| DB01118 | Amiodarone | approved, investigational | yes | inhibitordownregulator | Details |
| DB00182 | Amphetamine | approved, illicit, investigational | unknown | agonist | Details |
| DB00540 | Nortriptyline | approved | unknown | antagonist | Details |
| DB00726 | Trimipramine | approved | unknown | binder | Details |
| DB00334 | Olanzapine | approved, investigational | no | inhibitor | Details |
| DB00217 | Bethanidine | approved | unknown | antagonist | Details |
| DB01365 | Mephentermine | approved | unknown | agonist | Details |
| DB06726 | Bufuralol | experimental | unknown | antagonist | Details |
| DB13345 | Dihydroergocristine | approved, experimental | yes | antagonistagonist | Details |
| DB01049 | Ergoloid mesylate | approved | yes | antagonistagonist | Details |
| DB11273 | Dihydroergocornine | approved | yes | antagonistagonist | Details |
| DB11278 | DL-Methylephedrine | approved | yes | agonist | Details |
| DB00715 | Paroxetine | approved, investigational | unknown | inhibitor | Details |
| DB00785 | Cryptenamine | approved | unknown | inhibitorpotentiator | Details |
| DB00867 | Ritodrine | approved, investigational | yes | agonistdownregulator | Details |
| DB00264 | Metoprolol | approved, investigational | unknown | inhibitor | Details |