| Atropine | A muscarinic antagonist used to treat poisoning by muscarinic agents, including organophosphates and other drugs. | |
| Betamethasone | A systemic corticosteroid used to relieve inflammation in various conditions, including but not limited to allergic states, dermatologic disorders, gastrointestinal diseases, and hematological disorders. | |
| Bosentan | A dual endothelin receptor antagonist used to treat pulmonary arterial hypertension. | |
| Bromfenac | An NSAID used to treat postoperative pain and inflammation of the eye. | |
| Bupivacaine | A local anesthetic used in a wide variety of superficial and invasive procedures. | |
| Chloramphenicol | A broad spectrum antibiotic that is effective against a variety of susceptible and serious bacterial infections but is not frequently used because of its high risk of bone marrow toxicity. | |
| Chlorhexidine | An antiseptic used to sterilize for surgeries and in healthcare practice, to reduce pocket depth in periodontitis, and to treat gingivitis. | |
| Desonide | A topical corticosteroid used for the symptomatic treatment of inflammatory and pruritic manifestations of corticosteroid responsive dermatoses. | |
| Dexamethasone | A glucocorticoid available in various modes of administration that is used for the treatment of various inflammatory conditions, including bronchial asthma, as well as endocrine and rheumatic disorders. | |
| Diclofenac | An NSAID used to treat the signs and symptoms of osteoarthritis and rheumatoid arthritis. | |
| Difluprednate | A topical corticosteroid used for the symptomatic treatment of inflammation and pain associated with ocular surgery. | |
| Fluorometholone | An ophthalmic corticosteroid used for the relief of inflammation located in both the palpebral and bulbar conjunctiva, the cornea, and the anterior segment of the globe of the eye. | |
| Gentamicin | An aminoglycoside used to treat a wide variety of aerobic infections in the body. | |
| Gramicidin D | A bactericidal antibiotic used in the treatment of dermatological and ophthalmic infections. | |
| Hydrocortisone acetate | A corticosteroid used to treat inflammatory and pruritic corticosteroid-responsive dermatoses and ulcerative colitis. | |
| Hydrocortisone phosphate | A corticosteroid used to treat congenital adrenal hyperplasia, for emergency asthma treatment, hypersensitivity, and inflammation. | |
| Loteprednol | A corticosteroid indicated in the treatment of pain and inflammation after cataract surgery. | No drug targets |
| Loteprednol etabonate | A corticosteroid used to treat allergic conjunctivitis as well as inflammation and pain after ocular surgery. | |
| Methylprednisolone | A corticosteroid used to treat inflammation or immune reactions across a variety of organ systems, endocrine conditions, and neoplastic diseases. | |
| Naphazoline | A sympathomimetic vasoconstrictor used for the symptomatic relief of redness and itching of the eye, and nasal congestion. | |
| Netilmicin | An aminoglycoside used to treat a wide variety of infections in the body. | |
| Phenylephrine | An alpha-1 adrenergic agonist used in the management of hypotension, generally in the surgical setting associated with the use of anesthetics. | |
| Polymyxin B | A polymyxin antibiotic used to treat a wide variety of infections in the body. | |
| Prednisolone | A glucocorticoid used to treat adrenocortical insufficiency, inflammatory conditions, and some cancers. | |
| Prednisolone acetate | A glucocorticoid used to treat a wide variety of endocrine, inflammatory, and immune conditions as well as for palliation of neoplastic conditions. | |
| Prednisolone phosphate | A corticosteroid used to treat inflammation, immune reactions, as well as endocrine or neoplastic conditions. | |
| Prednisone | A corticosteroid used to treat inflammation or immune-mediated reactions and to treat endocrine or neoplastic diseases. | |
| Rimexolone | A glucocorticoid used to treat inflammation of the eye. | |
| Spaglumic acid | The β-aspartyl isoform of N-Acetyl-l-aspartylglutamate, a naturally occurring neurotransmitter, used in allergic eye conditions due to its ability to stabilize mast cells. | |
| Tetryzoline | An alpha-adrenergic agonist used in the temporary symptomatic relief of discomfort and redness of the eyes due to minor irritations, as well as alleviate nasal congestion. | |
| Tobramycin | An aminoglycoside antibiotic used to treat cystic fibrosis-associated bacterial, lower respiratory tract, urinary tract, eye, skin, bone, and skin structure infections. | |
| Triamcinolone | A glucocorticoid used to treat a wide variety of inflammatory conditions of organ systems and tissues. | |