Neuromuscular Blocking Agents

Name
Neuromuscular Blocking Agents
Accession Number
DBCAT000511
Description

Drugs that interrupt transmission of nerve impulses at the skeletal neuromuscular junction. They can be of two types, competitive, stabilizing blockers (NEUROMUSCULAR NONDEPOLARIZING AGENTS) or noncompetitive, depolarizing agents (NEUROMUSCULAR DEPOLARIZING AGENTS). Both prevent acetylcholine from triggering the muscle contraction and they are used as anesthesia adjuvants, as relaxants during electroshock, in convulsive states, etc.

Drugs
DrugDrug Description
AlcuroniumA non-depolarizing skeletal muscle relaxant similar to tubocurarine. It is used as an anesthesia adjuvant.
AtracuriumA neuromuscular blocker indicated to relax muscles during mechanical ventilation under general anesthesia or intubation.
Atracurium besylateA non-depolarizing neuromuscular blocker used to facilitate endotracheal intubation and relax skeletal muscles during surgery.
Botulinum toxin type AA purified form of botulinum toxin type A used to block acetylcholine release in the treatment of chronic sialorrhea, muscle spasticity, and dystonia, as well as in cosmetic applications.
CisatracuriumA skeletal muscle relaxant used to facilitate tracheal intubation, muscle relaxation in surgery, or mechanical ventilation.
DaxibotulinumtoxinAA botulinum toxin used to treat glabellar lines and cervical dystonia in adults.
DecamethoniumFor use as a skeletal muscle relaxant
DoxacuriumA nondepolarizing neuromuscular blocking agent used as an adjunct to general anesthesia to facilitate tracheal intubation, and to provide skeletal muscle relaxation during surgical procedures.
GallamineNot Annotated
Gallamine triethiodideA nondepolarizing nerve blocker used in addition to anesthesia to cause skeletal muscle relaxation.
LetibotulinumtoxinAA purified type A botulinum neurotoxin protein complex used to improve the appearance of glabellar lines.
MetocurineMetocurine is a muscle relaxant.
Metocurine iodideFor use as an anesthesia adjunct to induce skeletal muscle relaxation and to reduce the intensity of muscle contractions in convulsive therapy.
MivacuriumA short-acting non-depolarizing neuromuscular blocking agent used to induce anesthesia during intubation and promote skeletal muscle relaxation during surgery or mechanical ventilation.
NeosaxitoxinNeosaxitoxin is under investigation in clinical trial NCT01786655 (Safety Study of Long-Acting Local Anesthetic).
PancuroniumA neuromuscular blocker used as an adjunct to general anesthesia to facilitate tracheal intubation and to provide skeletal muscle relaxation during surgery or mechanical ventilation.
PipecuroniumA nondepolarizing neuromuscular blocking agent used to relax muscles during anesthesia and surgical procedures.
PyrantelAn anthelmintic used to treat helminth infections.
RapacuroniumA nondepolarizing neuromuscular blocking agent used as an adjunct to general anesthesia to facilitate tracheal intubation, and to provide skeletal muscle relaxation during surgical procedures.
RocuroniumA vecuronium analog used to facilitate tracheal intubation and to relax skeletal muscles during surgery.
SuccinylcholineA depolarizing skeletal muscle relaxant used adjunctly to anesthesia and for skeletal muscle relaxation during intubation, mechanical ventilation, and surgical procedures.
TubocurarineTubocurarine is a non-depolarizing neuromuscular blocking agent and the first identified curare alkaloid. Curare is one of the names used to describe plant-derived poisons used by indigenous South Americans to...
VecuroniumA nondepolarizing neuromuscular blocking agent used to relax muscles or as an adjunct in general anesthesia during surgical procedures.
Drugs & Drug Targets
DrugTargetType
AlcuroniumNeuronal acetylcholine receptor subunit alpha-7target
AlcuroniumMuscarinic acetylcholine receptor M2target
AtracuriumHuman Carboxylesterasesenzyme
AtracuriumCholinesteraseenzyme
AtracuriumAcetylcholinesteraseenzyme
AtracuriumNeuronal acetylcholine receptor subunit alpha-7target
AtracuriumNeuronal Acetylcholine (nACh) Receptor Subunitstarget
AtracuriumMas-related G protein-coupled receptor member X2target
Atracurium besylateNeuronal acetylcholine receptor subunit alpha-2target
Botulinum toxin type AAlbumincarrier
Botulinum toxin type ARho-related GTP-binding protein RhoBtarget
Botulinum toxin type ASynaptosomal-associated protein 25target
CisatracuriumNeuronal Acetylcholine (nACh) Receptor Subunitstarget
CisatracuriumAcetylcholine receptor subunit alphatarget
CisatracuriumMuscarinic acetylcholine receptor M2target
CisatracuriumNeuronal acetylcholine receptor subunit alpha-2target
DaxibotulinumtoxinASynaptosomal-associated protein 25target
DecamethoniumAcetylcholine receptor subunit alphatarget
DecamethoniumNeuronal acetylcholine receptor subunit beta-2target
DecamethoniumNeuronal acetylcholine receptor subunit alpha-4target
DecamethoniumCholinesteraseenzyme
DecamethoniumNeuronal acetylcholine receptor subunit alpha-2target
DecamethoniumAcetylcholinesterasetarget
DoxacuriumNeuronal acetylcholine receptor subunit alpha-2target
DoxacuriumMuscarinic acetylcholine receptor M2target
DoxacuriumCholinesteraseenzyme
GallamineMuscle nicotinic acetylcholine receptortarget
GallamineAcetylcholinesterasetarget
GallamineMuscarinic acetylcholine receptor M2target
Gallamine triethiodideNeuronal acetylcholine receptor subunit alpha-2target
Gallamine triethiodideMuscarinic acetylcholine receptor M2target
Gallamine triethiodideAcetylcholinesterasetarget
Gallamine triethiodideMuscarinic acetylcholine receptor M1target
Gallamine triethiodideMuscarinic acetylcholine receptor M5target
LetibotulinumtoxinASynaptosomal-associated protein 25target
MetocurineMuscarinic acetylcholine receptor M2target
MetocurineNeuronal acetylcholine receptor subunit alpha-2target
Metocurine iodideNeuronal acetylcholine receptor subunit alpha-2target
Metocurine iodideNeuronal acetylcholine receptor subunit alpha-4target
Metocurine iodideNeuronal acetylcholine receptor subunit beta-2target
MivacuriumMuscarinic acetylcholine receptor M2target
MivacuriumNeuronal acetylcholine receptor subunit alpha-2target
MivacuriumMuscarinic acetylcholine receptor M3target
MivacuriumCholinesterasetarget
MivacuriumCholinesteraseenzyme
NeosaxitoxinSodium channel protein type 9 subunit alphatarget
NeosaxitoxinVoltage-gated sodium channel alpha subunittarget
PancuroniumMuscarinic acetylcholine receptor M3target
PancuroniumNeuronal acetylcholine receptor subunit alpha-2target
PancuroniumMuscarinic acetylcholine receptor M2target
PancuroniumCholinesteraseenzyme
PancuroniumSolute carrier family 22 member 2transporter
PancuroniumSolute carrier family 22 member 1transporter
PipecuroniumNeuronal acetylcholine receptor subunit alpha-2target
PipecuroniumMuscarinic acetylcholine receptor M2target
PipecuroniumMuscarinic acetylcholine receptor M3target
PipecuroniumCholinesteraseenzyme
PyrantelG protein-coupled receptor 35target
PyrantelMuscarinic acetylcholine receptor M1target
PyrantelCytochrome P450 4A11enzyme
RapacuroniumMuscarinic acetylcholine receptor M2target
RocuroniumSolute carrier organic anion transporter family member 1A2transporter
RocuroniumSolute carrier family 22 member 1transporter
Rocuronium5-hydroxytryptamine receptor 3Atarget
RocuroniumMuscarinic acetylcholine receptor M2target
RocuroniumNeuronal acetylcholine receptor subunit alpha-2target
SuccinylcholineCholinesteraseenzyme
SuccinylcholineNeuronal Acetylcholine (nACh) Receptor Subunitstarget
SuccinylcholineMuscarinic acetylcholine receptor M3target
SuccinylcholineMuscarinic acetylcholine receptor M2target
TubocurarineNeuronal acetylcholine receptor subunit alpha-7target
TubocurarineSolute carrier family 22 member 2transporter
TubocurarineSolute carrier family 22 member 1transporter
Tubocurarine5-hydroxytryptamine receptor 3Atarget
TubocurarineAcetylcholinesterasetarget
TubocurarineNeuronal acetylcholine receptor subunit alpha-2target
TubocurarineCholinesteraseenzyme
VecuroniumNeuronal acetylcholine receptor subunit alpha-2target
VecuroniumATP-dependent translocase ABCB1transporter