| DB00711 | Diethylcarbamazine | approved, investigational, vet_approved | yes | inhibitor | Details |
| DB00471 | Montelukast | approved | unknown | other/unknown | Details |
| DB00744 | Zileuton | approved, investigational, withdrawn | yes | inhibitor | Details |
| DB00939 | Meclofenamic acid | approved, vet_approved | yes | inhibitor | Details |
| DB01017 | Minocycline | approved, investigational | unknown | inhibitor | Details |
| DB01892 | Hyperforin | nutraceutical | unknown | inhibitor | Details |
| DB04725 | Licofelone | investigational | unknown | | Details |
| DB00163 | Vitamin E | approved, nutraceutical, vet_approved | unknown | | Details |
| DB00179 | Masoprocol | approved, investigational | yes | inhibitor | Details |
| DB05431 | MLN-977 | investigational | unknown | | Details |
| DB01014 | Balsalazide | approved, investigational | yes | inhibitor | Details |
| DB00244 | Mesalazine | approved | yes | inhibitor | Details |
| DB00795 | Sulfasalazine | approved | yes | inhibitor | Details |
| DB00233 | Aminosalicylic acid | approved | unknown | inhibitor | Details |
| DB13174 | Rhein | experimental | unknown | inhibitor | Details |
| DB11994 | Diacerein | approved, investigational | unknown | inhibitor | Details |
| DB11133 | Omega-3 fatty acids | approved, nutraceutical | unknown | substrate | Details |
| DB13168 | Omega-6 fatty acids | nutraceutical | unknown | substrate | Details |
| DB02709 | Resveratrol | investigational | unknown | | Details |
| DB09061 | Cannabidiol | approved, investigational | unknown | inhibitor | Details |
| DB09285 | Morniflumate | experimental | unknown | antagonist | Details |
| DB09285 | Morniflumate | experimental | unknown | inhibitor | Details |
| DB14001 | alpha-Tocopherol succinate | approved, nutraceutical, vet_approved | unknown | | Details |
| DB14002 | D-alpha-Tocopherol acetate | approved, nutraceutical, vet_approved | unknown | | Details |
| DB14011 | Nabiximols | investigational | unknown | inhibitor | Details |
| DB14009 | Medical Cannabis | experimental, investigational | unknown | inhibitor | Details |
| DB12010 | Fostamatinib | approved, investigational | unknown | inhibitor | Details |
| DB00586 | Diclofenac | approved, vet_approved | unknown | potentiator | Details |
| DB00159 | Icosapent | approved, nutraceutical | unknown | substrate | Details |