| DB00145 | Glycine | approved, nutraceutical, vet_approved | unknown | ligand | Details |
| DB00753 | Isoflurane | approved, vet_approved | yes | agonist | Details |
| DB00898 | Ethanol | approved | yes | agonist | Details |
| DB01028 | Methoxyflurane | approved, investigational, vet_approved, withdrawn | yes | agonist | Details |
| DB01159 | Halothane | approved, vet_approved | unknown | allosteric modulator | Details |
| DB01189 | Desflurane | approved | yes | agonist | Details |
| DB01236 | Sevoflurane | approved, vet_approved | yes | agonist | Details |
| DB03929 | D-Serine | approved, experimental | unknown | | Details |
| DB05417 | GW 468816 | investigational | unknown | | Details |
| DB01381 | Ginkgo biloba | approved, investigational, nutraceutical | unknown | antagonist | Details |
| DB00431 | Lindane | approved, withdrawn | unknown | antagonist | Details |
| DB11582 | Thiocolchicoside | experimental | unknown | antagonist | Details |
| DB00572 | Atropine | approved, vet_approved | unknown | antagonist | Details |
| DB00466 | Picrotoxin | experimental | unknown | antagonist | Details |
| DB01956 | Taurine | approved, nutraceutical | unknown | agonist | Details |
| DB09130 | Copper | approved, investigational | unknown | | Details |
| DB01593 | Zinc | approved, investigational | unknown | | Details |
| DB09061 | Cannabidiol | approved, investigational | unknown | | Details |
| DB14011 | Nabiximols | investigational | unknown | | Details |
| DB14009 | Medical Cannabis | experimental, investigational | unknown | | Details |
| DB14487 | Zinc acetate | approved, investigational | unknown | | Details |
| DB14533 | Zinc chloride | approved, investigational | unknown | inhibitor | Details |
| DB14548 | Zinc sulfate, unspecified form | approved, experimental | unknown | inhibitor | Details |
| DB00228 | Enflurane | approved, investigational, vet_approved | yes | potentiator | Details |