| DB00184 | Nicotine | approved | unknown | agonist | Details |
| DB00416 | Metocurine iodide | approved, withdrawn | yes | antagonist | Details |
| DB00483 | Gallamine triethiodide | approved | unknown | antagonist | Details |
| DB00657 | Mecamylamine | approved, investigational | yes | antagonist | Details |
| DB00728 | Rocuronium | approved | yes | antagonist | Details |
| DB00732 | Atracurium besylate | approved | yes | antagonist | Details |
| DB01135 | Doxacurium | approved | yes | antagonist | Details |
| DB01199 | Tubocurarine | approved | yes | antagonist | Details |
| DB01226 | Mivacurium | approved | yes | antagonist | Details |
| DB01245 | Decamethonium | approved | yes | partial agonist | Details |
| DB00411 | Carbamoylcholine | approved | yes | agonist | Details |
| DB00514 | Dextromethorphan | approved | unknown | antagonist | Details |
| DB01338 | Pipecuronium | approved | yes | antagonist | Details |
| DB01337 | Pancuronium | approved | yes | antagonist | Details |
| DB01336 | Metocurine | approved | yes | antagonist | Details |
| DB05740 | RPI-78M | investigational | unknown | | Details |
| DB00721 | Procaine | approved, investigational, vet_approved | unknown | antagonist | Details |
| DB01339 | Vecuronium | approved, investigational | yes | antagonist | Details |
| DB00898 | Ethanol | approved | unknown | | Details |
| DB07720 | Epibatidine | experimental | unknown | agonist | Details |
| DB08960 | Hexamethonium | experimental | yes | antagonist | Details |
| DB00472 | Fluoxetine | approved, vet_approved | unknown | antagonist | Details |