| DB00363 | Clozapine | approved | unknown | antagonist | Details |
| DB00246 | Ziprasidone | approved | unknown | antagonist | Details |
| DB00334 | Olanzapine | approved, investigational | unknown | antagonist | Details |
| DB00714 | Apomorphine | approved, investigational | yes | agonist | Details |
| DB00413 | Pramipexole | approved, investigational | yes | agonist | Details |
| DB00268 | Ropinirole | approved, investigational | unknown | agonist | Details |
| DB04908 | Flibanserin | approved, investigational | yes | antagonistagonist | Details |
| DB12061 | Pardoprunox | investigational | unknown | | Details |
| DB06216 | Asenapine | approved | unknown | antagonist | Details |
| DB06477 | Sumanirole | investigational | unknown | | Details |
| DB01186 | Pergolide | approved, investigational, vet_approved, withdrawn | yes | agonist | Details |
| DB01200 | Bromocriptine | approved, investigational, withdrawn | unknown | antagonist | Details |
| DB00589 | Lisuride | approved, investigational | yes | agonist | Details |
| DB00248 | Cabergoline | approved | unknown | agonist | Details |
| DB05271 | Rotigotine | approved | yes | agonist | Details |
| DB01267 | Paliperidone | approved | yes | antagonist | Details |
| DB01238 | Aripiprazole | approved, investigational | unknown | antagonistpartial agonist | Details |
| DB01224 | Quetiapine | approved | unknown | ligand | Details |
| DB01403 | Methotrimeprazine | approved, investigational | unknown | antagonist | Details |
| DB00409 | Remoxipride | approved, withdrawn | unknown | antagonist | Details |
| DB00988 | Dopamine | approved | yes | agonist | Details |
| DB01235 | Levodopa | approved | yes | agonist | Details |
| DB04946 | Iloperidone | approved | unknown | antagonist | Details |
| DB00477 | Chlorpromazine | approved, investigational, vet_approved | unknown | binder | Details |
| DB00408 | Loxapine | approved | unknown | binder | Details |
| DB00543 | Amoxapine | approved | unknown | antagonist | Details |
| DB08922 | Perospirone | experimental | unknown | antagonist | Details |
| DB09286 | Pipamperone | investigational | unknown | antagonist | Details |
| DB14185 | Aripiprazole lauroxil | approved, investigational | unknown | | Details |
| DB00490 | Buspirone | approved, investigational | unknown | antagonist | Details |
| DB00875 | Flupentixol | approved, investigational, withdrawn | unknown | antagonist | Details |
| DB00391 | Sulpiride | approved, investigational | unknown | antagonist | Details |
| DB00320 | Dihydroergotamine | approved, investigational | unknown | agonist | Details |