Aticaprant

DB12341InvestigationalSmall molecule

Aticaprant has been used in trials studying the health services research and basic science of Anxiety Disorders and Alcohol Dependence.

Chemical structure of Aticaprant
Mechanism
Curator reviewed
Formula / weight
C26H27FN2O2 · 418.512 g/mol (avg)
Also known as
BENZAMIDE, 4-(4-(((2S)-2-(3,5-DIMETHYLPHENYL)-1-PYRROLIDINYL)METHYL)PHENOXY)-3-FLUORO-
Code names
CERC-501 · JNJ-67953964 · JSPA-0658 · LY-2456302

Resolves to

Compound
UNIIDE4G8X55F5CAS1174130-61-0ChEMBLCHEMBL1921847PubChem44129648
Structure
InChIKeyZHPMYDSXGRRERG-DEOSSOPVSA-NSMILESCC1=CC(=CC(C)=C1)[C@@H]1CCCN1CC1=CC=C(OC2=CC=C(C=C2F)C(N)=O)C=C1
Targets
P41145OPRK1

What you can answer from here — as of June 15, 2026

1Protein targetEach mapped to UniProt, with action and pharmacological action
Listed above
54Drug interactionsStructured to mechanism, not free text
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13Clinical trialsPhase, status and sponsor resolved per trial
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4+ReferencesStructured and connected to the statements they support
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Which drugs share a target with Aticaprant, and which of those have an active Phase 3 trial?

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