| DB00002 | Cetuximab | approved | yes | binder | Details |
| DB00317 | Gefitinib | approved, investigational | yes | antagonist | Details |
| DB00530 | Erlotinib | approved, investigational | yes | antagonist | Details |
| DB01259 | Lapatinib | approved, investigational | yes | antagonist | Details |
| DB01269 | Panitumumab | approved, investigational | yes | suppressor | Details |
| DB00281 | Lidocaine | approved, vet_approved | unknown | antagonist | Details |
| DB03496 | Alvocidib | experimental, investigational | unknown | | Details |
| DB04988 | IGN311 | investigational | unknown | | Details |
| DB05294 | Vandetanib | approved | unknown | inhibitor | Details |
| DB05374 | Rindopepimut | investigational | unknown | | Details |
| DB05101 | Matuzumab | investigational | unknown | | Details |
| DB05424 | Canertinib | investigational | unknown | | Details |
| DB05944 | Varlitinib | investigational | unknown | | Details |
| DB06021 | AV-412 | investigational | unknown | | Details |
| DB05524 | Pelitinib | investigational | unknown | | Details |
| DB07602 | S-{3-[(4-ANILINOQUINAZOLIN-6-YL)AMINO]-3-OXOPROPYL}-L-CYSTEINE | experimental | unknown | | Details |
| DB07662 | PD-168393 | experimental | unknown | | Details |
| DB08916 | Afatinib | approved | yes | inhibitor | Details |
| DB09559 | Necitumumab | approved, investigational | yes | antagonist | Details |
| DB09330 | Osimertinib | approved | yes | inhibitorregulator | Details |
| DB11737 | Icotinib | experimental, investigational | unknown | antagonist | Details |
| DB13164 | Olmutinib | investigational | yes | inhibitor | Details |
| DB12202 | Zalutumumab | investigational | yes | antagonist | Details |
| DB11731 | Depatuxizumab mafodotin | investigational | no | antibody | Details |
| DB11828 | Neratinib | approved, investigational | yes | inhibitor | Details |
| DB12267 | Brigatinib | approved, investigational | yes | inhibitor | Details |
| DB10772 | Foreskin keratinocyte (neonatal) | approved | yes | agonist | Details |
| DB12010 | Fostamatinib | approved, investigational | unknown | inhibitor | Details |
| DB11963 | Dacomitinib | approved, investigational | yes | inhibitor | Details |
| DB15035 | Zanubrutinib | approved, investigational | unknown | inhibitor | Details |
| DB15327 | Abivertinib | investigational | yes | inhibitor | Details |
| DB16695 | Amivantamab | approved, investigational | yes | antibodydownregulator | Details |
| DB16390 | Mobocertinib | approved, investigational | yes | inhibitor | Details |
| DB00530 | Erlotinib | approved, investigational | unknown | inhibitor | Details |
| DB12114 | Poziotinib | investigational | unknown | inhibitorbinder | Details |