| DB00535 | Cefdinir | approved | no | inhibitor | Details |
| DB01065 | Melatonin | approved, nutraceutical, vet_approved | unknown | inhibitor | Details |
| DB01065 | Melatonin | approved, nutraceutical, vet_approved | unknown | substrateinhibitor | Details |
| DB00250 | Dapsone | approved, investigational | unknown | substrate | Details |
| DB00208 | Ticlopidine | approved | unknown | substrate | Details |
| DB01225 | Enoxaparin | approved | unknown | other | Details |
| DB00583 | Levocarnitine | approved, investigational | unknown | | Details |
| DB04821 | Nomifensine | approved, withdrawn | unknown | | Details |
| DB00006 | Bivalirudin | approved, investigational | unknown | inhibitor | Details |
| DB02300 | Calcipotriol | approved | unknown | inhibitor | Details |
| DB06774 | Capsaicin | approved | unknown | inhibitor | Details |
| DB04827 | Urethane | approved, withdrawn | unknown | inducer | Details |
| DB06468 | Cariporide | investigational | unknown | inhibitor | Details |
| DB00833 | Cefaclor | approved | unknown | inducer | Details |
| DB00847 | Cysteamine | approved, investigational | unknown | substrate | Details |
| DB06111 | AB192 | experimental | unknown | inhibitor | Details |
| DB05161 | Elafin | investigational | unknown | inhibitor | Details |
| DB00461 | Nabumetone | approved | unknown | inhibitor | Details |
| DB00104 | Octreotide | approved, investigational | unknown | inhibitor | Details |
| DB00233 | Aminosalicylic acid | approved | unknown | inhibitor | Details |
| DB00515 | Cisplatin | approved | unknown | inducer | Details |
| DB00550 | Propylthiouracil | approved, investigational | unknown | inhibitor | Details |
| DB06823 | Tiopronin | approved, investigational | unknown | inhibitor | Details |
| DB00500 | Tolmetin | approved | unknown | inhibitor | Details |
| DB00958 | Carboplatin | approved | unknown | substrate | Details |
| DB00526 | Oxaliplatin | approved, investigational | unknown | substrate | Details |