The Future of Drug Discovery: Tackling the Undruggable with New Biotechnologies
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Displaying targets
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Drug Name
Type
Name
target
enzyme
carrier
transporter
Clear
(21S)-1AZA-4,4-DIMETHYL-6,19-DIOXA-2,3,7,20-TETRAOXOBICYCLO[19.4.0] PENTACOSANE
target
Peptidyl-prolyl cis-trans isomerase FKBP1A
Details
4-[4-(4-Fluorophenyl)-2-[4-[(R)-methylsulfinyl]phenyl]-1H-imidazol-5-yl]pyridine
target
Mitogen-activated protein kinase 14
Details
4-[4-(4-Fluorophenyl)-2-[4-[(R)-methylsulfinyl]phenyl]-1H-imidazol-5-yl]pyridine
target
Mitogen-activated protein kinase 1
Details
4-(4-FLUOROPHENYL)-1-CYCLOROPROPYLMETHYL-5-(4-PYRIDYL)-IMIDAZOLE
target
Mitogen-activated protein kinase 14
Details
[HYDROXY(3-PHENYLPROPYL)AMINO]METHANOL
target
Peptide deformylase
Details
[HYDROXY(3-PHENYLPROPYL)AMINO]METHANOL
target
Peptide deformylase
Details
[HYDROXY(3-PHENYLPROPYL)AMINO]METHANOL
target
Peptide deformylase
Details
2-(3-BENZOYLPHENOXY)ETHYL(HYDROXY)FORMAMIDE
target
Peptide deformylase
Details
2-(3-BENZOYLPHENOXY)ETHYL(HYDROXY)FORMAMIDE
target
Peptide deformylase
Details
HYDROXY[3-(6-METHYLPYRIDIN-2-YL)PROPYL]FORMAMIDE
target
Peptide deformylase
Details
HYDROXY[3-(6-METHYLPYRIDIN-2-YL)PROPYL]FORMAMIDE
target
Peptide deformylase
Details
CARBOBENZYLOXY-(L)-LEUCINYL-(L)LEUCINYL METHOXYMETHYLKETONE
target
Pro-cathepsin H
Details
1-[4-(AMINOSULFONYL)PHENYL]-1,6-DIHYDROPYRAZOLO[3,4-E]INDAZOLE-3-CARBOXAMIDE
target
Cyclin-A2
Details
1-[4-(AMINOSULFONYL)PHENYL]-1,6-DIHYDROPYRAZOLO[3,4-E]INDAZOLE-3-CARBOXAMIDE
target
Cyclin-dependent kinase 2
Details
2-AMINO-6-(3,5-DIMETHYLPHENYL)SULFONYLBENZONITRILE
target
Gag-Pol polyprotein
Details
(6E,11E)-HEPTADECA-6,11-DIENE-9,9-DIYLBIS(PHOSPHONIC ACID)
target
Geranylgeranyl pyrophosphate synthase
Details
7-BENZYL-1,3-DIMETHYL-8-PIPERAZIN-1-YL-3,7-DIHYDRO-PURINE-2,6-DIONE
target
Dipeptidyl peptidase 4
Details
5-(2,3-dichlorophenyl)-N-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
target
Cyclin-dependent kinase 2
Details
6-(2-fluorophenyl)-N-(pyridin-3-ylmethyl)imidazo[1,2-a]pyrazin-8-amine
target
Cyclin-dependent kinase 2
Details
3-methyl-N-(pyridin-4-ylmethyl)imidazo[1,2-a]pyrazin-8-amine
target
Cyclin-dependent kinase 2
Details
5-(2-fluorophenyl)-N-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
target
Cyclin-dependent kinase 2
Details
3-bromo-5-phenyl-N-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
target
Cyclin-dependent kinase 2
Details
3-bromo-5-phenyl-N-(pyrimidin-5-ylmethyl)pyrazolo[1,5-a]pyridin-7-amine
target
Cyclin-dependent kinase 2
Details
3-bromo-6-phenyl-N-(pyrimidin-5-ylmethyl)imidazo[1,2-a]pyridin-8-amine
target
Cyclin-dependent kinase 2
Details
N-((2-aminopyrimidin-5-yl)methyl)-5-(2,6-difluorophenyl)-3-ethylpyrazolo[1,5-a]pyrimidin-7-amine
target
Cyclin-dependent kinase 2
Details
3-cyclopropyl-5-phenyl-N-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
target
Cyclin-dependent kinase 2
Details
2-[4-(2H-1,4-BENZOTHIAZINE-3-YL)-PIPERAZINE-1-LY]-1,3-THIAZOLE-4-CARBOXYLIC ACID ETHYLESTER
target
Genome polyprotein
Details
[(3S)-9-hydroxy-1-methyl-10-oxo-4,10-dihydro-3H-benzo[g]isochromen-3-yl]acetic acid
target
ActII protein
Details
3,4-dihydroxy-9,10-secoandrosta-1(10),2,4-triene-9,17-dione
target
Iron-dependent extradiol dioxygenase
Details
1-[2-HYDROXY-3-(4-CYCLOHEXYL-PHENOXY)-PROPYL]-4-(2-PYRIDYL)-PIPERAZINE
target
Genome polyprotein
Details
Displaying targets
23551 - 23580
of
33504
in total
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