Staurosporine

DB02010ExperimentalSmall molecule

An indolocarbazole that is a potent protein kinase C inhibitor which enhances cAMP-mediated responses in human neuroblastoma cells. (Biochem Biophys Res Commun 1995;214(3):1114-20).

Chemical structure of Staurosporine
Formula / weight
C28H26N4O3 · 466.531 g/mol (avg)
Code names
AM-2282 · CGP-39360

Resolves to

Clinical / RWD
Structure
InChIKeyHKSZLNNOFSGOKW-FYTWVXJKSA-NSMILES[H][C@]1(C[C@@]2([H])O[C@](C)(N3C4=CC=CC=C4C4=C5CNC(=O)C5=C5C6=CC=CC=C6N2C5=C34)[C@]1([H])OC)NC
Transporters

What you can answer from here — as of September 12, 2026

15Protein targetsEach mapped to UniProt, with action and pharmacological action
Listed above
1TransporterSubstrate / inhibitor direction, not just membership
Listed above
28+ReferencesStructured and connected to the statements they support
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