P450 2C8enzyme
Mometasone furoateProgesterone receptortarget
Mometasone furoateCytochrome P450 3A4enzyme
NedocromilCysteinyl leukotriene receptor 1target
NedocromilCysteinyl leukotriene receptor 2target
NedocromilProstaglandin D2 receptortarget
NedocromilN-formyl peptide receptor 1target
OlopatadineHistamine H1 receptortarget
OlopatadineProtein S100-A1target
OlopatadineHistamine H3 receptortarget
OlopatadineHistamine H2 receptortarget
OlopatadineATP-dependent translocase ABCB1transporter
OlopatadineFlavin-containing monooxygenase 3enzyme
OlopatadineFlavin-containing monooxygenase 1enzyme
OlopatadineAlbumincarrier
OlopatadineCytochrome P450 3A4enzyme
OlopatadineProtein S100-A2target
OlopatadineProtein S100-A13target
OlopatadineProtein S100-Btarget
OlopatadineProtein S100-A12target
OmalizumabHigh affinity immunoglobulin epsilon receptor subunit gammatarget
OmalizumabImmunoglobulin heavy constant epsilontarget
OxatomideHistamine H1 receptortarget
PheniramineHistamine H4 receptortarget
PheniramineNuclear receptor subfamily 1 group I member 3target
PheniramineHistamine H1 receptortarget
PromethazineATP-binding cassette sub-family C member 3transporter
PromethazineNMDA receptortarget
PromethazineCalmodulintarget
PromethazineAlbumincarrier
PromethazineATP-binding cassette sub-family C member 4transporter
PromethazineVoltage-gated Potassium Channelstarget
PromethazineD(2) dopamine receptortarget
PromethazineHistamine H1 receptortarget
PromethazineMuscarinic acetylcholine receptor M4target
PromethazineMuscarinic acetylcholine receptor M1target
PromethazineMuscarinic acetylcholine receptor M5target
PromethazineMuscarinic acetylcholine receptor M2target
PromethazineMuscarinic acetylcholine receptor M3target
PromethazineCytochrome P450 2D6enzyme
PromethazineCytochrome P450 2B6enzyme
PromethazineATP-dependent translocase ABCB1transporter
PromethazineCytochrome P450 2C9enzyme
PromethazineHistamine H2 receptortarget
PromethazineAlpha adrenergic receptortarget
PromethazineP2 Purinoceptorstarget
PromethazineVoltage-gated sodium channel alpha subunittarget
TixocortolGlucocorticoid receptortarget
TixocortolHistone deacetylase 2target
TranilastHematopoietic prostaglandin D synthasetarget
TranilastCytochrome P450 3A4enzyme
TranilastCytochrome P450 2C9enzyme
TranilastHistamine H1 receptortarget
TranilastSteryl-sulfatasetarget
TripelennamineAlbumincarrier
TripelennamineHistamine H1 receptortarget
TripelennamineCytochrome P450 2D6enzyme
TriprolidineHistamine H1 receptortarget
TriprolidineAlbumincarrier